CymitQuimica logo
Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

Show 3 more subcategories

Found 984 products of "Proteases/Proteasome"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • PKSI-527

    CAS:
    PKSI-527 inhibits plasma kallikrein (Ki=0.81μM), selective vs. glandular kallikrein/thrombin/urokinase/Xa, reduces bradykinin, affects clotting times.
    Formula:C25H32ClN3O4
    Color and Shape:Solid
    Molecular weight:473.99

    Ref: TM-T35579

    2mg
    81.00€
  • Ilomastat

    CAS:
    Formula:C20H28N4O4
    Purity:>95.0%(HPLC)(qNMR)
    Color and Shape:White to Light yellow powder to crystal
    Molecular weight:388.47

    Ref: 3B-I1202

    10mg
    119.00€
  • Tomeglovir

    CAS:
    Tomeglovir is a potent anti-CMV agent, inhibiting the processing of viral DNA-concatemers (IC50s: 0.34/0.039 μM for HCMV and MCMV).
    Formula:C23H27N3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:441.54

    Ref: TM-TQ0030

    2mg
    54.00€
  • Tilpisertib

    CAS:
    Tilpisertib is a serine/threonine kinase inhibitor (WO2017007689).
    Formula:C33H33ClN8O
    Color and Shape:Solid
    Molecular weight:593.13

    Ref: TM-T39466

    5mg
    873.00€
  • Dabigatran ethyl ester

    CAS:
    Dabigatran ethyl ester (Dabigatran (ethyl ester)) is an emerging oral anticoagulant and it also is a direct inhibitor of thrombin activity.
    Formula:C27H29N7O3
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:499.56

    Ref: TM-T15046

    2mg
    38.00€
    5mg
    51.00€
    10mg
    94.00€
    25mg
    155.00€
    50mg
    261.00€
    100mg
    410.00€
  • BAY-677

    CAS:
    BAY-677, an inactive counterpart to BAY-678, inhibits human neutrophil elastase with 20 nM IC50 and is an SGC-nominated probe.
    Formula:C20H15F3N4O2
    Color and Shape:Solid
    Molecular weight:400.35

    Ref: TM-T10473L

    2mg
    85.00€
  • Thrombin inhibitor 5

    CAS:
    Thrombin inhibitor 5 (compound 385), IC50: 0.1-1 μM, used in venous thromboembolism studies.
    Formula:C11H9FN4O3
    Purity:99.58%
    Color and Shape:Solid
    Molecular weight:264.21

    Ref: TM-T9845

    2mg
    35.00€
    5mg
    56.00€
    10mg
    86.00€
    25mg
    154.00€
    50mg
    224.00€
    100mg
    320.00€
    200mg
    434.00€
    1mL*10mM (DMSO)
    55.00€
  • H-Arg-4MβNA

    CAS:
    H-Arg-4MβNA (H-Arg-4MbNA) is a peptide that serves as a substrate for cathepsin H. The enzyme activity is often detected in gel electrophoresis.
    Formula:C17H23N5O2
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:329.4

    Ref: TM-T19347

    5mg
    33.00€
  • PD-166793

    CAS:
    PD-166793 is an MMP inhibitor with inhibitory effects on MMP-2, MMP-3 and MMP-13.PD-166793 improves myocardial ischemia in a rat heart failure model.
    Formula:C17H18BrNO4S
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:412.3

    Ref: TM-T20563

    5mg
    42.00€
    10mg
    60.00€
    25mg
    112.00€
    50mg
    175.00€
    100mg
    261.00€
    200mg
    368.00€
    1mL*10mM (DMSO)
    46.00€
  • (Arg)9

    CAS:
    (Arg)9 (Nona-L-arginine;Peptide R9) is a cell-penetrating peptide,and exhibits neuroprotective activity(IC50 of 0.78 μM, in the glutamic acid model).
    Formula:C54H110N36O10
    Color and Shape:Solid
    Molecular weight:1423.69

    Ref: TM-T13976

    100mg
    To inquire
    500mg
    To inquire
  • DMP 777

    CAS:
    DMP 777 is an orally active inhibitor of human leukocyte elastase.
    Formula:C31H40N4O6
    Color and Shape:Solid
    Molecular weight:564.67

    Ref: TM-T15144

    2mg
    88.00€
    5mg
    152.00€
    1mL*10mM (DMSO)
    205.00€
  • Ubenimex Hydrochloride [for Biochemical Research]

    CAS:
    Formula:C16H24N2O4·HCl
    Purity:>97.0%(HPLC)
    Color and Shape:White to Almost white powder to crystal
    Molecular weight:344.84

    Ref: 3B-B4000

    25mg
    135.00€
  • Trisodium Hydrogen Ethylenediaminetetraacetate Hydrate [for Biochemical Research]

    CAS:
    Formula:C10H13N2Na3O8·xH2O
    Purity:>98.0%(T)
    Color and Shape:White to Almost white powder to crystal
    Molecular weight:358.19 (as Anhydrous)

    Ref: 3B-T2599

    5g
    22.00€
    25g
    35.00€
  • Teneligliptin D8

    CAS:
    Teneligliptin D8 a deuterium labeled Teneligliptin (MP-513). Teneligliptin is a potent, orally available, competitive, and long-lasting inhibitor of DPP-4.
    Formula:C22H30N6OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:434.63

    Ref: TM-T13121

    1mg
    595.00€
    5mg
    1,431.00€
    10mg
    1,963.00€
    25mg
    2,907.00€
  • Daclatasvir dihydrochloride

    CAS:
    Daclatasvir dihydrochloride is an oral antiviral that treats chronic hepatitis C by inhibiting HCV's NS5A; rare liver enzyme elevation, seldom causes jaundice.
    Formula:C40H52Cl2N8O6
    Purity:99.67%
    Color and Shape:Solid
    Molecular weight:811.8

    Ref: TM-T1786

    1g
    230.00€
    5mg
    39.00€
    10mg
    48.00€
    25mg
    57.00€
    50mg
    67.00€
    100mg
    77.00€
    500mg
    161.00€
    1mL*10mM (DMSO)
    49.00€
  • 4-Butylresorcinol

    CAS:
    4-Butylresorcinol (Butylresorcinol) is a potent inhibitor of tyrosinase(IC50 : 11.27 μM), and is used in cosmetics as a depigmenting agent.
    Formula:C10H14O2
    Purity:99.48% - ≥95%
    Color and Shape:Light Beige Solid Powder
    Molecular weight:166.22

    Ref: TM-T7125

    200mg
    33.00€
    1mL*10mM (DMSO)
    33.00€
  • L-006235

    CAS:
    L-006235 is a potent and reversible inhibitor of cathepsin K with IC50 of 0.25 nM.
    Formula:C24H30N6O2S
    Purity:99.37%
    Color and Shape:Solid
    Molecular weight:466.6

    Ref: TM-T21616

    2mg
    39.00€
    5mg
    60.00€
    10mg
    92.00€
    25mg
    177.00€
    50mg
    299.00€
    100mg
    432.00€
    200mg
    602.00€
    1mL*10mM (DMSO)
    62.00€
  • Balicatib

    CAS:
    Balicatib (AAE581) is a potent and selective inhibitor of cathepsin K, used in trials studying the treatment of osteoporosis.
    Formula:C23H33N5O2
    Purity:97.78% - 98.17%
    Color and Shape:White To Off-White Solid Powder
    Molecular weight:411.54

    Ref: TM-T1850

    2mg
    39.00€
    5mg
    58.00€
    10mg
    94.00€
    25mg
    212.00€
    50mg
    358.00€
    100mg
    572.00€
    200mg
    803.00€
    1mL*10mM (DMSO)
    64.00€
  • Paritaprevir

    CAS:

    Paritaprevir (ABT450) 是一种非结构蛋白 3/4A 蛋白酶抑制剂,对 HCV 1a 和 HCV 1b 的 EC50 值分别为 1 和 0.21 nM。它也是SARS-CoV 3CLpro 的抑制剂,IC50为 1.31 μM。

    Formula:C40H43N7O7S
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:765.88

    Ref: TM-T22394

    5mg
    50.00€
    10mg
    64.00€
    25mg
    88.00€
  • GW280264X

    CAS:
    GW280264X (Carbamic acid) is an inhibitor of ADAM17 .
    Formula:C28H41N5O6S
    Purity:99.51%
    Color and Shape:Solid
    Molecular weight:575.72

    Ref: TM-T8961

    1mg
    156.00€
    5mg
    319.00€
    10mg
    477.00€
    25mg
    773.00€
    50mg
    1,063.00€
    100mg
    1,431.00€
    1mL*10mM (DMSO)
    404.00€