
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase(38 products)
- Cysteine Protease(111 products)
- DPP-4(27 products)
- Glutaminase(46 products)
- HIV Protease(507 products)
- PAI-1(26 products)
- Protease Inhibitors(50 products)
- Protease-activated Receptor(55 products)
- Proteasome(86 products)
- Serine Protease(54 products)
- p97(15 products)
Show 3 more subcategories
Found 979 products of "Proteases/Proteasome"
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SP-Chymostatin B
CAS:SP-Chymostatin B inhibits proteases like chymotrypsin and papain; less effective on human elastase; works at 100-200 μg/ml.Formula:C30H41N7O6Purity:98%Color and Shape:SolidMolecular weight:595.69DPP-IV-IN-1
CAS:DPP-IV-IN-1 is an effective inhibitor of dipeptidyl peptidase IV (DPP-IV), a serine protease (IC50: 4.6 nM).Formula:C11H18FN3O2Purity:98%Color and Shape:SolidMolecular weight:243.28Garvagliptin
CAS:Garvagliptin has antidiabetic activity.Formula:C18H23F2N3O3SPurity:98%Color and Shape:SolidMolecular weight:399.46(Rac)-Tanomastat
CAS:Tanomastat (BAY 12-9566) is an oral biphenyl MMP inhibitor; blocks MMP-2, -3, -9, -13, with anti-invasive and anti-metastatic properties.Formula:C23H19ClO3SColor and Shape:SolidMolecular weight:410.91GSK2793660 HCl
CAS:GSK2793660 is a irreversible covalent α,β-unsaturated amide based DPP1 inhibitor.Formula:C22H32ClN3O3Color and Shape:SolidMolecular weight:421.96Cysteine Protease inhibitor
CAS:Cysteine protease inhibitors are inhibitors of cysteine proteases. Target: Cysteine ProteaseFormula:C18H14N4OPurity:98%Color and Shape:SolidMolecular weight:302.33Elastase-IN-1
CAS:Elastase-IN-1 (Compound Q11) is a non-toxic elastase inhibitor with an IC 50 of 0.897 μM [1].Formula:C17H12N4O3Color and Shape:SolidMolecular weight:320.3Plasma kallikrein-IN-3
CAS:Plasma kallikrein-IN-3 is a potent inhibitor (IC50: 0.15 μM) used in hereditary angioedema and diabetic eye disease research.Formula:C20H23N5O2Color and Shape:SolidMolecular weight:365.43HCV-IN-3
CAS:HCV-IN-3 is a hepatitis C virus (HCV) NS3/4a protein inhibitor (IC50: 20 μM; Kd: 29 μM).Formula:C13H11F2NOPurity:98%Color and Shape:SolidMolecular weight:235.23Cathepsin L/S-IN-1
Cathepsin L/S-IN-1 inhibits Cathepsin L & S (IC50: 4.10 & 1.79 μM) and reduces metastasis in pancreatic cancer cells.Formula:C29H33BrN4O4SColor and Shape:SolidMolecular weight:613.57Ro 09-1679
CAS:Ro 09-1679 is a thrombin inhibitor.Formula:C22H39N9O6Purity:98%Color and Shape:SolidMolecular weight:525.6JPM-OEt
CAS:JPM-OEt: broad-spectrum, covalent cysteine cathepsin inhibitor with antitumor effects.Formula:C20H28N2O6Purity:98%Color and Shape:SolidMolecular weight:392.45OM-189
CAS:OM-189 is a selective inhibitor of synthetic thrombin.Formula:C24H36N6O3SPurity:98%Color and Shape:SolidMolecular weight:488.65Grazoprevir sodium salt
CAS:Grazoprevir sodium salt is a selective Hepatitis C virus NS3/4a protease inhibitor with broad activity across genotypes and resistant variants.Formula:C38H50N6NaO9SPurity:98%Color and Shape:SolidMolecular weight:789.9Prodipine hydrochloride
CAS:Prodipine hydrochloride for purified and plasma Dipeptidyl peptidase IV (DPP IV) from the rabbit (IC50 of 4.5 μM and 30 μM, respectively).Formula:C20H26ClNPurity:98%Color and Shape:SolidMolecular weight:315.88DTS
CAS:DTS is a selective and isoform-specific RSK1 kinase inhibitor. It also has broad cancer therapeutic potential.Formula:C14H14S3Purity:98%Color and Shape:SolidMolecular weight:278.46Cyclophilin inhibitor 3
CAS:Cyclophilin inhibitor 3 (compound 7c), a potent inhibitor of cyclophilin A (CypA), exhibited potent anti-HCV effects with an EC50 value of 4.2 μM.Formula:C34H38N4O6Color and Shape:SolidMolecular weight:598.69Desirudin
CAS:Desirudin (CGP 39393) inhibits thrombin, prevents thrombosis, and is used in thrombocytopenia research.Color and Shape:SolidAA9 TG2 inhibitor
CAS:AA9 is a novel transglutaminase (TG2) inhibitor.Formula:C32H36N4O5Color and Shape:SolidMolecular weight:556.65STOCK2S-26016
CAS:WNK-IN-B, a cell-permeable diaminoacridine, selectively inhibits WNK signaling in mpkDCT/MOVAS by targeting SPAK/OSR1 CCT domain.Formula:C20H19N3O2Color and Shape:SolidMolecular weight:333.38
