
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase(34 products)
- Cysteine Protease(96 products)
- DPP-4(20 products)
- Glutaminase(40 products)
- HIV Protease(449 products)
- PAI-1(25 products)
- Protease Inhibitors(50 products)
- Protease-activated Receptor(53 products)
- Proteasome(94 products)
- Serine Protease(50 products)
- p97(14 products)
Show 3 more subcategories
Found 1044 products of "Proteases/Proteasome"
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Elastase-IN-1
CAS:<p>Elastase-IN-1 (Compound Q11) is a non-toxic elastase inhibitor with an IC 50 of 0.897 μM [1].</p>Formula:C17H12N4O3Color and Shape:SolidMolecular weight:320.3HCV-IN-36
CAS:<p>HCV-IN-36: oral HCV inhibitor, EC50 0.016 μM, CC50 8.78 μM, potent antiviral.</p>Formula:C30H36ClN5Color and Shape:SolidMolecular weight:502.09BRD-8899
CAS:<p>BRD-8899 is a STK33 inhibitor, with an IC 50 of 11 nM [1].</p>Formula:C17H22N4O3SColor and Shape:SolidMolecular weight:362.45Tyrosinase-IN-5
CAS:<p>Tyrosinase-IN-5 (16c) inhibits tyrosinase with 0.02 μM IC50, reduces melanogenesis, and is low-toxicity.</p>Formula:C18H13N3O6Color and Shape:SolidMolecular weight:367.31BMS-363131
CAS:<p>BMS-363131 (BMS363131) is a potent and selective trypsin inhibitor with an IC50 value of <1.7 nM.</p>Formula:C28H40N6O5Purity:97.99%Color and Shape:SolidMolecular weight:540.65α-Glucosidase-IN-5
CAS:<p>α-Glucosidase-IN-5 (compound 8) is isolated from a twig extract of Polyalthia cinnamomea which is a potent α-glucosidase inhibitor with an IC50 of 57.9 µM.</p>Formula:C15H13NO3Color and Shape:SolidMolecular weight:255.27SAP2-IN-1
CAS:<p>SAP2-IN-1 inhibits secreted aspartate protease 2 (IC50: 0.92 μM), doesn't work in vitro, and helps research infections.</p>Formula:C34H29NO7Color and Shape:SolidMolecular weight:563.6Elasnin
CAS:<p>Elasnin is a reversible inhibitor of elastase for human granulocyte and pancreatic enzymes with IC50 values of 1.3 and 30 µg/ml, respectively.</p>Formula:C24H40O4Color and Shape:SolidMolecular weight:392.57MMP2-IN-2
CAS:<p>MMP2-IN-2 is an MMP-2 inhibitor that inhibits MMP-13, MMP-9, and MMP-8, and can be used in the study of cancer and immune diseases.</p>Formula:C13H8N4O4Purity:98.09%Color and Shape:SolidMolecular weight:284.23Glutaminase-IN-4
CAS:<p>Glutaminase-IN-4 (compound 2a) is a glutaminase (GLS) inhibitor (IC50: 2.3 μM).</p>Formula:C23H22N6O2S2Color and Shape:SolidMolecular weight:478.59L 658758
CAS:<p>L 658758 is an inhibitor of serine proteinase.</p>Formula:C16H20N2O9SColor and Shape:SolidMolecular weight:416.4ASPER-29
CAS:<p>ASPER-29, an Asperphenamate analog, inhibits cathepsins L/S with IC50s of 6.03/5.02 μM, useful in cancer migration/invasion research.</p>Formula:C31H29BrN2O5SColor and Shape:SolidMolecular weight:621.54CAY10704
CAS:<p>CAY10704: Potent HCV inhibitor, EC50=17 nM, low cytotoxicity, good in mice, liver-targeted, not hepatotoxic, weak against dengue.</p>Formula:C18H20Cl2N2Color and Shape:SolidMolecular weight:335.27DPP-4-IN-1
CAS:<p>DPP-4-IN-1 inhibits DPP-4 with 49 nM IC50, ideal for diabetes study, akin to Alogliptin.</p>Formula:C19H19ClN6Color and Shape:SolidMolecular weight:366.85AA10 TG2 inhibitor
CAS:<p>AA10 is an irreversible inhibitor of transglutaminase 2 (TG2).</p>Formula:C32H36N4O5Color and Shape:SolidMolecular weight:556.65BAY8040
CAS:<p>BAY8040 is a potent selective human neutrophilic elastase inhibitor with excellent potency and selectivity with promising pharmacokinetic characteristics.</p>Formula:C21H16F3N5O2Color and Shape:SolidMolecular weight:427.38PK44 phosphate
CAS:<p>PK44 phosphate is a potent inhibitor of dipeptidyl peptidase IV (DPP-IV) (IC50: 15.8 nM).</p>Formula:C17H19F5N7O5PColor and Shape:SolidMolecular weight:527.349VEL-0230
CAS:<p>VEL-0230 (NC-2300) is a cathespin K inhibitor boosting bone growth and reducing loss, targeting bone diseases and developed by Velcura Therapeutics.</p>Formula:C14H24NNaO5Color and Shape:SolidMolecular weight:309.33Alicapistat
CAS:<p>Alicapistat (ABT-957) is a human calpains 1 and 2 inhibitor. It can potentially be used to treat Alzheimer's disease (AD).</p>Formula:C25H27N3O4Purity:98%Color and Shape:SolidMolecular weight:433.5Tyrosinase-IN-6
CAS:<p>Tyrosinase-IN-6 (4B) is a potent tyrosinase inhibitor (IC50=3.80 μM) with good antioxidant activity.</p>Formula:C24H31N3O2Color and Shape:SolidMolecular weight:393.52
