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Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

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Found 987 products of "Proteases/Proteasome"

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  • ABT-770

    CAS:
    ABT-770: an orally potent and selective MMP inhibitor, shown to reduce tumor growth in animal models.
    Formula:C22H22F3N3O6
    Color and Shape:Solid
    Molecular weight:481.42

    Ref: TM-T29532

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Antiviral agent 30

    CAS:
    Antiviral Agent 30 (Example 118) is an active compound against HCV and RSV with an inhibitory concentration (IC 50) of greater than 25μM [1].
    Formula:C21H32N2O3S
    Color and Shape:Solid
    Molecular weight:392.56

    Ref: TM-T79128

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A-933548

    CAS:
    A-933548: potent calpain inhibitor, selective vs. cathepsins, stable, effective in cell assays.
    Formula:C25H21N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:439.47

    Ref: TM-T23596

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • SP-Chymostatin B

    CAS:
    SP-Chymostatin B inhibits proteases like chymotrypsin and papain; less effective on human elastase; works at 100-200 μg/ml.
    Formula:C30H41N7O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:595.69

    Ref: TM-T26202

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • DPP-IV-IN-1

    CAS:
    DPP-IV-IN-1 is an effective inhibitor of dipeptidyl peptidase IV (DPP-IV), a serine protease (IC50: 4.6 nM).
    Formula:C11H18FN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:243.28

    Ref: TM-T10082

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (Rac)-Tanomastat

    CAS:
    Tanomastat (BAY 12-9566) is an oral biphenyl MMP inhibitor; blocks MMP-2, -3, -9, -13, with anti-invasive and anti-metastatic properties.
    Formula:C23H19ClO3S
    Color and Shape:Solid
    Molecular weight:410.91

    Ref: TM-T62090

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GSK2793660 HCl

    CAS:
    GSK2793660 is a irreversible covalent α,β-unsaturated amide based DPP1 inhibitor.
    Formula:C22H32ClN3O3
    Color and Shape:Solid
    Molecular weight:421.96

    Ref: TM-T27468

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Cysteine Protease inhibitor

    CAS:
    Cysteine protease inhibitors are inhibitors of cysteine proteases. Target: Cysteine Protease
    Formula:C18H14N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:302.33

    Ref: TM-T10925

    25mg
    610.00€
  • Elastase-IN-1

    CAS:
    Elastase-IN-1 (Compound Q11) is a non-toxic elastase inhibitor with an IC 50 of 0.897 μM [1].
    Formula:C17H12N4O3
    Color and Shape:Solid
    Molecular weight:320.3

    Ref: TM-T60855

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Plasma kallikrein-IN-3

    CAS:
    Plasma kallikrein-IN-3 is a potent inhibitor (IC50: 0.15 μM) used in hereditary angioedema and diabetic eye disease research.
    Formula:C20H23N5O2
    Color and Shape:Solid
    Molecular weight:365.43

    Ref: TM-T61403

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • HCV-IN-3

    CAS:
    HCV-IN-3 is a hepatitis C virus (HCV) NS3/4a protein inhibitor (IC50: 20 μM; Kd: 29 μM).
    Formula:C13H11F2NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:235.23

    Ref: TM-T11540

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Cathepsin L/S-IN-1


    Cathepsin L/S-IN-1 inhibits Cathepsin L & S (IC50: 4.10 & 1.79 μM) and reduces metastasis in pancreatic cancer cells.
    Formula:C29H33BrN4O4S
    Color and Shape:Solid
    Molecular weight:613.57

    Ref: TM-T72569

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ro 09-1679

    CAS:
    Ro 09-1679 is a thrombin inhibitor.
    Formula:C22H39N9O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:525.6

    Ref: TM-T28553

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • JPM-OEt

    CAS:
    JPM-OEt: broad-spectrum, covalent cysteine cathepsin inhibitor with antitumor effects.
    Formula:C20H28N2O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:392.45

    Ref: TM-T15626

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Grazoprevir sodium salt

    CAS:
    Grazoprevir sodium salt is a selective Hepatitis C virus NS3/4a protease inhibitor with broad activity across genotypes and resistant variants.
    Formula:C38H50N6NaO9S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:789.9

    Ref: TM-T12065

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Prodipine hydrochloride

    CAS:
    Prodipine hydrochloride for purified and plasma Dipeptidyl peptidase IV (DPP IV) from the rabbit (IC50 of 4.5 μM and 30 μM, respectively).
    Formula:C20H26ClN
    Purity:98%
    Color and Shape:Solid
    Molecular weight:315.88

    Ref: TM-T13826

    50mg
    715.00€
    100mg
    1,071.00€
  • DTS

    CAS:
    DTS is a selective and isoform-specific RSK1 kinase inhibitor. It also has broad cancer therapeutic potential.
    Formula:C14H14S3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:278.46

    Ref: TM-T24020

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Cyclophilin inhibitor 3

    CAS:
    Cyclophilin inhibitor 3 (compound 7c), a potent inhibitor of cyclophilin A (CypA), exhibited potent anti-HCV effects with an EC50 value of 4.2 μM.
    Formula:C34H38N4O6
    Color and Shape:Solid
    Molecular weight:598.69

    Ref: TM-T64220

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Desirudin

    CAS:
    Desirudin (CGP 39393) inhibits thrombin, prevents thrombosis, and is used in thrombocytopenia research.
    Color and Shape:Solid

    Ref: TM-T64250

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AA9 TG2 inhibitor

    CAS:
    AA9 is a novel transglutaminase (TG2) inhibitor.
    Formula:C32H36N4O5
    Color and Shape:Solid
    Molecular weight:556.65

    Ref: TM-T69878

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • STOCK2S-26016

    CAS:
    WNK-IN-B, a cell-permeable diaminoacridine, selectively inhibits WNK signaling in mpkDCT/MOVAS by targeting SPAK/OSR1 CCT domain.
    Formula:C20H19N3O2
    Color and Shape:Solid
    Molecular weight:333.38

    Ref: TM-T29161

    25mg
    1,396.00€
    50mg
    1,815.00€
    100mg
    2,375.00€
  • Desethyl KBT-3022

    CAS:
    Desethyl KBT-3022 is an active metabolite of the antiplatelet compound KBT-3022.
    Formula:C23H20N2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:420.48

    Ref: TM-T10083

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • IMB-26

    CAS:
    IMB-26 is an HCV inhibitor (EC50: 2.1 μM) and has shown potent anti-HCV effects.
    Formula:C20H23BrN2O6
    Color and Shape:Solid
    Molecular weight:467.31

    Ref: TM-T62993

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • MDL-101146, (S)-

    CAS:
    MDL-101146, (S)- is an effective orally active inhibitor of human neutrophil elastase.
    Formula:C29H37F5N4O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:632.62

    Ref: TM-T25784L

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • U 27391

    CAS:
    U 27391 is a metalloproteinase inhibitor. It acts by inhibits the action of human recombinant interleukin-1beta and glycosaminoglycan synthesis.
    Formula:C23H36N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:448.56

    Ref: TM-T26304

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LB-30057

    CAS:
    LB-30057 is used as an oral thrombin inhibitor.
    Formula:C26H31N5O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:493.62

    Ref: TM-T25646

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • BMS-986094

    CAS:
    INX 08189 is an RNA-directed RNA polymerase (NS5B) inhibitor.
    Formula:C30H39N6O9P
    Color and Shape:Solid
    Molecular weight:658.64

    Ref: TM-T27616

    2mg
    93.00€
    50mg
    642.00€
    100mg
    1,116.00€
  • FK-448 Free base

    CAS:
    FK-448 Free base is an effective and specific inhibitor of chymotrypsin, with an IC50 of 720 nM.
    Formula:C25H30N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:406.52

    Ref: TM-T11290

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • KIN1400

    CAS:
    KIN1400 activates IRF3, boosts antiviral immunity, stimulates IFNbeta, and inhibits WNV, DV, and HCV.
    Formula:C24H17F2N3O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:449.47

    Ref: TM-T27732

    5mg
    310.00€
  • HCV-IN-37

    CAS:
    HCV-IN-37: potent HCV inhibitor, stable in rat plasma post-oral dose (15 mg/kg), blocks virus entry phase.
    Formula:C31H35F2N5
    Color and Shape:Solid
    Molecular weight:515.64

    Ref: TM-T63585

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LY 135305

    CAS:
    LY 135305 is a inhibition of spontaneous metastasis.
    Formula:C19H20ClN
    Purity:98%
    Color and Shape:Solid
    Molecular weight:297.82

    Ref: TM-T27874

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Thrombin inhibitor 6

    CAS:
    Thrombin Inhibitor 6, with an IC 50 of 1 nM, acts as a potent anticoagulant by inhibiting thrombin.
    Formula:C18H19ClN4O2S
    Color and Shape:Solid
    Molecular weight:390.89

    Ref: TM-T72448

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ono-3307 mesylate

    CAS:
    no-3307 mesylate is a protease inhibitor that inhibits a variety of proteases and may be used to study pancreatitis.
    Formula:C15H18N4O7S2
    Purity:97.60% - 98.16%
    Color and Shape:Solid
    Molecular weight:430.46

    Ref: TM-T28248

    1mg
    279.00€
    5mg
    685.00€
    10mg
    938.00€
    25mg
    1,444.00€
    50mg
    1,882.00€
  • RS-104966

    CAS:
    RS-104966 is an inhibitor of collagenase that acts by inducing the conformational change in the side-chains of the S1 pocket of MMP-1.
    Formula:C19H21NO6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:391.44

    Ref: TM-T24740

    25mg
    1,786.00€
    50mg
    2,860.00€
    100mg
    4,576.00€
  • BR351 precursor

    CAS:
    BR351 precursor is a precursor of BR351. BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).
    Formula:C27H32N2O8S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:576.68

    Ref: TM-T10598

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • WNK-IN-7

    CAS:
    WNK-IN-7 is a potent and selective WNK1 kinase inhibitor.
    Formula:C26H29N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.53

    Ref: TM-T24049

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BAY-678 racemate

    CAS:
    BAY-678 racemate: orally active, selective cell-permeable HNE inhibitor with IC50 of 20 nM.
    Formula:C20H15F3N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:400.35

    Ref: TM-T19202

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PTIQ

    CAS:
    MMP-3 expression inhibitor
    Formula:C13H17NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:235.28

    Ref: TM-T23206

    25mg
    224.00€
    50mg
    424.00€
    100mg
    802.00€
    250mg
    1,890.00€
  • K 579

    CAS:
    K 579 is a dipeptidyl peptidase IV inhibitor.
    Formula:C17H24N6O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:328.41

    Ref: TM-T22886

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • TNK2-IN-1

    CAS:
    TNK2-IN-1 is a TNK2 inhibitor (IC50: 224 nM) that can be used in cancer research.
    Formula:C23H24N6O2
    Color and Shape:Solid
    Molecular weight:416.48

    Ref: TM-T62164

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GSK-2793660

    CAS:
    GSK-2793660, an oral, irreversible CTSC inhibitor, aids bronchiectasis research.
    Formula:C20H27N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:357.45

    Ref: TM-T11466

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Epostatin

    CAS:
    Epostatin is a new dipeptidyl peptidase II (DPP-II, EC 3.4.14.2) inhibitor.
    Formula:C23H33N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:431.53

    Ref: TM-T25382

    25mg
    1,369.00€
  • WAY-151693

    CAS:
    WAY-151693 is an inhibitor of human collagenase-3 (MMP-13).
    Formula:C21H22ClN3O5S
    Color and Shape:Solid
    Molecular weight:463.93

    Ref: TM-T29150

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Nucleoside-Analog-1

    CAS:
    Nucleoside-Analog-1 is a 4′-Azidocytidine analogue, used to against Hepatitis C virus replication.
    Formula:C9H9N5O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.2

    Ref: TM-T19485

    2mg
    178.00€
    5mg
    313.00€
    25mg
    1,026.00€
    50mg
    1,341.00€
    100mg
    1,791.00€
  • YM-53601

    CAS:
    YM-53601 is an SQS inhibitor that inhibits adipogenic biosynthesis and lipid secretion in rodents.YM-53601 is a cholesterol-lowering agent that inhibits FDFT1.
    Formula:C21H22ClFN2O
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:372.86

    Ref: TM-T26345

    1mg
    152.00€
    5mg
    371.00€
    10mg
    595.00€
    25mg
    1,189.00€
    50mg
    1,935.00€
    1mL*10mM (DMSO)
    409.00€
  • ND-336

    CAS:
    ND-336 selectively inhibits MMP-2, MMP-9, MMP-14, boosts diabetic wound healing, reduces inflammation, and promotes angiogenesis and skin repair.
    Formula:C16H18ClNO3S2
    Color and Shape:Solid
    Molecular weight:371.9

    Ref: TM-T28146

    1mg
    268.00€
    5mg
    1,108.00€
    10mg
    1,953.00€
    500µg
    148.00€
  • Bz-D-Arg-pNA hydrochloride

    CAS:
    Bz-D-Arg-pNA hydrochloride is a competitive trypsin inhibitor.
    Formula:C19H23ClN6O4
    Color and Shape:Solid
    Molecular weight:434.88

    Ref: TM-T62464

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • NVP DPP 728 dihydrochloride

    CAS:
    NVP-DPP728 is a reversible DPP-IV inhibitor with a K i of 11 nM, enhancing insulin release by preventing GLP-1 degradation, used for diabetes research.
    Formula:C15H18N6O
    Color and Shape:Solid
    Molecular weight:298.34

    Ref: TM-T21691

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GLS1 Inhibitor

    CAS:
    GLS1 inhibitor blocks glutaminase 1 (IC50=0.021 μM), hinders NCI H1703 NSCLC cell growth in vitro (GI50=0.011 μM), and suppresses tumors in mice.
    Formula:C19H21N7O2S
    Color and Shape:Solid
    Molecular weight:411.48

    Ref: TM-T37222

    1mg
    105.00€
    5mg
    304.00€
    10mg
    444.00€
  • Nucleoside-Analog-2

    CAS:
    Nucleoside-Analog-2 is a 4'-Azidocytidine analogue, used to against Hepatitis C virus (HCV) replication.
    Formula:C9H11N5O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:285.21

    Ref: TM-T19486

    2mg
    178.00€
    5mg
    313.00€
    25mg
    1,026.00€
    50mg
    1,341.00€
    100mg
    1,791.00€
    1mL*10mM (DMSO)
    344.00€