Transferase
Transferases are a large class of enzymes that catalyze the transfer of functional groups, such as methyl, glycosyl, and phosphate groups, from one molecule to another. Inhibitors of transferases are used to study a wide range of biological processes, including signal transduction, metabolism, and gene expression. These inhibitors are essential tools in research areas such as cancer, metabolic diseases, and epigenetics, where dysregulation of transferase activity is implicated. At CymitQuimica, we offer a comprehensive selection of transferase inhibitors to support your research in enzymology, cell signaling, and disease mechanisms.
Found 29 products of "Transferase"
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Cycloleucine
CAS:Cycloleucine is an antagonist of NMDA receptor associated glycine receptor with a Ki of 600 μM.Formula:C6H11NO2Purity:99.90%Color and Shape:SolidMolecular weight:129.16Opicapone
CAS:Opicapone (BIA 9-1067), a potent COMT inhibitor for Parkinson's studies, lowers cell ATP (IC50: 98 μM).Formula:C15H10Cl2N4O6Purity:98.17% - 99.36%Color and Shape:SolidMolecular weight:413.17ST6 Sialyltransferase 5
ST6Sialyltransferase5 (EC:2.4.3.3, ST6GALNAC5, SIAT7E, ST6 N-acetylgalactosaminide alpha-2,6-sialyltransferase 5) transfers sialic acid to N-acetylgalactosamine (GalNAc) residues. It may serve as a biomarker in cervical screening samples.Sinbaglustat
CAS:Sinbaglustat (OGT2378), an oral N-alkyl iminosugar, inhibits GCS/GBA2 and treats lysosomal storage and neurodegenerative disorders.
Formula:C11H23NO4Purity:99.93%Color and Shape:SolidMolecular weight:233.3Histamine glutarimide
CAS:Histamine glutarimide is a novel QPCT inhibitor that targets inflammatory processes like eosinophil migration, showing anti-asthmatic effects in animal models.Formula:C10H13N3O2Purity:99.79%Color and Shape:SolidMolecular weight:207.23Ref: TM-T202353
1mg185.00€5mg459.00€10mg657.00€25mg1,026.00€50mg1,415.00€100mg1,863.00€200mg2,547.00€L-739750 2HCl
L-739750 2HCl is a potent inhibitor of peptidomimetic farnesyltransferase, a novel pseudopeptide mimetic with potential anticancer activity.Formula:C23H41Cl2N3O6S2Purity:98.69% - 99.16%Color and Shape:SoildMolecular weight:590.62FUT8-IN-1
FUT8-IN-1 (Compound 37) is an inhibitor of α-1,6-fucosyltransferase (FUT8), with a dissociation constant (KD) of 49 nM and an IC50 around 50 µM. In the presence of FUT8, FUT8-IN-1 forms a highly active naphthoquinone imine intermediate, thereby inhibiting FUT8's enzymatic activity.Formula:C23H25ClN2OColor and Shape:SolidMolecular weight:380.91β-1,4-GALT1-IN-1
β-1,4-GALT1-IN-1 (Compound 6) is a β-1,4-GALT1 inhibitor with an IC50 value of 6.2 μM. It is applicable in studying various pathological conditions, including cancer, autoimmune diseases, and viral infections.Formula:C29H23NO10Color and Shape:SolidMolecular weight:545.494Ibiglustat
CAS:Ibiglustat (GZ402671) inhibits Glucosylceramide synthase, may treat Fabry disease by preventing GL-3 synthesis.Formula:C20H24FN3O2SPurity:97.97% - 98.81%Color and Shape:SolidMolecular weight:389.49Nitecapone
CAS:Nitecapone is a reversible inhibitor of S-COMT (IC50 values of 300 nM in rat liver)Formula:C12H11NO6Purity:98.39%Color and Shape:SolidMolecular weight:265.22Entacapone
CAS:Entacapone (OR-611) is a selective and reversible inhibitor of catechol-O-methyltransferase (COMT).Formula:C14H15N3O5Purity:98.80% - >99.99%Color and Shape:Yellow Crystalline SolidMolecular weight:305.29Ref: TM-T2216
5mg34.00€10mg49.00€25mg75.00€50mg90.00€100mg137.00€200mg197.00€500mg333.00€1mL*10mM (DMSO)50.00€Tipifarnib
CAS:Tipifarnib (IND 58359), a quinolinone, inhibits farnesyl transferase, blocks Ras activation, arrests cell growth, and curbs angiogenesis.Formula:C27H22Cl2N4OPurity:97.1% - 99.22%Color and Shape:Off-White To Pale Beige SolidMolecular weight:489.4PD 128042
CAS:PD 128042 (CI 976) is a potent orally active and selective ACAT inhibitor(IC50: 73 nM) and a potent lysophospholipid acyltransferase(LPAT) inhibitor.Formula:C23H39NO4Purity:99.79%Color and Shape:SolidMolecular weight:393.56CP-609754
CAS:CP-609754 shows selective inhibition of farnesyltransferase.Formula:C29H22ClN3O2Purity:99.86% - 99.87%Color and Shape:SolidMolecular weight:479.96Ref: TM-T38050
1mg55.00€5mg116.00€10mg187.00€25mg319.00€50mg449.00€100mg638.00€200mg840.00€1mL*10mM (DMSO)134.00€Tipifarnib (S enantiomer)
CAS:Tipifarnib S enantiomer ((S)-(-)-R-115777) is the S-enantiomer of Tipifarnib. Tipifarnib is a potent and specific farnesyltransferase inhibitor (IC50: 0.6 nM).Formula:C27H22Cl2N4OPurity:99.05%Color and Shape:SolidMolecular weight:489.4Ref: TM-T17102
1mg49.00€5mg102.00€10mg163.00€25mg284.00€50mg409.00€100mg577.00€200mg778.00€1mL*10mM (DMSO)109.00€Ervogastat
CAS:Ervogastat (PF-06865571) is a potent and well-tolerated diacylglycerol acyltransferase 2 inhibitor.Formula:C21H21N5O4Purity:99.97%Color and Shape:SolidMolecular weight:407.42Ref: TM-T9186
1mg123.00€5mg290.00€10mg485.00€25mg782.00€50mg1,063.00€100mg1,431.00€1mL*10mM (DMSO)301.00€3-O-Methyltolcapone
CAS:3-O-Methyltolcapone (Ro 40-7591) is a metabolite of Tolcapone which is a potent COMT inhibitor.Formula:C15H13NO5Purity:98%Color and Shape:SolidMolecular weight:287.27Lucerastat
CAS:Lucerastat（NBDGJ） is an orally available inhibitor of GCS for Fabry disease by reducing harmful substrates.. GCS is a key enzyme in sphingolipid synthesiss.Formula:C10H21NO4Purity:98%Color and Shape:SolidMolecular weight:219.28α-2,3-sialyltransferase-IN-1
CAS:α-2,3-sialyltransferase-IN-1 is a noncompetitive inhibitor of α-2,3-sialyltransferase(IC50 of 6 μM).Formula:C28H45NO6Purity:98% - 98%Color and Shape:SolidMolecular weight:491.66Prenyl-IN-1
CAS:Prenyl-IN-1 inhibits prenylation selectively, counters oxidative stress in Parkinson's.Formula:C28H24ClN5O2Purity:>99.99%Color and Shape:SolidMolecular weight:497.98
