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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2280 products of "Membrane Transporter/Ion Channel"

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  • 264W94

    CAS:
    <p>264W94 robustly inhibits IBAT, induces CYP7A1, and significantly reduces cholesterol.</p>
    Formula:C23H31NO4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:417.56
  • URAT1 inhibitor 3


    <p>URAT1 inhibitor 3: potent oral URAT1 blocker, IC50=0.8 nM, for gout/hyperuricemia study.</p>
    Formula:C14H8Cl2N2O2
    Color and Shape:Solid
    Molecular weight:307.13
  • NMD670

    CAS:
    <p>NMD670 is an orally active, partial inhibitor of the skeletal muscle-specific chloride channel ClC-1. It enhances muscle excitability and neuromuscular transmission, restoring muscle function and mobility. NMD670 has a favorable safety profile and improves muscle function in rats, particularly in an MG rat model [1].</p>
    Formula:C12H10BrNO4
    Color and Shape:Solid
    Molecular weight:312.12
  • ML-SI1

    CAS:
    <p>ML-SI1, a racemic mixture of diastereoisomers, is a TRPML inhibitor and acts on TRPML1 (IC50: 15 μM).</p>
    Formula:C23H26Cl2N2O3
    Color and Shape:Solid
    Molecular weight:449.37
  • Unoprostone

    CAS:
    <p>Unoprostone is a prostaglandin F2α analogs (PGAs), and reduces intraocular pressure and is used topically for glaucoma or ocular hypertension.</p>
    Formula:C22H38O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:382.53
  • Blixeprodil

    CAS:
    <p>Blixeprodil (GM-1020) is an orally active NMDA receptor antagonist with an affinity of Ki = 3.25 µM in rat cortical tissue. It inhibits NR1/2A-NMDAR-mediated currents in HEK293 cells with an IC50 of 1.192 µM. Blixeprodil demonstrates antidepressant effects in rat models and exhibits blood-brain barrier permeability.</p>
    Formula:C13H16FNO
    Color and Shape:Solid
    Molecular weight:221.271
  • Insecticidal agent 21

    CAS:
    <p>Insecticidal agent 21 (Compound 6) is an insecticide targeting Culex pipiens larvae with an LC50 of 0.4 μg/mL. It achieves multi-target neurotoxicity by inhibiting acetylcholinesterase (AChE) and simultaneously targeting other neural receptors, including nicotinic acetylcholine receptors (nAChR), voltage-gated sodium channels (VGSC), and γ-aminobutyric acid receptors (GABAAR). Insecticidal agent 21 shows potent insecticidal activity and can be utilized in the development of new insecticides to combat mosquito resistance to conventional agents.</p>
    Formula:C37H40ClN3O2
    Color and Shape:Solid
    Molecular weight:594.185
  • Cav 3.2 inhibitor 1


    <p>Cav 3.2 inhibitor 1 targets T-type calcium channels, weakly binds D2 receptors, and aids physical and visceral pain research.</p>
    Formula:C32H39N3O
    Color and Shape:Solid
    Molecular weight:481.67
  • SC-435 mesylate

    CAS:
    <p>SC-435 is an ileal apical sodium co-dependent bile acid transporter (ASBT). SC-435 inhibits plasma cholesterol.</p>
    Formula:C37H59N3O7S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:722.01
  • EF1502 free base

    CAS:
    <p>EF1502 is a potent and selective GABA transporter inhibitor.</p>
    Formula:C22H26N2O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:414.58
  • V-ATPase-IN-1

    CAS:
    <p>V-ATPase-IN-1 (Compound 3b-03) is an inhibitor of Vacuolar-type H+-ATPases (V-ATPase), exhibiting an inhibition constant (IC50) of 194.80 μM and effectively targeting the V-ATPase subunit A with a dissociation constant (Kd) of 0.803 μM. This compound demonstrates insecticidal activity against M. separata (LC50 = 2.64 mM), aiding in the development of chemical insecticides.</p>
    Formula:C21H20ClNO2
    Color and Shape:Solid
    Molecular weight:353.84
  • ABCG2-IN-4

    CAS:
    <p>ABCG2-IN-4 (Compound K31) is an orally active ABCG2 inhibitor that reduces the release of Protoporphyrin IX (PPIX) from red blood cells into the plasma and prevents phototoxicity. In mouse models, ABCG2-IN-4 also demonstrates anti-inflammatory and antioxidant properties.</p>
    Formula:C24H32N4O4
    Color and Shape:Solid
    Molecular weight:440.535
  • P-gp/BCRP-IN-1

    CAS:
    <p>P-gp/BCRP-IN-1, safe and oral, inhibits P-gp/BCRP transporters, enhancing Paclitaxel bioavailability.</p>
    Formula:C27H25ClN4O3
    Color and Shape:Solid
    Molecular weight:488.97
  • Olorigliflozin

    CAS:
    <p>Olorigliflozin is a sodium glucose co-transporter (SGLT) inhibitor with antihyperglycemic properties.</p>
    Formula:C23H27ClO7
    Color and Shape:Solid
    Molecular weight:450.909
  • ARN23765

    CAS:
    <p>ARN23765 is an F508del-CFTR corrector with an EC50 of 38 pM in human bronchial epithelial cells. It enhances the maturation and function of F508del-CFTR at the cell membrane, influencing ion transport and secretion, thereby addressing the pathological mechanisms of cystic fibrosis (CF).</p>
    Formula:C30H22F5N3O6
    Color and Shape:Solid
    Molecular weight:615.504
  • Dehydelone

    CAS:
    <p>Dehydelone(KOS-1584, R-1645, SK-10088) is a microtubule stabilizer that may be used in the treatment of non-small cell lung cancer.</p>
    Formula:C27H39NO5S
    Color and Shape:Solid
    Molecular weight:489.67
  • ATPase-IN-5

    CAS:
    <p>ATPase-IN-5 (Compound 11) is an antifungal Pma1p (H+ -ATPase) inhibitor (IC50 = 12.7 μM) that inhibits the growth of Candida albicans and Saccharomyces cerevisiae.</p>
    Formula:C10H10N4O3S
    Purity:99.19%
    Color and Shape:Solid
    Molecular weight:266.28
  • (S)-Albuterol

    CAS:
    <p>(S)-Albuterol functions as a muscarinic receptor and phospholipase C activator, enhancing the intracellular free calcium concentration in airway smooth muscle cells.</p>
    Formula:C13H21NO3
    Color and Shape:Solid
    Molecular weight:239.311
  • P-gp modulator 3


    <p>P-gp modulator 3 (Compound 37) is a potent, competitive, metabotropic P-glycoprotein (P-gp) modulator.</p>
    Formula:C31H37N3O5
    Color and Shape:Solid
    Molecular weight:531.64
  • Pyrimidinone 8

    CAS:
    <p>Pyrimidinone 8 is a reversible, linear non-competitive inhibitor of divalent metal transporter 1 (DMT1) with a Ki of 20 μM (hDMT1). It does not affect the surface expression of hDMT1 and is not influenced by extracellular pH. Pyrimidinone 8 inhibits hDMT1-mediated iron uptake, with an IC50 of 13.8 μM.</p>
    Formula:C10H12N4O
    Color and Shape:Solid
    Molecular weight:204.229
  • NYX-2925

    CAS:
    <p>NYX-2925, an oral NMDAR modulator, enhances Src in mPFC. No CAMKII impact or addictive/sedative effects. Useful for CNS disorder studies.</p>
    Formula:C14H23N3O4
    Color and Shape:Solid
    Molecular weight:297.35
  • Opakalim

    CAS:
    <p>Opakalim is an activator of potassium channels (potassium channel) and exhibits anticonvulsant activity.</p>
    Formula:C18H22F2N4O
    Color and Shape:Solid
    Molecular weight:348.39
  • GABA-IN-4

    CAS:
    <p>GABA-IN-4 (Compound 17) is a derivative of N-(indol-3-ylglyoxylyl)benzylamine. It exhibits high affinity for the benzodiazepine receptor (BzR), the binding site within the GABAA receptor complex, with a Ki value of 67 nM. Benzodiazepines are widely used as anxiolytic, sedative-hypnotic, and anticonvulsant agents.</p>
    Formula:C17H13ClN2O2
    Color and Shape:Solid
    Molecular weight:312.75
  • CRM1-IN-3

    CAS:
    <p>CRM1-IN-3 (B28), a noncovalent inhibitor of CRM1, is utilized in the research of protein localization and tumor studies [1].</p>
    Formula:C26H26ClN3O3
    Color and Shape:Solid
    Molecular weight:463.96
  • Suloctidil HCl

    CAS:
    <p>Suloctidil HCl is a peripheral vascular dilator.</p>
    Formula:C20H36ClNOS
    Color and Shape:Solid
    Molecular weight:374.02
  • Sp-8-Br-cGMPS

    CAS:
    <p>Sp-8-Br-cGMPS, an analogue of cGMP, acts as an agonist for cGMP gated cation channels (CNG channels) with an EC50 of 106.5 μM. While Sp-8-Br-cGMPS can induce currents, it does not stabilize channel open states as effectively as a full agonist.</p>
    Formula:C10H11BrN5O6PS
    Color and Shape:Solid
    Molecular weight:440.17
  • 3-Bromoamphetamine hydrochloride

    CAS:
    <p>3-Bromoamphetamine hydrochloride is a para-substituted amphetamine that functions as a monoamine releaser.</p>
    Formula:C9H13BrClN
    Color and Shape:Solid
    Molecular weight:250.563
  • (2S,3S,11bR)-Dihydrotetrabenazine

    CAS:
    <p>(2S,3S,11bR)-Dihydrotetrabenazine ((2S,3S,11bR)-DHTBZ) is a highly selective inhibitor of vesicular monoamine transporter 2 (VMAT2) with a Ki value of 593 nM. It suppresses the vesicular transport of monoamine neurotransmitters, such as dopamine and serotonin, leading to reduced release into the synaptic cleft. This compound holds potential for research in Huntington's disease and other hyperkinetic movement disorders.</p>
    Formula:C19H29NO3
    Color and Shape:Solid
    Molecular weight:319.44
  • Zilvetrigine

    CAS:
    <p>Zilvetrigine is a sodium channel (sodium channel) blocker. It can be used as an analgesic.</p>
    Formula:C20H20ClN3O2
    Color and Shape:Solid
    Molecular weight:369.845
  • NMDA agonist 1

    CAS:
    <p>NMDA agonist 1 (compound 42d) is a potent NMDA agonist with a Ki value of 96 nM. It acts as a partial agonist of the GluN1/GluN2B complex, exhibiting an EC50 value of 78 nM.</p>
    Formula:C12H13N3O3S
    Color and Shape:Solid
    Molecular weight:279.315
  • Tamitinol

    CAS:
    <p>Tamitinol is a neurotropic drug. It has been found to help symptoms of obsessive rumination in conjunction with maprotiline.</p>
    Formula:C12H20N2OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:240.37
  • Cav 3.2 inhibitor 2


    <p>Cav 3.2 inhibitor 2 blocks T-type Ca2+ channels (IC50=0.09339 μM) and reduces mouse somatic/visceral pain. Used for intractable pain studies.</p>
    Formula:C32H37F2N3O
    Color and Shape:Solid
    Molecular weight:517.65
  • KCa2 channel modulator 2


    Compound 2q is a potent, subtype-selective K/Ca 2 modulator, effective on human K Ca 2.3 and rat K Ca 2.2a with EC50s of 0.60 μM and 0.64 μM.
    Formula:C16H15ClFN5
    Color and Shape:Solid
    Molecular weight:331.78
  • PDE1-IN-4


    <p>PDE1-IN-4: inhibits PDE1C/A/B with IC50s 10/145/354 nM, may help study idiopathic pulmonary fibrosis.</p>
    Formula:C33H33N3O4
    Color and Shape:Solid
    Molecular weight:535.63
  • GABAA receptor agonist 2


    <p>Compound 4c, a potent GABAA agonist with anti-depressive effects in mouse FST/TST, shows promise in depression research.</p>
    Formula:C22H36O5
    Color and Shape:Solid
    Molecular weight:380.52
  • YY-23

    CAS:
    <p>YY-23 is a selective NMDAR (containing GluN2C or GluN2D) inhibitor. By inhibiting NMDARs with GluN2D on GABAergic interneurons in the prefrontal cortex, YY-23 suppresses GABAergic neurotransmission and enhances excitatory transmission. YY-23 exhibits antidepressant activity and is useful for neurological disease research.</p>
    Formula:C33H54O8
    Color and Shape:Solid
    Molecular weight:578.777
  • S-8510 phosphate

    CAS:
    <p>S-8510 phosphate is an agonist of inverse Benzodiazepine (BDZ) receptor(Kis of 34.6 nM, 36.2 nM for –GABA and +GABA respectively).</p>
    Formula:C12H13N4O6P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:340.23
  • Leualacin

    CAS:
    <p>Leualacin is a novel calcium blocker from Hapsidospora irregularis.</p>
    Formula:C31H47N3O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:573.72
  • Antidepressant agent 9

    CAS:
    <p>Antidepressant agent 9 (Compound 24) is an orally active inhibitor of NMDAR and SERT, with IC50 values of 3.50 μM and 1044 nM, respectively. It exhibits good metabolic stability and plasma exposure, and demonstrates antidepressant-like effects in the forced swim test in mice.</p>
    Formula:C17H24N2
    Color and Shape:Solid
    Molecular weight:256.386
  • Suzetrigine

    CAS:
    <p>Suzetrigine (VX-548) is an oral NaV1.8 inhibitor with analgesic properties for acute pain research.</p>
    Formula:C21H20F5N3O4
    Purity:98.08% - 99.27%
    Color and Shape:Solid
    Molecular weight:473.39
  • (+)-Tetrabenazine

    CAS:
    <p>(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-fold</p>
    Formula:C19H27NO3
    Purity:98.31%
    Color and Shape:Solid
    Molecular weight:317.42
  • SYM2206

    CAS:
    <p>SYM2206 is a low affinity non-competitive AMPA receptor antagonist with an IC50 value of 1.6 μM.SYM2206 exhibits anticancer activity by blocking Nav1.6-mediated</p>
    Formula:C20H22N4O3
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:366.41
  • Odevixibat

    CAS:
    <p>Odevixibat (A4250) is a selective oral inhibitor for ileal bile acid transport, potentially treating primary biliary cirrhosis.</p>
    Formula:C37H48N4O8S2
    Purity:99.53% - 99.83%
    Color and Shape:Solid
    Molecular weight:740.93
  • SDZ 220-040

    CAS:
    <p>SDZ 220-040 是一种选择性哺乳动物 NMDA 受体拮抗剂,可诱导根系生长的部分无重力模式 。</p>
    Formula:C16H16Cl2NO6P
    Purity:98.13%
    Color and Shape:Solid
    Molecular weight:420.18
  • Umbellulone

    CAS:
    <p>Umbellulone is a natural product isolated from Umbellularia californica, and stimulates the TRPA1 channel in a subset of peptidergic, nociceptive neurons, activating the trigeminovascular system via this mechanism.</p>
    Formula:C10H14O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:150.22

    Ref: TM-T13953

    1mg
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  • 5-Hydroxylansoprazole

    CAS:
    <p>5-Hydroxylansoprazole (AG1908) is the active metabolite of plasma Lansoprazole, inhibits the proton pump, and is used in the study of peptic ulcers.</p>
    Formula:C16H14F3N3O3S
    Purity:99.00%
    Color and Shape:Solid
    Molecular weight:385.36

    Ref: TM-T14051

    1mg
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  • (-)-Bicuculline methobromide

    CAS:
    <p>(-)-Bicuculline methobromide is a potent antagonist of GABAA receptor .</p>
    Formula:C21H20BrNO6
    Color and Shape:White
    Molecular weight:462.29

    Ref: TM-T12043

    1mg
    Discontinued
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  • A-887826

    CAS:
    <p>A-887826 is a selective, orally bioavailable, and voltage-dependent Na(v1.8) channel blocker (IC50: 11 nM). It attenuates neuropathic tactile allodynia in vivo.</p>
    Formula:C26H29ClN4O3
    Color and Shape:Solid
    Molecular weight:480.99

    Ref: TM-T10209

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  • Indapamide

    CAS:
    <p>Indapamide (Noranat) is a non-thiazide sulphonamide diuretic compound, generally used in the treatment of hypertension, as well as decompensated cardiac failure.</p>
    Formula:C16H16ClN3O3S
    Purity:98.97% - 99.83%
    Color and Shape:Solid
    Molecular weight:365.83

    Ref: TM-T1498

    1g
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  • Dexivacaine

    CAS:
    Dexivacaine is an type of anesthetic.
    Formula:C15H22N2O
    Color and Shape:Solid
    Molecular weight:246.35

    Ref: TM-T31400

    ne
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  • Verapamil EP Impurity C hydrochloride

    CAS:
    <p>NSC-609249 hydrochloride, an impurity of Verapamil, is a calcium channel blocker with potent orally active properties. It also functions as a first-generation P-glycoprotein (P-gp) inhibitor.</p>
    Formula:C12H20ClNO2
    Color and Shape:Solid
    Molecular weight:245.75

    Ref: TM-T40591

    ne
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  • Zastaprazan

    CAS:
    <p>Zastaprazan (JP-1366, compound 6) is a potassium-competitive acid blocker and proton pump inhibitor that suppresses gastric acid secretion, indicated for GERD.</p>
    Formula:C22H26N4O
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:362.48

    Ref: TM-T39583

    ne
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  • L-Cysteine S-sulfate sodium salt sesquihydrate

    CAS:
    <p>L-Cysteine S-sulfate sodium salt sesquihydrate is a useful organic compound for research related to life sciences. The catalog number is T64782 and the CAS number is 150465-29-5.</p>
    Formula:C9H25N3Na3O17S6
    Color and Shape:Solid
    Molecular weight:708.63

    Ref: TM-T64782

    ne
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  • GNE-9278

    CAS:
    <p>GNE-9278 is a highly selective NMDAR orthosteric modulator that targets the GluN1 transmembrane structural domain (TMD), enhancing peak current and agonist affinity in activated NMDAR.</p>
    Formula:C21H27N5O3S
    Color and Shape:Solid
    Molecular weight:429.54

    Ref: TM-T62376

    ne
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  • PF-06761281

    CAS:
    <p>PF-06761281 is a partially selective sodium-coupled citrate transporter protein (NaCT/SLC13A5) inhibitor, oral, reducing plasma glucose concentration.</p>
    Formula:C13H17NO6
    Color and Shape:Solid
    Molecular weight:283.28

    Ref: TM-T60547

    ne
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  • 3-Methylglutaconic acid

    CAS:
    <p>3-Methylglutaconic acid, a primary metabolite accumulating in 3-Methylglutaconic aciduria (MGTA), induces lipid and protein oxidation, while diminishing non-enzymatic antioxidant defenses in cerebral cortex supernatants, thereby promoting oxidative stress in the cerebral cortex. This compound is utilized in research concerning brain damage diseases [1].</p>
    Formula:C6H8O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:144.13

    Ref: TM-T78071

    1mg
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  • (±)​-​Vasicine

    CAS:
    <p>(±)-Vasicine, the racemate of Vasicine, is isolated from Peganum harmala seeds and exhibits anti-ulcer activity.</p>
    Formula:C11H12N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:188.23

    Ref: TM-T12681

    25mg
    Discontinued
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  • Alfadolone acetate

    CAS:
    <p>Alfadolone acetate is a gamma-aminobutyric acid (GABA) receptor agonist.</p>
    Formula:C23H34O5
    Color and Shape:Solid
    Molecular weight:390.51

    Ref: TM-T26592

    ne
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  • Filapixant

    CAS:
    <p>Filapixant, a purinoreceptor antagonist. This compound serves as the active reference substance for Eliapixant.</p>
    Formula:C24H26F3N5O3S
    Color and Shape:Solid
    Molecular weight:521.56

    Ref: TM-T39357

    ne
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  • 2-AEMP TFA

    CAS:
    <p>2-AEMP TFA is a potent and rapidly acting antagonist of GABA(A)-ρ1 receptors. 2-AEMP is an analog of GABA.</p>
    Formula:C3H10NO3P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:139.091

    Ref: TM-T26380

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  • Apcin A HCL

    CAS:
    <p>Apcin A HCL is an Apcin derivative. Apcin A HCL is an anaphase-promoting complex (APC) inhibitor. Apcin-A HCL interacts strongly with Cdc20, and inhibits the ubiquitination of Cdc20 substrates. Apcin-A HCL can be used to synthesize the PROTAC CP5V [1].</p>
    Formula:C10H15Cl4N5O2
    Purity:99.30%
    Color and Shape:Solid
    Molecular weight:379.07

    Ref: TM-T001

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  • Indoxacarb

    CAS:
    <p>Indoxacarb is an Oxadiazine insecticide.</p>
    Formula:C22H17ClF3N3O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:527.83

    Ref: TM-T20895

    50mg
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  • (Rac)-Lanicemine

    CAS:
    <p>(Rac)-Lanicemine ((Rac)-AZD6765) is the racemate of Lanicemine. Lanicemine (AZD6765) is a low-trapping NMDA channel blocker with a Ki of 0.56-2.1 μM for the NMDA receptor and IC50 values of 4-7 μM and 6.4 μM in CHO and Xenopus oocyte cells, respectively. Lanicemine shows antidepressant effects [1].</p>
    Formula:C13H14N2
    Color and Shape:Solid
    Molecular weight:198.26

    Ref: TM-T60235

    ne
    Discontinued
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  • Pazinaclone

    CAS:
    <p>Pazinaclone is a non-benzodiazepine (GABAA) partial agonist with sedative and anxiolytic activity.</p>
    Formula:C25H23ClN4O4
    Purity:97.79% - 99.07%
    Color and Shape:Solid
    Molecular weight:478.93

    Ref: TM-T28303

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  • Fostedil

    CAS:
    <p>Fostedil enhances heart function, maintains blood flow during partial/total coronary occlusions, and lowers aortic pressure.</p>
    Formula:C18H20NO3PS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:361.4

    Ref: TM-T27351

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  • Motugivatrep

    CAS:
    <p>Motugivatrep is a potent and selective TRPV1 antagonist that can be used to study TRPV1-related respiratory diseases.</p>
    Formula:C22H20F3NO3
    Purity:99.22%
    Color and Shape:Solid
    Molecular weight:403.39

    Ref: TM-T64312

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  • Pipequaline

    CAS:
    <p>Pipequaline (PK-8165) is an anticonflict &amp; anticonvulsant quinoline derivative. It is an anxiolytic drug that was never marketed. It possesses a novel chemical structure that is not closely related to other drugs of this type. The drug has a similar pharmacological profile to the benzodiazepine family of drugs, but with mainly anxiolytic properties and very little sedative, amnestic or anticonvulsant effects, and so is classified as a nonbenzodiazepine anxiolytic.</p>
    Formula:C22H24N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:316.44

    Ref: TM-T4655

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  • CMPDA

    CAS:
    <p>CMPDA is a positive allosteric modulator of AMPA receptors [EC50s: 45.4 nM/63.4 nM for GluA2i/GluA2o receptor].</p>
    Formula:C16H28N2O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:376.53

    Ref: TM-TQ0114

    50mg
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  • CGP 44532

    CAS:
    <p>CGP 44532 a GABAB receptor agonist.</p>
    Formula:C4H12NO3P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:153.12

    Ref: TM-T26991

    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • T16A(inh)-C01

    CAS:
    <p>T16A(inh)-C01 is the Ca(2+)-activated Cl(-) Channel, Ano1 class C inhibitor.</p>
    Formula:C18H16O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:312.32

    Ref: TM-T24846

    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • Gacyclidine

    CAS:
    <p>Gacyclidine (OTO311), an NMDA receptor blocker, treats tinnitus and injuries in the brain and spinal cord.</p>
    Formula:C16H25NS
    Purity:99.85% - 99.92%
    Color and Shape:Solid
    Molecular weight:263.44

    Ref: TM-T27397

    1mg
    Discontinued
    5mg
    Discontinued
    10mg
    Discontinued
    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    500mg
    Discontinued
    Discontinued product
  • Tifenazoxide

    CAS:
    <p>Tifenazoxide is an effective and SUR1/Kir6.2 selective KATP channels opener. Tifenazoxide has an anti-diabetic effect, can inhibit glucose-stimulated insulin release in vitro and in vivo.</p>
    Formula:C9H10ClN3O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:291.78

    Ref: TM-T17094

    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • Phenamil methanesulfonate

    CAS:
    <p>TRPP3 channel inhibitor</p>
    Formula:C13H16ClN7O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:401.83

    Ref: TM-T23148

    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • Belfosdil

    CAS:
    <p>Belfosdil is a blocker of antihypertensive calcium channel.</p>
    Formula:C27H50O7P2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:548.63

    Ref: TM-T26764

    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • LFS-1107

    CAS:
    <p>LFS-1107, a reversible CRM1 inhibitor (Kd: 12.5 pM), selectively targets and eliminates ENKTL cells, offering potential for cancer research applications [1].</p>
    Formula:C12H11N5OS2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:305.38

    Ref: TM-T81936

    5mg
    Discontinued
    50mg
    Discontinued
    Discontinued product
  • Bumetanide sodium

    CAS:
    <p>Bumetanide sodium, a potent diuretic, blocks NKCC1 (IC50: 0.68 μM) and NKCC2 (IC50: 4.0 μM).</p>
    Formula:C17H19N2NaO5S
    Color and Shape:Solid
    Molecular weight:386.4

    Ref: TM-T61713

    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • VMAT2-IN-2 tosylate

    CAS:
    <p>VMAT2-IN-2 tosylate is a potent inhibitor of VMAT2 and is applicable in the research of tardive dyskinesia [1].</p>
    Formula:C27H36F3NO6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:559.64

    Ref: TM-T79061

    5mg
    Discontinued
    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • CGP 56999A

    CAS:
    CGP 56999A is a GABA(B) receptor antagonist; it boosts BDNF and reduces dopamine loss in rat striatum.
    Formula:C19H30NO5P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:383.42

    Ref: TM-T26993

    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • HMR 1556

    CAS:
    <p>HMR 1556 is a chromanol derivative and is an IKs blocker (IC50s of 10.5 nM and 34 nM in canine and guinea pig left ventricular myocytes, respectively).</p>
    Formula:C17H24F3NO5S
    Color and Shape:Solid
    Molecular weight:411.44

    Ref: TM-T15487

    1mg
    Discontinued
    Discontinued product
  • Xilmenolone

    CAS:
    <p>Xilmenolone acts as a positive allosteric modulator of the GABA_A receptor [1].</p>
    Formula:C26H37N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:423.59

    Ref: TM-T78670

    5mg
    Discontinued
    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product