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Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

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Found 985 products of "Proteases/Proteasome"

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  • Azo-Resveratrol

    CAS:
    Azo-Resveratrol is an analog of Resveratrol used as a potent tyrosinase inhibitor.
    Formula:C12H10N2O3
    Color and Shape:Solid
    Molecular weight:230.22

    Ref: TM-T70783

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • HCV-IN-34

    CAS:
    HCV-IN-35, an oral HCV blocker, has an EC50 of 0.010 μM and a CC50 of 7.5 μM, indicating strong antiviral effects.
    Formula:C31H36ClN5
    Color and Shape:Solid
    Molecular weight:514.1

    Ref: TM-T63567

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Tyrosinase-IN-7

    CAS:
    Tyrosinase-IN-7 is a small-molecule tyrosinase inhibitor (IC50 1.57 μM) that suppresses melanin activity and cell growth with low cytotoxicity.
    Formula:C15H10O5
    Purity:99%
    Color and Shape:Solid
    Molecular weight:270.24

    Ref: TM-T72786

    1mg
    60.00€
    5mg
    130.00€
    10mg
    200.00€
    25mg
    401.00€
    50mg
    645.00€
    100mg
    1,018.00€
    200mg
    1,378.00€
  • BC-05

    CAS:
    BC-05, an orally active inhibitor targeting CD13 and the proteasome, displays potent inhibition with IC50 values of 0.13 μM against human CD13 and 1.39 μM for
    Formula:C21H29BN2O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:464.27

    Ref: TM-T78847

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • RID-F

    CAS:
    RID-F is an inhibitor of the nonpeptidic proteasome.
    Formula:C38H50N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:566.82

    Ref: TM-T26082

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AL-9

    CAS:
    AL-9 is a GT-1b and GT-2a replication inhibitor.
    Formula:C23H22N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:402.45

    Ref: TM-T25020

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PMPA sodium

    CAS:
    PMPA sodium is a potent and selective glutamate carboxypeptidase 2 (GCP II/N-acetylated a-linked dipeptidase/NAALADase) inhibitor.
    Formula:C6H11Na4O7P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:318.08

    Ref: TM-T25968

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Tyrosinase-IN-11

    CAS:
    Tyrosinase-IN-11: potent inhibitor, IC50 - 50nM/64nM (L-tyrosinase/L-dopa), antioxidant, low toxicity, for hyperpigmentation study.
    Formula:C15H14O5
    Color and Shape:Solid
    Molecular weight:274.27

    Ref: TM-T72703

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Kallikrein 5-IN-2

    CAS:
    Kallikrein 5-IN-2 inhibits KLK5 (pIC50=7.1); may normalize skin shedding, lessen inflammation & itching.
    Formula:C23H22N6O
    Color and Shape:Solid
    Molecular weight:398.46

    Ref: TM-T72624

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • VA4 TG2 inhibitor

    CAS:
    VA4 is a novel irreversible TG2 transamidase site-specific inhibitor.
    Formula:C33H41N5O6S
    Color and Shape:Solid
    Molecular weight:635.77

    Ref: TM-T69933

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AZD5248

    CAS:
    AZD-5248 is a potent, selective, first generation, oral inhibitor of dipeptidyl peptidase 1 (DPP1).
    Formula:C22H22N4O2
    Color and Shape:Solid
    Molecular weight:374.44

    Ref: TM-T71117

    1mg
    682.00€
  • BMS-363131

    CAS:
    BMS-363131 (BMS363131) is a potent and selective trypsin inhibitor with an IC50 value of <1.7 nM.
    Formula:C28H40N6O5
    Purity:97.99%
    Color and Shape:Solid
    Molecular weight:540.65

    Ref: TM-T30519

    1mg
    81.00€
  • α-Glucosidase-IN-5

    CAS:
    α-Glucosidase-IN-5 (compound 8) is isolated from a twig extract of Polyalthia cinnamomea which is a potent α-glucosidase inhibitor with an IC50 of 57.9 µM.
    Formula:C15H13NO3
    Color and Shape:Solid
    Molecular weight:255.27

    Ref: TM-T60389

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SAP2-IN-1

    CAS:
    SAP2-IN-1 inhibits secreted aspartate protease 2 (IC50: 0.92 μM), doesn't work in vitro, and helps research infections.
    Formula:C34H29NO7
    Color and Shape:Solid
    Molecular weight:563.6

    Ref: TM-T63986

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Glutaminase-IN-4

    CAS:
    Glutaminase-IN-4 (compound 2a) is a glutaminase (GLS) inhibitor (IC50: 2.3 μM).
    Formula:C23H22N6O2S2
    Color and Shape:Solid
    Molecular weight:478.59

    Ref: TM-T63137

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • L 658758

    CAS:
    L 658758 is an inhibitor of serine proteinase.
    Formula:C16H20N2O9S
    Color and Shape:Solid
    Molecular weight:416.4

    Ref: TM-T24311

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • BC-23

    CAS:
    BC-23 (NSC 45382) is a proteasome inhibitor with antitumor and antimicrobial activity for the study of leukemia and small cell lung cancer.
    Formula:C21H14ClN3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:439.87

    Ref: TM-T26754

    1mg
    99.00€
    5mg
    187.00€
    10mg
    303.00€
    25mg
    547.00€
    50mg
    817.00€
    100mg
    1,225.00€
  • AGLME

    CAS:
    AGLME is used in a direct enzymatic assay for activated Hageman factor measuring the ability of Hageman factor to hydrolyze the cpd.
    Formula:C11H21N3O4
    Color and Shape:Solid
    Molecular weight:259.3

    Ref: TM-T25007

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BI-L 45XX

    CAS:
    BI-L 45XX, an anti-inflammatory benzimidazole derivative, has inhibitory effects on neutrophil function.
    Formula:C10H9F3N2O2S
    Color and Shape:Solid
    Molecular weight:278.25

    Ref: TM-T26813

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Tyrphostin 47

    CAS:
    Tyrphostin 47 inhibits the protein-tyrosine kinase activity of EGF-R.
    Formula:C10H8N2O2S
    Color and Shape:Solid
    Molecular weight:220.25

    Ref: TM-T24908

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Levovirin valinate HCl

    CAS:
    Levovirin valinate HCl is a valine ester prodrug of levovirin as a new investigational drug for the therapy of the hepatitis C virus.
    Formula:C13H22ClN5O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:379.8

    Ref: TM-T25702L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ici 186756

    CAS:
    Ici 186756 is a novel, effective, and selective inhibitor of human neutrophil elastase.
    Formula:C33H49N5O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:659.77

    Ref: TM-T25518

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Chymase-IN-2

    CAS:
    Chymase-IN-2 is a modulator of chymase.
    Formula:C19H15ClF2NO3PS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:441.82

    Ref: TM-T12450

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A-953227

    CAS:
    A-953227: Selective calpain inhibitor with improved cathepsin selectivity, strong microsomal stability, and cellular efficacy.
    Formula:C25H20FN5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:457.46

    Ref: TM-T23598

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Duazomycin

    CAS:
    Duazomycin, an antitumor substance and glutamine antagonist, is used as a chemotherapeutic agent.
    Formula:C8H11N3O4
    Color and Shape:Solid
    Molecular weight:213.19

    Ref: TM-T27217

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Moxicoumone

    CAS:
    Moxicoumone is an anticoagulant agent.
    Formula:C22H30N2O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:418.48

    Ref: TM-T25835

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Tyrphostin A46

    CAS:
    Tyrphostin A46 is an antagonist of the epidermal growth factor-urogastrone receptor.
    Formula:C10H8N2O3
    Purity:98%
    Color and Shape:Off-White Solid
    Molecular weight:204.18

    Ref: TM-T24910

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MDK0734

    CAS:
    MDK0734 is a selective inhibitor of cathepsin B endopeptidase and exopeptidase activities.
    Formula:C15H17N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:271.31

    Ref: TM-T27989

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • FQ

    CAS:
    FQ is a novel reversible inhibitor of mixed-type tyrosinase.
    Formula:C14H9FN2O
    Color and Shape:Solid
    Molecular weight:240.23

    Ref: TM-T27358

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ADAMTS-5 Inhibitor

    CAS:
    ADAMTS-5 Inhibitor is an inhibitor of ADAMTS-5 with an IC50 of 1.1 µM and can be used in studies about cartilage destruction in arthritis.
    Formula:C16H11ClF3N3OS3
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:449.92

    Ref: TM-T14124

    1mg
    46.00€
    5mg
    93.00€
    10mg
    122.00€
    25mg
    193.00€
    50mg
    289.00€
    100mg
    414.00€
    200mg
    580.00€
    1mL*10mM (DMSO)
    96.00€
  • TNIK-IN-1

    CAS:
    TNIK-IN-1 is an inhibitor of Traf2- and Nck-interacting kinase (TNIK).
    Formula:C19H17N5O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:395.43

    Ref: TM-T26282

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Diethyl pyimDC

    CAS:
    Diethyl pyimDC is an inhibitor of human collagen prolyl 4-hydroxylase 1 (CP4H1).
    Formula:C14H15N3O4
    Color and Shape:Solid
    Molecular weight:289.29

    Ref: TM-T27170

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Aldumastat

    CAS:
    Aldumastat (GLPG1972) is a highly potent, specific and orally active inhibitor of ADAMTS-5.Aldumastat is used for the study of osteoarthritis of the knee.
    Formula:C20H24F2N4O3
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:406.43

    Ref: TM-T35859

    1mg
    269.00€
  • MK-4882

    CAS:
    MK-4882 is an effective inhibitor of HCV NS5A.
    Formula:C42H50N8O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:778.9

    Ref: TM-T24475

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Sortin1

    CAS:
    Sortin1, a chemical genetic-hit compound, specifically induces mislocalization of both soluble and membrane-associated vacuolar markers in plants and yeast.
    Formula:C26H19NO6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:441.43

    Ref: TM-T16912

    25mg
    2,570.00€
    50mg
    3,352.00€
    100mg
    5,089.00€
  • MDK7677

    CAS:
    MDK7677 is a selective inhibitor of cathepsin B endopeptidase and exopeptidase activities.
    Formula:C12H10N4O3
    Color and Shape:Solid
    Molecular weight:258.23

    Ref: TM-T28003

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Furaprofen

    CAS:
    Furaprofen is an HCV inhibitor with anti-inflammatory activity that inhibits carrageenan-induced paw edema in rats.
    Formula:C17H14O3
    Purity:98.49% - 99.52%
    Color and Shape:Solid
    Molecular weight:266.29

    Ref: TM-T16715

    1mg
    260.00€
    5mg
    620.00€
    10mg
    888.00€
    25mg
    1,369.00€
    50mg
    1,783.00€
  • GEMSA

    CAS:
    GEMSA is a potent inhibitor of enkephalin convertase ( K i =8.8 nM) with analgesic effect[1].
    Formula:C7H13N3O4S
    Color and Shape:Solid
    Molecular weight:235.26

    Ref: TM-T21843

    5mg
    597.00€
  • AK 275

    CAS:
    AK 275 is a calpain inhibitor that prevents degradation of cytoskeletal and myelin proteins in spinal cord in vitro.
    Formula:C20H31N3O4
    Color and Shape:Solid
    Molecular weight:377.48

    Ref: TM-T25009

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AZD-9684

    CAS:
    AZD-9684, a carboxypeptidase U inhibitor, is used potentially for the prevention of thrombosis.
    Formula:C10H14N2O2S
    Color and Shape:Solid
    Molecular weight:226.3

    Ref: TM-T26725

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • ITX-4520

    CAS:
    ITX-4520 novel highly potent, orally bioavailable inhibitor of hepatitis C virus (HCV) entry.
    Formula:C24H23F2N3OS
    Color and Shape:Solid
    Molecular weight:439.52

    Ref: TM-T27641

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • L 722151

    CAS:
    L 722151 is an FXIIIa inhibitor.
    Formula:C8H9ClN2O5S3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:344.82

    Ref: TM-T24349

    25mg
    1,783.00€
  • Chymase-IN-1

    CAS:
    Chymase-IN-1 is a selective, orally active inhibitor of human mast cell chymase (IC50: 29 nM).
    Formula:C20H15ClNO4PS
    Purity:99.17%
    Color and Shape:Solid
    Molecular weight:431.83

    Ref: TM-T10811

    1mg
    155.00€
    5mg
    369.00€
    10mg
    525.00€
    25mg
    787.00€
    50mg
    1,054.00€
    100mg
    1,415.00€
    500mg
    2,802.00€
    1mL*10mM (DMSO)
    404.00€
  • ADAMTS-5-IN-2

    CAS:
    ADAMTS-5-IN-2 is a potent inhibitor of ADAMTS-5, exhibiting an IC50 of 0.71 µM, and holds potential for osteoarthritis research.
    Formula:C17H15N3OS
    Color and Shape:Solid
    Molecular weight:309.39

    Ref: TM-T72868

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Safironil

    CAS:
    Safironil, a novel antifibrotic, competitively inhibits collagen synthesis and modulates fibrosis, impacting type I/III collagen levels.
    Formula:C15H23N3O4
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:309.36

    Ref: TM-T67961

    1mg
    64.00€
    5mg
    136.00€
    10mg
    192.00€
    25mg
    334.00€
    50mg
    477.00€
    100mg
    662.00€
    200mg
    892.00€
    1mL*10mM (DMSO)
    137.00€
  • RWJ-58643 HCl

    CAS:
    RWJ 58643 inhibits beta-tryptase & trypsin; at 100µg with budesonide 200µg, reduces symptoms & IL-5; high doses cause late eosinophilia.
    Formula:C20H27ClN6O4S
    Color and Shape:Solid
    Molecular weight:482.984

    Ref: TM-T68474

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CA 074

    CAS:

    CA 074 is a potent inhibitor of cathepsin B with a Ki value of 2 to 5 nM.CA 074 inhibits ischemic hippocampal neuronal death in primates and attenuates

    Formula:C18H29N3O6
    Purity:97.80%
    Color and Shape:Solid
    Molecular weight:383.44

    Ref: TM-T21509

    1mg
    80.00€
    5mg
    210.00€
    10mg
    329.00€
    25mg
    660.00€
    50mg
    917.00€
    100mg
    1,216.00€
  • XMU-MP-2

    CAS:

    XMU-MP-2 is a potent and selective protease inhibitor with anticancer activity that inhibits the growth of oncogenic BRK-driven tumors in a mouse xenograft

    Formula:C32H33F3N8O2
    Purity:99.29%
    Color and Shape:Solid
    Molecular weight:618.65

    Ref: TM-T69980

    1mg
    185.00€
    5mg
    459.00€
    10mg
    657.00€
    25mg
    1,026.00€
    50mg
    1,415.00€
    100mg
    1,872.00€
    500mg
    3,734.00€
  • 2',5-Difluoro-2'-deoxycytidine

    CAS:
    2',5-Difluoro-2'-deoxycytidine has potent anti-HCV activity and toxicity to rRNA.
    Formula:C9H11F2N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:263.2

    Ref: TM-T10067

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • EI-1

    CAS:
    EI-1 is an inhibitor of Hepatitis C virus entry.
    Formula:C16H19F3N6O3
    Color and Shape:Solid
    Molecular weight:400.36

    Ref: TM-T71871

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€