CymitQuimica logo
Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

Show 3 more subcategories

Found 1045 products of "Proteases/Proteasome"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • Z-LLF-CHO

    CAS:
    <p>Z-LLF-CHO (Z-Leu-Leu-Phe-CHO) effectively inhibits the chymotrypsin-like activity of the pituitary multicatalytic proteinase complex with a Ki value of 460 nM.</p>
    Formula:C29H39N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:509.64
  • SJA6017

    CAS:
    <p>SJA6017: inhibits calpain-1/2, cathepsins B/L; prevents apoptosis, protects spinal cord, boosts function. IC50s: 7.5-78 nM.</p>
    Formula:C17H25FN2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:372.45
  • AA9 TG2 inhibitor

    CAS:
    <p>AA9 is a novel transglutaminase (TG2) inhibitor.</p>
    Formula:C32H36N4O5
    Color and Shape:Solid
    Molecular weight:556.65
  • GS-9256

    CAS:
    <p>GS-9256 is a selective inhibitor of the HCV NS3 protease, exhibiting favorable pharmacokinetic properties and antiviral activity [1].</p>
    Formula:C46H56ClF2N6O8PS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:957.46
  • Cysteine Protease inhibitor

    CAS:
    <p>Cysteine protease inhibitors are inhibitors of cysteine proteases. Target: Cysteine Protease</p>
    Formula:C18H14N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:302.33
  • SQ 32602

    CAS:
    <p>SQ 32602 is a cathepsin E inhibitor.</p>
    Formula:C32H52N3O7P
    Color and Shape:Solid
    Molecular weight:621.74
  • Tyrosinase-IN-8


    <p>Tyrosinase-IN-8, a potent inhibitor of tyrosinase, demonstrates an inhibitory concentration (IC 50) value of 1.6 µM and exhibits low cytotoxicity while</p>
    Formula:C16H12O4
    Color and Shape:Solid
    Molecular weight:268.26
  • Alicapistat

    CAS:
    <p>Alicapistat (ABT-957) is a human calpains 1 and 2 inhibitor. It can potentially be used to treat Alzheimer's disease (AD).</p>
    Formula:C25H27N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:433.5
  • VEL-0230

    CAS:
    <p>VEL-0230 (NC-2300) is a cathespin K inhibitor boosting bone growth and reducing loss, targeting bone diseases and developed by Velcura Therapeutics.</p>
    Formula:C14H24NNaO5
    Color and Shape:Solid
    Molecular weight:309.33
  • JNJ-10329670

    CAS:
    <p>JNJ 10329670 is a highly potent (Ki of approximately 30 nM), nonpeptidic, noncovalent inhibitor of human cathepsin S with immunosuppressive activity.</p>
    Formula:C30H34ClF3N6O3S
    Color and Shape:Solid
    Molecular weight:651.14
  • BMS-488043

    CAS:
    <p>BMS-488043 is a novel and unique oral small molecule HIV fusion inhibitor that inhibits the attachment of Human Immunodeficiency Virus type 1 (HIV-1) to CD4(+)</p>
    Formula:C22H22N4O5
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:422.43
  • BAY-43-9695

    CAS:
    <p>BAY-43-9695 is a non-nucleoside compound with anti-human cytomegalovirus (HCMV) activity. It is the major metabolite of BAY-38-4766.</p>
    Formula:C22H25N3O4S
    Purity:99.50% - 99.65%
    Color and Shape:Solid
    Molecular weight:427.52
  • BMS-929075

    CAS:
    <p>BMS-929075 is an orally active HCV NS5B replicase (HCV NS5B replicase) palm site variant inhibitor with potency, high oral bioavailability and pharmacokinetic</p>
    Formula:C31H24F2N4O3
    Purity:98.44% - 99.94%
    Color and Shape:Solid
    Molecular weight:538.54
  • NP-313

    CAS:
    <p>NP-313 (NSC-4264) is a potent antithrombotic that blocks platelet aggregation via thromboxane A2 synthesis inhibition and targets SOCC-mediated Ca2+ efflux.</p>
    Formula:C12H8ClNO3
    Purity:98.97%
    Color and Shape:Solid
    Molecular weight:249.65
  • TY-51469

    CAS:
    <p>TY-51469 is an inhibitor of chymase (IC50s for simian and human chymases: 0.4 and 7.0 nM, respectively).</p>
    Formula:C20H15FN2O6S4
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:526.6
  • CZL55

    CAS:
    <p>CZL55 is a potent caspase-1 inhibitor with an IC50 value of 0.024 μM.CZL55 has low cytotoxicity and can be used in the study of febrile seizures (FS).</p>
    Formula:C20H22N2O6
    Purity:98.19%
    Color and Shape:Solid
    Molecular weight:386.4
  • (2RS)-FPMPA

    CAS:
    <p>(2RS)-FPMPA(FPMPA) has antiviral activity with an IC50 value of 1.85 μM measured in human MT12 cells infected with SHIV (DH4R).</p>
    Formula:C9H13FN5O4P
    Purity:99.9% - >99.99%
    Color and Shape:Solid
    Molecular weight:305.2
  • GSK-364735

    CAS:
    <p>GSK-364735 is an HIV-1 IN inhibitor.</p>
    Formula:C19H18FN3O4
    Purity:97.73%
    Color and Shape:Solid
    Molecular weight:371.36
  • TG2-IN-3h

    CAS:
    <p>TG2-IN-3h is a highly selective, potent, cell-permeable fluorescent irreversible tissue transglutaminase (tg2) inhibitor</p>
    Formula:C21H26N4O4S
    Purity:99.34% - 99.76%
    Color and Shape:Solid
    Molecular weight:430.52
  • UPGL00004

    CAS:
    <p>UPGL00004: potent GAC inhibitor, IC50=29 nM, Kd=27 nM, suppresses triple-negative breast cancer cell growth.</p>
    Formula:C25H26N8O2S2
    Purity:97.93%
    Color and Shape:Solid
    Molecular weight:534.66