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Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

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Found 1044 products of "Proteases/Proteasome"

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  • STOCK2S-26016

    CAS:
    <p>WNK-IN-B, a cell-permeable diaminoacridine, selectively inhibits WNK signaling in mpkDCT/MOVAS by targeting SPAK/OSR1 CCT domain.</p>
    Formula:C20H19N3O2
    Color and Shape:Solid
    Molecular weight:333.38
  • Efegatran sulfate

    CAS:
    <p>Efegatran sulfate (LY294468 sulfate) is a potent thrombin inhibitor used in the treatment of thrombotic disorders.</p>
    Formula:C21H34N6O7S
    Purity:≥98% - ≥98%
    Color and Shape:Solid
    Molecular weight:514.6
  • AA9 TG2 inhibitor

    CAS:
    <p>AA9 is a novel transglutaminase (TG2) inhibitor.</p>
    Formula:C32H36N4O5
    Color and Shape:Solid
    Molecular weight:556.65
  • Desirudin

    CAS:
    <p>Desirudin (CGP 39393) inhibits thrombin, prevents thrombosis, and is used in thrombocytopenia research.</p>
    Color and Shape:Solid
  • GS-9256

    CAS:
    <p>GS-9256 is a selective inhibitor of the HCV NS3 protease, exhibiting favorable pharmacokinetic properties and antiviral activity [1].</p>
    Formula:C46H56ClF2N6O8PS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:957.46
  • Z-LLF-CHO

    CAS:
    <p>Z-LLF-CHO (Z-Leu-Leu-Phe-CHO) effectively inhibits the chymotrypsin-like activity of the pituitary multicatalytic proteinase complex with a Ki value of 460 nM.</p>
    Formula:C29H39N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:509.64
  • MMP13-IN-4

    CAS:
    <p>MMP13-IN-4 (compound 13) is a potent, selective MMP-13 inhibitor with an IC50 of 14.6 μM, implicated in the pathology of osteoarthritis (OA) [1].</p>
    Formula:C21H17BrN4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:485.29
  • Cyclophilin inhibitor 3

    CAS:
    <p>Cyclophilin inhibitor 3 (compound 7c), a potent inhibitor of cyclophilin A (CypA), exhibited potent anti-HCV effects with an EC50 value of 4.2 μM.</p>
    Formula:C34H38N4O6
    Color and Shape:Solid
    Molecular weight:598.69
  • ND-322 HCl

    CAS:
    <p>ND-322 HCl (ND 322 Hydrochloride) is a selective inhibitor of MT1-MMP and MMP2 and reduces in vitro melanoma cell growth, migration and invasion.</p>
    Formula:C15H16ClNO3S2
    Purity:99.49%
    Color and Shape:Solid
    Molecular weight:357.88
  • DTS

    CAS:
    <p>DTS is a selective and isoform-specific RSK1 kinase inhibitor. It also has broad cancer therapeutic potential.</p>
    Formula:C14H14S3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:278.46
  • Prodipine hydrochloride

    CAS:
    <p>Prodipine hydrochloride for purified and plasma Dipeptidyl peptidase IV (DPP IV) from the rabbit (IC50 of 4.5 μM and 30 μM, respectively).</p>
    Formula:C20H26ClN
    Purity:98%
    Color and Shape:Solid
    Molecular weight:315.88
  • SLK/STK10-IN-1

    CAS:
    <p>SLK/STK10-IN-1 is a selective and potent inhibitor of SLK and STK10 with potential antitumor activity.</p>
    Formula:C17H13ClN2O3
    Purity:99.34%
    Color and Shape:Solid
    Molecular weight:328.75
  • ZD-0892

    CAS:
    <p>ZD-0892: potent, selective neutrophil elastase inhibitor; Ki 6.7 nM (human), 200 nM (porcine).</p>
    Formula:C24H32F3N3O5
    Purity:95% - 99.53%
    Color and Shape:Solid
    Molecular weight:499.52
  • Grazoprevir sodium salt

    CAS:
    <p>Grazoprevir sodium salt is a selective Hepatitis C virus NS3/4a protease inhibitor with broad activity across genotypes and resistant variants.</p>
    Formula:C38H50N6NaO9S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:789.9
  • Tyrosinase-IN-4

    CAS:
    <p>Tyrosinase-IN-4, a potent inhibitor, has uses in skin-whitening, food preservation, cosmetics, agriculture, and medicine.</p>
    Formula:C15H9ClO3
    Color and Shape:Solid
    Molecular weight:272.68
  • JPM-OEt

    CAS:
    <p>JPM-OEt: broad-spectrum, covalent cysteine cathepsin inhibitor with antitumor effects.</p>
    Formula:C20H28N2O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:392.45
  • N-Phenylthiourea

    CAS:
    <p>N-Phenylthiourea (Phenylthiocarbamide) is EC 1.14.18.1 (tyrosinase) inhibitor, a diphenolase inhibitor, and a non-competitive inhibitor of the PvdP tyrosinase.</p>
    Formula:C7H8N2S
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:152.22
  • (S)-BI-1001

    CAS:
    <p>(S)-BI-1001 is an active S-enantiomer of BI-1001. (S)-BI-1001 has antiviral potency against HIV-1 integrase (IC50: 28 nM, and EC50: 450 nM and a Kd: 4.7 μM).</p>
    Formula:C19H15BrClNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:420.68
  • p-Aminobenzamidine dihydrochloride

    CAS:
    <p>4-Aminobenzamidine dihydrochloride (p-Aminobenzamidine dihydrochloride) is a strong trypsin inhibitor and a relatively weak inhibitor of urokinase type</p>
    Formula:C7H11Cl2N3
    Purity:99.00% - 99.56%
    Color and Shape:Solid
    Molecular weight:208.088
  • PF-00356231 hydrochloride

    CAS:
    <p>PF-00356231 hydrochloride is an inhibitor of matrix metalloproteinase MMP-12 with IC50 of 1.4 μM.</p>
    Formula:C25H21ClN2O3S
    Purity:98.39%
    Color and Shape:Solid
    Molecular weight:464.96