
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase(38 products)
- Cysteine Protease(111 products)
- DPP-4(27 products)
- Glutaminase(46 products)
- HIV Protease(506 products)
- PAI-1(26 products)
- Protease Inhibitors(50 products)
- Protease-activated Receptor(55 products)
- Proteasome(86 products)
- Serine Protease(54 products)
- p97(15 products)
Show 3 more subcategories
Found 985 products of "Proteases/Proteasome"
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Azo-Resveratrol
CAS:Azo-Resveratrol is an analog of Resveratrol used as a potent tyrosinase inhibitor.Formula:C12H10N2O3Color and Shape:SolidMolecular weight:230.22HCV-IN-34
CAS:HCV-IN-35, an oral HCV blocker, has an EC50 of 0.010 μM and a CC50 of 7.5 μM, indicating strong antiviral effects.Formula:C31H36ClN5Color and Shape:SolidMolecular weight:514.1Tyrosinase-IN-7
CAS:Tyrosinase-IN-7 is a small-molecule tyrosinase inhibitor (IC50 1.57 μM) that suppresses melanin activity and cell growth with low cytotoxicity.Formula:C15H10O5Purity:99%Color and Shape:SolidMolecular weight:270.24BC-05
CAS:BC-05, an orally active inhibitor targeting CD13 and the proteasome, displays potent inhibition with IC50 values of 0.13 μM against human CD13 and 1.39 μM forFormula:C21H29BN2O9Purity:98%Color and Shape:SolidMolecular weight:464.27RID-F
CAS:RID-F is an inhibitor of the nonpeptidic proteasome.Formula:C38H50N2O2Purity:98%Color and Shape:SolidMolecular weight:566.82AL-9
CAS:AL-9 is a GT-1b and GT-2a replication inhibitor.Formula:C23H22N4O3Purity:98%Color and Shape:SolidMolecular weight:402.45PMPA sodium
CAS:PMPA sodium is a potent and selective glutamate carboxypeptidase 2 (GCP II/N-acetylated a-linked dipeptidase/NAALADase) inhibitor.Formula:C6H11Na4O7PPurity:98%Color and Shape:SolidMolecular weight:318.08Tyrosinase-IN-11
CAS:Tyrosinase-IN-11: potent inhibitor, IC50 - 50nM/64nM (L-tyrosinase/L-dopa), antioxidant, low toxicity, for hyperpigmentation study.Formula:C15H14O5Color and Shape:SolidMolecular weight:274.27Kallikrein 5-IN-2
CAS:Kallikrein 5-IN-2 inhibits KLK5 (pIC50=7.1); may normalize skin shedding, lessen inflammation & itching.Formula:C23H22N6OColor and Shape:SolidMolecular weight:398.46VA4 TG2 inhibitor
CAS:VA4 is a novel irreversible TG2 transamidase site-specific inhibitor.Formula:C33H41N5O6SColor and Shape:SolidMolecular weight:635.77AZD5248
CAS:AZD-5248 is a potent, selective, first generation, oral inhibitor of dipeptidyl peptidase 1 (DPP1).Formula:C22H22N4O2Color and Shape:SolidMolecular weight:374.44BMS-363131
CAS:BMS-363131 (BMS363131) is a potent and selective trypsin inhibitor with an IC50 value of <1.7 nM.Formula:C28H40N6O5Purity:97.99%Color and Shape:SolidMolecular weight:540.65α-Glucosidase-IN-5
CAS:α-Glucosidase-IN-5 (compound 8) is isolated from a twig extract of Polyalthia cinnamomea which is a potent α-glucosidase inhibitor with an IC50 of 57.9 µM.Formula:C15H13NO3Color and Shape:SolidMolecular weight:255.27SAP2-IN-1
CAS:SAP2-IN-1 inhibits secreted aspartate protease 2 (IC50: 0.92 μM), doesn't work in vitro, and helps research infections.Formula:C34H29NO7Color and Shape:SolidMolecular weight:563.6Glutaminase-IN-4
CAS:Glutaminase-IN-4 (compound 2a) is a glutaminase (GLS) inhibitor (IC50: 2.3 μM).Formula:C23H22N6O2S2Color and Shape:SolidMolecular weight:478.59L 658758
CAS:L 658758 is an inhibitor of serine proteinase.Formula:C16H20N2O9SColor and Shape:SolidMolecular weight:416.4BC-23
CAS:BC-23 (NSC 45382) is a proteasome inhibitor with antitumor and antimicrobial activity for the study of leukemia and small cell lung cancer.Formula:C21H14ClN3O4SPurity:98%Color and Shape:SolidMolecular weight:439.87AGLME
CAS:AGLME is used in a direct enzymatic assay for activated Hageman factor measuring the ability of Hageman factor to hydrolyze the cpd.Formula:C11H21N3O4Color and Shape:SolidMolecular weight:259.3BI-L 45XX
CAS:BI-L 45XX, an anti-inflammatory benzimidazole derivative, has inhibitory effects on neutrophil function.Formula:C10H9F3N2O2SColor and Shape:SolidMolecular weight:278.25Tyrphostin 47
CAS:Tyrphostin 47 inhibits the protein-tyrosine kinase activity of EGF-R.Formula:C10H8N2O2SColor and Shape:SolidMolecular weight:220.25Levovirin valinate HCl
CAS:Levovirin valinate HCl is a valine ester prodrug of levovirin as a new investigational drug for the therapy of the hepatitis C virus.Formula:C13H22ClN5O6Purity:98%Color and Shape:SolidMolecular weight:379.8Ici 186756
CAS:Ici 186756 is a novel, effective, and selective inhibitor of human neutrophil elastase.Formula:C33H49N5O9Purity:98%Color and Shape:SolidMolecular weight:659.77Chymase-IN-2
CAS:Chymase-IN-2 is a modulator of chymase.Formula:C19H15ClF2NO3PSPurity:98%Color and Shape:SolidMolecular weight:441.82A-953227
CAS:A-953227: Selective calpain inhibitor with improved cathepsin selectivity, strong microsomal stability, and cellular efficacy.Formula:C25H20FN5O3Purity:98%Color and Shape:SolidMolecular weight:457.46Duazomycin
CAS:Duazomycin, an antitumor substance and glutamine antagonist, is used as a chemotherapeutic agent.Formula:C8H11N3O4Color and Shape:SolidMolecular weight:213.19Moxicoumone
CAS:Moxicoumone is an anticoagulant agent.Formula:C22H30N2O6Purity:98%Color and Shape:SolidMolecular weight:418.48Tyrphostin A46
CAS:Tyrphostin A46 is an antagonist of the epidermal growth factor-urogastrone receptor.Formula:C10H8N2O3Purity:98%Color and Shape:Off-White SolidMolecular weight:204.18MDK0734
CAS:MDK0734 is a selective inhibitor of cathepsin B endopeptidase and exopeptidase activities.Formula:C15H17N3O2Purity:98%Color and Shape:SolidMolecular weight:271.31FQ
CAS:FQ is a novel reversible inhibitor of mixed-type tyrosinase.Formula:C14H9FN2OColor and Shape:SolidMolecular weight:240.23ADAMTS-5 Inhibitor
CAS:ADAMTS-5 Inhibitor is an inhibitor of ADAMTS-5 with an IC50 of 1.1 µM and can be used in studies about cartilage destruction in arthritis.Formula:C16H11ClF3N3OS3Purity:99.66%Color and Shape:SolidMolecular weight:449.92Ref: TM-T14124
1mg46.00€5mg93.00€10mg122.00€25mg193.00€50mg289.00€100mg414.00€200mg580.00€1mL*10mM (DMSO)96.00€TNIK-IN-1
CAS:TNIK-IN-1 is an inhibitor of Traf2- and Nck-interacting kinase (TNIK).Formula:C19H17N5O3SPurity:98%Color and Shape:SolidMolecular weight:395.43Diethyl pyimDC
CAS:Diethyl pyimDC is an inhibitor of human collagen prolyl 4-hydroxylase 1 (CP4H1).Formula:C14H15N3O4Color and Shape:SolidMolecular weight:289.29Aldumastat
CAS:Aldumastat (GLPG1972) is a highly potent, specific and orally active inhibitor of ADAMTS-5.Aldumastat is used for the study of osteoarthritis of the knee.Formula:C20H24F2N4O3Purity:99.87%Color and Shape:SolidMolecular weight:406.43MK-4882
CAS:MK-4882 is an effective inhibitor of HCV NS5A.Formula:C42H50N8O7Purity:98%Color and Shape:SolidMolecular weight:778.9Sortin1
CAS:Sortin1, a chemical genetic-hit compound, specifically induces mislocalization of both soluble and membrane-associated vacuolar markers in plants and yeast.Formula:C26H19NO6Purity:98%Color and Shape:SolidMolecular weight:441.43MDK7677
CAS:MDK7677 is a selective inhibitor of cathepsin B endopeptidase and exopeptidase activities.Formula:C12H10N4O3Color and Shape:SolidMolecular weight:258.23Furaprofen
CAS:Furaprofen is an HCV inhibitor with anti-inflammatory activity that inhibits carrageenan-induced paw edema in rats.Formula:C17H14O3Purity:98.49% - 99.52%Color and Shape:SolidMolecular weight:266.29GEMSA
CAS:GEMSA is a potent inhibitor of enkephalin convertase ( K i =8.8 nM) with analgesic effect[1].Formula:C7H13N3O4SColor and Shape:SolidMolecular weight:235.26AK 275
CAS:AK 275 is a calpain inhibitor that prevents degradation of cytoskeletal and myelin proteins in spinal cord in vitro.Formula:C20H31N3O4Color and Shape:SolidMolecular weight:377.48AZD-9684
CAS:AZD-9684, a carboxypeptidase U inhibitor, is used potentially for the prevention of thrombosis.Formula:C10H14N2O2SColor and Shape:SolidMolecular weight:226.3ITX-4520
CAS:ITX-4520 novel highly potent, orally bioavailable inhibitor of hepatitis C virus (HCV) entry.Formula:C24H23F2N3OSColor and Shape:SolidMolecular weight:439.52L 722151
CAS:L 722151 is an FXIIIa inhibitor.Formula:C8H9ClN2O5S3Purity:98%Color and Shape:SolidMolecular weight:344.82Chymase-IN-1
CAS:Chymase-IN-1 is a selective, orally active inhibitor of human mast cell chymase (IC50: 29 nM).Formula:C20H15ClNO4PSPurity:99.17%Color and Shape:SolidMolecular weight:431.83Ref: TM-T10811
1mg155.00€5mg369.00€10mg525.00€25mg787.00€50mg1,054.00€100mg1,415.00€500mg2,802.00€1mL*10mM (DMSO)404.00€ADAMTS-5-IN-2
CAS:ADAMTS-5-IN-2 is a potent inhibitor of ADAMTS-5, exhibiting an IC50 of 0.71 µM, and holds potential for osteoarthritis research.Formula:C17H15N3OSColor and Shape:SolidMolecular weight:309.39Safironil
CAS:Safironil, a novel antifibrotic, competitively inhibits collagen synthesis and modulates fibrosis, impacting type I/III collagen levels.Formula:C15H23N3O4Purity:99.83%Color and Shape:SolidMolecular weight:309.36Ref: TM-T67961
1mg64.00€5mg136.00€10mg192.00€25mg334.00€50mg477.00€100mg662.00€200mg892.00€1mL*10mM (DMSO)137.00€RWJ-58643 HCl
CAS:RWJ 58643 inhibits beta-tryptase & trypsin; at 100µg with budesonide 200µg, reduces symptoms & IL-5; high doses cause late eosinophilia.Formula:C20H27ClN6O4SColor and Shape:SolidMolecular weight:482.984CA 074
CAS:CA 074 is a potent inhibitor of cathepsin B with a Ki value of 2 to 5 nM.CA 074 inhibits ischemic hippocampal neuronal death in primates and attenuates
Formula:C18H29N3O6Purity:97.80%Color and Shape:SolidMolecular weight:383.44XMU-MP-2
CAS:XMU-MP-2 is a potent and selective protease inhibitor with anticancer activity that inhibits the growth of oncogenic BRK-driven tumors in a mouse xenograft
Formula:C32H33F3N8O2Purity:99.29%Color and Shape:SolidMolecular weight:618.652',5-Difluoro-2'-deoxycytidine
CAS:2',5-Difluoro-2'-deoxycytidine has potent anti-HCV activity and toxicity to rRNA.Formula:C9H11F2N3O4Purity:98%Color and Shape:SolidMolecular weight:263.2EI-1
CAS:EI-1 is an inhibitor of Hepatitis C virus entry.Formula:C16H19F3N6O3Color and Shape:SolidMolecular weight:400.36
