5-HT Receptor
5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.
Found 1025 products of "5-HT Receptor"
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3-Hydroxy agomelatine D3
CAS:3-Hydroxy agomelatine D3 is a deuterated metabolite of Agomelatine and a 5-HT2C antagonist (IC50: 3.2 μM, Ki: 1.8 μM).Formula:C15H17NO3Purity:98%Color and Shape:SolidMolecular weight:262.32Olanzapine D3
CAS:Olanzapine D3 is the deuterium labeled Olanzapine.Formula:C17H20N4SPurity:98%Color and Shape:SolidMolecular weight:315.45BW 723C86
CAS:BW 723C86 is a 5-HT2B receptor agonist with anxiolytic effects, inducing overeating and reduced grooming in rats, useful in studying neurological disorders.Formula:C16H19ClN2OSPurity:99.35%Color and Shape:SolidMolecular weight:322.85Flibanserin-d4
CAS:Flibanserin: Serotonin 5-HT1A agonist (Ki=1 nM), 5-HT2A antagonist (49 nM). Flibanserin D4 is deuterium-labeled.Formula:C20H21F3N4OPurity:98%Color and Shape:SolidMolecular weight:394.43Aramisulpride
CAS:Aramisulpride is a dual antagonist of the dopamine D2 receptor and serotonin receptor, primarily utilized for investigating metabolic disorders.Formula:C17H27N3O4SColor and Shape:SolidMolecular weight:369.48Paliperidone Palmitate
CAS:Paliperidone: atypical antipsychotic, dopamine & serotonin antagonist, affects α1/α2 adrenergic and H1 histamine receptors.Formula:C39H57FN4O4Purity:98%Color and Shape:SolidMolecular weight:664.89Granisetron
CAS:Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.
Formula:C18H24N4OColor and Shape:SolidMolecular weight:312.41Agomelatine (L(+)-Tartaric acid)
CAS:Agomelatine (L(+)-Tartaric acid) is an MT1/MT2 agonist and selective 5-HT2C antagonist, supporting melatonergic and serotonergic signaling studies in neuroscience.Formula:C19H23NO8Purity:99.79%Color and Shape:SolidMolecular weight:393.39Asenapine hydrochloride
CAS:Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors with antipsychotic effects.Formula:C17H17Cl2NOColor and Shape:SolidMolecular weight:322.23cis-(Z)-Flupentixol dihydrochloride
CAS:cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.Formula:C23H27Cl2F3N2OSPurity:98.07%Color and Shape:SolidMolecular weight:507.441-Phenylbiguanide HCl
CAS:Compound PDK0269, as 5-HT3 receptor agonists(3–100 μM, pEC50 5.05±0.06), acutely increased XII (hypoglossal) burst frequency and regularity, and decreased bursts/episode . Phenylbiguanide produced a dose-related (10-500 microM) increase in the release of dopamine (280-2000%). When nomifensine (5 microM) was included in the Ringer solution, the effect of Compound PDK0269 on the release of dopamine was ameliorated or inhibited.Formula:C8H12ClN5Purity:99.31%Color and Shape:SolidMolecular weight:213.67Levomepromazine
CAS:Levomepromazine (Methotrimeprazine) is a Ca2+ release inducer with antiviral, anti-inflammatory, neuroprotective, sedative, and anti-nociceptive activities.Formula:C19H24N2OSPurity:99.15%Color and Shape:SolidMolecular weight:328.47Eplivanserin (mixture)
CAS:Eplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist,Formula:C19H21FN2O2Color and Shape:SolidMolecular weight:328.387WAY-100635
CAS:WAY-100635 is a potent 5-HT 1A receptor antagonist pyramidal neuron firing frequency during conditioned reflexes; a dopamine D4 receptor agonist .Formula:C25H34N4O2Purity:98.972%Color and Shape:SolidMolecular weight:422.56(Rac)-Rotigotine hydrochloride
CAS:(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, a partial the 5-HT1A receptor agonist.Formula:C19H26ClNOSColor and Shape:SolidMolecular weight:351.93SB-200646A
CAS:SB-200646A: oral 5-HT2B/2C antagonist; higher affinity than 5-HT2A (pKi: 7.5, 6.9 vs 5.2); anxiolytic with in vivo effects.Formula:C15H15ClN4OPurity:98%Color and Shape:SolidMolecular weight:302.76Alosetron D3 Hydrochloride
CAS:Alosetron D3 (GR 68755 D3) Hydrochloride is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.Formula:C17H19ClN4OPurity:98%Color and Shape:SolidMolecular weight:333.83Sumatriptan
CAS:Sumatriptan (GR 43175 free base) is a 5-HT1 receptor agonist with anti-inflammatory activity used in acute migraine and acute myocardial infarction.Formula:C14H21N3O2SPurity:99.93%Color and Shape:White To Off-White Crystalline PowderMolecular weight:295.4Cariprazine D6
CAS:Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).Formula:C21H26D6Cl2N4OPurity:98%Color and Shape:SolidMolecular weight:433.45Vilazodone-d8
CAS:Vilazodone D8 is a deuterium-labeled vilazodone. Vilazodone is a combined inhibitor of serotonin specific reuptake (SSRI) and agonist of 5-HT1A receptor partial.Formula:C26H27N5O2Purity:98%Color and Shape:SolidMolecular weight:449.57Fluvoxamine
CAS:Fluvoxamine (DU-23000) is a selective, orally available 5-HT and serotonin reuptake inhibitor (SSRI) exhibiting antidepressant effects.Formula:C15H21F3N2O2Purity:99.91%Color and Shape:SolidMolecular weight:318.33Spiroxatrine
CAS:Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the study of diseases related to the cardiovascular system.Formula:C22H25N3O3Purity:99.94%Color and Shape:SolidMolecular weight:379.453-Hydroxy agomelatine
CAS:3-Hydroxy agomelatine (3-Hydroxyagomelatine) is a 5-HT2C receptor antagonist used in the study of neurological disorders.Formula:C15H17NO3Color and Shape:SolidMolecular weight:259.3LY310762
CAS:LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.Formula:C24H27FN2O2·HClPurity:99.8%Color and Shape:SolidMolecular weight:430.94Sarpogrelate hydrochloride
CAS:Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.Formula:C24H32ClNO6Purity:99.73%Color and Shape:Colorless LiquidMolecular weight:465.97Cyclopiazonic acid
CAS:Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.Formula:C20H20N2O3Purity:99.27% - 99.80%Color and Shape:SolidMolecular weight:336.38m-Chlorophenylbiguanide hydrochloride
CAS:m-Chlorophenylbiguanide hydrochloride is a 5-HT3 receptor agonist.Formula:C8H11Cl2N5Purity:99.43% - 99.87%Color and Shape:SolidMolecular weight:248.11Cinitapride
CAS:Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.Formula:C21H30N4O4Purity:99.52%Color and Shape:SolidMolecular weight:402.49Ref: TM-T21385
1mg73.00€5mg155.00€10mg240.00€25mg479.00€50mg692.00€100mg973.00€1mL*10mM (DMSO)177.00€Piboserod hydrochloride
CAS:Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.Formula:C22H32ClN3O2Color and Shape:SolidMolecular weight:405.96SB 204741
CAS:SB 204741 is a selective 5-HT2B antagonist with high affinity and pKi value of 7.1.Formula:C14H14N4OSPurity:99.83%Color and Shape:SolidMolecular weight:286.35Ref: TM-T23312
1mg38.00€2mg50.00€5mg84.00€10mg119.00€25mg234.00€50mg439.00€100mg600.00€200mg837.00€1mL*10mM (DMSO)84.00€Amitriptyline
CAS:Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.Formula:C20H23NPurity:98.24% - 99.64%Color and Shape:Crystals SolidMolecular weight:277.4Buclizine dihydrochloride
CAS:Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic andFormula:C28H33ClN2·2HClPurity:98.05%Color and Shape:Off-White PowderMolecular weight:505.95Tandospirone citrate
CAS:Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : 27 nM)Formula:C27H37N5O9Purity:97.84% - 99.90%Color and Shape:SolidMolecular weight:575.61Brexpiprazole HCl
CAS:Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.Formula:C25H27N3O2S·xHClPurity:99.05%Color and Shape:SolidMolecular weight:433.6Ref: TM-T8690
1mg124.00€5mg271.00€10mg408.00€25mg672.00€50mg945.00€100mg1,279.00€500mg2,547.00€1mL*10mM (DMSO)319.00€Ansofaxine hydrochloride
CAS:Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).Formula:C24H32ClNO3Purity:99.57% - 99.77%Color and Shape:SolidMolecular weight:417.97Tropisetron
CAS:Tropisetron (ICS 205-930) is an α7-nicotinic receptor agonist and 5-HT3 receptor antagonist with Kis of 6.9 nM and 5.3 nM, respectively.Formula:C17H20N2O2Purity:99.68%Color and Shape:White SolidMolecular weight:284.354F 4PP oxalate
CAS:4F 4PP oxalate is a 5-HT2A antagonist.
Formula:C22H26FNO·C2H2O4Purity:97.34%Color and Shape:SolidMolecular weight:429.49Sarpogrelate
CAS:Sarpogrelate (MCI-9042), an oral 5-HT2 antagonist, boosts platelet aggregation and aids in studying Buerger's disease.Formula:C24H31NO6Color and Shape:SolidMolecular weight:429.51Harmine hydrochloride
CAS:Harmine hydrochloride (telepathine hydrochloride) is extracted from Peganum Harmala Genus.Formula:C13H13ClN2OPurity:99.61% - >99.99%Color and Shape:Yellow To Slightly Green Crystalline PowderMolecular weight:248.71Nelotanserin
CAS:Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).Formula:C18H15BrF2N4O2Purity:98.42% - 99.88%Color and Shape:SolidMolecular weight:437.24Ref: TM-T7350
1mg38.00€2mg50.00€5mg84.00€10mg113.00€25mg178.00€50mg333.00€100mg495.00€500mg1,071.00€1mL*10mM (DMSO)80.00€Ondansetron
CAS:Ondansetron (GR 38032) is a serotonin 5-HT3 receptor antagonist used mainly as an antiemetic.Formula:C18H19N3OPurity:99.92%Color and Shape:White To Yellow CrystalsMolecular weight:293.36SB 242084 dihydrochloride
CAS:SB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively.Formula:C21H21Cl3N4O2Color and Shape:SolidMolecular weight:467.78S1RA hydrochloride
CAS:S1RA hydrochloride (E-52862 hydrochloride) is an effective and specific sigma-1 receptor(σ1R, Ki: 17 nM) antagonist, and has good selectivity against σ2R (Ki >Formula:C20H24ClN3O2Purity:98% - 99.84%Color and Shape:SolidMolecular weight:373.87Ref: TM-T4229
1mg35.00€5mg75.00€10mg105.00€25mg205.00€50mg334.00€100mg492.00€500mg973.00€1mL*10mM (DMSO)84.00€Sevoflurane
CAS:Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.Formula:C4H3F7OPurity:98%Color and Shape:Less Oil Colorless OilMolecular weight:200.05Ref: TM-T22425
2mg39.00€5mg54.00€10mg75.00€25mg110.00€50mg158.00€100mg226.00€200mg339.00€1mL*10mM (DMSO)56.00€Geissoschizine methyl ether
CAS:Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.Formula:C22H26N2O3Purity:99.24% - 99.68%Color and Shape:SolidMolecular weight:366.45Ref: TM-TN1032
1mg130.00€2mg187.00€5mg319.00€10mg485.00€25mg770.00€50mg1,035.00€100mg1,395.00€1mL*10mM (DMSO)326.00€Spiperone hydrochloride
CAS:5-HT2A serotonin and selective D2-like dopamine receptor antagonistFormula:C23H27ClFN3O2Purity:98%Color and Shape:SolidMolecular weight:431.93SKF-83566
CAS:SKF-83566: Blood-brain permeable, orally active D1 dopamine antagonist; weaker 5-HT2 antagonist, Ki=11 nM.Formula:C17H18BrNOPurity:95.00% - 99.82%Color and Shape:SolidMolecular weight:332.23MK 212 hydrochloride
CAS:MK 212 hydrochloride is a 5-HT2C receptor agonistFormula:C8H11ClN4·HClPurity:99.88%Color and Shape:SolidMolecular weight:235.12Lurasidone hydrochloride
CAS:Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.Formula:C28H36N4O2S·HClPurity:99.51%Color and Shape:SolidMolecular weight:529.14Ref: TM-T1735
5mg39.00€10mg59.00€25mg75.00€50mg90.00€100mg137.00€200mg213.00€500mg447.00€1mL*10mM (DMSO)54.00€ML 10302
CAS:ML 10302 is a potent 5-HT4 agonist with Ki of 1.07 nM, boosts bowel movement, and may aid in neurology research.Formula:C15H21ClN2O3Color and Shape:SolidMolecular weight:312.79SAX-187
CAS:SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.Formula:C15H13ClN4O2S2Purity:97.82% - 98%Color and Shape:SolidMolecular weight:380.87Ref: TM-T3183
1mg79.00€5mg152.00€10mg245.00€25mg398.00€50mg532.00€100mg735.00€200mg973.00€1mL*10mM (DMSO)166.00€Perospirone
CAS:Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.Formula:C23H30N4O2SPurity:99.23%Color and Shape:White PowderMolecular weight:426.57Desvenlafaxine succinate hydrate
CAS:Desvenlafaxine succinate hydrate (WY 45233 Succinate) is an antidepressant of the serotonin-norepinephrine reuptake inhibitor (SNRI).Formula:C20H33NO7Purity:99.26%Color and Shape:White Crystalline PowdeMolecular weight:399.48SB399885
CAS:SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.Formula:C18H21Cl2N3O4SPurity:98.94%Color and Shape:SolidMolecular weight:446.35Ref: TM-T19669
1mg67.00€5mg123.00€10mg177.00€25mg291.00€50mg393.00€100mg553.00€200mg743.00€1mL*10mM (DMSO)150.00€Zotepine
CAS:Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,Formula:C18H18ClNOSPurity:99.78%Color and Shape:SolidMolecular weight:331.86Metoclopramide
CAS:Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.Formula:C14H22ClN3O2Purity:99.75%Color and Shape:SolidMolecular weight:299.80Piboserod
CAS:Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.Formula:C22H31N3O2Purity:97.21% - 99.49%Color and Shape:SolidMolecular weight:369.5Ref: TM-T2278
1mg38.00€2mg50.00€5mg84.00€10mg118.00€25mg220.00€50mg403.00€100mg582.00€500mg1,198.00€1mL*10mM (DMSO)120.00€Eptapirone
CAS:Eptapirone (F 11440) is a highly effective and selective 5-HT1A receptor agonist with marked antidepressant and anxiolytic potential.Formula:C16H23N7O2Purity:99.39% - 99.65%Color and Shape:SolidMolecular weight:345.4Harmine
CAS:Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.Formula:C13H12N2OPurity:98.29% - 99.92%Color and Shape:Off-White SolidMolecular weight:212.25Ramosetron hydrochloride
CAS:Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.Formula:C17H18ClN3OPurity:99.95%Color and Shape:SolidMolecular weight:315.8Alprenolol benzoate
CAS:Alprenolol benzoate is the benzoate salt of Alprenolol -- a beta blocker.Formula:C22H29NO4Color and Shape:SolidMolecular weight:371.48Trazodone
CAS:Trazodone (AF-1161), a 5-HT 2A/2C receptor antagonist, is used as an antidepressant for treating major anxiety disorders and depressive disorder.Formula:C19H22ClN5OPurity:99.79% - 99.92%Color and Shape:White To Off-White Crystalline PowderMolecular weight:371.861-(1-Naphthyl) piperazine hydrochloride
CAS:1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multipleFormula:C14H17ClN2Purity:98.27%Color and Shape:SolidMolecular weight:248.75A-582941 dihydrochloride
CAS:A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partialFormula:C17H22Cl2N4Purity:99.55%Color and Shape:SolidMolecular weight:353.29Ref: TM-T22016
1mg42.00€5mg88.00€10mg120.00€25mg235.00€50mg354.00€100mg533.00€200mg743.00€1mL*10mM (DMSO)87.00€Sertindole
CAS:Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).Formula:C24H26ClFN4OPurity:99.87% - 99.92%Color and Shape:Off-White To Pale Yellow SolidMolecular weight:440.94Flibanserin hydrochloride
CAS:Flibanserin HCl: oral 5-HT1A agonist & 5-HT2A antagonist, Ki values 1 nM & 49 nM, for HSDD, has antidepressant/anxiolytic properties.Formula:C20H22ClF3N4OColor and Shape:SolidMolecular weight:426.87Rizatriptan benzoate
CAS:Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraineFormula:C22H25N5O2Purity:99% - 99.79%Color and Shape:White To Off-White Crystalline PowderMolecular weight:391.47Ref: TM-T1512
10mg44.00€25mg74.00€50mg119.00€100mg173.00€200mg259.00€500mg437.00€1mL*10mM (DMSO)48.00€PU02
CAS:PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.Formula:C16H12N4SPurity:99.35%Color and Shape:SolidMolecular weight:292.36Rotigotine Hydrochloride
CAS:Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.
Formula:C19H26ClNOSPurity:99.53% - 99.56%Color and Shape:Almost White To White Crystalline PowderMolecular weight:351.93LY334370
CAS:LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nMFormula:C21H22FN3OPurity:99.32%Color and Shape:SolidMolecular weight:351.42Anpirtoline free base
CAS:Anpirtoline: potent 5-HT1B agonist; lowers serotonin synthesis; reduces aggression; 5-HT3 antagonist; crosses blood-brain barrier.Formula:C10H13ClN2SColor and Shape:SolidMolecular weight:228.74Almotriptan Malate
CAS:Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.Formula:C17H25N3O2S·C4H6O5Purity:99.95%Color and Shape:Pale Yellow SolidMolecular weight:469.55Escitalopram Oxalate
CAS:Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.Formula:C22H23FN2O5Purity:97.39% - 99.73%Color and Shape:White SolidMolecular weight:414.43Ref: TM-T6493
1g268.00€10mg37.00€25mg52.00€50mg63.00€100mg86.00€200mg118.00€500mg187.00€1mL*10mM (DMSO)42.00€NLX-204 hydrochloride(2170405-10-2 free base)
NLX-204 hydrochloride is a potent and selective ERK1/2 phosphorylation-preferring serotonin 5 HT1A receptor agonist(pKi = 10.19).Formula:C20H23Cl2F2N3O2Purity:99.59%Color and Shape:SolidMolecular weight:446.32Serotonin hydrochloride
CAS:Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (Formula:C10H13ClN2OPurity:98.05% - 99.93%Color and Shape:White To Cream PowderMolecular weight:212.676Rotigotine-
CAS:Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.Formula:C19H25NOSPurity:98.08% - 99.59%Color and Shape:SolidMolecular weight:315.47Ref: TM-T6647
5mg50.00€10mg73.00€25mg138.00€50mg241.00€100mg358.00€200mg523.00€500mg822.00€1mL*10mM (DMSO)52.00€5-HT1A modulator 2 hydrochloride
CAS:5-HT1A modulator 2 hydrochloride is a modulator of 5-HT1A showing an affinity of 53 nM for 5-HT1A binding.Formula:C11H16ClNOPurity:98.5%Color and Shape:SolidMolecular weight:213.7Metadoxine
CAS:Metadoxine (Metadoxil) is a neurotransmitter stimulant.Formula:C8H11NO3·C5H7NO3Purity:99.19%Color and Shape:Off-White PowderMolecular weight:298.29Azaphen
CAS:Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.Formula:C16H21Cl2N5OPurity:97.62%Color and Shape:SolidMolecular weight:370.28PRX-07034 hydrochloride
CAS:PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.Formula:C21H29Cl2N3O4SPurity:98.5%Color and Shape:SolidMolecular weight:490.44Pergolide mesylate
CAS:Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.Formula:C20H30N2O3S2Purity:99.70%Color and Shape:White To Off-White SolidMolecular weight:410.59Cariprazine
CAS:Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderateFormula:C21H32Cl2N4OPurity:99.68% - 99.87%Color and Shape:SolidMolecular weight:427.41Ref: TM-T4577
1mg49.00€5mg92.00€10mg145.00€25mg281.00€50mg394.00€100mg550.00€200mg780.00€1mL*10mM (DMSO)103.00€7-Amino-4-(trifluoromethyl)coumarin
CAS:7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.Formula:C10H6F3NO2Purity:97.31% - 97.84%Color and Shape:Yellow PowderMolecular weight:229.16Sumatriptan hydrochloride
CAS:Sumatriptan hydrochloride (GR 43175), an oral 5-HT1 receptor agonist, treats migraines; Ki: 5-HT1D - 17 nM, 5-HT1B - 27 nM, 5-HT1A - 100 nM.Formula:C14H22ClN3O2SColor and Shape:SolidMolecular weight:331.86Phenylbiguanide
CAS:Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)Formula:C8H11N5Purity:99.54%Color and Shape:SolidMolecular weight:177.21Pirenperone
CAS:Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.Formula:C23H24FN3O2Purity:99.2%Color and Shape:SolidMolecular weight:393.45F-15599
CAS:F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).Formula:C19H21ClF2N4OPurity:98.72%Color and Shape:SolidMolecular weight:394.85Ref: TM-T7281
1mg49.00€5mg92.00€10mg152.00€25mg295.00€50mg477.00€100mg715.00€200mg982.00€1mL*10mM (DMSO)104.00€Olanzapine HCl
CAS:Olanzapine HCl, an FDA-approved atypical antipsychotic for schizophrenia and bipolar disorder, resembles clozapine and quetiapine.Formula:C17H21ClN4SColor and Shape:SolidMolecular weight:348.89Cilansetron Hydrochloride
CAS:Cilansetron Hydrochloride can be used for irritable Bowel Syndrome (IBS) with Diarrhea Predominance.Formula:C20H24ClN3O2Color and Shape:SolidMolecular weight:373.88Lurasidone
CAS:Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6Formula:C28H36N4O2SPurity:99.78% - 99.91%Color and Shape:SolidMolecular weight:492.68WAY-100635 Monomaleate
CAS:WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.Formula:C25H34N4O2·C4H4O4Purity:98.44% - 99.46%Color and Shape:SolidMolecular weight:538.64Ref: TM-T2631
2mg43.00€5mg63.00€10mg89.00€25mg170.00€50mg315.00€100mg470.00€200mg680.00€500mg1,054.00€1mL*10mM (DMSO)74.00€Eltoprazine
CAS:Eltoprazine(DU28853) is a serenic or antiaggressive agent which as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.Formula:C12H16N2O2Color and Shape:SolidMolecular weight:220.27Renzapride hydrochloride
CAS:Renzapride is a 5-HT3 antagonist and 5-HT4 agonist. Renzapride also functions as a 5-HT2B antagonist and has some affinity for the 5-HT2A and 5-HT2C receptors.Formula:C16H23Cl2N3O2Color and Shape:SolidMolecular weight:360.28Loxapine hydrochloride
CAS:Loxapine hydrochloride, an oral anti-psychotic, inhibits dopamine and blocks 5-HT receptors.Formula:C18H19Cl2N3OColor and Shape:SolidMolecular weight:364.27Adoprazine hydrochloride
CAS:Adoprazine hydrochloride is a dopamine D2 receptor antagonist and 5-HT1A receptor agonist potential antipsychotic drug.Formula:C24H25ClFN3O2Color and Shape:SolidMolecular weight:441.93ARC-239
CAS:ARC-239 is an agonist of α2-adrenergic receptor.Formula:C24H29N3O3Color and Shape:SolidMolecular weight:407.51(E)-3,4,5-Trimethoxycinnamic acid
CAS:(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.Formula:C12H14O5Purity:99.83%Color and Shape:SolidMolecular weight:238.24VUF 10166
CAS:VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.Formula:C13H15ClN4Purity:99.66%Color and Shape:SolidMolecular weight:262.74(S)-Amisulpride
CAS:(S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist.Formula:C17H27N3O4SPurity:98.38%Color and Shape:SolidMolecular weight:369.48Ref: TM-T26375
1mg34.00€5mg84.00€10mg123.00€25mg225.00€50mg358.00€100mg485.00€200mg622.00€1mL*10mM (DMSO)94.00€Cerlapirdine hydrochloride
CAS:Cerlapirdine/SAM-531, potent 5-HT6 antagonist, targets Alzheimer's and schizophrenia cognitive issues; phase II trials, promising efficacy, safe profile.Formula:C22H24ClN3O3SColor and Shape:SolidMolecular weight:445.96
