JAK
JAK (Janus kinase) inhibitors are compounds that target the JAK-STAT signaling pathway, which is involved in cell growth, immune response, and angiogenesis. By inhibiting JAK, these compounds can reduce the signaling that leads to the formation of new blood vessels in tumors, thereby inhibiting tumor growth. JAK inhibitors are important in the treatment of cancers and inflammatory diseases. At CymitQuimica, we offer a diverse range of high-quality JAK inhibitors to support your research in oncology, immunology, and angiogenesis.
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Gusacitinib
CAS:1425381-60-7
Gusacitinib (ASN-002) (ASN-002) is spleen tyrosine kinase (SYK) and janus kinase (JAK) inhibitor (IC50: 5-46 …
Formula:
C24H28N8O2
Purity:
98.06% - 99.94%
Color and Shape:
Solid
Molecular weight:
460.53
Ref: TM-T14331
| 1mg | 42.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 188.00 € | ||
| 50mg | 350.00 € | ||
| 100mg | 522.00 € | ||
| 200mg | 750.00 € | ||
| 1mL*10mM (DMSO) | 116.00 € |
Estimated delivery in United States, on Monday 7 Jul 2025
Ilginatinib
CAS:1239358-86-1
Ilginatinib (NS-018) is a highly active and orally bioavailable inhibitor of JAK2.
Formula:
C21H20FN7
Purity:
98.4% - 99.01%
Color and Shape:
Solid
Molecular weight:
389.43
Ref: TM-T12266
| 1mg | 64.00 € | ||
| 5mg | 138.00 € | ||
| 10mg | 187.00 € | ||
| 25mg | 273.00 € | ||
| 50mg | 393.00 € | ||
| 100mg | 562.00 € | ||
| 200mg | 743.00 € | ||
| 1mL*10mM (DMSO) | 133.00 € |
Estimated delivery in United States, on Monday 7 Jul 2025
Golidocitinib
CAS:2091134-68-6
Golidocitinib (AZD4205) is a selective JAK1 inhibitor (IC50: 73 nM) and weakly inhibits JAK2/JAK3 (IC50: …
Formula:
C25H31N9O2
Purity:
98.87% - 99.88%
Color and Shape:
Solid
Molecular weight:
489.57
Ref: TM-T10431
| 2mg | 96.00 € | ||
| 5mg | 163.00 € | ||
| 10mg | 268.00 € | ||
| 25mg | 465.00 € | ||
| 50mg | 618.00 € | ||
| 100mg | 880.00 € | ||
| 1mL*10mM (DMSO) | 170.00 € |
Estimated delivery in United States, on Monday 7 Jul 2025
Delgocitinib
CAS:1263774-59-9
Delgocitinib is a potent JAK inhibitor (IC50: 2.8-58 nM), treats inflammatory diseases, and is the …
Formula:
C16H18N6O
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
310.35
Ref: TM-T15096
| 1mg | 169.00 € | ||
| 5mg | 311.00 € | ||
| 10mg | 487.00 € | ||
| 25mg | 929.00 € | ||
| 50mg | 1,415.00 € | ||
| 100mg | 2,062.00 € | ||
| 200mg | 2,775.00 € | ||
| 1mL*10mM (DMSO) | 349.00 € |
Estimated delivery in United States, on Monday 7 Jul 2025
Ilginatinib hydrochloride
CAS:1239358-85-0
Ilginatinib hydrochloride (NS-018 hydrochloride) is a highly active and orally bioavailable inhibitor of JAK2.
Formula:
C21H21ClFN7
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
425.89
Ref: TM-T12266L2
| 1mg | 77.00 € | ||
| 5mg | 165.00 € | ||
| 10mg | 240.00 € | ||
| 25mg | 408.00 € | ||
| 50mg | 562.00 € | ||
| 100mg | 800.00 € | ||
| 200mg | 1,074.00 € | ||
| 1mL*10mM (DMSO) | 177.00 € |
Estimated delivery in United States, on Monday 7 Jul 2025
Ilginatinib maleate
CAS:1354799-87-3
Ilginatinib maleate (NS-018 maleate) is a highly active and orally bioavailable inhibitor of JAK2.
Formula:
C25H24FN7O4
Purity:
99.74% - 99.82%
Color and Shape:
Solid
Molecular weight:
505.5
Ref: TM-T12266L
| 1mg | 64.00 € | ||
| 5mg | 138.00 € | ||
| 10mg | 187.00 € | ||
| 25mg | 273.00 € | ||
| 50mg | 393.00 € | ||
| 100mg | 562.00 € | ||
| 200mg | 743.00 € | ||
| 1mL*10mM (DMSO) | 153.00 € |
Estimated delivery in United States, on Monday 7 Jul 2025
JAK2 Inhibitor V
CAS:195371-52-9
JAK2 Inhibitor V (JAK2 Inhibitor V Z3) is a novel specific inhibitor of Jak2, inhibiting …
Formula:
C23H24N2O
Purity:
98.36% - 99.15%
Color and Shape:
Solid
Molecular weight:
344.45
Ref: TM-T3042
| 2mg | 39.00 € | ||
| 5mg | 57.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 157.00 € | ||
| 50mg | 274.00 € | ||
| 100mg | 505.00 € | ||
| 500mg | 1,121.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Monday 7 Jul 2025
WHI-P154
CAS:211555-04-3
Formula:
C16H14BrN3O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
376.2047
Ref: IN-DA00BF57
| 1g | 597.00 € | ||
| 10mg | 68.00 € | ||
| 50mg | 118.00 € | ||
| 100mg | 187.00 € | ||
| 250mg | 224.00 € |
Estimated delivery in United States, on Monday 7 Jul 2025
Brepocitinib P-Tosylate
CAS:2140301-96-6
Brepocitinib P-Tosylate (PF-06700841 P-Tosylate) is a potent dual inhibitor of Janus kinase 1 (JAK1) and …
Formula:
C25H29F2N7O4S
Purity:
99.82% - 99.97%
Color and Shape:
Solid
Molecular weight:
561.6
Ref: TM-T12427
| 1mg | 35.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 104.00 € | ||
| 25mg | 216.00 € | ||
| 50mg | 393.00 € | ||
| 100mg | 628.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Monday 7 Jul 2025
(E)-N-Benzyl-2-cyano-3-(3,4-dihydroxyphenyl)acrylamide；AG 490
CAS:133550-30-8
Formula:
C17H14N2O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
294.3047
Ref: IN-DA0038YC
| 1g | 510.00 € | ||
| 10mg | 64.00 € | ||
| 20mg | 91.00 € | ||
| 50mg | 120.00 € | ||
| 250mg | 305.00 € |
Estimated delivery in United States, on Monday 7 Jul 2025
Tyk2-IN-22
CAS:933667-23-3
Tyk2-IN-22 (Compound A8) is a selective inhibitor of tyrosine kinase 2 (Tyk2), effectively inhibiting Tyk2, …
Formula:
C16H16ClN5O2
Color and Shape:
Solid
Molecular weight:
345.78
Ref: TM-T203504
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Jul 2025
TAK-901
CAS:934541-31-8
TAK-901 has been used in trials studying the treatment of Lymphoma, Myelofibrosis, Multiple Myeloma, Myeloid …
Formula:
C28H32N4O3S
Purity:
99.02% - 99.59%
Color and Shape:
Solid
Molecular weight:
504.64
Ref: TM-T2709
| 5mg | 72.00 € | ||
| 25mg | 213.00 € | ||
| 50mg | 371.00 € |
Estimated delivery in United States, on Tuesday 8 Jul 2025
WDR5-IN-6
CAS:326901-92-2
WDR5-IN-6 is a WDR5 inhibitor targeting the WBM locus.WDR5-IN-6 is highly synergistic with OICR-9429, a …
Formula:
C13H8Cl2N2O2S
Purity:
99.69%
Color and Shape:
Soild
Molecular weight:
327.19
Ref: TM-T77495
| 1mg | 46.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 144.00 € | ||
| 25mg | 281.00 € | ||
| 50mg | 454.00 € | ||
| 100mg | 725.00 € | ||
| 500mg | 1,473.00 € |
Estimated delivery in United States, on Tuesday 8 Jul 2025
Nimucitinib
CAS:2740557-24-6
Nimucitinib is a Janus kinase (JAK) inhibitor that can be used to treat dry eye …
Formula:
C25H26F2N6O2
Purity:
98.71%
Color and Shape:
Soild
Molecular weight:
480.51
Ref: TM-T67907
| 1mg | 96.00 € | ||
| 2mg | 139.00 € | ||
| 5mg | 227.00 € | ||
| 10mg | 354.00 € | ||
| 25mg | 653.00 € | ||
| 50mg | 938.00 € | ||
| 100mg | 1,454.00 € | ||
| 500mg | 2,822.00 € |
Estimated delivery in United States, on Tuesday 8 Jul 2025
JAK3-IN-15
JAK3-IN-15 (compound 22) is a JAK3 inhibitor that reduces the secretion of p-JAK3 induced by …
Color and Shape:
Odour Solid
Ref: TM-T200631
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Jul 2025
JAK2-IN-6
CAS:353512-04-6
JAK2-IN-6: A potent JAK2-specific inhibitor (IC50=22.86μg/mL), blocks JAK2 signaling, has anticancer properties, and is inactive …
Formula:
C14H10ClN3OS2
Purity:
99.38%
Color and Shape:
Solid
Molecular weight:
335.83
Ref: TM-T40443
| 1mg | 38.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 188.00 € | ||
| 50mg | 281.00 € | ||
| 100mg | 426.00 € | ||
| 200mg | 617.00 € |
Estimated delivery in United States, on Tuesday 8 Jul 2025
JAK-IN-33
JAK-IN-33 (Compound 3 (R)) is a selective inhibitor of the Janus kinase (JAK) family [1].
Purity:
98%
Color and Shape:
Odour Solid
Ref: TM-T82018
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Jul 2025
JAK/HDAC-IN-4
JAK/HDAC-IN-4 (compound 11 i) is a dual inhibitor targeting both JAK2 and HDAC6, with IC50 …
Formula:
C30H32N8O5S
Color and Shape:
Solid
Molecular weight:
616.69
Ref: TM-T201233
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Jul 2025
JAK1/STAT3-IN-1
JAK1/STAT3-IN-1 (compound 4f) functions as an anti-atopic dermatitis (AD) agent by inhibiting the JAK1/STAT3 signaling …
Formula:
C30H33FN4O3S
Color and Shape:
Solid
Molecular weight:
548.67
Ref: TM-T205385
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Jul 2025
Povorcitinib phosphate
CAS:1637677-33-8
Povorcitinib phosphate is a selective JAK1 inhibitor and can be used in studies about the …
Formula:
C23H25F5N7O5P
Purity:
99.57%
Color and Shape:
Solid
Molecular weight:
605.45
Ref: TM-T39113L
| 1mg | 65.00 € | ||
| 2mg | 95.00 € | ||
| 5mg | 145.00 € | ||
| 10mg | 212.00 € | ||
| 25mg | 359.00 € | ||
| 50mg | 512.00 € | ||
| 100mg | 695.00 € | ||
| 200mg | 937.00 € |
Estimated delivery in United States, on Tuesday 8 Jul 2025
