
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase(38 products)
- Cysteine Protease(111 products)
- DPP-4(27 products)
- Glutaminase(46 products)
- HIV Protease(506 products)
- PAI-1(26 products)
- Protease Inhibitors(50 products)
- Protease-activated Receptor(55 products)
- Proteasome(85 products)
- Serine Protease(54 products)
- p97(15 products)
Show 3 more subcategories
Found 984 products of "Proteases/Proteasome"
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PKSI-527
CAS:PKSI-527 inhibits plasma kallikrein (Ki=0.81μM), selective vs. glandular kallikrein/thrombin/urokinase/Xa, reduces bradykinin, affects clotting times.Formula:C25H32ClN3O4Color and Shape:SolidMolecular weight:473.99Ilomastat
CAS:Formula:C20H28N4O4Purity:>95.0%(HPLC)(qNMR)Color and Shape:White to Light yellow powder to crystalMolecular weight:388.47Tomeglovir
CAS:Tomeglovir is a potent anti-CMV agent, inhibiting the processing of viral DNA-concatemers (IC50s: 0.34/0.039 μM for HCMV and MCMV).Formula:C23H27N3O4SPurity:98%Color and Shape:SolidMolecular weight:441.54Tilpisertib
CAS:Tilpisertib is a serine/threonine kinase inhibitor (WO2017007689).Formula:C33H33ClN8OColor and Shape:SolidMolecular weight:593.13Dabigatran ethyl ester
CAS:Dabigatran ethyl ester (Dabigatran (ethyl ester)) is an emerging oral anticoagulant and it also is a direct inhibitor of thrombin activity.Formula:C27H29N7O3Purity:99.98%Color and Shape:SolidMolecular weight:499.56BAY-677
CAS:BAY-677, an inactive counterpart to BAY-678, inhibits human neutrophil elastase with 20 nM IC50 and is an SGC-nominated probe.Formula:C20H15F3N4O2Color and Shape:SolidMolecular weight:400.35Thrombin inhibitor 5
CAS:Thrombin inhibitor 5 (compound 385), IC50: 0.1-1 μM, used in venous thromboembolism studies.Formula:C11H9FN4O3Purity:99.58%Color and Shape:SolidMolecular weight:264.21Ref: TM-T9845
2mg35.00€5mg56.00€10mg86.00€25mg154.00€50mg224.00€100mg320.00€200mg434.00€1mL*10mM (DMSO)55.00€H-Arg-4MβNA
CAS:H-Arg-4MβNA (H-Arg-4MbNA) is a peptide that serves as a substrate for cathepsin H. The enzyme activity is often detected in gel electrophoresis.Formula:C17H23N5O2Purity:99.98%Color and Shape:SolidMolecular weight:329.4PD-166793
CAS:PD-166793 is an MMP inhibitor with inhibitory effects on MMP-2, MMP-3 and MMP-13.PD-166793 improves myocardial ischemia in a rat heart failure model.Formula:C17H18BrNO4SPurity:99.86%Color and Shape:SolidMolecular weight:412.3Ref: TM-T20563
5mg42.00€10mg60.00€25mg112.00€50mg175.00€100mg261.00€200mg368.00€1mL*10mM (DMSO)46.00€(Arg)9
CAS:(Arg)9 (Nona-L-arginine;Peptide R9) is a cell-penetrating peptide,and exhibits neuroprotective activity(IC50 of 0.78 μM, in the glutamic acid model).Formula:C54H110N36O10Color and Shape:SolidMolecular weight:1423.69DMP 777
CAS:DMP 777 is an orally active inhibitor of human leukocyte elastase.Formula:C31H40N4O6Color and Shape:SolidMolecular weight:564.67Ubenimex Hydrochloride [for Biochemical Research]
CAS:Formula:C16H24N2O4·HClPurity:>97.0%(HPLC)Color and Shape:White to Almost white powder to crystalMolecular weight:344.84Trisodium Hydrogen Ethylenediaminetetraacetate Hydrate [for Biochemical Research]
CAS:Formula:C10H13N2Na3O8·xH2OPurity:>98.0%(T)Color and Shape:White to Almost white powder to crystalMolecular weight:358.19 (as Anhydrous)Teneligliptin D8
CAS:Teneligliptin D8 a deuterium labeled Teneligliptin (MP-513). Teneligliptin is a potent, orally available, competitive, and long-lasting inhibitor of DPP-4.Formula:C22H30N6OSPurity:98%Color and Shape:SolidMolecular weight:434.63Daclatasvir dihydrochloride
CAS:Daclatasvir dihydrochloride is an oral antiviral that treats chronic hepatitis C by inhibiting HCV's NS5A; rare liver enzyme elevation, seldom causes jaundice.Formula:C40H52Cl2N8O6Purity:99.67%Color and Shape:SolidMolecular weight:811.8Ref: TM-T1786
1g230.00€5mg39.00€10mg48.00€25mg57.00€50mg67.00€100mg77.00€500mg161.00€1mL*10mM (DMSO)49.00€4-Butylresorcinol
CAS:4-Butylresorcinol (Butylresorcinol) is a potent inhibitor of tyrosinase(IC50 : 11.27 μM), and is used in cosmetics as a depigmenting agent.Formula:C10H14O2Purity:99.48% - ≥95%Color and Shape:Light Beige Solid PowderMolecular weight:166.22L-006235
CAS:L-006235 is a potent and reversible inhibitor of cathepsin K with IC50 of 0.25 nM.Formula:C24H30N6O2SPurity:99.37%Color and Shape:SolidMolecular weight:466.6Ref: TM-T21616
2mg39.00€5mg60.00€10mg92.00€25mg177.00€50mg299.00€100mg432.00€200mg602.00€1mL*10mM (DMSO)62.00€Balicatib
CAS:Balicatib (AAE581) is a potent and selective inhibitor of cathepsin K, used in trials studying the treatment of osteoporosis.Formula:C23H33N5O2Purity:97.78% - 98.17%Color and Shape:White To Off-White Solid PowderMolecular weight:411.54Ref: TM-T1850
2mg39.00€5mg58.00€10mg94.00€25mg212.00€50mg358.00€100mg572.00€200mg803.00€1mL*10mM (DMSO)64.00€Paritaprevir
CAS:Paritaprevir (ABT450) 是一种非结构蛋白 3/4A 蛋白酶抑制剂,对 HCV 1a 和 HCV 1b 的 EC50 值分别为 1 和 0.21 nM。它也是SARS-CoV 3CLpro 的抑制剂,IC50为 1.31 μM。
Formula:C40H43N7O7SPurity:99.72%Color and Shape:SolidMolecular weight:765.88GW280264X
CAS:GW280264X (Carbamic acid) is an inhibitor of ADAM17 .Formula:C28H41N5O6SPurity:99.51%Color and Shape:SolidMolecular weight:575.72Ref: TM-T8961
1mg156.00€5mg319.00€10mg477.00€25mg773.00€50mg1,063.00€100mg1,431.00€1mL*10mM (DMSO)404.00€

