CymitQuimica logo
Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

Show 3 more subcategories

Found 985 products of "Proteases/Proteasome"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • Acetyl-Calpastatin (184-210)(human) acetate


    Acetyl-Calpastatin acetate inhibits µ-calpain (Ki=0.2nM) and cathepsin L (Ki=6μM) selectively and reversibly.

    Formula:C144H234N36O46S
    Purity:97.84% - 98.16%
    Color and Shape:Solid
    Molecular weight:3237.68

    Ref: TM-TP2056L

    1mg
    115.00€
    5mg
    255.00€
    10mg
    375.00€
    25mg
    562.00€
    50mg
    792.00€
    100mg
    1,064.00€
    200mg
    1,444.00€
  • Acetyl-Calpastatin(184-210)(human) TFA


    Acetyl-Calpastatin(184-210)(human) TFA inhibits μ-calpain (Ki 0.2 nM) and cathepsin L (Ki 6 μM) selectively and reversibly.
    Formula:C144H231F3N36O46S
    Color and Shape:Solid
    Molecular weight:3291.65

    Ref: TM-T75794

    5mg
    To inquire
    50mg
    To inquire
  • α 1 Antichymotrypsin, Human Plasma

    CAS:
    Alpha 1 Antichymotrypsin, Human Plasma is an inhibitor of serine proteases. This compound is present in amyloid lesions associated with Alzheimer's disease and can be utilized in Alzheimer's research.
    Color and Shape:Solid

    Ref: TM-TP3129

    10mg
    To inquire
    50mg
    To inquire
  • Sulodexide

    CAS:
    Sulodexide is an orally administered combination of glycosaminoglycans, consisting of low molecular weight heparin (80%) and dermatan sulfate (20%). It demonstrates antithrombotic properties by interacting with antithrombin III (AT III) and heparin cofactor II (HC II), and by inhibiting thrombin formation. Additionally, sulodexide enhances profibrinolytic activity by releasing tissue plasminogen activator (tPA). It also offers endothelial protection, possesses anti-inflammatory effects, and alleviates chronic venous disease.
    Color and Shape:Solid

    Ref: TM-T88323

    10mg
    To inquire
    50mg
    To inquire
  • Atecegatran TFA

    CAS:
    Atecegatran TFA is often used as an anticoagulant and can be used to treat cardiovascular disease.
    Formula:C23H22ClF5N4O6
    Purity:97.47% - 99.77%
    Color and Shape:Solid
    Molecular weight:580.89

    Ref: TM-T30191L

    1mg
    185.00€
    5mg
    459.00€
    50mg
    1,415.00€
    100mg
    1,872.00€
  • L-Methionine-DL-sulfoximine

    CAS:
    MSO blocks glutamine synthetase, impacts astroglia, and is used in convulsant research.
    Formula:C5H12N2O3S
    Purity:99.56% - ≥98%
    Color and Shape:White Crystalline Powder
    Molecular weight:180.23

    Ref: TM-T41299

    50mg
    39.00€
    100mg
    52.00€
  • Proteasome-IN-7


    Proteasome-IN-7 (Compound 6f) is a macrolactam-based epoxyketone proteasome inhibitor with an IC50 value of 37.92 nM against the 20S proteasome ChT-L subunit. It exhibits potent antiproliferative effects on multiple myeloma, acute lymphoblastic leukemia, and non-small cell lung cancer.
    Formula:C48H56N6O10S
    Color and Shape:Solid
    Molecular weight:909.06

    Ref: TM-T205355

    10mg
    To inquire
    50mg
    To inquire
  • GSK2336805

    CAS:
    GSK-2336805, an HCV NS5A inhibitor, is effective against genotypes 1, 4, 5, and some of 6.
    Formula:C42H52N8O8
    Color and Shape:Solid
    Molecular weight:796.91

    Ref: TM-T27461

    25mg
    2,178.00€
    50mg
    2,862.00€
    100mg
    3,870.00€
  • PF 00356231

    CAS:

    PF 00356231 is a selectivity inhibitor MMP-12 and can be used in studies about the treatment of emphysema and chronic obstructive pulmonary disease (COPD).

    Formula:C25H20N2O3S
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:428.5

    Ref: TM-T60071

    1mg
    185.00€
    5mg
    415.00€
    10mg
    622.00€
    25mg
    1,119.00€
    50mg
    1,679.00€
    100mg
    2,520.00€
    200mg
    3,780.00€
  • Ac-Phe-Gly-pNA

    CAS:
    Ac-Phe-Gly-pNA is the chymotrypsin specific substrate [1] .
    Formula:C19H20N4O5
    Color and Shape:Solid
    Molecular weight:384.39

    Ref: TM-T74692

    5mg
    To inquire
    50mg
    To inquire
  • HCV-IN-47

    CAS:
    Compound PDK0173, with CAS No. 300543-56-0, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0173 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.
    Formula:C17H19ClN2
    Color and Shape:Solid
    Molecular weight:286.79

    Ref: TM-PDK0173

    200mg
    36.00€
  • Diaminopropionoyl tripeptide-33

    CAS:
    Diaminopropionoyl Tripeptide-33 is a bioactive peptide that safeguards skin cells against UVA-induced DNA damage and is utilized as a cosmetic ingredient [1].
    Formula:C17H27N7O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:425.44

    Ref: TM-T80203

    5mg
    To inquire
    50mg
    To inquire
  • Aristololactam IIIa

    CAS:
    Aristololactam IIIa inhibits superoxide and elastase generation; IC50: 0.12 μg/mL and 0.20 μg/mL.
    Formula:C16H9NO4
    Color and Shape:Solid
    Molecular weight:279.25

    Ref: TM-T75619

    5mg
    To inquire
    50mg
    To inquire
  • Sadopeptins A


    Sadopeptins A, a natural product isolated from Streptomyces sp., is a potent proteasome inhibitor [1].
    Formula:C49H71N9O13S
    Color and Shape:Solid
    Molecular weight:1026.21

    Ref: TM-T75623

    5mg
    To inquire
    50mg
    To inquire
  • HIV-1 inhibitor-6 

    CAS:
    HIV-1 inhibitor-6 (3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo-) is a potent HIV-1 pre-mRNA selective splicing
    Formula:C14H10N4O4S
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:330.32

    Ref: TM-T9854

    1mg
    75.00€
    5mg
    169.00€
    10mg
    284.00€
    25mg
    452.00€
    50mg
    645.00€
    100mg
    867.00€
    500mg
    To inquire
  • Apovincamine

    CAS:
    Apovincamine is a vinca alkaloid and a chemical precursor of Vinpocetine, which is a derivative of Vincamine with vasodilating activity.
    Formula:C21H24N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:336.44

    Ref: TM-T21047

    25mg
    1,369.00€
  • TFLLRNPNDK-NH2

    CAS:
    TFLLRNPNDK-NH2 is a biologically active peptide and a thrombin receptor activating peptide (TRAP).
    Formula:C54H89N17O15
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1216.39

    Ref: TM-T80239

    5mg
    To inquire
    50mg
    To inquire
  • 5-Amino-8-hydroxyquinoline

    CAS:
    5-Amino-8-hydroxyquinoline(5A8HQ),Proteasome inhibitor. Potential anticancer agent.
    Formula:C9H8N2O
    Purity:99.69%
    Color and Shape:Solid
    Molecular weight:160.17

    Ref: TM-T60234

    25mg
    34.00€
    50mg
    44.00€
    100mg
    56.00€
    500mg
    113.00€
    1mL*10mM (DMSO)
    44.00€
  • Glutaminase-IN-3

    CAS:
    Glutaminase-IN-3 is a potent Glutaminase 1 inhibitor with potential antitumor activity and inhibits GLS1 for cancer research.
    Formula:C19H19F3N6O2S
    Purity:98.51%
    Color and Shape:Solid
    Molecular weight:452.45

    Ref: TM-T37385

    5mg
    59.00€
    10mg
    84.00€
    25mg
    119.00€
    50mg
    170.00€
    100mg
    251.00€
    1mL*10mM (DMSO)
    73.00€
  • Diprotin A TFA

    CAS:
    Diprotin A (TFA) is an inhibitor of dipeptidyl peptidase IV (DPP-IV).
    Formula:C19H32F3N3O6
    Color and Shape:Solid
    Molecular weight:455.47

    Ref: TM-T11049

    2mg
    51.00€