
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase(34 products)
- Cysteine Protease(96 products)
- DPP-4(20 products)
- Glutaminase(40 products)
- HIV Protease(449 products)
- PAI-1(25 products)
- Protease Inhibitors(50 products)
- Protease-activated Receptor(53 products)
- Proteasome(94 products)
- Serine Protease(50 products)
- p97(14 products)
Show 3 more subcategories
Found 1044 products of "Proteases/Proteasome"
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STOCK2S-26016
CAS:<p>WNK-IN-B, a cell-permeable diaminoacridine, selectively inhibits WNK signaling in mpkDCT/MOVAS by targeting SPAK/OSR1 CCT domain.</p>Formula:C20H19N3O2Color and Shape:SolidMolecular weight:333.38Efegatran sulfate
CAS:<p>Efegatran sulfate (LY294468 sulfate) is a potent thrombin inhibitor used in the treatment of thrombotic disorders.</p>Formula:C21H34N6O7SPurity:≥98% - ≥98%Color and Shape:SolidMolecular weight:514.6AA9 TG2 inhibitor
CAS:<p>AA9 is a novel transglutaminase (TG2) inhibitor.</p>Formula:C32H36N4O5Color and Shape:SolidMolecular weight:556.65Desirudin
CAS:<p>Desirudin (CGP 39393) inhibits thrombin, prevents thrombosis, and is used in thrombocytopenia research.</p>Color and Shape:SolidGS-9256
CAS:<p>GS-9256 is a selective inhibitor of the HCV NS3 protease, exhibiting favorable pharmacokinetic properties and antiviral activity [1].</p>Formula:C46H56ClF2N6O8PSPurity:98%Color and Shape:SolidMolecular weight:957.46Z-LLF-CHO
CAS:<p>Z-LLF-CHO (Z-Leu-Leu-Phe-CHO) effectively inhibits the chymotrypsin-like activity of the pituitary multicatalytic proteinase complex with a Ki value of 460 nM.</p>Formula:C29H39N3O5Purity:98%Color and Shape:SolidMolecular weight:509.64MMP13-IN-4
CAS:<p>MMP13-IN-4 (compound 13) is a potent, selective MMP-13 inhibitor with an IC50 of 14.6 μM, implicated in the pathology of osteoarthritis (OA) [1].</p>Formula:C21H17BrN4O5Purity:98%Color and Shape:SolidMolecular weight:485.29Cyclophilin inhibitor 3
CAS:<p>Cyclophilin inhibitor 3 (compound 7c), a potent inhibitor of cyclophilin A (CypA), exhibited potent anti-HCV effects with an EC50 value of 4.2 μM.</p>Formula:C34H38N4O6Color and Shape:SolidMolecular weight:598.69ND-322 HCl
CAS:<p>ND-322 HCl (ND 322 Hydrochloride) is a selective inhibitor of MT1-MMP and MMP2 and reduces in vitro melanoma cell growth, migration and invasion.</p>Formula:C15H16ClNO3S2Purity:99.49%Color and Shape:SolidMolecular weight:357.88DTS
CAS:<p>DTS is a selective and isoform-specific RSK1 kinase inhibitor. It also has broad cancer therapeutic potential.</p>Formula:C14H14S3Purity:98%Color and Shape:SolidMolecular weight:278.46Prodipine hydrochloride
CAS:<p>Prodipine hydrochloride for purified and plasma Dipeptidyl peptidase IV (DPP IV) from the rabbit (IC50 of 4.5 μM and 30 μM, respectively).</p>Formula:C20H26ClNPurity:98%Color and Shape:SolidMolecular weight:315.88SLK/STK10-IN-1
CAS:<p>SLK/STK10-IN-1 is a selective and potent inhibitor of SLK and STK10 with potential antitumor activity.</p>Formula:C17H13ClN2O3Purity:99.34%Color and Shape:SolidMolecular weight:328.75ZD-0892
CAS:<p>ZD-0892: potent, selective neutrophil elastase inhibitor; Ki 6.7 nM (human), 200 nM (porcine).</p>Formula:C24H32F3N3O5Purity:95% - 99.53%Color and Shape:SolidMolecular weight:499.52Grazoprevir sodium salt
CAS:<p>Grazoprevir sodium salt is a selective Hepatitis C virus NS3/4a protease inhibitor with broad activity across genotypes and resistant variants.</p>Formula:C38H50N6NaO9SPurity:98%Color and Shape:SolidMolecular weight:789.9Tyrosinase-IN-4
CAS:<p>Tyrosinase-IN-4, a potent inhibitor, has uses in skin-whitening, food preservation, cosmetics, agriculture, and medicine.</p>Formula:C15H9ClO3Color and Shape:SolidMolecular weight:272.68JPM-OEt
CAS:<p>JPM-OEt: broad-spectrum, covalent cysteine cathepsin inhibitor with antitumor effects.</p>Formula:C20H28N2O6Purity:98%Color and Shape:SolidMolecular weight:392.45N-Phenylthiourea
CAS:<p>N-Phenylthiourea (Phenylthiocarbamide) is EC 1.14.18.1 (tyrosinase) inhibitor, a diphenolase inhibitor, and a non-competitive inhibitor of the PvdP tyrosinase.</p>Formula:C7H8N2SPurity:99.71%Color and Shape:SolidMolecular weight:152.22(S)-BI-1001
CAS:<p>(S)-BI-1001 is an active S-enantiomer of BI-1001. (S)-BI-1001 has antiviral potency against HIV-1 integrase (IC50: 28 nM, and EC50: 450 nM and a Kd: 4.7 μM).</p>Formula:C19H15BrClNO3Purity:98%Color and Shape:SolidMolecular weight:420.68p-Aminobenzamidine dihydrochloride
CAS:<p>4-Aminobenzamidine dihydrochloride (p-Aminobenzamidine dihydrochloride) is a strong trypsin inhibitor and a relatively weak inhibitor of urokinase type</p>Formula:C7H11Cl2N3Purity:99.00% - 99.56%Color and Shape:SolidMolecular weight:208.088PF-00356231 hydrochloride
CAS:<p>PF-00356231 hydrochloride is an inhibitor of matrix metalloproteinase MMP-12 with IC50 of 1.4 μM.</p>Formula:C25H21ClN2O3SPurity:98.39%Color and Shape:SolidMolecular weight:464.96
