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5-HT Receptor

5-HT Receptor

5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.

Found 940 products of "5-HT Receptor"

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  • Cyclopiazonic acid

    CAS:
    <p>Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.</p>
    Formula:C20H20N2O3
    Purity:99.27% - 99.80%
    Color and Shape:Solid
    Molecular weight:336.38
  • m-Chlorophenylbiguanide hydrochloride

    CAS:
    <p>m-Chlorophenylbiguanide hydrochloride is a 5-HT3 receptor agonist.</p>
    Formula:C8H11Cl2N5
    Purity:99.43% - 99.87%
    Color and Shape:Solid
    Molecular weight:248.11
  • Piperacetazine

    CAS:
    <p>Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.</p>
    Formula:C24H30N2O2S
    Purity:99.9% - 99.92%
    Color and Shape:Solid
    Molecular weight:410.57
  • Piboserod hydrochloride

    CAS:
    <p>Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.</p>
    Formula:C22H32ClN3O2
    Color and Shape:Solid
    Molecular weight:405.96
  • SB 204741

    CAS:
    <p>SB 204741 is a selective 5-HT2B antagonist with high affinity and pKi value of 7.1.</p>
    Formula:C14H14N4OS
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:286.35
  • Buclizine dihydrochloride

    CAS:
    <p>Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and</p>
    Formula:C28H33ClN2·2HCl
    Purity:98.05%
    Color and Shape:Off-White Powder
    Molecular weight:505.95
  • Tandospirone citrate

    CAS:
    <p>Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : 27 nM)</p>
    Formula:C27H37N5O9
    Purity:97.84% - 99.90%
    Color and Shape:Solid
    Molecular weight:575.61
  • NGB 2904

    CAS:
    <p>NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).</p>
    Formula:C28H29Cl2N3O
    Purity:98.79%
    Color and Shape:Solid
    Molecular weight:494.46
  • Zacopride hydrochloride

    CAS:
    <p>Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.</p>
    Formula:C15H20ClN3O2·HCl
    Purity:98.32%
    Color and Shape:Solid
    Molecular weight:346.26
  • 5-Benzyloxygramine

    CAS:
    <p>5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.</p>
    Formula:C18H20N2O
    Purity:99.13%
    Color and Shape:Solid
    Molecular weight:280.36
  • N-Desmethylclozapine

    CAS:
    <p>N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.</p>
    Formula:C17H17ClN4
    Purity:97.25% - 99.83%
    Color and Shape:Yellow Crystalline Solid
    Molecular weight:312.8
  • 4F 4PP oxalate

    CAS:
    <p>4F 4PP oxalate is a 5-HT2A antagonist.</p>
    Formula:C22H26FNO·C2H2O4
    Purity:97.34%
    Color and Shape:Solid
    Molecular weight:429.49
  • Sarpogrelate

    CAS:
    <p>Sarpogrelate (MCI-9042), an oral 5-HT2 antagonist, boosts platelet aggregation and aids in studying Buerger's disease.</p>
    Formula:C24H31NO6
    Color and Shape:Solid
    Molecular weight:429.51
  • Spiperone hydrochloride

    CAS:
    <p>5-HT2A serotonin and selective D2-like dopamine receptor antagonist</p>
    Formula:C23H27ClFN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:431.93
  • Harmine hydrochloride

    CAS:
    <p>Harmine hydrochloride (telepathine hydrochloride) is extracted from Peganum Harmala Genus.</p>
    Formula:C13H13ClN2O
    Purity:99.61% - >99.99%
    Color and Shape:Yellow To Slightly Green Crystalline Powder
    Molecular weight:248.71
  • Ondansetron

    CAS:
    <p>Ondansetron (GR 38032) is a serotonin 5-HT3 receptor antagonist used mainly as an antiemetic.</p>
    Formula:C18H19N3O
    Purity:99.92%
    Color and Shape:White To Yellow Crystals
    Molecular weight:293.36
  • SB 242084 dihydrochloride

    CAS:
    <p>SB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively.</p>
    Formula:C21H21Cl3N4O2
    Color and Shape:Solid
    Molecular weight:467.78
  • S1RA hydrochloride

    CAS:
    <p>S1RA hydrochloride (E-52862 hydrochloride) is an effective and specific sigma-1 receptor(σ1R, Ki: 17 nM) antagonist, and has good selectivity against σ2R (Ki &gt;</p>
    Formula:C20H24ClN3O2
    Purity:98% - 99.84%
    Color and Shape:Solid
    Molecular weight:373.87
  • SKF-83566

    CAS:
    <p>SKF-83566: Blood-brain permeable, orally active D1 dopamine antagonist; weaker 5-HT2 antagonist, Ki=11 nM.</p>
    Formula:C17H18BrNO
    Purity:95.00% - 99.82%
    Color and Shape:Solid
    Molecular weight:332.23
  • Dasotraline hydrochloride

    CAS:
    <p>Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.</p>
    Formula:C16H16Cl3N
    Purity:98.92% - 99.6%
    Color and Shape:Solid
    Molecular weight:328.66
  • ML 10302

    CAS:
    <p>ML 10302 is a potent 5-HT4 agonist with Ki of 1.07 nM, boosts bowel movement, and may aid in neurology research.</p>
    Formula:C15H21ClN2O3
    Color and Shape:Solid
    Molecular weight:312.79
  • SAX-187

    CAS:
    <p>SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.</p>
    Formula:C15H13ClN4O2S2
    Purity:97.82% - 98%
    Color and Shape:Solid
    Molecular weight:380.87
  • L-745870 trihydrochloride

    CAS:
    <p>L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.</p>
    Formula:C18H22Cl4N4
    Purity:97.52%
    Color and Shape:Solid
    Molecular weight:436.21
  • Rotigotine-

    CAS:
    <p>Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.</p>
    Formula:C19H25NOS
    Purity:98.08% - 99.59%
    Color and Shape:Solid
    Molecular weight:315.47
  • Zotepine

    CAS:
    <p>Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,</p>
    Formula:C18H18ClNOS
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:331.86
  • Metoclopramide

    CAS:
    <p>Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.</p>
    Formula:C14H22ClN3O2
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:299.80
  • Desvenlafaxine succinate hydrate

    CAS:
    <p>Desvenlafaxine succinate hydrate (WY 45233 Succinate) is an antidepressant of the serotonin-norepinephrine reuptake inhibitor (SNRI).</p>
    Formula:C20H33NO7
    Purity:99.26%
    Color and Shape:White Crystalline Powde
    Molecular weight:399.48
  • Harmine

    CAS:
    <p>Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.</p>
    Formula:C13H12N2O
    Purity:98.29% - 99.92%
    Color and Shape:Off-White Solid
    Molecular weight:212.25
  • Rotigotine Hydrochloride

    CAS:
    <p>Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.</p>
    Formula:C19H26ClNOS
    Purity:99.53% - 99.56%
    Color and Shape:Almost White To White Crystalline Powder
    Molecular weight:351.93
  • Ramosetron hydrochloride

    CAS:
    <p>Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.</p>
    Formula:C17H18ClN3O
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:315.8
  • Pergolide mesylate

    CAS:
    <p>Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.</p>
    Formula:C20H30N2O3S2
    Purity:99.70%
    Color and Shape:White To Off-White Solid
    Molecular weight:410.59
  • Trazodone

    CAS:
    <p>Trazodone (AF-1161), a 5-HT 2A/2C receptor antagonist, is used as an antidepressant for treating major anxiety disorders and depressive disorder.</p>
    Formula:C19H22ClN5O
    Purity:99.79% - 99.92%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:371.86
  • 1-(1-Naphthyl) piperazine hydrochloride

    CAS:
    <p>1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple</p>
    Formula:C14H17ClN2
    Purity:98.27%
    Color and Shape:Solid
    Molecular weight:248.75
  • A-582941 dihydrochloride

    CAS:
    <p>A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partial</p>
    Formula:C17H22Cl2N4
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:353.29
  • Sertindole

    CAS:
    <p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>
    Formula:C24H26ClFN4O
    Purity:99.87% - 99.92%
    Color and Shape:Off-White To Pale Yellow Solid
    Molecular weight:440.94
  • Rizatriptan benzoate

    CAS:
    <p>Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraine</p>
    Formula:C22H25N5O2
    Purity:99% - 99.79%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:391.47
  • PU02

    CAS:
    <p>PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.</p>
    Formula:C16H12N4S
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:292.36
  • Cinitapride

    CAS:
    <p>Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.</p>
    Formula:C21H30N4O4
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:402.49
  • Lurasidone hydrochloride

    CAS:
    <p>Lurasidone HCl: Atypical antipsychotic, treats schizophrenia &amp; bipolar, affects dopamine, serotonin &amp; adrenergic receptors.</p>
    Formula:C28H36N4O2S·HCl
    Purity:99.51%
    Color and Shape:Solid
    Molecular weight:529.14
  • Sarpogrelate hydrochloride

    CAS:
    <p>Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.</p>
    Formula:C24H32ClNO6
    Purity:99.73%
    Color and Shape:Colorless Liquid
    Molecular weight:465.97
  • Clozapine N-Oxide

    CAS:
    <p>View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.</p>
    Formula:C18H19ClN4O
    Purity:98.43% - 99.94%
    Color and Shape:Solid
    Molecular weight:342.82
  • Flibanserin hydrochloride

    CAS:
    <p>Flibanserin HCl: oral 5-HT1A agonist &amp; 5-HT2A antagonist, Ki values 1 nM &amp; 49 nM, for HSDD, has antidepressant/anxiolytic properties.</p>
    Formula:C20H22ClF3N4O
    Color and Shape:Solid
    Molecular weight:426.87
  • 5-HT1A modulator 2 hydrochloride

    CAS:
    <p>5-HT1A modulator 2 hydrochloride is a modulator of 5-HT1A showing an affinity of 53 nM for 5-HT1A binding.</p>
    Formula:C11H16ClNO
    Purity:98.5%
    Color and Shape:Solid
    Molecular weight:213.7
  • MK 212 hydrochloride

    CAS:
    <p>MK 212 hydrochloride is a 5-HT2C receptor agonist</p>
    Formula:C8H11ClN4·HCl
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:235.12
  • Eptapirone

    CAS:
    <p>Eptapirone (F 11440) is a highly effective and selective 5-HT1A receptor agonist with marked antidepressant and anxiolytic potential.</p>
    Formula:C16H23N7O2
    Purity:99.39% - 99.65%
    Color and Shape:Solid
    Molecular weight:345.4
  • Brexpiprazole HCl

    CAS:
    <p>Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.</p>
    Formula:C25H27N3O2S·xHCl
    Purity:99.05%
    Color and Shape:Solid
    Molecular weight:433.6
  • Nemifitide acetate(173240-15-8 free base)


    <p>Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.</p>
    Formula:C35H47FN10O8
    Purity:97.97%
    Color and Shape:Solid
    Molecular weight:754.85
  • Brexpiprazole

    CAS:
    <p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>
    Formula:C25H27N3O2S
    Purity:99.06% - 99.96%
    Color and Shape:Solid
    Molecular weight:433.57
  • 8-Hydroxy-DPAT hydrobromide

    CAS:
    <p>8-Hydroxy-DPAT hydrobromide (8-OH-DPAT hydrobromide) (8-OH-DPAT hydrobromide) is a potent and selective 5-HT1A agonist with a pIC50 of 8.19.</p>
    Formula:C16H26BrNO
    Purity:98.90% - 99.09%
    Color and Shape:Solid
    Molecular weight:328.29
  • Ansofaxine hydrochloride

    CAS:
    <p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>
    Formula:C24H32ClNO3
    Purity:99.57% - 99.77%
    Color and Shape:Solid
    Molecular weight:417.97
  • Geissoschizine methyl ether

    CAS:
    <p>Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.</p>
    Formula:C22H26N2O3
    Purity:99.24% - 99.68%
    Color and Shape:Solid
    Molecular weight:366.45
  • Tropisetron

    CAS:
    <p>Tropisetron (ICS 205-930) is an α7-nicotinic receptor agonist and 5-HT3 receptor antagonist with Kis of 6.9 nM and 5.3 nM, respectively.</p>
    Formula:C17H20N2O2
    Purity:99.68%
    Color and Shape:White Solid
    Molecular weight:284.35
  • Sevoflurane

    CAS:
    <p>Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.</p>
    Formula:C4H3F7O
    Purity:98%
    Color and Shape:Less Oil Colorless Oil
    Molecular weight:200.05
  • SB399885

    CAS:
    <p>SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.</p>
    Formula:C18H21Cl2N3O4S
    Purity:98.94%
    Color and Shape:Solid
    Molecular weight:446.35
  • LY334370

    CAS:
    <p>LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nM</p>
    Formula:C21H22FN3O
    Purity:99.32%
    Color and Shape:Solid
    Molecular weight:351.42
  • Lurasidone

    CAS:
    <p>Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6</p>
    Formula:C28H36N4O2S
    Purity:99.78% - 99.91%
    Color and Shape:Solid
    Molecular weight:492.68
  • Eltoprazine

    CAS:
    <p>Eltoprazine(DU28853) is a serenic or antiaggressive agent which as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.</p>
    Formula:C12H16N2O2
    Color and Shape:Solid
    Molecular weight:220.27
  • Perospirone

    CAS:
    <p>Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.</p>
    Formula:C23H30N4O2S
    Purity:99.23%
    Color and Shape:White Powder
    Molecular weight:426.57
  • ARC-239

    CAS:
    <p>ARC-239 is an agonist of α2-adrenergic receptor.</p>
    Formula:C24H29N3O3
    Color and Shape:Solid
    Molecular weight:407.51
  • VUF 10166

    CAS:
    <p>VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.</p>
    Formula:C13H15ClN4
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:262.74
  • (S)-Amisulpride

    CAS:
    <p>(S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist.</p>
    Formula:C17H27N3O4S
    Purity:98.38%
    Color and Shape:Solid
    Molecular weight:369.48
  • Puerarin

    CAS:
    <p>Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known as isoflavonoid C-glycosides. It is a 5-HT2C receptor antagonist.</p>
    Formula:C21H20O9
    Purity:98.90% - 99.21%
    Color and Shape:Yellow Brown Fine Powder
    Molecular weight:416.38
  • Nelotanserin

    CAS:
    <p>Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).</p>
    Formula:C18H15BrF2N4O2
    Purity:98.42% - 99.88%
    Color and Shape:Solid
    Molecular weight:437.24
  • S 14506 HCl

    CAS:
    <p>S 14506 HCl: Strong 5-HT1A agonist; pKi - 9.0 (5-HT1A), 6.6 (5-HT1B/C), &lt;6.0 (5-HT3).</p>
    Formula:C24H26FN3O2
    Color and Shape:Solid
    Molecular weight:407.48
  • RU 24969 free base

    CAS:
    <p>RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.</p>
    Formula:C14H16N2O
    Purity:97.38%
    Color and Shape:Solid
    Molecular weight:228.29
  • Azaphen

    CAS:
    <p>Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.</p>
    Formula:C16H21Cl2N5O
    Purity:97.62%
    Color and Shape:Solid
    Molecular weight:370.28
  • Alosetron (Hydrochloride(1:X))

    CAS:
    <p>Alosetron Hydrochloride is a selective 5-HT3 antagonist for treating IBS.</p>
    Formula:C17H18ClN4O
    Color and Shape:Solid
    Molecular weight:329.11691
  • (E)-3,4,5-Trimethoxycinnamic acid

    CAS:
    <p>(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.</p>
    Formula:C12H14O5
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:238.24
  • Loxapine hydrochloride

    CAS:
    <p>Loxapine hydrochloride, an oral anti-psychotic, inhibits dopamine and blocks 5-HT receptors.</p>
    Formula:C18H19Cl2N3O
    Color and Shape:Solid
    Molecular weight:364.27
  • Cinanserin

    CAS:
    <p>Cinanserin is a serotonin 5-HT2 antagonist.</p>
    Formula:C20H24N2OS
    Color and Shape:Solid
    Molecular weight:340.48
  • Serotonin hydrochloride

    CAS:
    <p>Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (</p>
    Formula:C10H13ClN2O
    Purity:98.05% - 99.93%
    Color and Shape:White To Cream Powder
    Molecular weight:212.676
  • WAY-100635 Monomaleate

    CAS:
    <p>WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.</p>
    Formula:C25H34N4O2·C4H4O4
    Purity:98.44% - 99.46%
    Color and Shape:Solid
    Molecular weight:538.64
  • Piboserod

    CAS:
    <p>Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.</p>
    Formula:C22H31N3O2
    Purity:97.21% - 99.49%
    Color and Shape:Solid
    Molecular weight:369.5
  • Almotriptan Malate

    CAS:
    <p>Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.</p>
    Formula:C17H25N3O2S·C4H6O5
    Purity:99.95%
    Color and Shape:Pale Yellow Solid
    Molecular weight:469.55
  • Risperidone hydrochloride

    CAS:
    <p>Risperidone hydrochloride blocks 5-HT2, inhibits P-glycoprotein, and antagonizes D2 receptors (Ki: 5-HT2A - 4.8 nM, D2 - 5.9 nM).</p>
    Formula:C23H28ClFN4O2
    Color and Shape:Solid
    Molecular weight:446.95
  • Ocaperidone

    CAS:
    <p>Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.</p>
    Formula:C24H25FN4O2
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:420.48
  • Phenylbiguanide

    CAS:
    <p>Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)</p>
    Formula:C8H11N5
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:177.21
  • Sumatriptan hydrochloride

    CAS:
    <p>Sumatriptan hydrochloride (GR 43175), an oral 5-HT1 receptor agonist, treats migraines; Ki: 5-HT1D - 17 nM, 5-HT1B - 27 nM, 5-HT1A - 100 nM.</p>
    Formula:C14H22ClN3O2S
    Color and Shape:Solid
    Molecular weight:331.86
  • Escitalopram Oxalate

    CAS:
    <p>Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.</p>
    Formula:C22H23FN2O5
    Purity:97.39% - 99.73%
    Color and Shape:White Solid
    Molecular weight:414.43
  • BRL-15572 hydrochloride

    CAS:
    <p>BRL-15572 hydrochloride: selective h5-HT1D antagonist with high affinity; useful for studying h5-HT1D responses.</p>
    Formula:C25H28Cl2N2O
    Color and Shape:Solid
    Molecular weight:443.41
  • 4i

    CAS:
    <p>4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.</p>
    Formula:C16H12ClN3O
    Purity:99.49%
    Color and Shape:Solid
    Molecular weight:297.74
  • SB 242084

    CAS:
    <p>SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.</p>
    Formula:C21H19ClN4O2
    Purity:99.75% - ≥98%
    Color and Shape:Solid
    Molecular weight:394.85
  • PNU 22394 hydrochloride

    CAS:
    <p>PNU 22394 hydrochloride is a 5-HT2C agonist and partial 5-HT2A/5-HT2B agonist</p>
    Formula:C13H17ClN2
    Purity:97.83%
    Color and Shape:Solid
    Molecular weight:236.74
  • Amitriptyline

    CAS:
    <p>Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.</p>
    Formula:C20H23N
    Purity:98.24% - 99.64%
    Color and Shape:Crystals Solid
    Molecular weight:277.4
  • Pirenperone

    CAS:
    <p>Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.</p>
    Formula:C23H24FN3O2
    Purity:99.2%
    Color and Shape:Solid
    Molecular weight:393.45
  • Quipazine

    CAS:
    <p>Quipazine: 5-HT agonist, Ki 1.4 nM at 5-HT3R, anti-SARS-CoV-2 (EC50 31.64 μM), for neurological research.</p>
    Formula:C13H15N3
    Color and Shape:Solid
    Molecular weight:213.28
  • SR 57227 hydrochloride

    CAS:
    <p>SR 57227A (SR 57227 hydrochloride) is a potent, orally active and selective 5-HT3 receptor agonist. It with ability to cross the blood brain barrier.</p>
    Formula:C10H14ClN3·HCl
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:248.15
  • Ramosetron

    CAS:
    <p>Ramosetron 是一种血清素 5-HT3 受体拮抗剂,用于治疗恶心和呕吐。它被认为比其他一代 5-HT3 拮抗剂如昂丹司琼具有更高的效力和更长的止吐作用。它还适用于治疗“男性以腹泻为主的肠易激综合征”。它仅获准在日本和选定的东南亚国家使用。</p>
    Formula:C17H17N3O
    Purity:98.84%
    Color and Shape:Solid
    Molecular weight:279.34
  • F-15599

    CAS:
    <p>F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).</p>
    Formula:C19H21ClF2N4O
    Purity:98.72%
    Color and Shape:Solid
    Molecular weight:394.85
  • 7-Amino-4-(trifluoromethyl)coumarin

    CAS:
    <p>7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.</p>
    Formula:C10H6F3NO2
    Purity:97.31% - 97.84%
    Color and Shape:Yellow Powder
    Molecular weight:229.16
  • Tiprenolol

    CAS:
    <p>Tiprenolol is a beta adrenergic receptor antagonist.[1]</p>
    Formula:C13H21NO2S
    Purity:99.43%
    Color and Shape:Solid
    Molecular weight:255.38
  • BMY 7378 dihydrochloride

    CAS:
    <p>BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.</p>
    Formula:C22H33Cl2N3O3
    Purity:97.32% - 99.08%
    Color and Shape:Solid
    Molecular weight:458.42
  • Tandospirone hydrochloride

    CAS:
    <p>Tandospirone (SM-3997) HCl: potent 5-HT1A partial agonist; Ki: 27 nM; anxiolytic, antidepressant, for CNS disorder research.</p>
    Formula:C21H30ClN5O2
    Color and Shape:Solid
    Molecular weight:419.95
  • γ-Mangostin

    CAS:
    <p>Gamma-Mangostin (Normangostin) has free radical scavenging activity, and antiproliferative and apoptotic activity. Gamma-Mangostin is an antihypertensive agent.</p>
    Formula:C23H24O6
    Purity:98.55% - 99.08%
    Color and Shape:Solid
    Molecular weight:396.43
  • Xanthotoxol

    CAS:
    <p>Xanthotoxol (Psoralen) is a bioactive furocoumarin with anti-inflammatory, antioxidant, 5-HT antagonist, and neuroprotective properties.</p>
    Formula:C11H6O4
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:202.16
  • TG6-10-1

    CAS:
    <p>TG6-10-1 is an EP2 antagonist.</p>
    Formula:C23H23F3N2O4
    Purity:99.66% - ≥95%
    Color and Shape:Solid
    Molecular weight:448.43
  • Cariprazine

    CAS:
    <p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>
    Formula:C21H32Cl2N4O
    Purity:99.68% - 99.87%
    Color and Shape:Solid
    Molecular weight:427.41
  • PRX-07034 hydrochloride

    CAS:
    <p>PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.</p>
    Formula:C21H29Cl2N3O4S
    Purity:98.5%
    Color and Shape:Solid
    Molecular weight:490.44
  • Aripiprazole monohydrate

    CAS:
    <p>Aripiprazole (OPC-14597) is a potent D2 partial agonist and inverse agonist of 5-HT2 receptors, used for schizophrenia and COVID-19 studies.</p>
    Formula:C23H29Cl2N3O3
    Color and Shape:Solid
    Molecular weight:466.4
  • MDL 100009

    CAS:
    <p>MDL 100009, the S-enantiomer of MDL 100151 and the opposite enantiomer of MDL 100907, is a selective antagonist of 5-HT2A.</p>
    Formula:C22H28FNO3
    Purity:98.96%
    Color and Shape:Solid
    Molecular weight:373.46