CymitQuimica logo
Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

Show 16 more subcategories

Found 66618 products of "Inhibitors"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • Samuraciclib

    CAS:
    <p>Samuraciclib (CT7001) is an oral CDK7 inhibitor with 41 nM IC50, notable for its high selectivity and potency against breast cancer cells.</p>
    Formula:C22H30N6O
    Color and Shape:Solid
    Molecular weight:394.51
  • CH-38083

    CAS:
    <p>CH-38083 is a selective and effective alpha-2 adrenoceptors antagonist.</p>
    Formula:C18H24ClNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:337.84
  • SCH-1473759

    CAS:
    SCH-1473759 is an inhibitor of the aurora (IC50s: 4 and 13 nM for Aurora A and B, respectively).
    Formula:C20H26N8OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:426.54
  • Menin-MLL inhibitor 4

    CAS:
    Menin-MLL inhibitor 4 has antitumor activity.Menin-MLL inhibitor 4 is an inhibitor of Menin- MLL (mixed-lineage leukemia protein) interaction .
    Formula:C32H38FN7O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:587.69
  • PRMT5-IN-1 hydrochloride


    <p>PRMT5 IN-1 hydrochloride is a potent PRMT5 inhibitor (IC50: 11 nM), forms covalent adduct with C449, and converts to an aldehyde in vivo.</p>
    Formula:C19H20Cl2N4O5
    Color and Shape:Solid
    Molecular weight:455.29
  • Udifitimod

    CAS:
    <p>Udifitimod (BMS-986166) is a potent, selective, and orally active modulator of the S1P1R receptor, showing potential for research in autoimmune diseases.</p>
    Formula:C25H33NO2
    Color and Shape:Solid
    Molecular weight:379.54
  • AZD 2066 hydrate


    <p>AZD 2066 hydrate is a selective, orally active, and brain-penetrant antagonist of mGluR5. It exhibits antinociceptive effects [1].</p>
    Formula:C19H18ClN5O3
    Color and Shape:Solid
    Molecular weight:386.33
  • CCR7 Ligand 1

    CAS:
    <p>CCR7-Cmp2105 is a thiadiazole-dioxide allosteric antagonist for CCR7 with a Kd of 3 nM and IC50 of 7.3 μM against arrestin binding.</p>
    Formula:C22H29N5O5S
    Color and Shape:Solid
    Molecular weight:475.56
  • Fosmanogepix

    CAS:
    Fosmanogepix (APX001) is a broad-spectrum oral antifungal that targets Gwt1 enzyme, transforming into active APX001A in the body.
    Formula:C22H21N4O6P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:468.40
  • FK-3657

    CAS:
    <p>FK-3657 is a non-peptide antagonist of bradykinin (BK)-B2 receptor.</p>
    Formula:C30H27Cl2N5O4
    Color and Shape:Solid
    Molecular weight:592.47
  • G-9791

    CAS:
    <p>G-9791 is an effective and selective inhibitor of group-I PAK.</p>
    Formula:C26H26ClFN6O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:508.98
  • Wikstrol A

    CAS:
    <p>Wikstrol A: antifungal, anti-mitotic, anti-HIV agent with various IC50/MDC values (67.8-131 µM) and deforms P. oryzae mycelia.</p>
    Formula:C30H22O10
    Color and Shape:Solid
    Molecular weight:542.49
  • Lapaquistat

    CAS:
    <p>Lapaquistat: active TAK-475 metabolite; reduces cholesterol synthesis and statin myotoxicity.</p>
    Formula:C31H39ClN2O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:603.1
  • CDK2-IN-9


    <p>CDK2-IN-9: potent CDK2 inhibitor (IC50: 0.63 μM), anti-proliferative, arrests S/G2M cell cycle, induces apoptosis, promising for melanoma study.</p>
    Formula:C21H16ClN3O4S
    Color and Shape:Solid
    Molecular weight:441.89
  • LP 12 hydrochloride hydrate


    <p>LP 12 hydrochloride hydrate: potent, selective 5-HT7 agonist (Ki: 0.13 nM); less affinity for D2, 5-HT1A/2A receptors.</p>
    Formula:C32H39N3O·HCl·xH2O
    Color and Shape:Solid
  • AS-1940477 hydrobromide

    CAS:
    <p>AS-1940477 hydrobromide is a p38 mitogen-activated protein kinase (MAPK) inhibitor.</p>
    Formula:C24H23BrFN5O2
    Color and Shape:Solid
    Molecular weight:512.38
  • Carbonic anhydrase inhibitor 10


    <p>CA inhibitor 10 targets MCF-7 cells, IC50: 11.9 μM; potent h CA IX inhibitor, Ki: 6.2 nM. Anti-cancer research.</p>
    Formula:C14H17N5O3S
    Color and Shape:Solid
    Molecular weight:335.38
  • FTO-IN-5

    CAS:
    <p>FTO-IN-5 is a potent, selective inhibitor targeting the fat mass obesity-associated protein (FTO).</p>
    Formula:C23H18Cl2N6O6
    Color and Shape:Solid
    Molecular weight:545.33
  • NK-1 Antagonist 1

    CAS:
    <p>NK-1 Antagonist 1 is a NK-1 receptor antagonist.</p>
    Formula:C25H23F6N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:539.47
  • PPI-2458

    CAS:
    <p>PPI-2458, a fumagillin derivative, irreversibly blocks MetAP2, hindering abnormal cell growth and angiogenesis with improved toxicity.</p>
    Formula:C22H36N2O6
    Color and Shape:Solid
    Molecular weight:424.53
  • UK-432097

    CAS:
    <p>UK 432097 is an adenosine A2A agonist.</p>
    Formula:C40H47N11O6
    Color and Shape:Solid
    Molecular weight:777.87
  • ATUX-1215

    CAS:
    <p>ATUX-1215, a protein phosphatase 2A (PP2A) activator, diminishes the phosphorylation of ERK, p38, JNK, and Akt, as well as decreases the secretion of IL-12p70,</p>
    Formula:C27H24F5NO4S
    Color and Shape:Solid
    Molecular weight:553.54
  • Galectin-8-IN-1


    <p>Galectin-8-IN-1 selectively binds galectin-8N with 48 μM affinity, 15x more than galectin-3.</p>
    Formula:C16H18N2O6
    Color and Shape:Solid
    Molecular weight:334.32
  • FT3967385


    <p>FT3967385: New USP30 inhibitor boosts mitochondrial ubiquitylation via PINK1-PARKIN.</p>
    Formula:C21H19N5O2
    Color and Shape:Solid
    Molecular weight:373.41
  • Complex III-IN-2


    <p>Complex III-IN-2 inhibits complex III, with antifungal EC50: 29.31 mg/L vs R. solani, 29.98 mg/L vs S. sclerotiorum.</p>
    Formula:C15H21ClN2O2S
    Color and Shape:Solid
    Molecular weight:328.86
  • Onalespib lactate

    CAS:
    <p>Onalespib lactate is a second-generation, potent and selective HSP90 Inhibitor with antitumor activity.</p>
    Formula:C27H37N3O6
    Color and Shape:Solid
    Molecular weight:499.6
  • CDK4-IN-1

    CAS:
    <p>CDK4 inhibitor is a novel and specific CDK4/Cyclin D1 inhibitor with an IC50 of 10 nM; 1500 and 500 fold than CDK1/Cyclin B (IC50&gt;15 uM) and CDK2/Cyclin A (IC50</p>
    Formula:C22H29ClN8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:440.97
  • 5-HT1A antagonist 1


    <p>Compound 6f is a potent, selective 5-HT1A receptor blocker (Ki: 35 nM), useful in CNS disorder research.</p>
    Formula:C23H29ClN6O2
    Color and Shape:Solid
    Molecular weight:456.97
  • CTX-712

    CAS:
    <p>CTX-712 is a potent inhibitor of cdc2-like kinase ( CLK ). CTX-712 inhibits inhibits cancer survival and cancer cell growth.</p>
    Formula:C19H17FN8O2
    Color and Shape:Solid
    Molecular weight:408.39
  • NMDA receptor antagonist-3


    <p>NMDA antagonist-3: recovery rate 40% at 100 μM, low toxicity in SH-SY5Y, human stem cells.</p>
    Formula:C13H19N3O6
    Color and Shape:Solid
    Molecular weight:313.31
  • EGFR-IN-34


    <p>EGFR-IN-34 is a low-toxicity, acrylamide derivative antitumor agent that is a potent inhibitor of EGFR.</p>
    Formula:C26H27ClN6O2
    Color and Shape:Solid
    Molecular weight:490.98
  • Antiangiogenic agent 3


    <p>Antiangiogenic agent 3 blocks HUVEC cell migration, chemotaxis, and lowers Src, cdc42, MAPK gene expression.</p>
    Formula:C19H20O7
    Color and Shape:Solid
    Molecular weight:360.36
  • Diospyrin

    CAS:
    <p>Diospyrin is a plant product that has significant inhibitory effect on the growth of Leishmania donovani promastigotes.</p>
    Formula:C22H14O6
    Color and Shape:Solid
    Molecular weight:374.34
  • RS 12254

    CAS:
    <p>RS 12254 is a dopamine agonist and antihypertensive agent.</p>
    Formula:C28H40N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:468.63
  • HPK1-IN-3


    <p>HPK1-IN-3: Selective HPK1 inhibitor, ATP-competitive, IC50=0.25nM; boosts IL-2 in PBMCs, EC50=108nM.</p>
    Formula:C23H22F4N6O2
    Color and Shape:Solid
    Molecular weight:490.45
  • Dyrk1A-IN-2


    <p>Dyrk1A-IN-2 is a DYRK1A inhibitor (EC50: 37 nM). dyrk1A-IN-2 exhibits efficient promotion of human β-cell replication, as well as low cytotoxicity.</p>
    Formula:C27H32N6O4
    Color and Shape:Solid
    Molecular weight:504.58
  • ATR-IN-12


    <p>ATR-IN-12, a potent ATR kinase inhibitor with IC50 of 0.007 μM, shows promise for drug development.</p>
    Formula:C22H27N5O3S
    Color and Shape:Solid
    Molecular weight:441.55
  • Xylarianaphthol-1

    CAS:
    <p>Xylarianaphthol-1 is an activator of p21 promoter in a p53-independent manner.</p>
    Formula:C16H20BrFN2O2
    Color and Shape:Solid
    Molecular weight:371.24
  • γ-secretase modulator 5


    <p>Compound 22d is a GSM that crosses the blood-brain barrier, inhibits Aβ42 production (IC50: 60 nM), and may help study Alzheimer's.</p>
    Color and Shape:Solid
  • GSK 932121

    CAS:
    <p>GSK 932121: potent antimalarial, targets P. falciparum by inhibiting cytochrome bc1 in the electron transport chain.</p>
    Formula:C20H15ClF3NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:425.79
  • Piceid 6″-O-azelaic acid ester


    <p>Piceid 6″-O-azelaic acid ester exhibited strong intracellular tyrosinase inhibition and decolorization activity.</p>
    Formula:C24H36O10
    Color and Shape:Solid
    Molecular weight:484.54
  • BAY-3153

    CAS:
    <p>BAY-3153 is a selective CCR1 ( C-C motif chemokine receptor 1 ) antagonist (human IC 50 =3 nM ; rat IC 50 =11 nM ; mice IC 50 =81 nM) .</p>
    Formula:C25H29Cl2N3O4
    Color and Shape:Solid
    Molecular weight:506.42
  • Rezatapopt

    CAS:
    <p>Rezatapopt (PC14586) is a p53 reactivator with antitumor activity for the study of locally advanced or metastatic solid tumors.</p>
    Formula:C28H31F4N5O2
    Purity:98.12%
    Color and Shape:Solid
    Molecular weight:545.57
  • Ganoderic acid R

    CAS:
    <p>Ganoderic acid R: potent anticancer, induces apoptosis, cytotoxic to MDR and sensitive tumor cells.</p>
    Formula:C34H50O6
    Color and Shape:Solid
    Molecular weight:554.76
  • MDK6465

    CAS:
    <p>MDK6465 (PCSK9-IN-8b), CAS#1900686-46-5, is a liver-targeted PCSK9 synthesis inhibitor.</p>
    Formula:C27H29ClFN9O4
    Color and Shape:Solid
    Molecular weight:598.03
  • Tamitinol

    CAS:
    <p>Tamitinol is a neurotropic drug. It has been found to help symptoms of obsessive rumination in conjunction with maprotiline.</p>
    Formula:C12H20N2OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:240.37
  • Nafarelin acetate hydrate

    CAS:
    <p>Nafarelin: a GnRH agonist used to treat endometriosis, precocious puberty, and control IVF. Delivered as a nasal spray. Marketed as Synarel by Pfizer.</p>
    Formula:C66H83N17O13·xC2H4O2·xH2O
    Color and Shape:Solid
    Molecular weight:1400.563
  • Heparastatin

    CAS:
    <p>Heparastatin is an inhibitor of heparanase.</p>
    Formula:C8H11F3N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:272.18
  • PSMA-1007

    CAS:
    <p>PSMA-1007 is a novel Glu-Ureido-type prostate-specific membrane antigen (PSMA) inhibitor.</p>
    Formula:C49H55FN8O16
    Color and Shape:Solid
    Molecular weight:1030.01
  • VEGFR-2-IN-13


    <p>VEGFR-2-IN-13 (Compound 19a) is a potent VEGFR-2 inhibitor (IC50: 3.4 nM). vEGFR-2-IN-13 arrests the HepG2 cell cycle in G2/M phase and induces apoptosis.</p>
    Formula:C24H18N6O2S
    Color and Shape:Solid
    Molecular weight:454.5
  • Factor B-IN-4

    CAS:
    <p>Factor B-IN-4 is a potent inhibitor (IC50: 1 μM) of complement factor B. Factor B-IN-4 can be used to study inflammatory and immune-related diseases.</p>
    Formula:C27H32N2O4
    Color and Shape:Solid
    Molecular weight:448.55
  • Ladirubicin

    CAS:
    <p>Ladirubicin, as an anthracyclines analog is the leading compound of alkylcyclines.</p>
    Formula:C29H31NO11S
    Color and Shape:Solid
    Molecular weight:601.62
  • PARP1/BRD4-IN-2


    <p>PARP1/BRD4-IN-2, a potent inhibitor of PARP1 and BRD4, halts cell cycle, triggers apoptosis, and has antitumor effects on TNBC.</p>
    Formula:C25H20N4O4
    Color and Shape:Solid
    Molecular weight:440.45
  • hTrkA-IN-2


    <p>hTrkA-IN-2 is a selective hTrkA metamorphosis inhibitor (IC50: 3.9 nM).</p>
    Formula:C24H22F3N5O3
    Color and Shape:Solid
    Molecular weight:485.46
  • Tazide


    <p>Tazide is an antitumor agent [1].</p>
    Formula:C12H16N4O
    Color and Shape:Solid
    Molecular weight:232.28
  • CGC 11144

    CAS:
    <p>CGC 11144 is a Polyamine analogue inhibit tumor growth in vitro and in vivo.</p>
    Formula:C40H100Cl10N10
    Color and Shape:Solid
    Molecular weight:1075.82
  • Aquayamycin

    CAS:
    <p>Aquayamycin is an anthraquinone derivative and inhibitor of the enzyme tyrosine hydroxylase..</p>
    Formula:C25H26O10
    Color and Shape:Solid
    Molecular weight:486.47
  • FPR2 agonist 2


    <p>Potent FPR2 agonist, crosses blood-brain barrier, EC50: 0.13 nM; reduces inflammation and mitochondrial dysfunction, inhibits caspase-3.</p>
    Formula:C25H20F2N4O2
    Color and Shape:Solid
    Molecular weight:446.45
  • KCa2 channel modulator 2


    Compound 2q is a potent, subtype-selective K/Ca 2 modulator, effective on human K Ca 2.3 and rat K Ca 2.2a with EC50s of 0.60 μM and 0.64 μM.
    Formula:C16H15ClFN5
    Color and Shape:Solid
    Molecular weight:331.78
  • Butaprost

    CAS:
    <p>Butaprost: EP2 receptor agonist, EC50=33 nM, Ki=2.4 μM (murine), reduces fibrosis via TGF-β/Smad2.</p>
    Formula:C24H40O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:408.57
  • IRAK4-IN-19


    <p>IRAK4-IN-19, an IRAK4 inhibitor (IC50: 4.3 nM), hampers IL23 synthesis and arthritis progression.</p>
    Formula:C25H26F2N8O
    Color and Shape:Solid
    Molecular weight:492.52
  • CK2 inhibitor 3


    <p>CK2 inhibitor 3: potent CK2 blocker, IC50 of 280 nM, suppresses tumor cell growth, highly selective among 320 kinases.</p>
    Formula:C13H9BrN4O3S
    Color and Shape:Solid
    Molecular weight:381.2
  • Antibiotic MA 144M1

    CAS:
    <p>Antibiotic MA 144M1, an anthracycline, targets gram-positive bacteria and animal tumors; derived from Streptomyces fermentation or aclacinomycin A conversion.</p>
    Formula:C42H55NO15
    Color and Shape:Solid
    Molecular weight:813.88
  • DJT06001

    CAS:
    <p>DJT06001 is a selective Factor Xa inhibitor, reducing thrombus formation with low risk of bleeding.</p>
    Formula:C21H20ClN3O5S
    Color and Shape:Solid
    Molecular weight:461.92
  • SGE-516

    CAS:
    <p>SGE516: neuroactive steroid, enhances GABAA, lowers neuronal activity, protects from seizures.</p>
    Formula:C23H35N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:385.54
  • Arterolane

    CAS:
    <p>Arterolane is an antimalarial compound. For against P. falciparum Ro73 and W2, the IC50s are both 1.1 nM.</p>
    Formula:C22H36N2O4
    Color and Shape:Solid
    Molecular weight:392.53
  • 5-HT7R antagonist 1


    <p>5-HT7R antagonist 1 is a G protein-biased antagonist with Ki of 6.5 nM for 5-HT 7R.</p>
    Formula:C14H18Cl2N4
    Color and Shape:Solid
    Molecular weight:313.23
  • α5β1 integrin agonist-1

    CAS:
    <p>α5β1 integrin agonist-1 is an α5β1 integrin agonist that selectively delivers 5-FU to tumour cells and induces tumour cell death.</p>
    Formula:C24H26FN5O9
    Color and Shape:Solid
    Molecular weight:547.49
  • L-365260 hemihydrate


    <p>L-365260 hemihydrate: selective oral CCK-B/gastrin blocker, Ki=1.9/2.0 nM, competes with guinea pig receptors.</p>
    Formula:C24H24N4O3
    Color and Shape:Solid
    Molecular weight:407.47
  • HDAC6-IN-12


    <p>HDAC6-IN-12 is a potent inhibitor of HDAC6 that binds in the DNA chain, causing DNA damage and exhibiting anticancer effects that can be used in cancer research</p>
    Formula:C24H39F2N3O5
    Color and Shape:Solid
    Molecular weight:487.58
  • EGFR-IN-44


    <p>EGFR-IN-44: potent EGFR kinase inhibitor, orally active, IC50 4.11 nM, 33.57% bioavailability, induces apoptosis, for lung cancer study.</p>
    Formula:C27H29ClN6O2S
    Color and Shape:Solid
    Molecular weight:537.08
  • H 218-54

    CAS:
    <p>H 218-54 is a renin inhibitor.</p>
    Formula:C37H56N2O5S
    Color and Shape:Solid
    Molecular weight:640.92
  • Tauro-ω-muricholic acid sodium


    <p>Tauro-ω-muricholic acid sodium (TωMCA sodium) is an analogue of tauro-α-muricholic acid, a bile acid of hepatic origin.</p>
    Formula:C26H44NNaO7S
    Color and Shape:Solid
    Molecular weight:537.68
  • Adafosbuvir

    CAS:
    <p>Adafosbuvir has antiviral activity.</p>
    Formula:C22H29FN3O10P
    Color and Shape:Solid
    Molecular weight:545.457
  • VEGFR-2-IN-17


    <p>VEGFR-2-IN-17 (15a) is a potent VEGFR-2 inhibitor with an IC50 of 67.25 nM, showing significant antitumor effects.</p>
    Formula:C21H14ClN3O2
    Color and Shape:Solid
    Molecular weight:375.81
  • Carbonic anhydrase inhibitor 3


    <p>Carbonic anhydrase inhibitor 3 (compound 11g) is an inhibitor of carbonic anhydrase II that reduces the intraocular pressure in glaucomatous rabbits [1].</p>
    Formula:C15H17N3O3S
    Color and Shape:Solid
    Molecular weight:319.38
  • SB 224289

    CAS:
    <p>SB 224289: selective 5-HT1B antagonist, pKi 8.2, 60x selectivity, effective orally.</p>
    Formula:C32H32N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:520.62
  • BRD-K25923209

    CAS:
    <p>BRD-K25923209 is a novel inhibitor of BAF transcriptional repression.</p>
    Formula:C29H36N4O3
    Color and Shape:Solid
    Molecular weight:488.62
  • iMDK quarterhydrate


    <p>iMDK quarterhydrate, PI3K inhibitor, blocks MDK growth; suppresses NSCLC safely with MEK inhibitor.</p>
    Formula:C21H15FN2O3S
    Color and Shape:Solid
    Molecular weight:380.91
  • PfPKG-IN-1


    <p>PfPKG-IN-1, an imidazole-based inhibitor, targets the Plasmodium falciparum cyclic guanosine monophosphate-dependent protein kinase (PfPKG).</p>
    Formula:C24H22ClN7OS
    Color and Shape:Solid
    Molecular weight:492
  • Anti-Influenza agent 3


    <p>Compound 11h: Potent, low-toxicity anti-influenza, inhibits M2 ion channels. EC50: 3.29μM (H3N2), 2.45μM (H1N1).</p>
    Formula:C16H22ClNOS
    Color and Shape:Solid
    Molecular weight:311.87
  • PLAP-IN-1

    CAS:
    <p>PLAP-IN-1: Potent, selective inhibitor of PLAP, IC50 of 32 nM; doesn't notably inhibit TNAP.</p>
    Formula:C25H21Cl2N3O5
    Color and Shape:Soild
    Molecular weight:514.36
  • ZM514


    <p>ZM514 inhibits CD73 (hCD73 IC50: 1.39 μM, mCD73 IC50: 14.65 μM) with low cytotoxicity, suitable for cancer research.</p>
    Formula:C36H57NO4
    Color and Shape:Solid
    Molecular weight:567.84
  • BI-4916

    CAS:
    <p>BI-4916 is a phosphoglycerate dehydrogenase (PHGDH) inhibitor that inhibits SSP and reduces cancer cell migration.</p>
    Formula:C23H24Cl2N2O6S
    Purity:98.55%
    Color and Shape:Solid
    Molecular weight:527.42
  • TH-6


    TH-6, a potent HDAC inhibitor (IC50: HDAC1-0.115, 2-0.135, 3-0.242, 6-0.138, 8-2.120 μM), blocks cell migration, invasion, and has anti-tumor properties.
    Formula:C22H24FN3O5
    Color and Shape:Solid
    Molecular weight:429.44
  • Protease-Activated Receptor-1 antagonist 1


    <p>Compound 13 is a PAR-1 antagonist with a 3 nM IC50, useful for thrombosis and heart disease research.</p>
    Formula:C25H24F2N2O3
    Color and Shape:Solid
    Molecular weight:438.47
  • Beloxepin

    CAS:
    <p>Beloxepin is an oral dual selective inhibitor of serotonin and norepinephrine uptake.</p>
    Formula:C19H21NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:295.38
  • PF-00489791

    CAS:
    <p>PF-00489791 (PF4634817) is a long-acting PDE5 inhibitor with hypotensive activity for the study of diabetic nephropathy.</p>
    Formula:C20H28N8O4S
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:476.55
  • Chitin synthase inhibitor 12


    <p>Chitin synthase inhibitor 12: potent CHS blocker (IC50: 0.16 mM), broad-spectrum antifungal, effective against resistant strains. Useful in IFI research.</p>
    Formula:C23H21ClFN3O5
    Color and Shape:Solid
    Molecular weight:473.88
  • MrgprX2 antagonist-6


    <p>MrgprX2 antagonist-6 is a potent antiallergic agent with inhibitory effects on mast cell degranulation.</p>
    Formula:C24H23F3N6O3
    Color and Shape:Solid
    Molecular weight:500.47
  • L 671776

    CAS:
    <p>L 671776 is an inositol monophosphatase inhibitor.</p>
    Formula:C23H32O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:388.5
  • MT-134


    <p>MT-134 is a SkMII -specific inhibitor and has excellent exposure in muscles.</p>
    Formula:C19H16N4O3
    Color and Shape:Solid
    Molecular weight:348.36
  • Antibacterial agent 99

    CAS:
    <p>Compound 7b (Antibacterial agent 99) is an effective agent with antibacterial, antifungal properties and no haemolytic activity.</p>
    Formula:C27H27BrN2
    Color and Shape:Solid
    Molecular weight:459.42
  • CYP2C9/CYP2C19-IN-1


    <p>CYP2C9/CYP2C19-IN-1 is a potent inhibitor of CYP2C9/CYP2C19 without liver toxicity or genotoxicity and can be used to study Zika virus (ZIKV) infection.</p>
    Formula:C27H28N2O6S
    Color and Shape:Solid
    Molecular weight:508.59
  • FPDT


    <p>FPDT combats glioblastoma by inhibiting the AKT pathway; IC50: &gt;100 μM (astrocytes), 45-68 μM (GBM cells).</p>
    Formula:C16H12FNO2S
    Color and Shape:Solid
    Molecular weight:301.34
  • ATX inhibitor 12


    <p>Oral ATX inhibitor 12 (IC50: 1.72 nM) at 60 mg/kg prevents lung damage in C57Bl/6J mice.</p>
    Formula:C30H34FN5O2
    Color and Shape:Solid
    Molecular weight:515.62
  • Longicoricin

    CAS:
    <p>Longicoricin is a monotetrahydrofuran Annonaceous acetogenin from Asimina longifolia.</p>
    Formula:C37H68O6
    Color and Shape:Solid
    Molecular weight:608.93
  • DC4SMe

    CAS:
    <p>DC4SMe, a prodrug for targeted tumor therapy and ADC synthesis, has IC50s: 1.9 nM (Ramos), 2.9 nM (Namalwa), 1.8 nM (HL60/s).</p>
    Formula:C35H31ClN5O7PS2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:764.21
  • 2,3-dinor-11β-Prostaglandin F2α

    CAS:
    <p>2,3-dinor-11β-Prostaglandin F2α (2,3-dinor-11β-PGF2α) was recovered from the urine of both normal monkeys and humans when infused with radiolabeled PGD2, where</p>
    Formula:C18H30O5
    Color and Shape:Solid
    Molecular weight:326.43
  • Taranabant

    CAS:
    <p>Taranabant: potent CB1 receptor inverse agonist; inhibits agonists with 0.13 nM Ki in vitro.</p>
    Formula:C27H25ClF3N3O2
    Purity:99.06% - 99.06%
    Color and Shape:Solid
    Molecular weight:515.96