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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2293 products of "Membrane Transporter/Ion Channel"

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  • Rufinamide
    Targetmol
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    Rufinamide

    CAS:
    <p>Rufinamide (E 2080), a triazole derivative, is used as voltage-gated sodium channel blocker for the treatment of seizure disorders.</p>
    Formula:C10H8F2N4O
    Purity:99.77% - >99.99%
    Color and Shape:White Powder
    Molecular weight:238.19

    Ref: TM-T2523

  • Ibutilide Fumarate
    Targetmol
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    Ibutilide Fumarate

    CAS:
    <p>Ibutilide Fumarate is a class III antiarrhythmic, prolonging action potentials by enhancing sodium influx, and can extend QT interval.</p>
    Formula:(C20H36N2O3S)2·C4H4O4
    Purity:99.68% - 99.74%
    Color and Shape:Solid
    Molecular weight:885.23

    Ref: TM-T6541

  • BAY-8002
    Targetmol
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    BAY-8002

    CAS:
    <p>BAY-8002 is a potent dual MCT1/2 inhibitor (IC50 values are 3, 8, and 12 nM at rat (C6), human (DLD-1) and mouse (4T1) MCT1 respectively).</p>
    Formula:C20H14ClNO5S
    Purity:98.7% - 99.13%
    Color and Shape:Solid
    Molecular weight:415.85

    Ref: TM-T5208

  • Ko 143
    Targetmol
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    Ko 143

    CAS:
    <p>Ko 143 is a selective inhibitor of ATP-binding cassette sub-family G member 2 (ABCG2; BCRP).</p>
    Formula:C26H35N3O5
    Purity:99.01% - 99.89%
    Color and Shape:Solid
    Molecular weight:469.57

    Ref: TM-TQ0186

  • Benzamil
    Targetmol
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    Benzamil

    CAS:
    <p>Benzamil blocks ENaC, inhibiting sodium transport (IC50=4 nM) and binds with Kd=5 nM to bovine kidney membranes.</p>
    Formula:C13H14ClN7O
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:319.75

    Ref: TM-T5850

  • Tetraethylammonium chloride
    Targetmol
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    Tetraethylammonium chloride

    CAS:
    <p>Tetraethylammonium chloride is a quaternary ammonium compound.</p>
    Formula:C8H20ClN
    Purity:≥95%
    Color and Shape:White Solid Solid Particulate/Powder
    Molecular weight:165.7

    Ref: TM-T7538

  • SAR7334 hydrochloride
    Targetmol
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    SAR7334 hydrochloride

    CAS:
    <p>SAR7334 hydrochloride is a potent and specific inhibitor of TRPC6(IC50 of 7.9 nM).</p>
    Formula:C21H24Cl3N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:440.79

    Ref: TM-T12849L

  • Pikamilone
    Targetmol
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    Pikamilone

    CAS:
    Pikamilone (Picamilon) is an intelligent medicine.
    Formula:C10H12N2O3
    Purity:99.38%
    Color and Shape:White Crystalline Powder
    Molecular weight:208.21

    Ref: TM-T3290

  • BRITE-338733
    Targetmol
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    BRITE-338733

    CAS:
    <p>BRITE-338733 is a novel inhibitor of ATPase. BRITE 338733 inhibits the expression of RecA in bacteria (IC50=4.7 μM) for the bacterial infections treatment.</p>
    Formula:C27H35N3O2
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:433.59

    Ref: TM-T22280

  • CTP disodium dihydrate
    Targetmol
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    CTP disodium dihydrate

    CAS:
    <p>CTP disodium dihydrate is an agonist of P2X4 purinergic receptor</p>
    Formula:C9H18N3Na2O16P3
    Purity:98.51%
    Color and Shape:White Crystalline Powder
    Molecular weight:563.15

    Ref: TM-T7881

  • AM92016
    Targetmol
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    AM92016

    CAS:
    <p>AM92016 is a specific blocker of the time dependent delayed rectifier potassium current. AM92016 does not show any β-adrenoceptor blocking activity.</p>
    Formula:C26H30Cl2N2O6S
    Color and Shape:Solid
    Molecular weight:569.49

    Ref: TM-T70194

  • Nicainoprol
    Targetmol
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    Nicainoprol

    CAS:
    <p>Nicainoprol (RU-42924) is a fast-sodium-channel blocking drug. Nicainoprol is a potent antiarrhythmic agent.</p>
    Formula:C21H27N3O3
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:369.46

    Ref: TM-T4539

  • Raxatrigine
    Targetmol
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    Raxatrigine

    CAS:
    Raxatrigine (CNV 1014802) has been investigated for the treatment of Bipolar Disorder and Bipolar Depression.
    Formula:C18H19FN2O2
    Purity:98% - 99.43%
    Color and Shape:Solid
    Molecular weight:314.35

    Ref: TM-T2342

  • Riluzole
    Targetmol
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    Riluzole

    CAS:
    <p>Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.</p>
    Formula:C8H5F3N2OS
    Purity:99.71% - 99.88%
    Color and Shape:Powder
    Molecular weight:234.2

    Ref: TM-T0349

  • Apinocaltamide
    Targetmol
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    Apinocaltamide

    CAS:
    Apinocaltamide (ACT-709478) is an orally available and selective T-type calcium channel blocker that cross BBB for Cav3.1, Cav3.2, and Cav3.3,epilepsy.
    Formula:C22H18F3N5O
    Purity:99.80%
    Color and Shape:Solid
    Molecular weight:425.41

    Ref: TM-T14120

  • Bupivacaine
    Targetmol
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    Bupivacaine

    CAS:
    <p>Bupivacaine (AH-250) is a NMDA receptor inhibitor.Bupivacaine can block sodium, L-calcium, and potassium channels.Bupivacaine potently blocks SCN5A channels</p>
    Formula:C18H28N2O
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:288.43

    Ref: TM-T0030L

  • SRI-41315
    Targetmol
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    SRI-41315

    CAS:
    <p>SRI-41315 is an eRF1 degrader that acts as a molecular glue at the ribosomal decoding center.SRI-41315 induces extended pauses at the termination codon.</p>
    Formula:C22H19N3O2
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:357.41

    Ref: TM-T61306

  • CX717
    Targetmol
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    CX717

    CAS:
    <p>CX 717 is a positive allosteric modulator of AMPA receptor which has an antidepressant-like effect.</p>
    Formula:C11H11N3O3
    Purity:99.81%
    Color and Shape:Soild
    Molecular weight:233.23

    Ref: TM-T60201

  • JNJ-28583113
    Targetmol
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    JNJ-28583113

    CAS:
    <p>JNJ-28583113 is a TRPM2 antagonist, inducing phosphorylation of GSK3α and β subunits, protecting cells from oxidative stress-induced cell death.</p>
    Formula:C19H21F3N2O2
    Purity:98.57%
    Color and Shape:Solid
    Molecular weight:366.38

    Ref: TM-T74779

  • Safinamide
    Targetmol
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    Safinamide

    CAS:
    <p>Safinamide: reversible MAO-B inhibitor, enhances dopamine, blocks glutamate release, sodium, calcium channels; may treat Parkinson's, RLS, epilepsy.</p>
    Formula:C17H19FN2O2
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:302.34

    Ref: TM-T6651L

  • Ro 25-6981 Maleate
    Targetmol
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    Ro 25-6981 Maleate

    CAS:
    <p>Ro 25-6981 Maleate is an NMDA receptor antagonist used in the study of neurological disorders such as Parkinson's and epilepsy.</p>
    Formula:C26H33NO6
    Purity:99.42%
    Color and Shape:Solid
    Molecular weight:455.54

    Ref: TM-T12758L

  • HUP30
    Targetmol
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    HUP30

    CAS:
    <p>HUP30 is a potent vasodilating agent. HUP30 can stimulate soluble guanylyl cyclase, activate K+ channels, and block extracellular Ca2+ influx.</p>
    Formula:C14H15N3O3S
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:305.35

    Ref: TM-TNU0864

  • ZT-1a
    Targetmol
    + Info

    ZT-1a

    CAS:
    <p>ZT-1a is a SPAK inhibitor.ZT-1a inhibits SPAK.ZT-1a can be used for the prevention and treatment of neurodegenerative and neurocognitive disorders.</p>
    Formula:C22H15Cl3N2O2
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:445.73

    Ref: TM-T39566

  • N-Methyl-L-leucin
    Targetmol
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    N-Methyl-L-leucin

    CAS:
    <p>N-Methyl-L-leucine ((S)-4-Methyl-2-(methylamino)pentanoic acid) is a novel calcium channel antagonist used in pain research.</p>
    Formula:C7H15NO2
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:145.2

    Ref: TM-T65918

  • PF 03716556
    Targetmol
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    PF 03716556

    CAS:
    PF 03716556 (PF-3716556) , an effective and specific P-CAB (potassium-competitive acid blocker), is utilized for the treatment of gastroesophageal reflux
    Formula:C22H26N4O3
    Purity:99.79% - 99.95%
    Color and Shape:Solid
    Molecular weight:394.47

    Ref: TM-T2093

  • Darigabat
    Targetmol
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    Darigabat

    CAS:
    <p>Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.</p>
    Formula:C22H21FN4O3S
    Purity:98.42% - 99.29%
    Color and Shape:Solid
    Molecular weight:440.49

    Ref: TM-T16489

  • Doxapram
    Targetmol
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    Doxapram

    CAS:
    Doxapram (Dopram) is a respiratory stimulant that inhibits TASK-1, TASK-3, and TASK-1/TASK-3 heterodimer channels.
    Formula:C24H30N2O2
    Purity:99.42%
    Color and Shape:Solid
    Molecular weight:378.51

    Ref: TM-T22315

  • VU590
    Targetmol
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    VU590

    CAS:
    <p>VU590 is an inhibitor of extrarenal medullary potassium ROMK.VU590 inhibits Kir7.1 and modulates uterine myometrial contractility and melanocortin signalling.</p>
    Formula:C24H32N4O7
    Purity:98.06%
    Color and Shape:Solid
    Molecular weight:488.53

    Ref: TM-T23516

  • VB124
    Targetmol
    + Info

    VB124

    CAS:
    <p>VB124 is an orally active, potent and selective MCT4 inhibitor. VB124 blocked lactate importand expor in MDA-MB-231 cells.Cost-effective and quality-assured.</p>
    Formula:C23H23ClN2O4
    Purity:99.21% - 99.57%
    Color and Shape:Soild
    Molecular weight:426.89

    Ref: TM-T60165

  • Mtb ATP synthase-IN-1
    Targetmol
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    Mtb ATP synthase-IN-1

    CAS:
    Mtb ATP synthase-IN-1 is a potent, low-toxicity M. tuberculosis inhibitor with good oral bioavailability and metabolic stability.
    Formula:C17H13N3O4
    Purity:98.28%
    Color and Shape:Solid
    Molecular weight:323.30

    Ref: TM-T60877

  • Propoxycaine hydrochloride
    Targetmol
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    Propoxycaine hydrochloride

    CAS:
    Propoxycaine hydrochloride is an ester local anesthetic that inhibits voltage-gated sodium channels, modulates nerve impulses, and induces loss of sensation.
    Formula:C16H27ClN2O3
    Purity:97.25%
    Color and Shape:Solid
    Molecular weight:330.85

    Ref: TM-T13830

  • Dimiracetam
    Targetmol
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    Dimiracetam

    CAS:
    <p>Dimiracetam, a NMDA-receptor antagonist, is used potentially for the treatment of neuropathic pain.</p>
    Formula:C6H8N2O2
    Purity:>99.99% - >99.99%
    Color and Shape:Solid
    Molecular weight:140.14

    Ref: TM-T27178

  • BL-1249
    Targetmol
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    BL-1249

    CAS:
    <p>BL-1249 is a selective and potent non-steroidal potassium channel activator with anti-inflammatory activity that activates K2P2.1 (TREK-1) and K2P10.1 (TREK-2).</p>
    Formula:C17H17N5
    Purity:98% - 98.25%
    Color and Shape:Solid
    Molecular weight:291.35

    Ref: TM-T14666

  • Methionine
    Targetmol
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    Methionine

    CAS:
    <p>Methionine (D-Methionine) (MRX-1024; D-Methionine) is an effective chemoprotective agent which can also inhibit the neuronal activity through GABAA receptor</p>
    Formula:C5H11NO2S
    Purity:99.13% - 99.62%
    Color and Shape:Solid
    Molecular weight:149.21

    Ref: TM-T19418L

  • Lanicemine dihydrochloride
    Targetmol
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    Lanicemine dihydrochloride

    CAS:
    <p>Lanicemine dihydrochloride (AZD-6765 dihydrochloride) is an NMDA channel blocker with antidepressant activity and can be used to study neurological diseases.</p>
    Formula:C13H16Cl2N2
    Purity:98.37%
    Color and Shape:Solid
    Molecular weight:271.19

    Ref: TM-T60471

  • Bupivacaine-d9
    Targetmol
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    Bupivacaine-d9

    CAS:
    Bupivacaine-d9 is a deuterated compound of Bupivacaine. Bupivacaine has a CAS number of 38396-39-3. Bupivacaine is a NMDA receptor inhibitor.Bupivacaine can block sodium, L-calcium, and potassium channels.Bupivacaine potently blocks SCN5A channels with the IC50 of 69.5 μM. Bupivacaine can be used for the research of chronic pain.
    Formula:C18H19D9N2O
    Color and Shape:Solid
    Molecular weight:297.48

    Ref: TM-TMIJ-0210

  • Eleclazine
    Targetmol
    + Info

    Eleclazine

    CAS:
    <p>Eleclazine (GS-6615) is a novel and selective voltage-gated sodium channel inhibitor with antiarrhythmic properties that reduces peak sodium current (INaP).</p>
    Formula:C21H16F3N3O3
    Purity:98.67%
    Color and Shape:Solid
    Molecular weight:415.37

    Ref: TM-T71945

  • SAR7334
    Targetmol
    + Info

    SAR7334

    CAS:
    <p>SAR7334 (TRCP6-IN-1) is a potent and specific inhibitor of TRPC6(IC50 of 7.9 nM).</p>
    Formula:C21H22ClN3O
    Purity:99.62% - 99.71%
    Color and Shape:Solid
    Molecular weight:367.87

    Ref: TM-T12849

  • Flavoxate
    Targetmol
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    Flavoxate

    CAS:
    <p>Flavoxate is an anticholinergic with antimuscarinic effects.</p>
    Formula:C24H25NO4
    Color and Shape:Solid
    Molecular weight:391.46

    Ref: TM-T0703L

  • Eperisone
    Targetmol
    + Info

    Eperisone

    CAS:
    <p>Eperisone: a muscle relaxant for stiffness and pain, relaxes muscles, improves circulation, and mitigates pain by inhibiting reflexes and vasodilation.</p>
    Formula:C17H25NO
    Color and Shape:Solid
    Molecular weight:259.39

    Ref: TM-T40744

  • Amlodipine besilate impurity G
    Targetmol
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    Amlodipine besilate impurity G

    CAS:
    <p>Amlodipine besilate impurity G is a Calcium Channel antagonist with potential application in the study of neurological diseases and is an impurity in the</p>
    Formula:C17H18ClNO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:335.78

    Ref: TM-T20994

  • Amlodipine hydrochloride
    Targetmol
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    Amlodipine hydrochloride

    CAS:
    <p>Amlodipine hydrochloride is a salt of Amlodipine --- a medication used to lower blood pressure and prevent chest pain.</p>
    Formula:C20H26Cl2N2O5
    Color and Shape:Solid
    Molecular weight:445.34

    Ref: TM-T0231L

  • Cinepazide
    Targetmol
    + Info

    Cinepazide

    CAS:
    <p>Cinepazide: a vasodilator targeting adenosine A2 receptors, treats various vascular diseases.</p>
    Formula:C22H31N3O5
    Color and Shape:White Powder
    Molecular weight:417.5

    Ref: TM-T0368L

  • MCT-IN-1
    Targetmol
    + Info

    MCT-IN-1

    CAS:
    <p>MCT-IN-1 (compound 2) acts as a potent inhibitor of the monocarboxylate transporter (MCT), demonstrating IC50 values of 9 nM for MCT1 and 14 nM for MCT4.</p>
    Formula:C19H26N2O3
    Color and Shape:Solid
    Molecular weight:330.42

    Ref: TM-T88656

  • VGSC blocker-1
    Targetmol
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    VGSC blocker-1

    CAS:
    <p>VGSC blocker-1 inhibits 34.9% INa in nNav1.5 at 1 μM, reduces MDA-MB-231 invasion by 0.3%, non-toxic.</p>
    Formula:C24H32F2N2
    Color and Shape:Solid
    Molecular weight:386.52

    Ref: TM-T39717

  • FSC231
    Targetmol
    + Info

    FSC231

    CAS:
    <p>FSC231 is a PICK1 inhibitor with analgesic activity, activating GSK-3β and ERK1/2.</p>
    Formula:C13H10Cl2N2O3
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:313.14

    Ref: TM-T86471

  • BAY-390
    Targetmol
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    BAY-390

    CAS:
    <p>BAY-390, a selective TRPA1 inhibitor, crosses species, penetrates brains, with IC50s: 16-82 nM. Used in inflammation research.</p>
    Formula:C13H15F4NO
    Color and Shape:Solid
    Molecular weight:277.26

    Ref: TM-T73432

  • PBFI-AM
    Targetmol
    + Info

    PBFI-AM

    CAS:
    <p>PBFI-AM is a useful tool to determine intracellular K + content [1] .</p>
    Formula:C58H62N2O24
    Color and Shape:Solid
    Molecular weight:1171.11

    Ref: TM-T74091

  • Dofetilide D4
    Targetmol
    + Info

    Dofetilide D4

    CAS:
    Dofetilide D4 (UK 68789 D4), a deuterium-labeled version of Dofetilide, is categorized as a Class III antiarrhythmic medication.
    Formula:C19H27N3O5S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:445.59

    Ref: TM-T11072

  • Topiramate D12
    Targetmol
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    Topiramate D12

    CAS:
    <p>Topiramate D12 is a deuterium labeled Topiramate. Topiramate is an agent of broad-spectrum antiepileptic. Topiramate is an antagonist of GluR5 receptor.</p>
    Formula:C12H21NO8S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:351.44

    Ref: TM-T13185