Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(100 products)
- Adiponectin receptor(5 products)
- CFTR(66 products)
- CGRP Receptor(54 products)
- Calcium Channel(545 products)
- Chloride channel(53 products)
- GABA Receptor(369 products)
- Monoamine Transporter(30 products)
- Monocarboxylate transporter(18 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(10 products)
- OAT(32 products)
- OCT(7 products)
- P-gp(55 products)
- Potassium Channel(283 products)
- Proton pump(41 products)
- SGLT(31 products)
- Sodium Channel(219 products)
- TRP/TRPV Channel(96 products)
Show 13 more subcategories
Found 2586 products of "Membrane Transporter/Ion Channel"
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NSC265473
CAS:NSC265473 is an ABCG2 substrate.Formula:C21H35N3O4SColor and Shape:SolidMolecular weight:425.58Conantokin G TFA
Conantokin G TFA, a 17-aa peptide, blocks NMDA receptors with 480 nM IC50 and is neuroprotective.Formula:C90H139F3N26O46Color and Shape:SolidMolecular weight:2378.21(S)-PF-03716556
CAS:(S)-PF-03716556 can be used as an acid pump inhibitor for the treatment of disease conditions mediated by acid pump inhibitory activity.Formula:C22H26N4O3Purity:99.75% - 99.91%Color and Shape:SoildMolecular weight:394.47Dihydroisopimaric acid
CAS:Dihydroisopimaric acid opens BKαβ1 channels - large Ca²⁺-activated K⁺ conductors, verified by whole-cell voltage clamp.Formula:C20H32O2Color and Shape:SolidMolecular weight:304.47TRPV1 activator-2
CAS:TRPV1 activator-2 (Compound 9), a capsaicin head analog, engages in targeted interactions with channel residues at the lipid-water interface [1].Formula:C19H29NO3Color and Shape:SolidMolecular weight:319.44Antidepressant agent 3
Agent 3: orally active, antidepressant, anxiolytic, boosts performance and cognition.Formula:C17H30ClN5O2SColor and Shape:SolidMolecular weight:403.97Charybdotoxin
CAS:Specific inhibitor of the big conductance Ca2+-activated K+ channel.Formula:C176H277N57O55S7Purity:98%Color and Shape:SolidMolecular weight:4295.95TRPV4 antagonist 4
CAS:<p>Potent TRPV4 blocker with 22.65 nM IC50; inhibits current and aids acute lung injury.</p>Formula:C28H32Cl2N6OColor and Shape:SolidMolecular weight:539.50Tertiapin LQ
Kir1.1 channel blocker, 250x selective; Kd: Kir1.1 (1.1 nM), Kir3.1/3.2 (274 nM), Kir3.1/3.4 (361 nM). Tertiapin-Q derivative.Formula:C106H179N33O24S4Purity:98%Color and Shape:SolidMolecular weight:2428.03RU-TRAAK-2
CAS:<p>RU-TRAAK-2 reversibly inhibits TWIK-related K+ channel, inactive on Kv1.2, GIRK2, Slo1.</p>Formula:C19H17N3OSPurity:99.81%Color and Shape:SolidMolecular weight:335.42Calcium Ionophore I
CAS:Calcium Ionophore I has a wide range of applications in life science related research.Formula:C38H72N2O8Color and Shape:SolidMolecular weight:685.0Conantokin-T
CAS:Non-competitive NMDA receptor antagonistFormula:C110H175N31O45SPurity:98%Color and Shape:SolidMolecular weight:2683.81H-Lys-Tyr-OH TFA
Lysyltyrosine TFA is a dipeptide that may enhance brain function by boosting noradrenaline and tyrosine release.Formula:C17H24F3N3O6Color and Shape:SolidMolecular weight:423.38Euphol acetate
CAS:Euphol acetate, a triterpene from Euphorbia broteri, inhibits liver transport proteins OATP1B1/3.Formula:C32H52O2Color and Shape:SolidMolecular weight:468.75BKCa activator-1
BKCa activator-1 (Compound 51b) is an orally active activator of BKCa calcium-activated potassium channels with an EC50 of 2.82 μM. It promotes K+ efflux, leading to cell membrane hyperpolarization and inhibition of smooth muscle contraction. In a spontaneous hypertensive rat (SHR) model, it alleviates urinary incontinence and exhibits antitussive effects in a guinea pig cough model.Formula:C22H23F7N2O3Color and Shape:SolidMolecular weight:496.418AR-C141990 hydrochloride
CAS:<p>AR-C141990 HCl inhibits MCT-1 (pKi 7.6) and MCT-2 (pKi 6.6), and has immunosuppressive effects.</p>Formula:C26H29ClN4O4SColor and Shape:SolidMolecular weight:529.05Linoleic Acid Amide
CAS:<p>Linoleic Acid Amide (Linoleamide) is derived from linoleic acid and regulates Ca2+ flux by inhibiting the sarco/endoplasmic reticulum Ca2+-ATPase.</p>Formula:C18H33NOPurity:98%Color and Shape:SolidMolecular weight:279.46Mutabilol
Mutabilol boosts P-gp in NCI-H460/R cells; natural from Plectranthus mutabilis.Formula:C19H24O5Color and Shape:SolidMolecular weight:332.39NF864
CAS:NF864, a suramin analog, is a P2X1 receptor inhibitor.Formula:C57H28N6Na12O41S12Purity:98%Color and Shape:SolidMolecular weight:2113.5α5-GABAA receptor modulator 1
α5-GABAA receptor modulator 1 (Compound A-4) is a selective silent allosteric modulator (SAM) targeting the α5 subunit of GABAA receptors, useful for research into central nervous system (CNS) disorders.Formula:C21H20FN3O4Color and Shape:SolidMolecular weight:397.4
