Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase(38 products)
- Cysteine Protease(111 products)
- DPP-4(27 products)
- Glutaminase(46 products)
- HIV Protease(506 products)
- PAI-1(26 products)
- Protease Inhibitors(50 products)
- Protease-activated Receptor(55 products)
- Proteasome(86 products)
- Serine Protease(54 products)
- p97(15 products)
Show 3 more subcategories
Found 984 products of "Proteases/Proteasome"
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HCV-IN-31
CAS:HCV-IN-31 is a HCV inhibitor with an EC50/EC95 of 15.7 μM.Formula:C12H17FN6O3Purity:99.83%Color and Shape:SolidMolecular weight:312.3Dabigatran
CAS:Dabigatran (BIBR 953ZW), a thrombin inhibitor, prevents thrombus formation, reducing stroke and embolism risk in nonvalvular atrial fibrillation patients.Formula:C25H25N7O3Purity:97.44% - 98.7%Color and Shape:Tan SolidMolecular weight:471.51NSC 405020
CAS:NSC 405020 is a noncatalytic inhibitor of MT1-MMP.Formula:C12H15Cl2NOPurity:96.93% - 99.07%Color and Shape:SolidMolecular weight:260.16Histatin 5 acetate
Histatin 5 acetate inhibits the activity of the host matrix metalloproteinases MMP-2 and MMP-9 with IC50s of 0.57 and 0.25 μM, respectively.Formula:C135H199N51O35Purity:98.72%Color and Shape:SolidMolecular weight:3096.35CTTHWGFTLC, CYCLIC acetate(244082-19-7 free base)
CTTHWGFTLC, CYCLIC acetate is an inhibitor for matrix metalloproteinases (MMP)-2 and MMP-9.Formula:C54H75N13O16S2Purity:99.71%Color and Shape:SolidMolecular weight:1226.39Bemnifosbuvir
CAS:Bemnifosbuvir (AT-511) is a novel phosphoramidate prodrug of 2'-fluoro-2'-C-methylguanosine-5'-monophosphate that has potent in vitro activity against HCV.Formula:C24H33FN7O7PPurity:99.35% - 99.54%Color and Shape:SolidMolecular weight:581.53Elbasvir
CAS:Elbasvir (MK-8742) is an NS5A inhibitor developed for chronic HCV treatment.Formula:C49H55N9O7Purity:98.95% - 99.85%Color and Shape:SolidMolecular weight:882.02Ref: TM-T4544
1mg42.00€2mg52.00€5mg79.00€10mg113.00€25mg200.00€50mg334.00€100mg537.00€1mL*10mM (DMSO)111.00€Proteinase K
CAS:Proteinase K (Protease K) is a non-specific serine protease. Proteinase K hydrolyzes peptide bonds and is used for protein digestion. Cost-effective and quality-assured.Formula:C29H27N2O12PPurity:98%Color and Shape:SolidMolecular weight:626.511(R)-MG-132
CAS:(R)-MG-132 (Z-Leu-D-leu-leu-al) is the enantiomer of MG-132. (R)-MG-132 stereoisomer is a more potent proteasome inhibitor than MG-132.Formula:C26H41N3O5Purity:99.90%Color and Shape:SolidMolecular weight:475.62Ref: TM-T12628
2mg38.00€5mg57.00€10mg79.00€25mg120.00€50mg177.00€100mg268.00€200mg398.00€1mL*10mM (DMSO)71.00€GW280264X
CAS:GW280264X (Carbamic acid) is an inhibitor of ADAM17 .Formula:C28H41N5O6SPurity:99.51%Color and Shape:SolidMolecular weight:575.72Ref: TM-T8961
1mg156.00€5mg319.00€10mg477.00€25mg773.00€50mg1,063.00€100mg1,431.00€1mL*10mM (DMSO)404.00€KKI-5 acetate(97145-43-2 free base)
KKI-5 acetate: Serine protease inhibitor, targets kallikrein/plasmin, potential anticancer and angioedema therapy.Formula:C37H59N11O11Purity:99.44%Color and Shape:SolidMolecular weight:833.95Coblopasvir
CAS:Coblopasvir is a pan-genotypic non-structural protein 5A (NS5A) inhibitor. It can be used to study chronic hepatitis C virus infection.Formula:C41H50N8O8Purity:99.33%Color and Shape:SolidMolecular weight:782.88Anagliptin hydrochloride
CAS:Anagliptin (SK-0403) hydrochloride: potent, selective oral DPP-4 inhibitor; IC50: DPP-4 3.8 nM, DPP-8 68 nM, DPP-9 60 nM.Formula:C19H26ClN7O2Color and Shape:SolidMolecular weight:419.91TAPI-1 trifluoroacetate (163847-77-6(free base))
TAPI-1 is an ADAM17/TACE inhibitor, which blocks shedding of cytokine receptors.Formula:C28H38F3N5O7Purity:98.06%Color and Shape:SolidMolecular weight:613.62Ivachtin
CAS:Ivachtin (Caspase-3 Inhibitor VII) is a nonpeptide, noncompetitive and reversibl caspase-3 inhibitor(IC50 = 23 nM) and is a modest inhibitor of the remaining
Formula:C20H21N3O7SPurity:99.74%Color and Shape:SolidMolecular weight:447.46Denagliptin tosylate
CAS:Denagliptin (GW823093 or GSK-823093) is a dipeptidyl peptidase IV (DPP-IV) inhibitor.Formula:C27H26F3N3O4SColor and Shape:SolidMolecular weight:545.57Balicatib
CAS:Balicatib (AAE581) is a potent and selective inhibitor of cathepsin K, used in trials studying the treatment of osteoporosis.Formula:C23H33N5O2Purity:97.78% - 98.17%Color and Shape:White To Off-White Solid PowderMolecular weight:411.54Ref: TM-T1850
2mg39.00€5mg58.00€10mg94.00€25mg212.00€50mg358.00€100mg572.00€200mg803.00€1mL*10mM (DMSO)64.00€Bemnifosbuvir hemisulfate
CAS:Bemnifosbuvir hemisulfate (AT-527) is a potent inhibitor of HCV virus replication.Formula:C48H68F2N14O18P2SPurity:99.98%Color and Shape:SolidMolecular weight:1261.15Proteasome inhibitor IX
CAS:Proteasome inhibitor IX (PS-IX) is an inhibitor of chymotrypsin-like activity of the 20S proteasome (IC50 ~1 μM).Formula:C20H21B2NO5Purity:99.77%Color and Shape:SolidMolecular weight:377.01Grazoprevir hydrate
CAS:Grazoprevir: Hepatitis C protease inhibitor effective against various genotypes, including drug-resistant strains.Formula:C38H52N6O10SPurity:98%Color and Shape:SolidMolecular weight:784.92
