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JAK
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Tyrphostin AG 490
CAS:133550-30-8
Formula:
C17H14N2O3
Purity:
>98.0%(T)(HPLC)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
294.31
Ref: 3B-T2962
1g | 778.00 € | ||
20mg | 47.00 € | ||
100mg | 131.00 € |
Estimated delivery in United States, on Friday 2 Aug 2024
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WHI-P154
CAS:211555-04-3
Formula:
C16H14BrN3O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
376.2047
Ref: AN-AG00BF57
1g | 589.00 € | ||
10mg | 55.00 € | ||
50mg | 143.00 € | ||
100mg | 172.00 € | ||
250mg | 274.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Ilginatinib hydrochloride
CAS:1239358-85-0
Ilginatinib hydrochloride (NS-018 hydrochloride) is a highly active and orally bioavailable inhibitor of JAK2.
Formula:
C21H21ClFN7
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
425.89
Ref: TM-T12266L2
1mg | 91.00 € | ||
1ml | 207.00 € | ||
5mg | 217.00 € | ||
10mg | 304.00 € | ||
25mg | 447.00 € | ||
50mg | 639.00 € | ||
100mg | 916.00 € | ||
500mg | 1,845.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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JAK2 Inhibitor V
CAS:195371-52-9
JAK2 Inhibitor V (JAK2 Inhibitor V Z3) is a novel specific inhibitor of Jak2, inhibiting …
Formula:
C23H24N2O
Purity:
99.15%
Color and Shape:
Solid
Molecular weight:
344.45
Ref: TM-T3042
1ml | 63.00 € | ||
2mg | 39.00 € | ||
5mg | 56.00 € | ||
10mg | 83.00 € | ||
25mg | 153.00 € | ||
50mg | 268.00 € | ||
100mg | 494.00 € | ||
500mg | 1,100.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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Ilginatinib
CAS:1239358-86-1
Ilginatinib (NS-018) is a highly active and orally bioavailable inhibitor of JAK2.
Formula:
C21H20FN7
Purity:
99.43%
Color and Shape:
Solid
Molecular weight:
389.43
Ref: TM-T12266
1mg | 93.00 € | ||
1ml | 213.00 € | ||
2mg | 133.00 € | ||
5mg | 218.00 € | ||
10mg | 303.00 € | ||
25mg | 444.00 € | ||
50mg | 639.00 € | ||
100mg | 916.00 € | ||
500mg | 1,838.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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Golidocitinib
CAS:2091134-68-6
Golidocitinib (AZD4205) is a selective JAK1 inhibitor (IC50: 73 nM) and weakly inhibits JAK2/JAK3 (IC50: …
Formula:
C25H31N9O2
Purity:
99.98%
Color and Shape:
Solid
Molecular weight:
489.57
Ref: TM-T10431
1ml | 168.00 € | ||
2mg | 94.00 € | ||
5mg | 160.00 € | ||
10mg | 262.00 € | ||
25mg | 457.00 € | ||
50mg | 605.00 € | ||
100mg | 861.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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Delgocitinib
CAS:1263774-59-9
Delgocitinib is a potent JAK inhibitor (IC50: 2.8-58 nM), treats inflammatory diseases, and is the …
Formula:
C16H18N6O
Purity:
99.90%
Color and Shape:
Solid
Molecular weight:
310.35
Ref: TM-T15096
1mg | 167.00 € | ||
1ml | 347.00 € | ||
5mg | 500.00 € | ||
10mg | 722.00 € | ||
25mg | 1,096.00 € | ||
50mg | 1,486.00 € | ||
100mg | 2,016.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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Brepocitinib P-Tosylate
CAS:2140301-96-6
Brepocitinib P-Tosylate (PF-06700841 P-Tosylate) is a potent dual inhibitor of Janus kinase 1 (JAK1) and …
Formula:
C25H29F2N7O4S
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
561.6
Ref: TM-T12427
1mg | 35.00 € | ||
1ml | 87.00 € | ||
5mg | 69.00 € | ||
10mg | 102.00 € | ||
25mg | 212.00 € | ||
50mg | 384.00 € | ||
100mg | 616.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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(E)-N-benzyl-2-cyano-3-(3,4-dihydroxyphenyl)prop-2-enamide
CAS:133550-30-8
Formula:
C17H14N2O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
294.3047
Ref: AN-AG0038YC
1g | 582.00 € | ||
10mg | 63.00 € | ||
20mg | 90.00 € | ||
50mg | 125.00 € | ||
250mg | 475.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Ilginatinib maleate
CAS:1354799-87-3
Ilginatinib maleate (NS-018 maleate) is a highly active and orally bioavailable inhibitor of JAK2.
Formula:
C25H24FN7O4
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
505.5
Ref: TM-T12266L
1mg | 93.00 € | ||
1ml | 245.00 € | ||
2mg | 134.00 € | ||
5mg | 217.00 € | ||
10mg | 303.00 € | ||
25mg | 444.00 € | ||
50mg | 642.00 € | ||
100mg | 917.00 € | ||
500mg | 1,839.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
Gusacitinib
CAS:1425381-60-7
Gusacitinib (ASN-002) (ASN-002) is spleen tyrosine kinase (SYK) and janus kinase (JAK) inhibitor (IC50: 5-46 …
Formula:
C24H28N8O2
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
460.53
Ref: TM-T14331
1mg | 47.00 € | ||
1ml | 116.00 € | ||
5mg | 94.00 € | ||
10mg | 121.00 € | ||
25mg | 185.00 € | ||
50mg | 343.00 € | ||
100mg | 510.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
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4-(3'-HYDROXYPHENYL)AMINO-6,7-DIMETHOXYQUINAZOLINE, HCL
CAS:153437-55-9
Formula:
C16H16ClN3O3
Purity:
≥97.0%
Molecular weight:
333.7695
Ref: AN-AG00AB8Z
5mg | 113.00 € | ||
10mg | 158.00 € | ||
25mg | 311.00 € | ||
50mg | 495.00 € | ||
100mg | To inquire |
Estimated delivery in United States, on Friday 9 Aug 2024
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JAK1-IN-11
CAS:2427608-43-1
JAK1-IN-11 (compound 11) serves as a potent inhibitor of Janus kinases, exhibiting nanomolar inhibitory concentrations …
Formula:
C26H36N6O4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
528.67
Ref: TM-T79079
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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Povorcitinib phosphate
CAS:1637677-33-8
Povorcitinib phosphate is a selective JAK1 inhibitor and can be used in studies about the …
Formula:
C23H25F5N7O5P
Purity:
97.71%
Color and Shape:
Solid
Molecular weight:
605.45
Ref: TM-T39113L
1mg | 95.00 € | ||
1ml | 313.00 € | ||
5mg | 231.00 € | ||
10mg | 346.00 € | ||
25mg | 587.00 € | ||
50mg | 833.00 € | ||
100mg | 1,133.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
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JAK-IN-25
CAS:2127110-22-7
JAK-IN-25 (compound 19), a potent JAK inhibitor, exhibits IC50 values of 6 nM for TYK2, …
Formula:
C19H17N5O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
379.37
Ref: TM-T78175
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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JAK-IN-27
CAS:2673176-36-6
JAK-IN-27, also known as compound 1, is an orally active, potent inhibitor of the JAKS …
Formula:
C20H21F2N7O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
413.42
Ref: TM-T79110
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
JAK kinase-IN-1
CAS:2698389-43-2
JAK kinase-IN-1 (Example 1) functions as a potent inhibitor targeting the JAK family, which includes …
Formula:
C17H19F2N7OS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
407.44
Ref: TM-T79807
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
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JAK/HDAC-IN-2
JAK/HDAC-IN-2, a potent 2-amino-4-phenylaminopyrimidine dual-target inhibitor, effectively suppresses JAK1/2 and HDAC3/6 at nanomolar concentrations.
Formula:
C28H38N6O5S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
570.7
Ref: TM-T78708
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Monday 12 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
WDR5-IN-6
CAS:326901-92-2
WDR5-IN-6 is a WDR5 inhibitor targeting the WBM locus.WDR5-IN-6 is highly synergistic with OICR-9429, a …
Formula:
C13H8Cl2N2O2S
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
327.19
Ref: TM-T77495
1mg | 45.00 € | ||
5mg | 96.00 € | ||
10mg | 142.00 € | ||
25mg | 275.00 € | ||
50mg | 447.00 € | ||
100mg | 708.00 € | ||
500mg | 1,439.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024
![discount label](https://static.cymitquimica.com/public/img/discount.png)
TAK-901
CAS:934541-31-8
TAK-901 has been used in trials studying the treatment of Lymphoma, Myelofibrosis, Multiple Myeloma, Myeloid …
Formula:
C28H32N4O3S
Purity:
99.1%
Color and Shape:
Solid
Molecular weight:
504.64
Ref: TM-T2709
5mg | 76.00 € | ||
25mg | 209.00 € | ||
50mg | 363.00 € |
Estimated delivery in United States, on Monday 12 Aug 2024