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Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

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Found 895 products for "Proteases/Proteasome".

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  • BJJF078

    CAS:
    BJJF078, an aminopiperidine, inhibits human/mouse TG2 (IC50: 41/54 nM) and TG1 (IC50: 0.16 μM), may be used in MS studies.
    Formula:C27H29N3O6S
    Purity:99.56%
    Color and Shape:Soild
    Molecular weight:523.6

    Ref: TM-T67865

    1mg
    50.00€
    5mg
    101.00€
    10mg
    142.00€
    25mg
    236.00€
    50mg
    353.00€
    100mg
    522.00€
    200mg
    743.00€
  • Retagliptin Phosphate

    CAS:
    Retagliptin Phosphate (SP 2086) is pharmaceutical composition of DPP-4 inhibitor, for treating type-2 diabetes.
    Formula:C19H21F6N4O7P
    Purity:98.70%
    Color and Shape:Solid
    Molecular weight:562.36

    Ref: TM-T12710

    100mg
    To inquire
    1mg
    34.00€
    2mg
    42.00€
    5mg
    60.00€
    1mL*10mM (DMSO)
    79.00€
    10mg
    87.00€
    25mg
    161.00€
    50mg
    245.00€
  • ML604440

    CAS:
    ML604440 is a cell permeable proteasome β1i (LMP2) subunit inhibitor.
    Formula:C17H24BF3N2O4
    Purity:97.06%
    Color and Shape:Solid
    Molecular weight:388.19

    Ref: TM-T12079

    1mg
    109.00€
    2mg
    158.00€
    5mg
    259.00€
    1mL*10mM (DMSO)
    285.00€
    10mg
    409.00€
    25mg
    677.00€
    50mg
    954.00€
    100mg
    1,288.00€
    200mg
    1,728.00€
  • ARP-100

    CAS:
    ARP-100 (MMP-2 Inhibitor III) is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM).
    Formula:C17H20N2O5S
    Purity:97.18%
    Color and Shape:White Solid
    Molecular weight:364.42

    Ref: TM-T14322

    1mg
    34.00€
    5mg
    66.00€
    1mL*10mM (DMSO)
    73.00€
    10mg
    92.00€
    25mg
    178.00€
    50mg
    334.00€
    100mg
    537.00€
  • midesteine

    CAS:
    Midesteine (MR-889) is a small molecule neutrophil elastase inhibitor used in the treatment of bronchitis, asthma and chronic lung disease.
    Formula:C12H13NO3S3
    Purity:99.87% - 99.98%
    Color and Shape:Solid
    Molecular weight:315.43

    Ref: TM-T68099

    1mg
    52.00€
    5mg
    105.00€
    10mg
    157.00€
    25mg
    253.00€
    50mg
    359.00€
    100mg
    512.00€
    200mg
    717.00€
  • BLT-1

    CAS:
    BLT-1 is a scavenger receptor BI (SR-BI)inhibitor.
    Formula:C12H23N3S
    Purity:97.97%
    Color and Shape:White Solid
    Molecular weight:241.4

    Ref: TM-T14667

    1mg
    43.00€
    2mg
    56.00€
    1mL*10mM (DMSO)
    90.00€
    5mg
    93.00€
    10mg
    152.00€
    25mg
    259.00€
    50mg
    409.00€
    100mg
    592.00€
  • DBPR108

    CAS:
    DBPR108 is an orally bioavailable dipeptide-derived DPP4 inhibitor (IC50: 15 nM) and it has no inhibition on DDP8 and DPP9.
    Formula:C16H25FN4O2
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:324.39

    Ref: TM-T15079

    1mg
    48.00€
    5mg
    100.00€
    1mL*10mM (DMSO)
    110.00€
    10mg
    133.00€
    25mg
    215.00€
    50mg
    306.00€
    100mg
    414.00€
    200mg
    573.00€
  • Ruzasvir

    CAS:
    Ruzasvir (MK-8408) is a novel and potent pan-genotypic inhibitor of hepatitis C virus NS5A with antiviral activity.
    Formula:C49H55FN10O7S
    Purity:96.87% - 99.93%
    Color and Shape:Solid
    Molecular weight:947.09

    Ref: TM-T68015

    1mg
    152.00€
    5mg
    380.00€
    10mg
    555.00€
    25mg
    863.00€
  • KW-2450 Formate


    KW-2450 Formate is an IGF-1R/IR tyrosine kinase inhibitor with antitumor effects that acts through inhibition of Aurora A and B kinases.KW-2450 Formate inhibits the growth of TNBC xenografts and induces tetraploid accumulation.
    Formula:C29H31N5O5S
    Purity:99.70%
    Color and Shape:Solid
    Molecular weight:561.65

    Ref: TM-T68405L

    1mg
    175.00€
    5mg
    434.00€
    10mg
    622.00€
    25mg
    973.00€
    50mg
    1,341.00€
    100mg
    1,773.00€
  • Cathepsin C-IN-6


    Cathepsin C-IN-6 (compound 2), an E-64c-hydrazideas-derived inhibitor of cathepsin C, possesses anti-inflammatory properties and impedes neutrophil elastase
    Formula:C24H35N5O4·xC2HF3O2
    Color and Shape:Solid

    Ref: TM-T79496

    5mg
    To inquire
    50mg
    To inquire
  • Histatin 5 (TFA)(115966-68-2,free)


    Histatin 5 (TFA)(115966-68-2,free) (Histatin 5 (TFA)) inhibits the activity of the host matrix metalloproteinases MMP-2 and MMP-9 with IC50s of 0.57 and 0.25 μM
    Formula:C135H196F3N51O35
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3150.32

    Ref: TM-TP1446

    1mg
    159.00€
    5mg
    532.00€
    10mg
    832.00€
    25mg
    1,489.00€
    50mg
    2,247.00€
  • Dihydrofuran-3(2H)-one

    CAS:
    Dihydrofuran-3(2H)-one, with CAS No. 22929-52-8, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Dihydrofuran-3(2H)-one provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.
    Formula:C4H6O2
    Purity:99.92%
    Molecular weight:86.09

    Ref: TM-T7228

    1mL*10mM (DMSO)
    33.00€
    200mg
    33.00€
  • Activated Protein C (390-404), human

    CAS:
    Human Activated Protein C (390-404) peptide derived from serine protease, suppresses APC anticoagulation.
    Formula:C91H130N22O23
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1900.14

    Ref: TM-TP1628

    100mg
    To inquire
    500mg
    To inquire
  • ADAM8-IN-1

    CAS:
    ADAM8-IN-1 is a potent ADAM8 inhibitor with an IC 50 value of 73 nM.
    Formula:C44H44Br4N6O12S2
    Color and Shape:Solid
    Molecular weight:1232.6

    Ref: TM-T73998

    5mg
    To inquire
    50mg
    To inquire
  • HCV-IN-4

    CAS:
    HCV-IN-4: Potent, oral HCV NS5A inhibitor; effective vs GT1a/b, GT2b, GT3a, Y93H, L31V; EC90s: 3 pM-0.02 nM.
    Formula:C52H58FN9O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:956.07

    Ref: TM-TP1468

    100mg
    To inquire
    500mg
    To inquire
  • Barbituric acid

    CAS:
    Barbituric acid is a pyrimidine derivative and the basic skeleton of barbiturate drugs, barbiturate drugs and other heterocyclic compounds.
    Formula:C4H4N2O3
    Purity:99.83%
    Molecular weight:128.09

    Ref: TM-T205940

    50mg
    58.00€
    100mg
    87.00€
  • Tyrosinase-IN-38


    Tyrosinase-IN-38 (compound 6b) is a competitive inhibitor of tyrosinase, demonstrating an IC50 of 25.82 μM and exhibits antioxidant activity.
    Color and Shape:Odour Solid

    Ref: TM-T200602

    10mg
    To inquire
    50mg
    To inquire
  • LXE408 fumarate


    LXE408 fumarate: orally available, selective kinetoplastid proteasome inhibitor with IC50/EC50 of 0.04 μM for L. donovani; potentially aids in VL research.
    Formula:C27H22FN7O6
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:559.51

    Ref: TM-T39214L

    1mg
    299.00€
    2mg
    447.00€
    5mg
    563.00€
    1mL*10mM (DMSO)
    830.00€
    10mg
    897.00€
    25mg
    1,324.00€
    50mg
    1,791.00€
    100mg
    2,412.00€
  • TMC647055 Choline salt


    TMC647055 choline salt is a selective and cell-permeating inhibitor of HCV NS5B (IC50: 34 nM).
    Formula:C37H53N5O8S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:727.91

    Ref: TM-T13170

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • BAY 1217224

    CAS:
    BAY 1217224 is a neutral, non-prodrug Thrombin inhibitor with good oral pharmacokinetics.
    Formula:C24H27ClFN3O5
    Color and Shape:Solid
    Molecular weight:491.94

    Ref: TM-T39124

    25mg
    7,192.00€