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Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

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Found 1045 products of "Proteases/Proteasome"

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  • Probenecid

    CAS:
    <p>Probenecid (Benemid) is a benzoic acid derivative with antihyperuricemic property.</p>
    Formula:C13H19NO4S
    Purity:98.95% - 99.84%
    Color and Shape:Crystals From Dil Alcohol Pleasant Aftertaste (Ntp 1992)
    Molecular weight:285.36
  • ARP-100

    CAS:
    <p>ARP-100 (MMP-2 Inhibitor III) is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM).</p>
    Formula:C17H20N2O5S
    Purity:97.18%
    Color and Shape:Solid
    Molecular weight:364.42
  • BRD-6929

    CAS:
    <p>BRD-6929, a brain-targeted HDAC1/2 inhibitor (IC50 1/8 nM), enhances gnidimacrin's anti-HIV effect, useful in mood behavior studies.</p>
    Formula:C19H17N3O2S
    Purity:98.01% - 99.05%
    Color and Shape:Solid
    Molecular weight:351.42
  • Hck-IN-1

    CAS:
    <p>Hck-IN-1 selectively inhibits Nef:Hck, IC50: 2.8 μM; &gt;20 μM for Hck alone. Potent HIV-1 Nef antagonist, IC50: 100-300 nM for HIV-1 replication.</p>
    Formula:C16H11ClN6O3S
    Purity:99.07%
    Color and Shape:Solid
    Molecular weight:402.81
  • PF-3450074

    CAS:
    <p>PF-3450074 (PF-74) is a specific HIV-1 inhibitor, blocking viral replication and uncoating at submicromolar EC50=8-640 nM.</p>
    Formula:C27H27N3O2
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:425.52
  • RA190

    CAS:
    <p>RA190 inhibits proteasome function by covalently binding to cysteine 88 of ubiquitin receptor RPN13.</p>
    Formula:C28H23Cl5N2O2
    Purity:97.7%
    Color and Shape:Solid
    Molecular weight:596.76
  • RAMB4

    CAS:
    <p>RAMB4 (PTP1B-IN-9) is a ubiquitin-proteasome system (UPS)-stressor,with anticancer activity.</p>
    Formula:C19H13Cl4NO
    Purity:98.89% - 99.38%
    Color and Shape:Solid
    Molecular weight:413.12
  • GSK2838232

    CAS:
    <p>GSK2838232 inhibit HIV reverse transcriptase activity across a broad panel of HIV-1 isolates,GSK2838232 is novel human immune virus (HIV) maturation inhibitor.</p>
    Formula:C48H73ClN2O6
    Purity:97.97%
    Color and Shape:Solid
    Molecular weight:809.56
  • DBPR108

    CAS:
    <p>DBPR108 is an orally bioavailable dipeptide-derived DPP4 inhibitor (IC50: 15 nM) and it has no inhibition on DDP8 and DPP9.</p>
    Formula:C16H25FN4O2
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:324.39
  • 3-Aminopropionitrile fumarate (2:1)

    CAS:
    <p>3-Aminopropionitrile fumarate (2:1) (β-Aminopropionitrile fumarate) is an organic compound and antirheumatic agent used in veterinary medicine.</p>
    Formula:C4H4O4·2C3H6N2
    Purity:99.76% - >99.99%
    Color and Shape:White Crystalline Powder
    Molecular weight:256.26
  • Ref: IN-DA0048C1

    1mg
    50.00€
    5mg
    50.00€
    25mg
    155.00€
    50mg
    197.00€
    100mg
    331.00€
    250mg
    531.00€
  • Islatravir

    CAS:
    <p>Islatravir (MK-8591) is an effective anti-HIV-1 agent.</p>
    Formula:C12H12FN5O3
    Purity:98.77%
    Color and Shape:Solid
    Molecular weight:293.25
  • Sofosbuvir impurity F

    CAS:
    <p>Sofosbuvir impurity F (Sofosbuvir 3',5'-Bis-(S)-phosphate) is both a diastereomer of Sofosbuvir and an impurity of Sofosbuvir which is an inhibitor of HCV RNA</p>
    Formula:C34H45FN4O13P2
    Purity:98.05%
    Color and Shape:Solid
    Molecular weight:798.69
  • Bivalirudin acetate


    <p>Bivalirudin acetate is a thrombin inhibitor, a peptide-based anticoagulant, used for research on acute coronary syndrome.</p>
    Formula:C100H142N24O35
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:2240.34
  • BJJF078

    CAS:
    <p>BJJF078, an aminopiperidine, inhibits human/mouse TG2 (IC50: 41/54 nM) and TG1 (IC50: 0.16 μM), may be used in MS studies.</p>
    Formula:C27H29N3O6S
    Purity:98.19%
    Color and Shape:Soild
    Molecular weight:523.6
  • Aprotinin

    CAS:
    <p>Aprotinin (Traskolan) is a broad-spectrum serine protease (BPTI) inhibitor. Aprotinin is an antifibrinolytic agent. Cost-effective and quality-assured.</p>
    Formula:C284H432N84O79S7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:6511.51
  • 6-Acetylnimbandiol

    CAS:
    <p>6-Acetylnimbandiol, a non-toxic agent, inhibits tyrosinase (IC50=69.85 μM), melanin, and MITF; useful in melanoma studies.</p>
    Formula:C28H34O8
    Color and Shape:Solid
    Molecular weight:498.56
  • α 1(I) Collagen (614-639), human

    CAS:
    <p>This is a peptide inhibitor of collagen fibrillar matrix assembly.</p>
    Formula:C134H189N37O39
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2942.16
  • EP 171

    CAS:
    <p>EP 171 is a potent agonist of TP-receptors.</p>
    Formula:C23H29FO5
    Color and Shape:Solid
    Molecular weight:404.47
  • Berotralstat

    CAS:
    <p>Berotralstat (BCX7353) is an oral, low-toxicity, specific kallikrein inhibitor for hereditary angioedema research, blocking bradykinin release.</p>
    Formula:C30H26F4N6O
    Color and Shape:Solid
    Molecular weight:562.56