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Casein Kinase

Casein Kinase

Casein kinases are a family of serine/threonine protein kinases that regulate various cellular processes, including DNA repair, circadian rhythms, and signal transduction. These kinases are involved in the phosphorylation of numerous proteins and are implicated in diseases such as cancer, neurodegenerative disorders, and metabolic syndromes. At CymitQuimica, we offer a selection of casein kinase inhibitors to support your research in signal transduction, cell cycle regulation, and therapeutic development.

Found 130 products of "Casein Kinase"

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  • Emodin

    CAS:
    <p>Emodin (Frangula emodin) is a selective 11β-HSD1 inhibitor,IC50 of 186 and 86 nM against 11β-HSD1 in humans and mice. High-Quality, Low-Cost!</p>
    Formula:C15H10O5
    Purity:98.37% - 99.53%
    Color and Shape:Physical Description Orange Needles Or Powder (Ntp 1992)
    Molecular weight:270.24
  • Ellagic acid

    CAS:
    <p>Ellagic acid (Gallogen), a thickened tetracyclic natural product, is a potent CK2 inhibitor. Ellagic acid is an antioxidant. Cost-effective and quality-assured.</p>
    Formula:C14H6O8
    Purity:97.11% - 99.75%
    Color and Shape:Cream Colored Needles From Pyridine 1992)
    Molecular weight:302.19
  • Silmitasertib sodium salt

    CAS:
    <p>Silmitasertib sodium salt (CX-4945 sodium salt) is a potent and orally bioavailable, highly selective inhibitor of CK2(IC50 of 1 nM, CK2α).</p>
    Formula:C19H11ClN3NaO2
    Purity:99.49% - 99.62%
    Color and Shape:Solid
    Molecular weight:371.75
  • A-3 hydrochloride

    CAS:
    <p>A-3 hydrochloride: potent, reversible kinase antagonist; permeable; inhibits PKC, CKI, PKA, CKII, MLCK; Ki: 4.3-80 μM.</p>
    Formula:C12H14Cl2N2O2S
    Purity:99.32%
    Color and Shape:Solid
    Molecular weight:321.22
  • NMS-P715

    CAS:
    <p>NMS-P715 is a highly selective and ATP-competitive MPS1 inhibitor(IC50 of 182 nM).</p>
    Formula:C35H39F3N8O3
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:676.73
  • CIGB-300

    CAS:
    <p>CIGB-300 (P15-Tat) is an anti-casein kinase 2 (CK2) peptide that exhibits anticancer properties by disrupting the phosphorylation activity of protein kinase CK2. The compound induces apoptosis in various tumor cell lines, making it valuable for research in cancer therapy.</p>
    Formula:C127H215N53O30S3
    Color and Shape:Solid
    Molecular weight:3060.6
  • CSNK2-IN-2


    <p>CSNK2-IN-2 (compound 2) is an orally active inhibitor of CSNK2. It is utilized in antiviral research.</p>
    Formula:C25H30FN9O
    Color and Shape:Solid
    Molecular weight:491.56
  • CK1-IN-4


    <p>CK1-IN-4 (Compound 59) is an inhibitor of casein kinase CK1δ with an IC50 of 2.74 μM. It exhibits neuroprotective activity in SH-SY5Y cells treated with Ethacrynic acid.</p>
    Color and Shape:Odour Solid
  • WAY-297174

    CAS:
    <p>WAY-297174 is a human protein kinase CK2 inhibitor with IC50 of &gt; 33 μM.</p>
    Formula:C11H12N2O2S2
    Purity:99.53%
    Color and Shape:Soild
    Molecular weight:268.36
  • Ellagic acid (hydrate)

    CAS:
    <p>Ellagic acid (hydrate) is a natural antioxidant and acts as a potent and ATP-competitive CK2 inhibitor (IC50:40 nM, Ki: 20 nM).</p>
    Formula:C14H8O9
    Purity:98%
    Color and Shape:Green To Beige Powder
    Molecular weight:320.21
  • AH078


    <p>AH078 (compound 37) is a selective PROTAC degrader targeting CK1δ and CK1ε with low selectivity for CK1α. AH078 consists of a PROTAC linker (black part) Monomethyl octanoate, a target protein ligand (red part) CK1δ/CK1ε ligand-1, and an E3 ligase ligand (blue part) E3 Ligase Ligand 58. The E3 ligase ligand combined with the linker forms the conjugate E3 Ligase Ligand-linker Conjugate 163.</p>
    Formula:C51H60F2N10O5S
    Color and Shape:Solid
    Molecular weight:963.15
  • GSK-3β/CK-1δ-IN-1


    <p>GSK-3β/CK-1δ-IN-1 (8d) is a dual inhibitor of GSK-3β and CK-1δ that can cross the blood-brain barrier, with IC50 values of 0.77 μM and 0.57 μM, respectively. GSK-3β/CK-1δ-IN-1 (8d) is applicable in neuroblastoma research.</p>
    Formula:C22H17F3N4O
    Color and Shape:Solid
    Molecular weight:410.39
  • Casein Kinase 2 Substrate Peptide

    CAS:
    <p>CK2 Substrate Peptide, C-terminus linked to EDANS, used for CK2 activity assays.</p>
    Formula:C45H73N19O24
    Color and Shape:Solid
    Molecular weight:1264.17
  • CK2-IN-13


    <p>CK2-IN-13 (compound 12c) is a potent inhibitor of CK2, with an IC50 value of 5.8 nM, playing a significant role in cancer research.</p>
    Formula:C19H13Br2NO3
    Color and Shape:Solid
    Molecular weight:463.119
  • Casein

    CAS:
    <p>Casein is a milk protein with multiple roles involved in novel drug delivery systems.</p>
    Purity:95%
    Color and Shape:Soild
  • Casein kinase 1δ-IN-14

    CAS:
    <p>Casein kinase 1δ-IN-14 (WAY-637081) can be used to study atherosclerosis-related cardiovascular disease.</p>
    Formula:C17H11ClN4O2
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:338.75
  • CK1-IN-3

    CAS:
    <p>WAY-296817 inhibits CK1, potential for circadian rhythm and inflammation research.</p>
    Formula:C17H16N2O3S
    Purity:99.18%
    Color and Shape:Solid
    Molecular weight:328.39
  • Casein kinase 1δ-IN-9

    CAS:
    <p>Casein kinase 1δ-IN-9 is a Quinone reductase 2 inhibitor with IC50 of 0.6μM.</p>
    Formula:C15H12ClN3
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:269.73
  • Casein Kinase Substrates 3

    CAS:
    <p>Casein Kinase Substrates 3 is a substrate of casein kinase.</p>
    Formula:C85H139N27O35S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2131.24
  • TBCA

    CAS:
    <p>TBCA: selective CK2 inhibitor, IC50=110 nM, Ki=77 nM, favors CK2 over CK1, DYRK1A, and 27 other kinases.</p>
    Formula:C9H4Br4O2
    Purity:99.3%
    Color and Shape:Solid
    Molecular weight:463.74
  • Casein kinase 1δ-IN-7

    CAS:
    <p>Casein kinase 1δ-IN-7 is a Casein kinase 1δ inhibitor for neurodegenerative diseases such as Alzheimer's disease.</p>
    Formula:C17H14N4O2S
    Purity:98.6%
    Color and Shape:Solid
    Molecular weight:338.38
  • Casein kinase 1δ-IN-8

    CAS:
    <p>Casein kinase 1δ-IN-8 is an inhibitor of casein kinase 1δ and is used to treat neurodegenerative diseases such as Alzheimer's disease type.</p>
    Formula:C19H14FN5OS
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:379.41
  • CK2-IN-14


    <p>CK2-IN-14 (Compound 10b) is an inhibitor of cyclin-dependent kinase 2α with an IC50 of 36.7 nM. It effectively hinders the growth of cancer cell lines 786-O and U937, with GI50 values of 7.3 μM and 7.5 μM, respectively.</p>
    Formula:C19H20ClN5S
    Color and Shape:Solid
    Molecular weight:385.91
  • Casein kinase 1δ-IN-6

    CAS:
    <p>CK1δ-IN-6: potent, selective CK-1δ inhibitor, IC50 23 nM, neuroprotective, anti-inflammatory, for neurodegenerative research.</p>
    Formula:C16H10ClF3N2OS
    Purity:99%
    Color and Shape:Soild
    Molecular weight:370.78
  • Casein kinase 1δ-IN-15

    CAS:
    <p>Casein kinase 1δ-IN-15, an inhibitor for casein kinase 1 (CK1δ), exhibits an IC50 of 0.045 μM [1].</p>
    Formula:C19H17FN6O
    Color and Shape:Solid
    Molecular weight:364.38
  • Casein kinase 1δ-IN-3

    CAS:
    <p>Casein kinase 1δ-IN-3 (Casein kinase 1δ-IN-3) (Compound 23a) is a casein kinase 1 delta (CK1d) inhibitor with a pIC50 of 6.5376 M.</p>
    Formula:C17H16N2O2S
    Purity:98.94%
    Color and Shape:Soild
    Molecular weight:312.39
  • QXG-6442


    <p>QXG-6442 is a molecular glue degrader targeting CK1α, demonstrating a degradation potency with a DC50 of 5.7 nM and a Dmax of 90%. In the MOLM-14 cell line, QXG-6442 induces antiproliferative effects.</p>
    Formula:C21H17N5O4
    Color and Shape:Solid
    Molecular weight:403.39
  • MU1742


    <p>MU1742 is a probe for CK1δ and CK1ε protein kinases [1] .</p>
    Formula:C22H22F2N6
    Color and Shape:Solid
    Molecular weight:408.45
  • CK1δ/CK1ε liagnd-1


    <p>CK1δ/CK1ε ligand-1 is a ligand of CK1δ/CK1ε and can serve as a target protein ligand for the synthesis of the CK1 PROTAC degrader AH078.</p>
    Formula:C21H20F2N6
    Color and Shape:Solid
    Molecular weight:394.42
  • CZP-IN-1


    <p>CZP-IN-1 (compound SH-1) is an inhibitor targeting the pathogen Trypanosoma cruzi protease (CZP) without affecting cathepsin L (IC50=28 nM). This compound is applicable in Chagas disease research.</p>
    Formula:C20H26N4O4S
    Color and Shape:Solid
    Molecular weight:418.51
  • FPFT-2216

    CAS:
    <p>FPFT-2216 is a "molecular glue" compound with potential anti-tumor activity that degrades IKZF6, IKZF1, DE1D and can be used to study immune system diseases.</p>
    Formula:C12H12N4O3S
    Purity:99.35% - 99.62%
    Color and Shape:Solid
    Molecular weight:292.31
  • PF-5006739

    CAS:
    <p>PF-5006739: potent, selective CK1δ/ε inhibitor (IC50: 3.9/17.0 nM); may treat psychiatric disorders, improves glucose tolerance, reduces opioid seeking.</p>
    Formula:C22H22FN7O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:419.45
  • MRT00033659

    CAS:
    <p>MRT00033659 inhibits CK1 (IC50=0.9 μM), CHK1 (IC50=0.23 μM), activates p53, and destabilizes E2F-1; it's a pyrazolo-pyridine.</p>
    Formula:C15H14N4O
    Color and Shape:Solid
    Molecular weight:266.3
  • SGC-CK2-1

    CAS:
    <p>SGC-CK2-1, a CK2 inhibitor, is a inducer of insulin production and secretion in pancreatic β-cells.</p>
    Formula:C20H21N7O
    Purity:99.41%
    Color and Shape:Solid
    Molecular weight:375.43
  • Longdaysin

    CAS:
    <p>Longdaysin is an inhibitor of CK1α and CK1δ (IC50s: 5.6/8.8 μM). It also can inhibit ERK2 (IC50: 52 μM).</p>
    Formula:C16H16F3N5
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:335.33
  • TA-01

    CAS:
    <p>TA-01 is a potent CK1 and p38 MAPK inhibitor, with IC50s of 6.4 nM, 6.8 nM, 6.7 nM for CK1ε, CK1δ and p38 MAPK, respectively.</p>
    Formula:C20H12F3N3
    Purity:99.55% - 99.94%
    Color and Shape:Solid
    Molecular weight:351.32
  • Epiblastin A

    CAS:
    <p>Epiblastin A inhibits CK1, targets its isoenzymes, and converts EpiSCs to cESCs.</p>
    Formula:C12H10ClN7
    Purity:99.45%
    Color and Shape:Solid
    Molecular weight:287.71
  • IWP-2

    CAS:
    <p>IWP-2 is a Wnt pathway inhibitor and an ATP-competitive CK1δ inhibitor. IWP-2 inhibits self-renewal of embryonic stem cells. Cost effective and quality assured.</p>
    Formula:C22H18N4O2S3
    Purity:96.1% - 99.49%
    Color and Shape:Solid
    Molecular weight:466.6
  • SR-3029

    CAS:
    <p>SR-3029 is a potent and highly specific CK1δ/CK1ε inhibitor.</p>
    Formula:C23H19F3N8O
    Purity:99.64%
    Color and Shape:Solid
    Molecular weight:480.45
  • TTP 22

    CAS:
    <p>TTP 22: ATP-competitive CK2 inhibitor; IC50/Ki: 0.1 μM/40 nM; &gt;250x selective over JNK3, ROCK1, MET.</p>
    Formula:C16H14N2O2S2
    Purity:97.08% - 97.78%
    Color and Shape:Solid
    Molecular weight:330.42
  • LY294002

    CAS:
    <p>LY294002 (SF 1101) is a broad-spectrum inhibitor of PI3K, inhibiting PI3Kα, PI3Kδ, and PI3Kβ (IC50=0.5/0.57/0.97 μM).</p>
    Formula:C19H17NO3
    Purity:98% - 99.96%
    Color and Shape:Pale Yellow Solid
    Molecular weight:307.34
  • CKI-7 free base

    CAS:
    <p>CKI-7 free base is a potent and ATP-competitive inhibitor of casein kinase 1 (CK1; IC50: 6 μM; Ki: 8.5 μM) and a selective Cdc7 kinase inhibitor.</p>
    Formula:C11H12ClN3O2S
    Color and Shape:Solid
    Molecular weight:285.75
  • IC261

    CAS:
    <p>IC261 (SU-5607) is a novel inhibitor of CK1, triggers the mitotic checkpoint control. The IC50 of IC261 for CK1 was 16 μM and for Cdk5 is 4.5 mM.</p>
    Formula:C18H17NO4
    Purity:99.45% - 99.91%
    Color and Shape:Solid
    Molecular weight:311.33
  • LY-294002 hydrochloride

    CAS:
    <p>LY-294002 HCl (NSC 697286) is a stable PI3K inhibitor (IC50: 0.5-0.97 µM) and prevents autophagosome formation.</p>
    Formula:C19H17NO3·HCl
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:343.81
  • LH846

    CAS:
    <p>LH846 is a selective inhibitor of CK1δ (IC50 values are 290 nM, 1.3 uM and 2.5 uM for CK1δ, ε and α); exhibits no inhibitory activity at CK2.</p>
    Formula:C16H13ClN2OS
    Purity:90% - 98.26%
    Color and Shape:Solid
    Molecular weight:316.81
  • PF-4800567

    CAS:
    <p>PF-4800567 is a selective inhibitor of casein kinase 1ε (CK1ε; IC50 = 32 nM) with greater than 20-fold selectivity over CK1δ.</p>
    Formula:C17H18ClN5O2
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:359.81
  • Orobol

    CAS:
    <p>Orobol (3’,4’,5,7-tetrahydroxy-isoflavon) is an inhibitor of tyrosine-specific protein kinase and phosphatidylinositol turnover.</p>
    Formula:C15H10O6
    Purity:98% - 98%
    Color and Shape:Solid
    Molecular weight:286.24
  • D4476

    CAS:
    <p>D4476 (Casein Kinase I Inhibitor) is an effective, selective, and cell-permeant CK1 (casein kinase 1) inhibitor( IC50=300 nM in a cell-free assay).</p>
    Formula:C23H18N4O3
    Purity:99.7% - 99.96%
    Color and Shape:Solid
    Molecular weight:398.41
  • AS-252424

    CAS:
    <p>AS-252424 is a potent and selective inhibitor of PI3Kγ with IC50 of 33 nM; &gt;10 fold selectivity for PI3Kγ versus PI3Kα.</p>
    Formula:C14H8FNO4S
    Purity:99.06% - 99.09%
    Color and Shape:Solid
    Molecular weight:305.28
  • (E/Z)-GO289

    CAS:
    <p>(E/Z)-GO289, which strongly lengthened circadian period, is a potent and selective inhibitor of CK2.</p>
    Formula:C17H15BrN4O2S
    Purity:98.1%
    Color and Shape:Solid
    Molecular weight:419.3
  • Umbralisib

    CAS:
    <p>Umbralisib (TGR 1202) is a PI3Kδ inhibitor.</p>
    Formula:C31H24F3N5O3
    Purity:99.56% - 99.56%
    Color and Shape:White Solid
    Molecular weight:571.55
  • TBB

    CAS:
    <p>TBB (NSC-231634)(NSC-231634) is a highly selective, ATP/GTP-competitive inhibitor of casein kinase-2 (CK2).</p>
    Formula:C6HBr4N3
    Purity:98.51% - 99.45%
    Color and Shape:Off-White Solid
    Molecular weight:434.71
  • CKI-7

    CAS:
    <p>CKI-7 is a potent and ATP-competitive inhibitor of casein kinase 1 (CK1; IC50: 6 μM; Ki: 8.5 μM) and a selective Cdc7 kinase inhibitor.</p>
    Formula:C11H14Cl3N3O2S
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:358.67
  • Umbralisib hydrochloride

    CAS:
    <p>Umbralisib hydrochloride: PI3Kδ inhibitor; IC50=22.2 nM, EC50=24.3 nM; active vs CK1ε, EC50=6.0 μM.</p>
    Formula:C31H25ClF3N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:608.01
  • MLN8054

    CAS:
    <p>MLN8054 is a potent and selective Aurora A kinase inhibitor with an IC50 of 4 nM.</p>
    Formula:C25H15ClF2N4O2
    Purity:98.07% - 98.26%
    Color and Shape:Solid
    Molecular weight:476.86
  • NCC007

    CAS:
    <p>NCC007 is a novel CKIα and CKIδ dual inhibitors by structural modification of N9 and C2 position of longdaysin.</p>
    Formula:C22H28F3N7
    Purity:98.88%
    Color and Shape:Solid
    Molecular weight:447.5
  • CK2-IN-1

    CAS:
    <p>CK2 inhibitor</p>
    Formula:C14H9NO3
    Purity:97.28%
    Color and Shape:Solid
    Molecular weight:239.23
  • CK1-IN-1

    CAS:
    <p>CK1-IN-1, a CK1 inhibitor with IC50: 15nM CK1δ, 16nM CK1ε, 73nM p38σ; patent WO2015119579A1.</p>
    Formula:C24H15F2N3
    Purity:98.79%
    Color and Shape:Solid
    Molecular weight:383.39
  • TAK-715

    CAS:
    <p>TAK-715 is a p38 MAPK inhibitor for p38α.</p>
    Formula:C24H21N3OS
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:399.51
  • DMAT

    CAS:
    <p>DMAT (Casein kinase II Inhibitor) is a potent and specific inhibitor of CK2(IC50 value of 130 nM).</p>
    Formula:C9H7Br4N3
    Purity:99.48%
    Color and Shape:Solid
    Molecular weight:476.79
  • Silmitasertib

    CAS:
    <p>Silmitasertib (CX-4945) is a potent, orally bioavailable inhibitor of casein kinase 2 (CK2; Ki: 0.38 nM).</p>
    Formula:C19H12ClN3O2
    Purity:98% - 99.90%
    Color and Shape:Solid
    Molecular weight:349.77
  • PF-670462

    CAS:
    <p>PF-670462 is a potent (IC50 = 7.7 ± 2.2 nM) and selective (&gt;30-fold with respect to 42 additional kinases) inhibitor of CK1ε in isolated enzyme preparations.</p>
    Formula:C19H22Cl2FN5
    Purity:99.42% - 99.72%
    Color and Shape:Solid
    Molecular weight:410.32
  • XL413

    CAS:
    <p>XL-413 is an oral CDC7 kinase inhibitor, potentially blocking DNA replication, mitosis, and cancer cell growth.</p>
    Formula:C14H12ClN3O2
    Purity:98.40% - >99.99%
    Color and Shape:Solid
    Molecular weight:289.72
  • SSTC3

    CAS:
    <p>SSTC3 is a casein kinase 1α (CK1α) activator with potential antitumor activity that inhibits WNT signaling.</p>
    Formula:C23H17F3N4O3S2
    Purity:98.65% - 99.94%
    Color and Shape:Solid
    Molecular weight:518.53
  • AMG-548

    CAS:
    <p>AMG-548, oral p38α inhibitor (Ki=0.5 nM), &gt;1000x selectivity over p38γ/δ, blocks TNFα (IC50=3 nM), also inhibits Wnt/Casein kinase 1δ/ε.</p>
    Formula:C29H27N5O
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:461.56
  • SR-1277

    CAS:
    <p>SR-1277 is a potent, highly selective and ATP-competitive CK1δ/ε inhibitor, regulating Wee1 activity at the G2/M cell-cycle interface, and antiproliferative.</p>
    Formula:C21H19N9O3S
    Color and Shape:Solid
    Molecular weight:477.5
  • CK2/PIM1-IN-1

    CAS:
    <p>CK2/PIM1-IN-1 inhibits CK2 &amp; PIM1 (IC50s: 3.787 &amp; 4.327 μM), aimed for cancer research.</p>
    Formula:C15H9NO4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:331.37
  • 4,5,6,7-Tetrabromobenzimidazole

    CAS:
    <p>4,5,6,7-Tetrabromobenzimidazole is a selective and ATP-competitive inhibitor of protein kinase CK2 [1].</p>
    Formula:C7H2Br4N2
    Color and Shape:Solid
    Molecular weight:433.72
  • CK2-IN-9

    CAS:
    <p>CK2-IN-9, a potent and selective CK2 kinase inhibitor, exhibits an inhibitory concentration (IC50) of 3 nM against its target enzyme and hampers Wnt reporter</p>
    Formula:C23H29N9O
    Color and Shape:Solid
    Molecular weight:447.54
  • Quinalizarin

    CAS:
    <p>Quinalizarin, the most selective CK2 inhibitor, is superior to CX-4945 which is the first-in-class CK2 inhibitor.</p>
    Formula:C14H8O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:272.21
  • Tyrphostin AG 1112

    CAS:
    <p>Tyrphostin AG 1112 is a Bcr-Abl kinase blocker. It can activate the terminal differentiation of K562 cells and the purging of Ph+ cells.</p>
    Formula:C15H10N6
    Color and Shape:Solid
    Molecular weight:274.28
  • PF 4800567 hydrochloride

    CAS:
    <p>casein kinase 1ε inhibitor</p>
    Formula:C17H19Cl2N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:396.27
  • IQA

    CAS:
    <p>IQA is a casein kinase 2 (CK2) inhibitor.</p>
    Formula:C17H12N2O3
    Color and Shape:Solid
    Molecular weight:292.29
  • (R)-DRF053 dihydrochloride

    CAS:
    <p>cdk/CK1 inhibitor,potent and ATP-competitive</p>
    Formula:C23H29Cl2N7O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:490.43
  • TMCB

    CAS:
    <p>CK2 and ERK8 inhibitor</p>
    Formula:C11H9Br4N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:534.82
  • CK2-IN-6

    CAS:
    <p>CK2-IN-6: Potent CK2 inhibitor for cancer, inflammation, pain, and immune research.</p>
    Formula:C19H16ClN7O2
    Color and Shape:Solid
    Molecular weight:409.83
  • SRPIN-803

    CAS:
    <p>SRPIN-803 is a selective dual SRPK1 and CK2 inhibitor.</p>
    Formula:C14H9F3N4O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:370.31
  • Umbralisib sulfate

    CAS:
    <p>Umbralisib sulfate, an oral dual PI3Kδ/CK1ε inhibitor (EC50: 22.2 nM/6.0 μM), targets CLL T cells for blood cancer research.</p>
    Formula:C31H26F3N5O7S
    Color and Shape:Solid
    Molecular weight:669.63
  • Umbralisib tosylate

    CAS:
    <p>Umbralisib tosylate, an oral PI3Kδ/CK1ε inhibitor (EC50: 22.2 nM/6.0 μM), shows promise for CLL research.</p>
    Formula:C38H32F3N5O6S
    Color and Shape:Solid
    Molecular weight:743.75
  • BTX161

    CAS:
    <p>BTX161: potent CKIα degrader, surpasses Lenalidomide in AML, triggers DDR + p53, stabilizes MDM2.</p>
    Formula:C15H16N2O3
    Color and Shape:Solid
    Molecular weight:272.3
  • HDAC/CK2-IN-1

    CAS:
    <p>HDAC/CK2-IN-1 (compound 38) acts as an inhibitor of HDAC1 (IC 50 = 1.46 μM), HDAC6 (IC 50 = 0.66 μM), and CK2 (IC 50 = 3.67 μM). It demonstrates promising antiproliferative effects on various cell lines, including Jurkat, MCF-7, HCT-116, and HL-60.</p>
    Formula:C15H18Br4N4O2
    Color and Shape:Solid
    Molecular weight:605.95
  • CK2-IN-4

    CAS:
    <p>CK2-IN-4 is a protein kinase (CK2) inhibitor with an IC50 value of 8.6 µM.</p>
    Formula:C18H11N3O4S
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:365.36
  • CK2α-IN-1

    CAS:
    <p>CK2α-IN-1 is a selective non-ATP-competitive CK2α inhibitor with an IC50 of 7.0 µM and a Ki of 1.6 µM.CK2α-IN-1 exhibits potential anticancer activity and can</p>
    Formula:C16H11N3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:341.34
  • CK1-IN-2

    CAS:
    <p>CK1-IN-2 (compound Nr.4) is a potent CK1 inhibitor p38a, and is used in DUX4 overexpression-associated diseases, such as muscular dystrophy.</p>
    Formula:C17H12FN3O2
    Purity:99.31%
    Color and Shape:Solid
    Molecular weight:309.29
  • PI-828

    CAS:
    <p>PI-828 (LY 294002), a PI3K inhibitor, researches PI3K function and aids stem cell differentiation into mesoderm.</p>
    Formula:C19H18N2O3
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:322.36
  • XL413 xHCl

    CAS:
    <p>BMS-863233 HCl is an ATP-competitive Cdc7 inhibitor (IC50: 3.4 nM) that is potent and selective.BMS-863233 HCl inhibited CK2 and PIM1 with IC50 values of 215</p>
    Formula:C14H12ClN3O2·xHCl
    Purity:99.37% - 99.67%
    Color and Shape:Solid
    Molecular weight:326.18
  • BioE-1115

    CAS:
    <p>BioE-1115 is a selective and potent inhibitor of serine-threonine protein kinase (PASK, IC50 = 4 nM). BioE-1115 is a potent inhibitor of CK2α (IC50 = 10 μM).</p>
    Formula:C19H18FN3O2
    Purity:97.54%
    Color and Shape:Solid
    Molecular weight:339.36
  • Casein kinase 1δ-IN-1

    CAS:
    <p>Casein kinase 1δ-IN-1 (WAY-643895) is an inhibitor of casein kinase 1δ (CK1δ), which inhibits CK1δ.</p>
    Formula:C11H7N3OS
    Purity:99.46%
    Color and Shape:Solid
    Molecular weight:229.26
  • Ac-VDVAD-CHO

    CAS:
    <p>Ac-VDVAD-CHO is an inhibitor of caspase-2 and caspase-3 (IC50: 46 nM for caspase-2 and 15 nM for caspase-3) [1].</p>
    Formula:C23H37N5O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:543.57
  • ON 108600

    CAS:
    <p>ON 108600 is a chemical inhibitor targeting CK2 (Casein Kinase 2), TNIK, and DYRK1, demonstrating IC50 values of 0.016 μM and 0.007 μM for DYRK1A and DYRK1B, 0.</p>
    Formula:C22H14Cl2N2O6S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:537.39
  • Casein kinase 1δ-IN-5

    CAS:
    <p>Casein kinase 1δ-IN-5 is a potent and selective CK-1δ inhibitor, exhibiting an IC50 of 47 nM, and demonstrates neuroprotective and anti-inflammatory effects in</p>
    Formula:C16H11F3N2OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:336.33
  • Casein kinase 1δ-IN-10

    CAS:
    <p>Casein kinase 1δ-IN-10 is an inhibitor of casein kinase 1δ (CK1δ).</p>
    Formula:C21H17N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:359.38
  • TID43

    CAS:
    <p>TID43, a CK2 inhibitor, exhibits potent inhibition with an IC50 value of 0.3 μM. It is applicable in anti-angiogenic research [1].</p>
    Formula:C10H3I4NO4
    Color and Shape:Solid
    Molecular weight:708.755
  • XL413 hydrochloride

    CAS:
    <p>XL413 hydrochloride (BMS-863233 Hydrochloride) is a potent, selective and ATP competitive inhibitor of Cdc7. XL413 hydrochloride also inhibits CK2 and PIM1.</p>
    Formula:C14H13Cl2N3O2
    Purity:98.81% - 99.8%
    Color and Shape:Solid
    Molecular weight:326.18
  • Casein kinase 1δ-IN-4

    CAS:
    <p>"Casein kinase 1δ-IN-4 (compound 567) is a potent inhibitor of casein kinase 1δ with potential application in Alzheimer's disease research [1]."</p>
    Formula:C16H12N6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:320.37
  • Casein Kinase II Inhibitor IV

    CAS:
    <p>Casein kinase II inhibitor IV is an effective small molecule inducer, which can be used to induce epidermal keratinocyte differentiation.</p>
    Formula:C24H23N5O3
    Purity:99.65% - 99.75%
    Color and Shape:Solid
    Molecular weight:429.47
  • Casein kinase 1δ-IN-13

    CAS:
    Casein kinase1δ-IN-13 (compound 401) is an inhibitor of Casein kinase1δ. It is utilized in the research of neurodegenerative diseases.
    Formula:C15H13N3O2S
    Color and Shape:Solid
    Molecular weight:299.35
  • Casein kinase 1δ-IN-28

    CAS:
    <p>Casein kinase1δ-IN-28 (Compound 4) is an inhibitor of CK1ε, with an IC50 of 0.0146 μM. The human liver microsome metabolism rate for Casein kinase1δ-IN-28 is 52%.</p>
    Formula:C23H23FN6
    Color and Shape:Solid
    Molecular weight:402.467
  • CK1δ-IN-6

    CAS:
    <p>CK1δ-IN-6 (Compound 303) is an inhibitor of Casein kinase 1δ, with potential applications in Alzheimer's disease research.</p>
    Formula:C23H17N3O4
    Color and Shape:Solid
    Molecular weight:399.399
  • WAY-606344

    CAS:
    <p>WAY-606344 (Compound 97) is an inhibitor of Casein kinase 1δ and shows potential for Alzheimer's disease research.</p>
    Formula:C14H8ClN3O2
    Color and Shape:Solid
    Molecular weight:285.685