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Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

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Found 1045 products of "Proteases/Proteasome"

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  • PROTAC 20S proteasome subunit β5 degrader 2


    <p>PROTAC 20S proteasome subunit β5 degrader 2 is a PROTAC degrader targeting the 20S proteasome subunit β5 (20Sproteasomesubunit β5), with a DC50 of 0.16 μM. It inhibits the proliferation of FaDu cancer cells, showcasing an IC50 of 0.23 μM. Additionally, PROTAC20Sproteasomesubunit β5 degrader 2 demonstrates antitumor activity in a mouse model.</p>
    Color and Shape:Odour Solid
  • GSK2818713

    CAS:
    <p>GSK2818713 is a novel Hepatitis C NS5A replication complex inhibitor.</p>
    Formula:C46H56N8O8
    Color and Shape:Solid
    Molecular weight:849.002
  • Procizumab


    <p>Procizumab is a humanized IgG1 antibody that targets dipeptidyl peptidase 3 (DPP3). It shows potential for investigating sepsis. For the isotype control, refer to HumanIgG1kappa, Isotype Control.</p>
    Color and Shape:Odour Liquid
  • BI-1230

    CAS:
    <p>BI-1230 is a potent inhibitor of HCV NS3 protease, exhibiting efficacy in the low nanomolar range, and notably suppresses viral replication.</p>
    Formula:C42H52N6O9S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:816.96
  • Ellipyrone B


    <p>Ellipyrone B, a γ-pyrone-based macrocyclic polyketide with antihyperglycemic properties, demonstrates inhibitory activity against dipeptidyl peptidase-4 (IC 50</p>
    Formula:C25H38O7
    Color and Shape:Solid
    Molecular weight:450.57
  • MMP-3 Inhibitor

    CAS:
    <p>MMP-3 Inhibitor is a peptide matrix metalloproteinase-3 (MMP-3) inhibitor with a Ki value of 95 nM.MMP-3 inhibitor has anticancer and antitumor activity.</p>
    Formula:C27H46N10O9S
    Purity:98.87%
    Color and Shape:Solid
    Molecular weight:686.78
  • HCV-IN-4

    CAS:
    <p>HCV-IN-4: Potent, oral HCV NS5A inhibitor; effective vs GT1a/b, GT2b, GT3a, Y93H, L31V; EC90s: 3 pM-0.02 nM.</p>
    Formula:C52H58FN9O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:956.07
  • DPP-4-IN-14


    <p>DPP-4-IN-14 (compound 30) is an inhibitor of DPP-4, with an IC50 value of 12.82 nM.</p>
    Formula:C33H27N7O3
    Color and Shape:Solid
    Molecular weight:569.613
  • HIV-1 protease-IN-14


    <p>HIV-1protease-IN-14 (compound 5ae) is an effective inhibitor of HIV-1protease, exhibiting Ki values of 0.28 nM and 56.9 nM against WTHIV-1PR and R41THIV-1PR, respectively. This compound also demonstrates low cytotoxicity.</p>
    Color and Shape:Odour Solid
  • Bictegravir Sodium

    CAS:
    <p>Bictegravir Sodium is an HIV-1 integrase inhibitor with 7.5 nM IC50, offering strong, selective anti-HIV effects and minimal toxicity.</p>
    Formula:C21H17F3N3NaO5
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:471.36
  • LXE408 fumarate


    <p>LXE408 fumarate: orally available, selective kinetoplastid proteasome inhibitor with IC50/EC50 of 0.04 μM for L. donovani; potentially aids in VL research.</p>
    Formula:C27H22FN7O6
    Purity:99.89%
    Color and Shape:Soild
    Molecular weight:559.51
  • PS 915

    CAS:
    <p>PS 915 is a substrate for colorimetric assay. It was used for plasma antithrombin.</p>
    Formula:C27H36ClN7O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:590.08
  • Ichorcumab

    CAS:
    <p>Ichorcumab (JNJ-375) is a fully human IgG4 antibody that targets thrombin. It binds to exosite 1 of thrombin, inhibiting substrate binding without affecting its catalytic activity. For isotype control, refer to HumanIgG1kappa, Isotype Control.</p>
    Color and Shape:Liquid
  • KKI-5

    CAS:
    <p>KKI 5: Serine protease inhibitor, blocks kallikrein &amp; plasmin, potential for cancer therapy &amp; angioedema treatment.</p>
    Formula:C35H55N11O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:773.88
  • Histargin

    CAS:
    <p>Histargin is an enzyme inhibitor separated from Streptomyces roseoviridis.</p>
    Formula:C14H25N7O4
    Color and Shape:Solid
    Molecular weight:355.39
  • Relacatib

    CAS:
    <p>Relacatib (SB-462795) is a potent cathepsins K, L, V inhibitor with high affinity (Ki: 41-68 pM) and reduces bone resorption effectively.</p>
    Formula:C27H32N4O6S
    Color and Shape:Solid
    Molecular weight:540.64
  • Tyrosinase-IN-38


    <p>Tyrosinase-IN-38 (compound 6b) is a competitive inhibitor of tyrosinase, demonstrating an IC50 of 25.82 μM and exhibits antioxidant activity.</p>
    Color and Shape:Odour Solid
  • Aristololactam IIIa

    CAS:
    <p>Aristololactam IIIa inhibits superoxide and elastase generation; IC50: 0.12 μg/mL and 0.20 μg/mL.</p>
    Formula:C16H9NO4
    Color and Shape:Solid
    Molecular weight:279.25
  • Tiprelestat

    CAS:
    <p>Tiprelestat: strong inhibitor of human neutrophil elastase, anti-inflammatory, antimicrobial, used in inflammation/immune research.</p>
    Formula:C254H416N72O75S10
    Color and Shape:Solid
    Molecular weight:5999.09
  • Lonodelestat TFA


    <p>Lonodelestat TFA, an oral peptide, selectively inhibits hNE, potentially aiding in CF research.</p>
    Formula:C73H112F3N15O21
    Color and Shape:Solid
    Molecular weight:1592.75
  • Cathepsin D and E FRET Substrate acetate(839730-93-7 Free base)


    <p>Fluorogenic substrate for cathepsins D &amp; E; cleaves at Phe-Phe bond; not for B, H, L. Useful for assays and studies.</p>
    Color and Shape:Odour Solid
  • Paritaprevir dihydrate

    CAS:
    <p>Paritaprevir dihydrate: potent oral HCV NS3/4A inhibitor (EC50: 0.21-1 nM), SARS-CoV-3CL blocker (IC50: 1.31 μM), metabolized by CYP3A, boosted by Ritonavir.</p>
    Formula:C40H47N7O9S
    Color and Shape:Solid
    Molecular weight:801.91
  • ADAM8-IN-1

    CAS:
    <p>ADAM8-IN-1 is a potent ADAM8 inhibitor with an IC 50 value of 73 nM.</p>
    Formula:C44H44Br4N6O12S2
    Color and Shape:Solid
    Molecular weight:1232.6
  • Ac-Phe-Gly-pNA

    CAS:
    <p>Ac-Phe-Gly-pNA is the chymotrypsin specific substrate [1] .</p>
    Formula:C19H20N4O5
    Color and Shape:Solid
    Molecular weight:384.39
  • Sulodexide

    CAS:
    <p>Sulodexide is an orally administered combination of glycosaminoglycans, consisting of low molecular weight heparin (80%) and dermatan sulfate (20%). It demonstrates antithrombotic properties by interacting with antithrombin III (AT III) and heparin cofactor II (HC II), and by inhibiting thrombin formation. Additionally, sulodexide enhances profibrinolytic activity by releasing tissue plasminogen activator (tPA). It also offers endothelial protection, possesses anti-inflammatory effects, and alleviates chronic venous disease.</p>
    Color and Shape:Solid
  • Cerpegin

    CAS:
    <p>Cerpegin, a pyridine ketone fused c-lactone, acts as an inhibitor of the 20S proteasome. It possesses pharmacological properties as a neuropsychiatric sedative, anti-inflammatory, analgesic, and exhibits anti-ulcer activity.</p>
    Formula:C10H11NO3
    Color and Shape:Solid
    Molecular weight:193.2
  • Carboxypeptidase C

    CAS:
    <p>Carboxypeptidase C removes COOH-terminal amino acids and others in peptides for biochemical studies.</p>
    Color and Shape:Solid
  • MMP-9-IN-6

    CAS:
    <p>MMP-9-IN-6: MMP-9 inhibitor, IC50 of 50 µM, anti-ulcer, potential anti-tumor, for tissue repair studies.</p>
    Formula:C25H19NO2
    Purity:99.75%
    Color and Shape:Soild
    Molecular weight:365.42
  • VAMP


    <p>VAMP is a tetrapeptide that acts as a competitive dipeptidyl peptidase IV (DPP-IV) inhibitor, exhibiting an IC50 of 1.00 μM and a Kd of 6.89 μM. It effectively targets the DPP-IV-GLP-1 axis and is utilized in the research of type 2 diabetes.</p>
    Formula:C18H32N4O5S
    Color and Shape:Solid
    Molecular weight:416.535
  • Ala-Phe-Pro-pNA TFA


    <p>Ala-Phe-Pro-pNA TFA serves as a chromogenic substrate for tripeptidyl peptidase and can be utilized to assess the enzyme's activity.</p>
    Color and Shape:Odour Solid
  • Chymotrypsinogen

    CAS:
    <p>Chymotrypsinogen is an inactive precursor of Chymotrypsin . Chymotrypsin is a serine protease produced by the pancreas [1] [2] .</p>
    Color and Shape:Solid
  • CTTHWGFTLC, CYCLIC

    CAS:
    <p>CTT Gelatinase Inhibitor peptide blocks MMP-2/9, hindering cancer by stopping tumor growth.</p>
    Formula:C52H71N13O14S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1166.33
  • Alisporivir

    CAS:
    <p>Alisporivir (Debio-025) is a cyclophilin A inhibitor that disrupts the interaction between CypA and NS5A. HCV activity in vivo and in vitro.</p>
    Formula:C63H113N11O12
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:1216.64
  • Histatin 5 TFA


    <p>Histatin 5 TFA effectively inhibits host matrix metalloproteinases (MMP-2) and (MMP-9), demonstrating inhibition concentrations (IC 50s) of 0.57 μM and 0.25 μM</p>
    Formula:C135H196N51F3O35
    Color and Shape:Solid
    Molecular weight:3150.31
  • Acetyl-Calpastatin(184-210)(human) TFA


    <p>Acetyl-Calpastatin(184-210)(human) TFA inhibits μ-calpain (Ki 0.2 nM) and cathepsin L (Ki 6 μM) selectively and reversibly.</p>
    Formula:C144H231F3N36O46S
    Color and Shape:Solid
    Molecular weight:3291.65
  • Gly-Pro-pNA hydrochloride

    CAS:
    <p>Gly-Pro-pNA hydrochloride (Gly-Pro p-nitroanilide hydrochloride) is a dipeptidyl peptidase inhibitor that inhibits dipeptidyl peptidase II, dipeptidyl peptidase</p>
    Formula:C13H17ClN4O4
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:328.75
  • Suc-AAP-Abu-pNA

    CAS:
    <p>Suc-AAP-Abu-pNA is a specific substrate for pancreatic elastase (Km = 100 μM; Kcat/Km = 35,300 s-1 M-1 for rat pancreatic elastase; Km = 30 μM; Kcat/Km = 351,</p>
    Formula:C25H34N6O9
    Color and Shape:Solid
    Molecular weight:562.57
  • TR-107

    CAS:
    <p>TR-107 (Anticancer agent 230) is a mitochondrial protease ClpP activator that inhibits tumor growth in the MDA-MB-231 xenograft model.</p>
    Formula:C22H19ClN4O
    Color and Shape:Soild
    Molecular weight:390.87
  • LMP7/LMP2-IN-1

    CAS:
    <p>LMP7/LMP2-IN-1 (Compound 19) is an orally effective inhibitor targeting the immunoproteasome subunits LMP7 and LMP2, with respective IC50 values of 257 and 10 nM. This compound reduces the production of antibodies and downregulates the B cells in the germinal centers of the spleen and plasma cells in NP-OVA immunized mice. It has potential applications in the study of autoimmune diseases.</p>
    Formula:C16H27BN4O3
    Color and Shape:Soild
    Molecular weight:334.22
  • Anticancer agent 114


    <p>Anticancer agent 114: oral dipeptide boronic acid, proteasome inhibitor, IC 50 = 2.2 nM, halts RPMI-8226 cell growth, for multiple myeloma research.</p>
    Formula:C28H33BF6N2O7
    Color and Shape:Solid
    Molecular weight:634.37
  • Phepropeptin C

    CAS:
    <p>Phepropeptin C is a microbial secondary metabolite that acts as a proteasome (proteasome) inhibitor, with an IC50 of 12.5 μg/mL.</p>
    Formula:C38H60N6O6
    Color and Shape:Solid
    Molecular weight:696.92
  • PD150606

    CAS:
    <p>PD150606 is a calpain inhibitor with neuroprotective activity that inhibits μ-calpains and interferes with excitotoxicity-dependent motor neuron death.</p>
    Formula:C9H7IO2S
    Purity:98.19%
    Color and Shape:Solid
    Molecular weight:306.12
  • TWH106


    <p>TWH106 is an inhibitor of the cyclophilin (Cyp) enzyme, exhibiting strong affinity for CypA and CypB with dissociation constants (KD) of 53 nM and 139 nM, respectively. It effectively inhibits the replication of HIV and HCV, demonstrating antiviral activity.</p>
    Color and Shape:Odour Solid
  • BMS-767778

    CAS:
    <p>BMS-767778, a DPP-4 inhibitor, is used potentially for the treatment of type 2 diabetes.</p>
    Formula:C19H20Cl2N4O2
    Color and Shape:Solid
    Molecular weight:407.29
  • Roseltide rT1

    CAS:
    <p>Roseltide rT1 is a neutrophil elastase inhibitor (IC50=0.47 μM) and is rich in cysteine, classified as one of the Roseltides (rT1-rT8). It has the potential to inhibit related diseases by improving neutrophil elastase-stimulated cAMP accumulation in vitro.</p>
    Formula:C110H177N31O31S6
    Color and Shape:Solid
    Molecular weight:2622.16
  • α 1(I) Collagen (614-639), human

    CAS:
    <p>This is a peptide inhibitor of collagen fibrillar matrix assembly.</p>
    Formula:C134H189N37O39
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2942.16
  • MMP-2 Inhibitor-4


    <p>MMP-2Inhibitor-4 (Compound 5g) is an MMP-2 inhibitor with an IC50 of 152.62 nM. It effectively reduces MMP-2 levels in K562 cell lines by stably binding to the active site of MMP-2 and exhibits strong anti-angiogenic effects in ACHN cell lines. MMP-2Inhibitor-4 shows potential for research in chronic myelogenous leukemia (CML).</p>
    Formula:C19H23N3O5S
    Color and Shape:Solid
    Molecular weight:405.468
  • NVP-DPP728 dihydrochloride

    CAS:
    <p>NVP-DPP728 dihydrochloride is a potent, selective DPP-IV inhibitor with a Ki of 11 nM, useful in diabetes research.</p>
    Formula:C15H20Cl2N6O
    Color and Shape:Solid
    Molecular weight:371.27
  • RJS308


    <p>RJS308 is a PROTAC degrader of cyclosporin A (cyclosporin A) with a DC50 of 284 nM. It exhibits antiviral activity by inhibiting the replication of HIV-1 and HCV. (Pink: ligand for target protein CypA ligand-2; Black: linker; Blue: ligand for E3 ligase VHL (S,R,S)-AHPC-Me)</p>
    Formula:C63H75N13O11S
    Color and Shape:Solid
    Molecular weight:1222.42
  • Stevia Powder


    <p>Stevia Powder, a natural sweetener, possesses antioxidant properties. It regulates antifibrotic pathways in cirrhotic rats, demonstrated by a reduction in hepatic stellate cells and decreased expression of matrix metalloproteinases MMP2 and MMP13. Furthermore, it increases the antifibrotic molecule Smad7, which helps prevent the elevation of serum necrosis and bile retention markers, thereby inhibiting the progression of liver fibrosis.</p>
    Color and Shape:Odour Solid
  • PR 39 (porcine) acetate


    <p>PR 39 (porcine) acetate is a noncompetitive, reversible and allosteric proteasome inhibitor.</p>
    Purity:98%
    Color and Shape:Liquid
    Molecular weight:N/A
  • 6-Acetylnimbandiol

    CAS:
    <p>6-Acetylnimbandiol, a non-toxic agent, inhibits tyrosinase (IC50=69.85 μM), melanin, and MITF; useful in melanoma studies.</p>
    Formula:C28H34O8
    Color and Shape:Solid
    Molecular weight:498.56
  • Zetomipzomib maleate

    CAS:
    <p>Zetomipzomib maleate (KZR-616) selectively targets LMP7/2 in immunoproteasomes, potential for autoimmune research.</p>
    Formula:C34H46N4O12
    Color and Shape:Solid
    Molecular weight:702.758
  • Rivulariapeptolides 988


    <p>Rivulariapeptolides 988 inhibits serine proteases: chymotrypsin (IC50 = 95.46 nM), elastase (15.29 nM), proteinase K (85.50 nM).</p>
    Formula:C50H68N8O13
    Color and Shape:Solid
    Molecular weight:989.12
  • L 659286

    CAS:
    <p>L 659286 is one kind of cephalosporin derivative.</p>
    Formula:C17H21N5O7S2
    Color and Shape:Solid
    Molecular weight:471.51
  • Pseudostellarin G

    CAS:
    <p>Pseudostellarin G, a naturally occurring cyclo-octapeptide, exhibits inhibitory activity against tyrosinase and suppresses melanin production.</p>
    Formula:C42H56N8O9
    Color and Shape:Solid
    Molecular weight:816.94
  • CRA-2059

    CAS:
    <p>CRA-2059 is a potent and selective inhibitor of tryptase, particularly targeting recombinant human tryptase-β (rHTβ), with a K i of 620 pM.</p>
    Formula:C34H46N12O8
    Purity:97.68%
    Color and Shape:Solid
    Molecular weight:750.818
  • Ellipyrone A


    <p>Ellipyrone A: γ-pyrone macrocycle, inhibits DPP-4 (IC50=0.35mM), α-glucosidase (IC50=0.74mM), α-amylase (IC50=0.59mM).</p>
    Formula:C25H34O8
    Color and Shape:Solid
    Molecular weight:462.53
  • Leptosin D

    CAS:
    <p>Leptosin D, a thiodiketopiperazine alkaloid derived from mushrooms, effectively inhibits tyrosinase activity, demonstrating an inhibition concentration (IC50)</p>
    Formula:C25H24N4O3S2
    Color and Shape:Solid
    Molecular weight:492.61
  • Emtricitabine S-oxide

    CAS:
    <p>Emtricitabine treats HIV; its degradation byproduct is Emtricitabine S-oxide.</p>
    Formula:C8H10FN3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:263.25
  • Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2

    CAS:
    <p>Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2, a melanotropin derivative and melanocyte-stimulating hormone, activates tyrosinase and demonstrates a thermoregulatory effect</p>
    Formula:C47H64N14O10
    Color and Shape:Solid
    Molecular weight:985.1
  • Peptide 74

    CAS:
    <p>Peptide 74 is a synthetic peptide. It also inhibits the activated form of this enzyme.</p>
    Formula:C62H107N23O20S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1558.79
  • Fotagliptin

    CAS:
    <p>Fotagliptin is a dipeptidyl peptidase IV inhibitor.</p>
    Formula:C17H19FN6O
    Color and Shape:Solid
    Molecular weight:342.37
  • Rivulariapeptolides 1121


    <p>Rivulariapeptolides 1121 inhibits serine proteases: chymotrypsin (IC50=35.52 nM), elastase (13.24 nM), proteinase K (48.05 nM).</p>
    Formula:C56H83N9O15
    Color and Shape:Solid
    Molecular weight:1122.31
  • E-64d [for Biochemical Research]

    CAS:
    Formula:C17H30N2O5
    Purity:>95.0%(HPLC)
    Color and Shape:White to Almost white powder to crystal
    Molecular weight:342.44

    Ref: 3B-E1337

    5mg
    127.00€
    25mg
    402.00€
  • CTS-1027

    CAS:
    <p>CTS-1027 is a small molecule inhibitor of MMPs (IC50s: 0.3 nM, 0.5 nM for MMP2, MMP13). It has &gt; 1,000 fold selectivity over MMP1.</p>
    Formula:C19H20ClNO6S
    Color and Shape:Solid
    Molecular weight:425.88
  • Tenofovir hydrate

    CAS:
    <p>Tenofovir hydrate (GS 1278 hydrate) is a nucleotide reverse transcriptase inhibitor with antiviral activity.</p>
    Formula:C9H16N5O5P
    Purity:99.63%
    Color and Shape:Solid
    Molecular weight:305.23
  • Ilomastat

    CAS:
    Formula:C20H28N4O4
    Purity:>95.0%(HPLC)(qNMR)
    Color and Shape:White to Light yellow powder to crystal
    Molecular weight:388.47

    Ref: 3B-I1202

    10mg
    189.00€
  • S-Methylglutathione

    CAS:
    <p>S-Methylglutathione (S-Methyl glutathione) is a 1-chloro-2,4-dinitrobenzene coupling inhibitor, an XOCl scavenger, and inhibitor of glyoxalase 1.</p>
    Formula:C11H19N3O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:321.35
  • Retagliptin

    CAS:
    <p>Retagliptin is a DPP-4 inhibitor potentially used to treat Type 2 diabetes.</p>
    Formula:C19H18F6N4O3
    Color and Shape:Solid
    Molecular weight:464.36
  • PSI-6206 13C,d3

    CAS:
    <p>PSI-6206 13CD3 is the deuterium labeled PSI-6206. PSI-6206 is a potent and selective HCV NS5B polymerase inhibitor.</p>
    Formula:C10H13FN2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:264.23
  • Tripeptide-32

    CAS:
    <p>Tripeptide-32 is a bioactive peptide recognized for its anti-aging properties, commonly utilized as an ingredient in cosmetics [1].</p>
    Formula:C12H22N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:302.33
  • Glutaminase-IN-3

    CAS:
    <p>Glutaminase-IN-3 is a potent Glutaminase 1 inhibitor with potential antitumor activity and inhibits GLS1 for cancer research.</p>
    Formula:C19H19F3N6O2S
    Purity:98.51%
    Color and Shape:Solid
    Molecular weight:452.45
  • MMP-8 Inhibitor I

    CAS:
    <p>MMP-8 Inhibitor I is a selective inhibitor of the neutrophil collagenase matrix metalloproteinase-8 (MMP-8) with an IC50 value of 4 nM.</p>
    Formula:C17H18N2O5S
    Color and Shape:Solid
    Molecular weight:362.4
  • Tilpisertib

    CAS:
    <p>Tilpisertib is a serine/threonine kinase inhibitor (WO2017007689).</p>
    Formula:C33H33ClN8O
    Color and Shape:Solid
    Molecular weight:593.13
  • Teneligliptin hydrobromide hydrate

    CAS:
    <p>Teneligliptin hydrobromide hydrate: potent, long-lasting DPP-4 inhibitor with ~1 nM IC50.</p>
    Formula:C22H33BrN6O2S
    Color and Shape:Solid
    Molecular weight:525.51
  • Sitagliptin fenilalanil

    CAS:
    <p>Sitagliptin fenilalanil is a dipeptidyl aminopeptidase (DPP-4) inhibitor.</p>
    Formula:C25H24F6N6O2
    Color and Shape:Solid
    Molecular weight:554.49
  • PKSI-527

    CAS:
    <p>PKSI-527 inhibits plasma kallikrein (Ki=0.81μM), selective vs. glandular kallikrein/thrombin/urokinase/Xa, reduces bradykinin, affects clotting times.</p>
    Formula:C25H32ClN3O4
    Color and Shape:Solid
    Molecular weight:473.99
  • H-Arg-4MβNA

    CAS:
    <p>H-Arg-4MβNA (H-Arg-4MbNA) is a peptide that serves as a substrate for cathepsin H. The enzyme activity is often detected in gel electrophoresis.</p>
    Formula:C17H23N5O2
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:329.4
  • BAY-677

    CAS:
    <p>BAY-677, an inactive counterpart to BAY-678, inhibits human neutrophil elastase with 20 nM IC50 and is an SGC-nominated probe.</p>
    Formula:C20H15F3N4O2
    Color and Shape:Solid
    Molecular weight:400.35
  • 5-Amino-8-hydroxyquinoline

    CAS:
    <p>5-Amino-8-hydroxyquinoline(5A8HQ),Proteasome inhibitor. Potential anticancer agent.</p>
    Formula:C9H8N2O
    Purity:99.69%
    Color and Shape:Solid
    Molecular weight:160.17
  • 6-Chloro-7-deazapurine-2F-β-D-arabinofuranose

    CAS:
    <p>6-Chloro-7-deazapurine-2F-β-D-arabinofuranose is a Nucleoside - 7-deazapurine nucleoside, fluoronucleoside, halo nucleoside; Arabino-nucleoside.</p>
    Formula:C11H11ClFN3O3
    Color and Shape:Solid
    Molecular weight:287.67
  • (Arg)9

    CAS:
    <p>(Arg)9 (Nona-L-arginine;Peptide R9) is a cell-penetrating peptide,and exhibits neuroprotective activity(IC50 of 0.78 μM, in the glutamic acid model).</p>
    Formula:C54H110N36O10
    Color and Shape:Solid
    Molecular weight:1423.69
  • Ubenimex Hydrochloride [for Biochemical Research]

    CAS:
    Formula:C16H24N2O4·HCl
    Purity:>97.0%(HPLC)
    Color and Shape:White to Almost white powder to crystal
    Molecular weight:344.84

    Ref: 3B-B4000

    25mg
    196.00€
  • Dabigatran ethyl ester

    CAS:
    <p>Dabigatran ethyl ester (Dabigatran (ethyl ester)) is an emerging oral anticoagulant and it also is a direct inhibitor of thrombin activity.</p>
    Formula:C27H29N7O3
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:499.56
  • Saquinavir mesylate

    CAS:
    <p>Saquinavir mesylate (Ro 31-8959/003) is an Inhibitor of HIV Proteaseused in antiretroviral therapy</p>
    Formula:C39H54N6O8S
    Purity:99.19%
    Color and Shape:White Or Pale Yellow Powder
    Molecular weight:766.9
  • Teneligliptin D8

    CAS:
    <p>Teneligliptin D8 a deuterium labeled Teneligliptin (MP-513). Teneligliptin is a potent, orally available, competitive, and long-lasting inhibitor of DPP-4.</p>
    Formula:C22H30N6OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:434.63
  • PD-166793

    CAS:
    <p>PD-166793 is an MMP inhibitor with inhibitory effects on MMP-2, MMP-3 and MMP-13.PD-166793 improves myocardial ischemia in a rat heart failure model.</p>
    Formula:C17H18BrNO4S
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:412.3
  • Tomeglovir

    CAS:
    Tomeglovir is a potent anti-CMV agent, inhibiting the processing of viral DNA-concatemers (IC50s: 0.34/0.039 μM for HCMV and MCMV).
    Formula:C23H27N3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:441.54
  • DMP 777

    CAS:
    DMP 777 is an orally active inhibitor of human leukocyte elastase.
    Formula:C31H40N4O6
    Color and Shape:Solid
    Molecular weight:564.67
  • Thrombin inhibitor 5

    CAS:
    <p>Thrombin inhibitor 5 (compound 385), IC50: 0.1-1 μM, used in venous thromboembolism studies.</p>
    Formula:C11H9FN4O3
    Purity:99.58%
    Color and Shape:Solid
    Molecular weight:264.21
  • H-Pro-Lys-OH TFA


    <p>H-Pro-Lys-OH TFA is a dipeptide composed of proline and lysine, serving as a substrate for imino dipeptidase (prolinase). Additionally, it can be utilized in peptide synthesis.</p>
    Formula:C13H22F3N3O5
    Color and Shape:Solid
    Molecular weight:357.33
  • 2'-β-C-Ethynyladenosine

    CAS:
    <p>2'-β-C-Ethynyladenosine is a nucleoside analog that potently inhibits hepatitis C virus (HCV) replication by targeting the viral NS5B polymerase.</p>
    Formula:C12H13N5O4
    Color and Shape:Solid
    Molecular weight:291.26
  • Sivelestat Sodium Tetrahydrate

    CAS:
    Formula:C20H21N2NaO7S·4H2O
    Purity:>95.0%(T)(HPLC)
    Color and Shape:White to Light yellow powder to crystal
    Molecular weight:528.50

    Ref: 3B-I1240

    25mg
    318.00€
  • Urokinase

    CAS:
    <p>Urokinase (uPA) is a serine protease that activates plasminogen to plasmin, crucial for thrombolysis and ECM degradation.</p>
    Color and Shape:Solid
  • Pentosan Polysulfate Sodium (W/W 43%)

    CAS:
    <p>Pentosan Polysulfate Sodium: anti-HIV, anti-inflammatory, aids cartilage, treats interstitial cystitis.</p>
    Purity:98%
    Color and Shape:Solid
    Molecular weight:N/A
  • Anguizole

    CAS:
    <p>Anguizole, a small molecule, effectively inhibits Hepatitis C Virus (HCV) replication by modifying the subcellular distribution of NS4B.</p>
    Formula:C17H11ClF2N4O2S
    Color and Shape:Solid
    Molecular weight:408.81
  • Pepstatin A

    CAS:
    Formula:C34H63N5O9
    Purity:>90.0%(HPLC)
    Color and Shape:White to Light yellow powder to crystal
    Molecular weight:685.90

    Ref: 3B-P3041

    10mg
    102.00€
  • (-)-Gallocatechin Gallate

    CAS:
    Formula:C22H18O11
    Purity:>95.0%(HPLC)
    Color and Shape:White to Light yellow powder to crystal
    Molecular weight:458.38

    Ref: 3B-G0628

    25mg
    290.00€
  • Tanaproget

    CAS:
    <p>Tanaproget is an orally available, high-affinity, non-steroidal progesterone receptor (PR) agonist with an IC50 of 1.7 nM for hPR.</p>
    Formula:C16H15N3OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:297.38