
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase(38 products)
- Cysteine Protease(111 products)
- DPP-4(27 products)
- Glutaminase(46 products)
- HIV Protease(506 products)
- PAI-1(26 products)
- Protease Inhibitors(50 products)
- Protease-activated Receptor(55 products)
- Proteasome(86 products)
- Serine Protease(54 products)
- p97(15 products)
Show 3 more subcategories
Found 984 products of "Proteases/Proteasome"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Cyclotheonellazole A
CAS:Cyclotheonellazole A inhibits elastase (IC50=0.034nM) & chymotrypsin (IC50=0.62nM), a natural macrocyclic peptide.Formula:C44H54N9NaO14S2Color and Shape:SolidMolecular weight:1020.07AA74-1
CAS:AA74-1 is a potent, selective APEH inhibitor that significantly enhances T-cell proliferation by inhibiting APEH activity [1].Formula:C16H28N4O2Purity:98%Color and Shape:SolidMolecular weight:308.42Inogatran
CAS:Inogatran is a synthetic thrombin inhibitor, developed for the possible treatment and prophylaxis of venous and arterial thrombotic diseases.Formula:C21H38N6O4Purity:98%Color and Shape:SolidMolecular weight:438.56JW 480
CAS:JW480 is a potent and selective inhibitor of KIAA1363, a serine hydrolase enzyme.Formula:C22H23NO2Purity:99.72%Color and Shape:SolidMolecular weight:333.42Ref: TM-T22883
2mg35.00€5mg49.00€10mg79.00€25mg160.00€50mg259.00€100mg416.00€200mg587.00€1mL*10mM (DMSO)57.00€NS5A-IN-3
CAS:NS5A-IN-3 is a potent NS5A inhibitor with high efficacy against HCV 1b, good activity on 3a, and strong metabolic stability; superior to daclatasvir.Formula:C44H44N6O8Purity:98%Color and Shape:SolidMolecular weight:784.86Petesicatib
CAS:Petesicatib is an inhibitor of cathepsin S. Petesicatib used in the research of immune diseases.Formula:C25H23F6N5O4SPurity:99.76%Color and Shape:SolidMolecular weight:603.54Ref: TM-T16474
1mg100.00€5mg236.00€10mg371.00€25mg735.00€50mg1,134.00€100mg1,468.00€200mg1,972.00€1mL*10mM (DMSO)314.00€LU-005i
CAS:LU-005i is a powerful inhibitor targeting the β5i subunit of immunoproteasomes, displaying a high potency with an IC 50 value of 6.6 nM, and exhibits selectivity by preferring β5i over the β5c subunit, which has an IC 50 value of 287 nM [1].Formula:C31H46N4O7Color and Shape:SolidMolecular weight:586.72LY52
CAS:LY52 is a matrix metalloproteinase-2 inhibitor. It acts by suppressing tumor invasion and metastasis.Formula:C22H24N4O6Purity:98%Color and Shape:SolidMolecular weight:440.45FK706
CAS:FK706, a human neutrophil elastase inhibitor (IC50: 83 nM, Ki: 4.2 nM), also blocks mouse and porcine elastases. Anti-inflammatory.Formula:C26H33F3N4NaO7Color and Shape:SolidMolecular weight:593.556XL-784
CAS:XL-784 is a selective MMP inhibitor with low IC50s for MMP-1,2,3,8,9,13, modulating extracellular matrix remodeling, tumor invasion, and metastasis in cancer.Formula:C42H42Cl2F4MgN6O16S2Purity:98%Color and Shape:SolidMolecular weight:1122.15BMS-538305 HCl
CAS:BMS-538305 is a potent, selective inhibitor of dipeptidyl peptidase IV (DPP-IV).Formula:C17H27ClN2O2Color and Shape:SolidMolecular weight:326.86(Rac)-Neurodegenerative Disorder-Targeting Compound 1
CAS:(Rac)-Neurodegenerative Disorder-Targeting Compound 1 is a calpain inhibitor.Formula:C28H28N4O4Color and Shape:SolidMolecular weight:484.55KCC009
CAS:KCC009 is a potent and selective Transglutaminase 2 Inhibitor.Formula:C21H22BrN3O5Color and Shape:SolidMolecular weight:476.32JTK-853
CAS:JTK-853: novel non-nucleoside HCV polymerase inhibitor with strong antiviral activity (EC50: 0.38 μM genotype 1a, 0.035 μM 1b).Formula:C28H23F7N6O4S2Purity:98%Color and Shape:SolidMolecular weight:704.64MMP-9-IN-8
CAS:MMP-9-IN-8 (Compound 3), an MMP-9 inhibitor, exhibits inhibitory activities of 42.16% at 10 μM and 58.28% at 50 μM.Formula:C20H21F4N7OColor and Shape:SolidMolecular weight:451.42Z-DEVD-CMK
CAS:Z-DEVD-CMK irreversibly inhibits various cathepsins in vitro [1].Formula:C27H35ClN4O12Color and Shape:SolidMolecular weight:643.04DCLK1-IN-2
CAS:DCLK1-IN-2 (Compound I-5) is a potent inhibitor of DCLK1, exhibiting an IC50 of 171.3 nM, and demonstrates significant antiproliferative effects on SW1990 cellFormula:C26H32N8O3SColor and Shape:SolidMolecular weight:536.65BMS-189664 HCl
CAS:BMS-189664 HCl is a selective and orally active thrombin active site inhibitor.Formula:C22H35ClN6O4SPurity:98%Color and Shape:SolidMolecular weight:515.07Ravidasvir HCl
CAS:Ravidasvir, also known as PPI-668 and ASC16, is a second-generation, orally active, potent and selective HCV NS5A protein inhibitor.Formula:C42H52Cl2N8O6Color and Shape:SolidMolecular weight:835.828Z-LVG
CAS:Z-LVG, an irreversible cysteine protease inhibitor and a tripeptide derivative of cystatin C, serves as an inhibitor of viral replication and is utilized inFormula:C21H31N3O6Color and Shape:SolidMolecular weight:421.49

