Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
Found 385 products of "Histamine Receptor"
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Triprolidine hydrochloride
CAS:Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.Formula:C19H23ClN2Color and Shape:SolidMolecular weight:314.852Triprolidine
CAS:Triprolidine: oral H1 receptor blocker with motor/sensory spinal effects, for allergy research.Formula:C19H22N2Color and Shape:SolidMolecular weight:278.39GSK189254A
CAS:GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).Formula:C21H25N3O2Purity:98.71% - 99.858%Color and Shape:SolidMolecular weight:351.44Ref: TM-TQ0066
1mg50.00€5mg84.00€10mg114.00€25mg205.00€50mg333.00€100mg477.00€200mg690.00€1mL*10mM (DMSO)64.00€Osthole
CAS:Osthole (Osthol), a potential inhibitor of histamine H1 receptor, has been shown to stimulate osteoblast proliferation and differentiation.Formula:C15H16O3Purity:99.93% - 99.96%Color and Shape:Fine White PowderMolecular weight:244.29Betazole
CAS:Betazole, an oral H2 receptor agonist, stimulates gastric acid and raises bile duct pressure, used for gastric secretory testing.Formula:C5H9N3Color and Shape:SolidMolecular weight:111.15Betazole dihydrochloride
CAS:Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor.
Formula:C5H11Cl2N3Purity:99.12%Color and Shape:SolidMolecular weight:184.067Mequitazine
CAS:Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.Formula:C20H22N2SPurity:99.98%Color and Shape:SolidMolecular weight:322.47Ciproxifan maleate
CAS:Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinityFormula:C20H22N2O6Purity:99.39%Color and Shape:SolidMolecular weight:386.4Ref: TM-T2004
1mg40.00€2mg52.00€5mg75.00€10mg101.00€25mg205.00€50mg380.00€100mg565.00€1mL*10mM (DMSO)82.00€Epinastine hydrochloride
CAS:Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.Formula:C16H15N3·HClPurity:99.26% - 99.62%Color and Shape:White SolidMolecular weight:285.77Mecamylamine hydrochloride
CAS:Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.Formula:C11H22ClNPurity:99.76% - >99.99%Color and Shape:White SolidMolecular weight:203.75JNJ-7777120
CAS:JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist, exhibits >1000-fold selectivity over the other histamin receptors.Formula:C14H16ClN3OPurity:99.83% - 99.96%Color and Shape:SolidMolecular weight:277.75Chlorcyclizine
CAS:CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.Formula:C18H21ClN2Purity:98.75%Color and Shape:SolidMolecular weight:300.83Chlorprothixene
CAS:Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.Formula:C18H18ClNSPurity:98.77% - 99.756%Color and Shape:Pale Yellow Crystals SolidMolecular weight:315.86VUF10460
CAS:VUF10460 is a non-imidazole histamine H4 receptor agonist.Formula:C15H19N5Purity:99.44% - 99.57%Color and Shape:SolidMolecular weight:269.34Dimaprit dihydrochloride
CAS:Dimaprit dihydrochloride: selective H2 agonist, inhibits nNOS (IC50: 49 μM), boosts gastric acid.Formula:C6H15N3S·2HClPurity:99.79%Color and Shape:SolidMolecular weight:234.19Talastine HCl
CAS:Talastine is an antihistamine drug.Formula:C19H22ClN3OPurity:98%Color and Shape:SolidMolecular weight:343.86C-Type Natriuretic Peptide (CNP) (1-22), human
CAS:C-Type Natriuretic Peptide (CNP) (1-22), human is the 1-22 fragment of C-Type Natriuretic Peptide.Formula:C93H157N27O28S3Purity:>99.99%Color and Shape:SolidMolecular weight:2197.6Ref: TM-TP1187
1mg119.00€5mg414.00€10mg658.00€25mg945.00€50mg1,264.00€100mg1,700.00€200mg2,270.00€500µg88.00€Tiaramide hydrochloride
CAS:Tiaramide hydrochloride (FK-1160) is an anti-inflammatory that blocks mast cell mediators and relaxes smooth muscles.Formula:C15H19Cl2N3O3SPurity:98.48%Color and Shape:SolidMolecular weight:392.3Ref: TM-T28972
1mg66.00€5mg130.00€10mg177.00€25mg299.00€50mg447.00€100mg623.00€200mg882.00€1mL*10mM (DMSO)137.00€Tribenoside
CAS:Tribenoside (BG-356) is a vasoprotectant with mild anti-inflammatory, analgesic, and wound healing properties.Formula:C29H34O6Purity:≥98%Color and Shape:LiquidMolecular weight:478.58cicloprofen
CAS:cicloprofen is Cell division cycle 7-related protein kinase (human) inhibitor.Formula:C16H14O2Purity:98.15%Color and Shape:SolidMolecular weight:238.2812Ref: TM-T8586
1mg62.00€5mg123.00€10mg180.00€25mg298.00€50mg419.00€100mg567.00€200mg752.00€1mL*10mM (DMSO)111.00€Acitazanolast
CAS:Acitazanolast (WP-871) is an anti-allergic drug candidate.
Formula:C9H7N5O3Purity:98.25%Color and Shape:SolidMolecular weight:233.182-Pyridylethylamine dihydrochloride
CAS:2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.Formula:C7H12Cl2N2Purity:99.42%Color and Shape:SolidMolecular weight:195.09Decloxizine
CAS:Decloxizine is a H1 receptor antagonistFormula:C21H28N2O2Purity:99.53%Color and Shape:White Or Similar To White PowderMolecular weight:340.46Zotepine
CAS:Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,Formula:C18H18ClNOSPurity:99.78%Color and Shape:SolidMolecular weight:331.86Pemirolast
CAS:Pemirolast: oral antiallergic, reduces paclitaxel reactions, inhibits neuropeptides, for asthma and conjunctivitis study.Formula:C10H8N6OColor and Shape:SolidMolecular weight:228.21Clemizole hydrochloride
CAS:Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.Formula:C19H21Cl2N3Purity:>99.99%Color and Shape:SolidMolecular weight:362.3Antazoline
CAS:Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias.Formula:C17H19N3Purity:≥95%Color and Shape:White Crystalline Powder SolidMolecular weight:265.35Psoralenoside
CAS:Psoralenoside: a compound from Psoralea fruit; has estrogenic, osteoblastic, antitumor, and antibacterial properties.Formula:C17H18O9Purity:99.03% - 99.49%Color and Shape:SolidMolecular weight:366.32Ref: TM-TN1008
1mg96.00€2mg139.00€5mg227.00€10mg364.00€25mg600.00€50mg845.00€100mg1,121.00€1mL*10mM (DMSO)235.00€Betahistine EP Impurity C
CAS:Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.Formula:C15H19N3Purity:≥95%Color and Shape:SolidMolecular weight:241.33Dioxopromethazine hydrochloride
CAS:Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.Formula:C17H20N2O2S·HClPurity:99.58%Color and Shape:SolidMolecular weight:352.88Betahistine
CAS:Betahistine treats vertigo and balance issues in Ménière's disease; it's a histamine analog and H1 receptor agonist.Formula:C8H12N2Purity:99.87% - 99.87%Color and Shape:Yellowish Liquid Liquid LiquidMolecular weight:136.19Buclizine dihydrochloride
CAS:Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic andFormula:C28H33ClN2·2HClPurity:98.05%Color and Shape:Off-White PowderMolecular weight:505.95S 38093
CAS:S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).Formula:C17H24N2O2Purity:99.95%Color and Shape:SolidMolecular weight:288.38Ref: TM-T4099
2mg35.00€5mg50.00€10mg75.00€25mg124.00€50mg198.00€100mg316.00€200mg442.00€1mL*10mM (DMSO)50.00€Dioxopromethazine
CAS:Dioxopromethazine (Dioxoprothazine) is a drug for the treatment of a cough and expectoration. It also can be used in local anesthesia.Formula:C17H20N2O2SPurity:98%Color and Shape:SolidMolecular weight:316.42Carcinine ditrifluoroacetate Acetate
Carcinine ditrifluoroacetate Acetate (β-Alanylhistamine dihydrochloride) is an H3 receptor antagonist.Formula:C14H20F6N4O7Purity:98.18%Color and Shape:SolidMolecular weight:470.32Decloxizine dihydrochloride
CAS:Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.Formula:C21H28N2O2·2ClHPurity:99.73%Color and Shape:SolidMolecular weight:413.39Histamine Phosphate
CAS:Histamine Phosphate (Histamine acid phosphate) acts directly on the blood vessels to dilate arteries and capillaries mediated by both H 1- and H 2-receptors.Formula:C5H9N·2H3O4PPurity:>99.99%Color and Shape:White Crystal PowderMolecular weight:307.14Alginic acid
CAS:Alginic acid, a polysaccharide from brown seaweed, has anti-anaphylactic and anti-inflammatory properties and is used in food industry.Formula:C14H22O13Purity:≥98%Color and Shape:SolidMolecular weight:398.317Betahistine dihydrochloride
CAS:Betahistine dihydrochloride (Betahistine 2HCl) is a histamine analog and H1 receptor agonist that serves as a vasodilator.Formula:C8H14Cl2N2Purity:99.22% - 99.88%Color and Shape:White To Light Yellow Crystalline PowderMolecular weight:209.12Thonzylamine
CAS:Thonzylamine is an antihistamine/anticholinergic, combined with Clofedanol or Phenylephrine for cold, hay fever, or allergy relief.Formula:C16H22N4OPurity:99.45%Color and Shape:SolidMolecular weight:286.37Alimemazine hemitartrate
CAS:Alimemazine hemitartrate (Trimeprazine hemitartrate) is aphenothiazine derivative that is used as an antipruritic.Formula:C18H22N2SC4H6O6Purity:98.16% - 99.69%Color and Shape:SolidMolecular weight:448.53JNJ-5207852
CAS:JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.Formula:C20H32N2OPurity:97.19%Color and Shape:SolidMolecular weight:316.48LML134
CAS:LML134 (LML-134) is an inverse agonist of Histamine 3 receptor (H3R)(hH3R cAMP and hH3R bdg with Kis of 0.3 nM and 12 nM).Formula:C19H29N5O3Purity:99.36%Color and Shape:SolidMolecular weight:375.47Ref: TM-T8514
1mg34.00€5mg78.00€10mg112.00€25mg203.00€50mg299.00€100mg447.00€200mg600.00€1mL*10mM (DMSO)86.00€S 38093 HCl
CAS:S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.Formula:C17H25ClN2O2Purity:97.91%Color and Shape:SolidMolecular weight:324.85Ref: TM-T4087
1mg37.00€5mg71.00€10mg92.00€25mg164.00€50mg225.00€100mg323.00€200mg437.00€1mL*10mM (DMSO)71.00€Hydroxyzine dihydrochloride
CAS:Hydroxyzine dihydrochloride treats allergies, pruritus, anxiety; causes drowsiness; also an antiemetic and sedative.Formula:C21H27ClN2O2·2HClPurity:99.46% - 99.79%Color and Shape:Oil PowderMolecular weight:447.83OXOMEMAZINE
CAS:Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.Formula:C18H22N2O2SPurity:99.58%Color and Shape:SolidMolecular weight:330.44Ranitidine
CAS:Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors).Formula:C13H22N4O3SPurity:99.52%Color and Shape:Solid SolidMolecular weight:314.40Bepotastine
CAS:Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.Formula:C21H25ClN2O3Purity:99.75%Color and Shape:SolidMolecular weight:388.89Ref: TM-T7893
2mg34.00€5mg50.00€10mg78.00€25mg141.00€50mg205.00€100mg313.00€200mg464.00€1mL*10mM (DMSO)56.00€Latrepirdine dihydrochloride
CAS:Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.Formula:C21H25N3·2HClPurity:98.45%Color and Shape:SolidMolecular weight:392.37Levocetirizine Dihydrochloride
CAS:Levocetirizine Dihydrochloride is a third-gen antihistamine targeting H1-receptors, treating allergies and urticaria.Formula:C21H27Cl3N2O3Purity:99.89%Color and Shape:White Or Off-White Crystalline PowderMolecular weight:461.81
