
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase(41 products)
- Cysteine Protease(117 products)
- DPP-4(26 products)
- Glutaminase(44 products)
- HIV Protease(473 products)
- PAI-1(27 products)
- Protease Inhibitors(49 products)
- Protease-activated Receptor(55 products)
- Proteasome(84 products)
- Serine Protease(55 products)
- p97(15 products)
Show 3 more subcategories
Found 895 products for "Proteases/Proteasome".
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
BJJF078
CAS:BJJF078, an aminopiperidine, inhibits human/mouse TG2 (IC50: 41/54 nM) and TG1 (IC50: 0.16 μM), may be used in MS studies.Formula:C27H29N3O6SPurity:99.56%Color and Shape:SoildMolecular weight:523.6Retagliptin Phosphate
CAS:Retagliptin Phosphate (SP 2086) is pharmaceutical composition of DPP-4 inhibitor, for treating type-2 diabetes.Formula:C19H21F6N4O7PPurity:98.70%Color and Shape:SolidMolecular weight:562.36Ref: TM-T12710
100mgTo inquire1mg34.00€2mg42.00€5mg60.00€1mL*10mM (DMSO)79.00€10mg87.00€25mg161.00€50mg245.00€ML604440
CAS:ML604440 is a cell permeable proteasome β1i (LMP2) subunit inhibitor.Formula:C17H24BF3N2O4Purity:97.06%Color and Shape:SolidMolecular weight:388.19Ref: TM-T12079
1mg109.00€2mg158.00€5mg259.00€1mL*10mM (DMSO)285.00€10mg409.00€25mg677.00€50mg954.00€100mg1,288.00€200mg1,728.00€ARP-100
CAS:ARP-100 (MMP-2 Inhibitor III) is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM).Formula:C17H20N2O5SPurity:97.18%Color and Shape:White SolidMolecular weight:364.42midesteine
CAS:Midesteine (MR-889) is a small molecule neutrophil elastase inhibitor used in the treatment of bronchitis, asthma and chronic lung disease.Formula:C12H13NO3S3Purity:99.87% - 99.98%Color and Shape:SolidMolecular weight:315.43BLT-1
CAS:BLT-1 is a scavenger receptor BI (SR-BI)inhibitor.Formula:C12H23N3SPurity:97.97%Color and Shape:White SolidMolecular weight:241.4Ref: TM-T14667
1mg43.00€2mg56.00€1mL*10mM (DMSO)90.00€5mg93.00€10mg152.00€25mg259.00€50mg409.00€100mg592.00€DBPR108
CAS:DBPR108 is an orally bioavailable dipeptide-derived DPP4 inhibitor (IC50: 15 nM) and it has no inhibition on DDP8 and DPP9.Formula:C16H25FN4O2Purity:99.68%Color and Shape:SolidMolecular weight:324.39Ref: TM-T15079
1mg48.00€5mg100.00€1mL*10mM (DMSO)110.00€10mg133.00€25mg215.00€50mg306.00€100mg414.00€200mg573.00€Ruzasvir
CAS:Ruzasvir (MK-8408) is a novel and potent pan-genotypic inhibitor of hepatitis C virus NS5A with antiviral activity.Formula:C49H55FN10O7SPurity:96.87% - 99.93%Color and Shape:SolidMolecular weight:947.09KW-2450 Formate
KW-2450 Formate is an IGF-1R/IR tyrosine kinase inhibitor with antitumor effects that acts through inhibition of Aurora A and B kinases.KW-2450 Formate inhibits the growth of TNBC xenografts and induces tetraploid accumulation.Formula:C29H31N5O5SPurity:99.70%Color and Shape:SolidMolecular weight:561.65Cathepsin C-IN-6
Cathepsin C-IN-6 (compound 2), an E-64c-hydrazideas-derived inhibitor of cathepsin C, possesses anti-inflammatory properties and impedes neutrophil elastaseFormula:C24H35N5O4·xC2HF3O2Color and Shape:SolidHistatin 5 (TFA)(115966-68-2,free)
Histatin 5 (TFA)(115966-68-2,free) (Histatin 5 (TFA)) inhibits the activity of the host matrix metalloproteinases MMP-2 and MMP-9 with IC50s of 0.57 and 0.25 μMFormula:C135H196F3N51O35Purity:98%Color and Shape:SolidMolecular weight:3150.32Dihydrofuran-3(2H)-one
CAS:Dihydrofuran-3(2H)-one, with CAS No. 22929-52-8, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Dihydrofuran-3(2H)-one provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formula:C4H6O2Purity:99.92%Molecular weight:86.09Activated Protein C (390-404), human
CAS:Human Activated Protein C (390-404) peptide derived from serine protease, suppresses APC anticoagulation.Formula:C91H130N22O23Purity:98%Color and Shape:SolidMolecular weight:1900.14ADAM8-IN-1
CAS:ADAM8-IN-1 is a potent ADAM8 inhibitor with an IC 50 value of 73 nM.Formula:C44H44Br4N6O12S2Color and Shape:SolidMolecular weight:1232.6HCV-IN-4
CAS:HCV-IN-4: Potent, oral HCV NS5A inhibitor; effective vs GT1a/b, GT2b, GT3a, Y93H, L31V; EC90s: 3 pM-0.02 nM.Formula:C52H58FN9O8Purity:98%Color and Shape:SolidMolecular weight:956.07Barbituric acid
CAS:Barbituric acid is a pyrimidine derivative and the basic skeleton of barbiturate drugs, barbiturate drugs and other heterocyclic compounds.Formula:C4H4N2O3Purity:99.83%Molecular weight:128.09Tyrosinase-IN-38
Tyrosinase-IN-38 (compound 6b) is a competitive inhibitor of tyrosinase, demonstrating an IC50 of 25.82 μM and exhibits antioxidant activity.Color and Shape:Odour SolidLXE408 fumarate
LXE408 fumarate: orally available, selective kinetoplastid proteasome inhibitor with IC50/EC50 of 0.04 μM for L. donovani; potentially aids in VL research.Formula:C27H22FN7O6Purity:99.89%Color and Shape:SolidMolecular weight:559.51Ref: TM-T39214L
1mg299.00€2mg447.00€5mg563.00€1mL*10mM (DMSO)830.00€10mg897.00€25mg1,324.00€50mg1,791.00€100mg2,412.00€TMC647055 Choline salt
TMC647055 choline salt is a selective and cell-permeating inhibitor of HCV NS5B (IC50: 34 nM).Formula:C37H53N5O8SPurity:98%Color and Shape:SolidMolecular weight:727.91BAY 1217224
CAS:BAY 1217224 is a neutral, non-prodrug Thrombin inhibitor with good oral pharmacokinetics.Formula:C24H27ClFN3O5Color and Shape:SolidMolecular weight:491.94

