CymitQuimica logo
Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

Show 3 more subcategories

Found 985 products of "Proteases/Proteasome"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • GLS-1-IN-1


    GLS-1-IN-1 (compound 1d) is a GLS-1 inhibitor that inhibits Hep G2, MCF 7 and MCF 10A cells.
    Formula:C26H25FN4OS
    Color and Shape:Solid
    Molecular weight:460.57

    Ref: TM-T62905

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Tilpisertib fosmecarbil

    CAS:
    Tilpisertib fosmecarbil is a potent inhibitor of serine/threonine kinases with anti-inflammatory properties.
    Formula:C35H36ClN8O7P
    Color and Shape:Solid
    Molecular weight:747.14

    Ref: TM-T72292

    25mg
    2,853.00€
    50mg
    3,763.00€
    100mg
    5,220.00€
  • RBx-0597

    CAS:
    RBx-0597 is a selective DPP-IV inhibitor with IC50 values of 32 nM, 31 nM, and 39 nM for human, mouse, and rat plasma DPP-IV, respectively. It is utilized in research focused on type 2 diabetes.
    Formula:C19H20F2N4O2
    Color and Shape:Solid
    Molecular weight:374.384

    Ref: TM-T206740

    10mg
    To inquire
    50mg
    To inquire
  • (1R,3S)-THCCA-Asn


    (1R,3S)-THCCA-Asn (4j) is a selective inhibitor of thrombin (IC50: 0.07-0.14 μM) with anti-thrombotic effects.
    Formula:C24H24N4O6
    Color and Shape:Solid
    Molecular weight:464.47

    Ref: TM-T62949

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • UK 356618

    CAS:
    UK 356618 is a potent and selective inhibitor of matrix metalloprotease-3 (IC50: 5.9 nM).
    Formula:C34H43N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:557.72

    Ref: TM-T17201

    5mg
    386.00€
    10mg
    673.00€
    25mg
    1,369.00€
  • GSK5852


    GSK5852, an HCV NS5B inhibitor, has IC50 of 50 nM; potently fights HCV with EC50 of 3.0 nM for GT1a and 1.7 nM for GT1b.
    Formula:C27H27BF2N2O6S
    Color and Shape:Solid
    Molecular weight:556.39

    Ref: TM-T63936

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 3-Aminobenzene-1,2-diol

    CAS:
    3-Aminobenzene-1,2-diol (compound C8) is an inhibitor of matrix metalloproteinases (MMP), with IC50 values of 20, 26, 16, and 16.3 μM against MMP-2, MMP-8, MMP-9, and MMP-14, respectively.
    Formula:C6H7NO2
    Color and Shape:Solid
    Molecular weight:125.13

    Ref: TM-T201595

    10mg
    To inquire
    50mg
    To inquire
  • HCV-IN-40

    CAS:
    HCV-IN-39 is a potent oral drug inhibiting HCV, effective on GT1a (EC50: 0.259μM), GT1b (EC50: 0.434μM), GT1b CES1 (EC50: 0.069μM) replicons.
    Formula:C21H26BrFN3O9P
    Color and Shape:Solid
    Molecular weight:594.32

    Ref: TM-T64202

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BAY-7598

    CAS:
    BAY-7598 is a potent, selective, and orally bioavailable MMP12 inhibitor (IC50s: 0.085, 0.67, and 1.1 nM for human/murine/rat MMP12).
    Formula:C28H31N3O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:505.56

    Ref: TM-T10474

    25mg
    3,348.00€
    50mg
    4,213.00€
    100mg
    5,580.00€
  • HCV NS5B polymerase-IN-2

    CAS:
    HCVNS5B polymerase-IN-2 (Compound 298) is an inhibitor of the Ns5b polymerase. It holds potential for research into the treatment of hepatitis C virus (HCV) infections.
    Formula:C26H24N2O4
    Color and Shape:Solid
    Molecular weight:428.48

    Ref: TM-T204671

    10mg
    To inquire
    50mg
    To inquire
  • Isobutylamido thiazolyl resorcinol

    CAS:
    Isobutylamido thiazolyl resorcinol is a tyrosinase (Tyrosinase) inhibitor that prevents pigment deposition induced by ultraviolet radiation.
    Formula:C13H14N2O3S
    Color and Shape:Solid
    Molecular weight:278.33

    Ref: TM-T201683

    10mg
    To inquire
    50mg
    To inquire
  • GW311616 hydrochloride

    CAS:
    GW-311616 hydrochloride is a long duration, orally bioavailable, and selective human neutrophil elastase (HNE) inhibitor (IC50: 22 nM; Ki: 0.31 nM).
    Formula:C19H32ClN3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:433.99

    Ref: TM-T11525L

    1mg
    273.00€
    5mg
    818.00€
    10mg
    1,359.00€
  • HCV-IN-38


    Potent oral HCV inhibitor HCV-IN-38 has 15 nM EC50, 431 SI, high efficacy, and low toxicity.
    Formula:C22H24ClF3N4O4
    Color and Shape:Solid
    Molecular weight:500.9

    Ref: TM-T63396

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SBI-581


    SBI-581: oral, potent TAO3 inhibitor, IC50=42nM, alters TKS5α at RAB11+ vesicles, blocks invadopodia, good mouse pharmacokinetics, anti-tumor.
    Formula:C24H21N3O2
    Color and Shape:Solid
    Molecular weight:383.44

    Ref: TM-T61663

    25mg
    1,305.00€
    50mg
    2,088.00€
    100mg
    3,357.00€
  • MK-8876

    CAS:
    MK-8876 is an Inhibitor of HCV NS5B Site D.
    Formula:C32H24F2N4O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:614.62

    Ref: TM-T28061

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Cathepsin C-IN-3


    Cathepsin C-IN-3 is a potent inhibitor of histone C (IC50: 61.79 nM) and also inhibits THP-1 cells (IC50: 101.5 nM) and U937 cells (IC50: 86.5 nM).
    Formula:C28H21F3N6OS
    Color and Shape:Solid
    Molecular weight:546.57

    Ref: TM-T63854

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Plasma kallikrein-IN-2


    Plasma kallikrein-IN-2: PKal inhibitor, IC50=0.1 nM. Used in angioedema, diabetic eye disease research.
    Formula:C28H24ClF3N8O3
    Color and Shape:Solid
    Molecular weight:612.99

    Ref: TM-T72337

    25mg
    2,718.00€
    50mg
    3,582.00€
    100mg
    4,950.00€
  • AMG-222 tosylate

    CAS:
    AMG-222 tosylate is a DPP-IV inhibitor in clinical development for type II diabetes.
    Formula:C39H47N9O6S
    Color and Shape:Solid
    Molecular weight:769.91

    Ref: TM-T71354

    25mg
    3,664.00€
    50mg
    4,843.00€
    100mg
    6,840.00€
  • Faldaprevir

    CAS:
    Faldaprevir is an orally effective, selective, non-covalent HCV NS3/4A protease inhibitor with high inhibitory activity against HCV 1a and 1b genotype.
    Formula:C40H49BrN6O9S
    Purity:99.04% - 99.19%
    Color and Shape:Solid
    Molecular weight:869.82

    Ref: TM-T19685

    1mg
    250.00€
    5mg
    610.00€
    10mg
    853.00€
    25mg
    1,243.00€
  • BI-1915

    CAS:

    BI-1915 is a selective inhibitor of Cathepsin S, with an IC50 of 17 nM. It is utilized in the research of autoimmune diseases.

    Formula:C21H37N5O3
    Color and Shape:Solid
    Molecular weight:407.55

    Ref: TM-T206466

    10mg
    To inquire
    50mg
    To inquire