Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,539 products)
- Apoptosis(5,812 products)
- Cell Cycle/Checkpoint(4,460 products)
- Chromatin/Epigenetics(2,245 products)
- Cytoskeletal Signaling(1,381 products)
- DNA Damage/DNA Repair(2,829 products)
- Endocrinology/Hormones(3,517 products)
- Enzyme(3,640 products)
- GPCR/G-Protein(8,357 products)
- Immunology and Inflammation(3,538 products)
- Influenza Virus(296 products)
- JAK/STAT signaling(405 products)
- MAPK Signaling(1,203 products)
- Membrane Transporter/Ion Channel(2,806 products)
- Metabolism(9,456 products)
- Microbiology/Virology(6,998 products)
- Neuroscience(9,938 products)
- Other Inhibitors(37,853 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,399 products)
- Proteases/Proteasome(1,600 products)
- Stem Cell and Derivatives(831 products)
- Tyrosine Kinase/Adaptors(2,016 products)
- Ubiquitination(1,650 products)
Show 16 more subcategories
Found 66626 products of "Inhibitors"
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WEHI-539
CAS:<p>WEHI-539 is a selective Bcl-XL inhibitor (IC50: 1.1 nM).</p>Formula:C31H29N5O3S2Purity:98%Color and Shape:SolidMolecular weight:583.72Antibacterial agent 77
<p>Antibacterial agent 77 (compound 12) is an antibacterial agent [1].</p>Formula:C22H27N3OSColor and Shape:SolidMolecular weight:381.53BChE-IN-5
<p>BChE-IN-5: potent, selective BChE inhibitor (IC50: 2.8 nM), more effective on hBChE, potential in Alzheimer's research.</p>Formula:C30H42N4OColor and Shape:SolidMolecular weight:474.68Plevitrexed
CAS:<p>Plevitrexed, an oral TS inhibitor (Ki: 0.44 nM), targets α-folate receptor & reduced folate carrier, treats gastric cancer.</p>Formula:C26H25FN8O4Purity:98%Color and Shape:SolidMolecular weight:532.53Mesulergine hydrochloride
CAS:<p>5-HT2A and 2C receptor antagonist</p>Formula:C18H27ClN4O2SPurity:98%Color and Shape:SolidMolecular weight:398.95Integrase-LEDGF/p75 allosteric inhibitor 1
CAS:<p>Oral HIV-1 allosteric integrase inhibitor, blocks DNA integration, antiviral, potent against NL432 (EC50: 3.9 nM).</p>Formula:C33H41NO6SColor and Shape:SolidMolecular weight:579.75BRD-9526
CAS:BRD-9526 is a potent and selective inhibitor of Sonic Hedgehog (Shh).Formula:C26H31Cl2N3O6SPurity:98%Color and Shape:SolidMolecular weight:584.51Tuberculosis inhibitor 4
<p>TB inhibitor 4, a spirothiazolidinone from mandelic acid, blocks 98% of M. tuberculosis H37Rv under 6 μg/mL.</p>Formula:C23H26N2O3SColor and Shape:SolidMolecular weight:410.53FY-56
<p>FY-56: potent, selective LSD1/KDM1A inhibitor (IC50=42nM); differentiates MOLM-13/MV4-11 cells; promising for AML research.</p>Formula:C23H19FN2O3Color and Shape:SolidMolecular weight:390.41rel-MDM2/4-p53-IN-3
<p>rel-MDM2/4-p53-IN-3 inhibits MDM2/4-p53 PPI, IC50: MDM2 18.5nM, MDM4 14.8nM, targets cancer research.</p>Formula:C25H24Cl2FN3O3Color and Shape:SolidMolecular weight:504.38Elongation factor P-IN-1
<p>EFP-IN-1: potent β-lysine derivative, inhibits EFP, slows E. coli growth.</p>Formula:C14H31N3O2Color and Shape:SolidMolecular weight:273.41Gamendazole
CAS:<p>Gamendazole is a novel drug candidate for male contraception. It has been shown to reduce fertility in male rats without affecting testosterone levels.</p>Formula:C18H11Cl2F3N2O2Purity:98%Color and Shape:SolidMolecular weight:415.19AEP-IN-1
<p>APE-IN-1, a potent AEP inhibitor (IC50: 89 nM), aids Alzheimer's diagnosis and drug research.</p>Formula:C18H27N3O3Color and Shape:SolidMolecular weight:333.43HDAC/HSP90-IN-4
<p>HDAC/HSP90-IN-4 inhibits HDAC (20 IC50=194nM, 26 IC50=360nM) & HSP90α (20 IC50=153nM, 26 IC50=77nM), affects cancer cell survival and invasion.</p>Formula:C20H23N3O6Color and Shape:SolidMolecular weight:401.15869Ici D1542
CAS:Ici D1542: potent TXS inhibitor & TXA2 receptor antagonist, effective thromboxane blocker in vitro.Formula:C25H30N2O7Purity:98%Color and Shape:SolidMolecular weight:470.51Atorvastatin 3-Deoxyhept-2E-Enoic Acid
CAS:Atorvastatin 3-Deoxyhept-2E-Enoic Acid, an impurity in Atorvastatin, lowers blood lipids as an HMG-CoA reductase inhibitor.Formula:C33H33FN2O4Purity:98%Color and Shape:SolidMolecular weight:540.62Nnc 09-0026
CAS:<p>Nnc 09-0026 is a neuronal calcium channel blocker</p>Formula:C25H35Cl2F3N2OColor and Shape:SolidMolecular weight:507.46G092
<p>G092 is a potent inhibitor of MsbA. MsbA is an ABC transporter protein. G092 has potential for antibacterial drug research.</p>Formula:C23H20Cl2N2O3Color and Shape:SolidMolecular weight:443.32LY 215840
CAS:<p>5-HT2/5-HT7 receptor antagonist</p>Formula:C24H33N3O2Purity:98%Color and Shape:SolidMolecular weight:395.54CCG258747
CAS:CCG258747 is a novel, selective inhibitor of the GRK2 subfamily.Formula:C28H27FN4O4Color and Shape:SolidMolecular weight:502.54XR8-89
CAS:<p>XR8-89, a potent PLpro inhibitor (IC50=0.1μM), blocks SARS-CoV-2 replication; useful for research.</p>Formula:C29H36N4O2SColor and Shape:SolidMolecular weight:504.69MM-589
CAS:<p>MM-589 is a potent WD repeat domain 5 (WDR5) inhibitor and mixed lineage leukemia (MLL) protein-protein interaction.</p>Formula:C28H44N8O5Purity:98%Color and Shape:SolidMolecular weight:572.70PF-07202954
CAS:<p>PF-07202954, a weakly basic diacylglycerol O-acyltransferase 2 (DGAT2) inhibitor, exhibits an inhibition concentration half-maximum (IC50) of 10 nM against</p>Formula:C22H23FN6O3Purity:98%Color and Shape:SolidMolecular weight:438.45(Rel)-Factor B-IN-5
CAS:<p>(Rel)-Factor B-IN-5 is a complement factor B inhibitor that can be used to study diseases associated with activation of the alternative complement pathway.</p>Formula:C27H32N2O4Purity:>99.99%Color and Shape:SolidMolecular weight:448.55XP5
<p>XP5 is an oral HDAC6 inhibitor, potent against cancer cells, including YCC3/7 (IC50=31 nM to 2.31 μM).</p>Formula:C19H25N3O5SColor and Shape:SolidMolecular weight:407.48Rostratin B
CAS:<p>Rostratin B, a cytotoxic disulfide, demonstrates in vitro cytotoxicity against human colon carcinoma (HCT-116), exhibiting an IC50 value of 1.9 μg/mL.</p>Formula:C18H20N2O6S2Color and Shape:SolidMolecular weight:424.49β-N-Acetyl-D-hexosaminidase-IN-1
<p>β-N-Acetyl-D-hexosaminidase-IN-1 is a newly discovered chemical compound that acts as an inhibitor for β-N-acetyl-D-hexosaminidase.</p>Formula:C18H13F2NO2SColor and Shape:SolidMolecular weight:345.36Beclabuvir
CAS:<p>Beclabuvir blocks HCV NS5B polymerase at thumb site 1, effective on genotypes 1, 3, 4, 5 with IC50 <28 nM.</p>Formula:C36H45N5O5SPurity:99.87% - 99.93%Color and Shape:SolidMolecular weight:659.84FW 34569
CAS:<p>FW 34569, an enkephalin analog, boosts growth hormones and prolactin, reduces cortisol and LH; FSH stable.</p>Formula:C30H43N5O7SPurity:98%Color and Shape:SolidMolecular weight:617.76Pamiparib maleate
CAS:<p>Pamiparib (BGB-290) is a selective PARP inhibitor that blocks DNA repair and promotes apoptosis.</p>Formula:C44H42F2N8O14Purity:98%Color and Shape:SolidMolecular weight:944.859Everafenib
<p>Everafenib: potent BRAF inhibitor, crosses blood-brain barrier, hinders MAPK, effective on V600EBRAF cells, outperforms other drugs in trials.</p>Formula:C20H23ClFN5O2S2Color and Shape:SolidMolecular weight:484.01ACT-672125
CAS:<p>ACT-672125: Potent CXCR3 blocker, may treat autoimmunity, safe with dose-dependent efficacy in lung inflammation.</p>Formula:C25H25F3N10O2SColor and Shape:SolidMolecular weight:586.59AP5 sodium
CAS:<p>AP5 sodium: potent oral GPR40 agonist, enhances ligands, may aid type II diabetes research.</p>Formula:C28H27FNNaO4Color and Shape:SolidMolecular weight:483.515ZLMT-12
<p>ZLMT-12: tacrine derivative, inhibits CDK2/CDK9, weak on AChE/BuChE, anti-proliferative, low toxicity, blocks S/G2/M phase, induces apoptosis.</p>Formula:C26H31ClN6OColor and Shape:SolidMolecular weight:479.02MAFP
CAS:MAFP (Methyl Arachidonyl Fluorophosphonate) is an effective irreversible inhibitor of anandamide amidase.Formula:C21H36FO2PColor and Shape:SolidMolecular weight:370.48DJT06001
CAS:<p>DJT06001 is a selective Factor Xa inhibitor, reducing thrombus formation with low risk of bleeding.</p>Formula:C21H20ClN3O5SColor and Shape:SolidMolecular weight:461.92Onfasprodil
CAS:<p>Onfasprodil, NR2B inhibitor & GABA regulator, potential for Alzheimer's research. (Patent CN111481543A)</p>Formula:C20H23FN2O3Color and Shape:SolidMolecular weight:358.41Dot1L-IN-1
CAS:<p>The Ki value of DOT1L-in-1 is 2pm.It is a highly effective, selective and novel Dot1L inhibitor.</p>Formula:C32H36ClN9O2SPurity:98%Color and Shape:SolidMolecular weight:646.21PROTAC FKBP Degrader-3
CAS:<p>PROTAC FKBP Degrader-3, with FKBP and VHL binding groups linked, is a potent FKBP degrader.</p>Formula:C68H90N6O17SPurity:98%Color and Shape:SolidMolecular weight:1295.54Complex III-IN-2
<p>Complex III-IN-2 inhibits complex III, with antifungal EC50: 29.31 mg/L vs R. solani, 29.98 mg/L vs S. sclerotiorum.</p>Formula:C15H21ClN2O2SColor and Shape:SolidMolecular weight:328.86FWM-1
<p>FWM-1 blocks SARS-CoV-2 NSP13, hinders ATP binding, with -328.6 kcal/mol binding energy.</p>Formula:C15H11ClN4O4S2Color and Shape:SolidMolecular weight:410.86GAT564
<p>GAT564, an allosteric CB1R modulator, shows EC50s of 87 nM (cAMP) & 320 nM (β-arrestin2) and lowers IOP effectively in glaucoma mice.</p>Formula:C20H16N2O2SColor and Shape:SolidMolecular weight:348.4222-HDHA
CAS:<p>22-HDHA is an oxidation product of docosahexaenoic acid .</p>Formula:C22H32O3Color and Shape:SolidMolecular weight:344.49Hypoglycemic agent 1
CAS:<p>Hypoglycemic agent 1 has an action for lowering blood sugar. It acts as a therapeutic and/or prophylactic agent for diabetes.</p>Formula:C25H24FN5O4Purity:98%Color and Shape:SolidMolecular weight:477.49HER2-IN-12
<p>HER2-IN-12 is an HER2 inhibitor with an IC50 value of 121 nM and can be used to study cancers such as breast cancer.</p>Formula:C17H18BrN5O2SColor and Shape:SolidMolecular weight:436.33Revamilast sodium
CAS:<p>Revamilast sodium, also known as GRC4039 sodium, is a phosphodiesterase IV inhibitor for potentially treating of asthma and rheumatoid arthritis</p>Formula:C18H8Cl2F2N3NaO4Color and Shape:SolidMolecular weight:462.17FPI-1465
CAS:<p>FPI-1465: Dual serine-β-lactamase & PBP inhibitor; IC50 PBP2=1.0 μg/mL; Kd CTX-M-15=0.011μM, OXA-48=5.3μM.</p>Formula:C11H18N4O7SColor and Shape:SolidMolecular weight:350.35Ascofuranone
CAS:<p>Ascofuranone is an inhibitor of the ubiquinol oxidase activity of Trypanosoma brucei mitochondrial alternative oxidase (TAO), as well as an inhibitor of HsDHODH</p>Formula:C23H29ClO5Color and Shape:SolidMolecular weight:420.935(S),6(S)-DiHETE
CAS:<p>5(S),6(S)-DiHETE: a 5,6-dihydroxy acid from LTA4 hydrolysis, lacks leukotriene activity.</p>Formula:C20H32O4Color and Shape:SolidMolecular weight:336.47Antiproliferative agent-8
<p>Compound 5a, an anticancer agent, enhances P53 and has antiproliferative effects.</p>Formula:C22H16ClN3O3Color and Shape:SolidMolecular weight:405.83CLK1/2-IN-1
CAS:<p>CLK1/2-IN-1 is a CLK1 and CLK2 inhibitor and it also inhibits SRPK1 and SRPK2.</p>Formula:C21H20F3N7OPurity:98%Color and Shape:SolidMolecular weight:443.42SB 258741 hydrochloride
<p>SB 258741 hydrochloride is a potent antagonist of the 5-HT 7 receptor, designed specifically for studying schizophrenia [1].</p>Formula:C19H31ClN2O2SColor and Shape:SolidMolecular weight:386.98Tubulin inhibitor 16
<p>Tubulin inhibitor 16 is a potent tubulin inhibitor with antiproliferative activity. Tubulin inhibitor 16 exhibits cytotoxicity in HepG2 cells [1].</p>Formula:C16H12FNO2Color and Shape:SolidMolecular weight:269.27BU09059
CAS:BU09059 is a potent, selective, short-acting antagonist of the κ-opioid receptor (KOR).Formula:C28H37N3O5Purity:98%Color and Shape:SolidMolecular weight:495.61RAD51-IN-8
<p>RAD51-IN-8 inhibits RAD51-BRCA2 interaction and H4A4 with EC50 of 19 μM; a micromolar PPI inhibitor.</p>Formula:C16H14Cl2FN3O2Color and Shape:SolidMolecular weight:370.21Zanapezil fumarate
CAS:<p>Zanapezil is an acetylcholinesterase (AChE) inhibitor. Zanapezil increases choline acetyltransferase activity in cultured rat septal cholinergic neurons.</p>Formula:C29H36N2O5Color and Shape:SolidMolecular weight:492.61MI-1481
CAS:<p>MI-1481: potent MML1 inhibitor, IC50 3.6 nM; disrupts menin-MLL1, active in MLL leukemia.</p>Formula:C29H30F3N7O2SPurity:98%Color and Shape:SolidMolecular weight:597.65EGFR/BRAF-IN-1
<p>EGFR/BRAF-IN-1 inhibits EGFR/BRAF (BRAFV600E IC50: 45 nM, GI50: 35 nM) and has antioxidant properties.</p>Formula:C26H28ClN3O4Color and Shape:SolidMolecular weight:481.97PI3K-IN-27
CAS:<p>PI3K-IN-27 is a potent PI3K inhibitor, relevant for cancer and immune disease research. See patent WO2021233227A1.</p>Formula:C30H26F2N6O2SColor and Shape:SolidMolecular weight:572.63GSK-3β inhibitor 6
<p>GSK-3β inhibitor 6 is a highly potent inhibitor of GSK-3β, with an IC50 value of 24.4 μM.</p>Formula:C20H17BrN4Color and Shape:SolidMolecular weight:393.28Netupitant metabolite Monohydroxy Netupitant
CAS:Monohydroxy Netupitant is a highly selective antagonist of NK1 receptor, and is Netupitant metabolite.Formula:C30H32F6N4O2Purity:98%Color and Shape:SolidMolecular weight:594.59JH-XVII-10
<p>JH-XVII-10: potent, oral DYRK1A/B inhibitor (IC50: 3/5 nM), shows antitumor activity in HNSCC.</p>Formula:C21H16F4N8OColor and Shape:SolidMolecular weight:472.4Ketomethylenebestatin
CAS:<p>Ketomethylenebestatin, a weaker carba-analog of aminopeptidase inhibitor bestatin, is 10x less potent.</p>Formula:C17H25NO4Purity:98%Color and Shape:SolidMolecular weight:307.38Hetrombopag olamine
CAS:<p>Hetrombopag olamine is a non-peptide thrombopoietin (TPO) receptor agonist with oral activity.</p>Formula:C29H36N6O7Purity:98%Color and Shape:SolidMolecular weight:580.63MEIS-IN-2
<p>MEIS-IN-2 is an inhibitor of MEIS1. MEIS-IN-2 can be used in studies of cardiac regeneration and haematopoietic stem cell (HSC) regulation.</p>Formula:C23H21ClN2O4Color and Shape:SolidMolecular weight:424.88Antifungal agent 28
<p>Antifungal 28 disrupts Candida, hits fluconazole-resistant strains, and inhibits biofilms.</p>Formula:C22H29N5OSColor and Shape:SolidMolecular weight:411.56IDH1 Inhibitor 1
CAS:<p>Oral, brain-penetrant mutant IDH1 inhibitor targeting R132H/C with IC50: 0.021/0.045μM; 2.52μM for IDH1WT.</p>Formula:C20H18F4N6O2Purity:98%Color and Shape:SolidMolecular weight:450.39Musettamycin
CAS:<p>Musettamycin triggers erythroid differentiation in blood cells, acts like anthracycline antibiotics, but only inhibits gram-positive bacteria.</p>Formula:C36H45NO14Color and Shape:SolidMolecular weight:715.74PARP1/BRD4-IN-2
<p>PARP1/BRD4-IN-2, a potent inhibitor of PARP1 and BRD4, halts cell cycle, triggers apoptosis, and has antitumor effects on TNBC.</p>Formula:C25H20N4O4Color and Shape:SolidMolecular weight:440.45Polvitolimod
CAS:<p>Polvitolimod is a TLR7 agonist used to treat infectious disease and cancer.</p>Formula:C13H14FN5O4Color and Shape:SolidMolecular weight:323.28OM-153
CAS:<p>OM-153 blocks tankyrase 1 (IC50: 13 nM) and 2 (IC50: 2 nM), stifling WNT signaling and COLO 320DM cell growth.</p>Formula:C28H24FN7O2Color and Shape:SolidMolecular weight:509.53BET-IN-6
CAS:<p>BET-IN-6: Potent BRD2/4 inhibitor and ligand for PROTAC BRD2/BRD4 degrader-1 synthesis.</p>Formula:C22H20N2O6SPurity:98%Color and Shape:SolidMolecular weight:440.47EP4 receptor antagonist 2
CAS:<p>EP4 receptor antagonist 2 (compound 2-13) is a potent agonist of the EP4 receptor (IC50: 7.8 nM) and has antitumour effects.</p>Formula:C27H29N3O5Color and Shape:SolidMolecular weight:475.54Glycotriosyl glutamine
CAS:<p>Glycotriosyl glutamine is a nephritogenoside analog.</p>Formula:C23H40N2O18Color and Shape:SolidMolecular weight:632.57Cbl-b-IN-2
CAS:<p>Cbl-b-IN-2 is an oral E3 enzyme inhibitor for immune-modulated diseases and cancer research.</p>Formula:C29H30F5N5O2Color and Shape:SolidMolecular weight:575.57A 70450
CAS:<p>A 70450, an inhibitor of aspartyl proteinase, can be used as an antifungal agent and may have a role in HIV protease inhibition therapy.</p>Formula:C42H71ClN6O5Purity:98%Color and Shape:SolidMolecular weight:775.50(±)-ANAP hydrochloride (1185251-08-4 free base)
<p>(±)-ANAP hydrochloride is the amino acid analog of prodan. It can be used as a fluorescent probes and enhance environmental sensitivity.</p>Formula:C15H17ClN2O3Purity:98%Color and Shape:SolidMolecular weight:308.76QPX7728 methoxy acetoxy methy ester
CAS:QPX7728 methoxy acetoxy methy ester is an inhibitor of boronic acid β-lactamase.Formula:C14H14BFO7Purity:98%Color and Shape:SolidMolecular weight:324.07SR121566A
CAS:SR121566A is a novel non-peptide antagonist of Glycoprotein IIb/IIIa (GP IIb-IIIa).Formula:C20H25N5O4SPurity:98%Color and Shape:SolidMolecular weight:431.51PDHK-IN-4
<p>PDHK-IN-4 inhibits PDHK2 (IC50: 0.0051 μM) & PDHK4 (IC50: 0.0122 μM), with potential for cancer research.</p>Formula:C24H25N5O3Color and Shape:SolidMolecular weight:431.49Heme Oxygenase-2-IN-1
<p>Heme Oxygenase-2-IN-1 is a selective HO-2 inhibitor with IC50s: 14.9 μM (HO-1), 0.9 μM (HO-2).</p>Formula:C19H17N3O2Color and Shape:SolidMolecular weight:319.36CU-2010
CAS:<p>CU-2010 is a synthetic compound that reduces blood loss and aids recovery post-cardiac surgery.</p>Formula:C37H42N6O6SColor and Shape:SolidMolecular weight:698.83(Rac)-PT2399
CAS:<p>(Rac)-PT2399 is a potent and specific inhibitor of hypoxia-inducible factor 2a (HIF-2α)(IC50 of 0.01 μM).</p>Formula:C17H10F5NO4SColor and Shape:SolidMolecular weight:419.32RXR antagonist 1
<p>RXR antagonist 1 is a Retinoid X Receptor (RXR) modulator that exhibits high RXR antagonism (pA2: 8.06). RXR antagonist 1 can be used to study type 2 diabetes.</p>Formula:C28H33F3N2O3Color and Shape:SolidMolecular weight:502.57DNA crosslinker 3 dihydrochloride
CAS:<p>Compound 1: a DNA minor groove binder with 1.4°C ΔTm; useful in cancer research.</p>Formula:C15H22Cl2N8OColor and Shape:SolidMolecular weight:401.29CDK7-IN-17
CAS:<p>CDK7-IN-17, a pyrimidine-based CDK7 inhibitor, shows promise for various cancers, especially with abnormal transcription.</p>Formula:C24H26F3N6OPColor and Shape:SolidMolecular weight:502.47RSK4-IN-1
CAS:<p>RSK4-IN-1 is a compound exhibiting potent inhibition of RSK4, demonstrated by an IC50 value of 9.5 nM.</p>Formula:C19H20F2N4O3Color and Shape:SolidMolecular weight:390.38Bcl-2-IN-6
<p>Bcl-2-IN-6 suppresses Bcl-2, upregulates p53/Bax/caspase-7, arrests cell cycle, and induces MCF-7 apoptosis; IC50s: MCF-7 20.91 μM, others <48 μM.</p>Formula:C25H24N4O5S2Color and Shape:SolidMolecular weight:524.61PDE4-IN-14
CAS:<p>PDE4-IN-14 (Compound 1) serves as an inhibitor of phosphodiesterase 4 (PDE4), applicable in research concerning diseases associated with PDE4, including</p>Formula:C19H20F2N4O3SColor and Shape:SolidMolecular weight:422.45LY503430
CAS:<p>LY503430: Oral AMPA enhancer with nootropic, neuroprotective properties, mitigates 6-OHDA/MPTP brain damage.</p>Formula:C20H25FN2O3SPurity:98%Color and Shape:SolidMolecular weight:392.49AXKO-0046
<p>AXKO-0046 is an indole derivative and small-molecule LDHB selective inhibitor.</p>Formula:C25H33N3Color and Shape:SolidMolecular weight:375.55S-HP210
<p>S-HP210: selective GR modulator, blocks NF-κB (IC50: 1.92 μM), non-toxic to mouse fibroblasts.</p>Formula:C22H19N3O2S2Color and Shape:SolidMolecular weight:421.54NSC381467
CAS:<p>NSC381467: Potent, oral EGFR-TK inhibitor with strong antiproliferative effects, promising for cancer research.</p>Formula:C20H16O7Color and Shape:SolidMolecular weight:368.34CYP11B1-IN-2
<p>CYP11B1-IN-2 selectively inhibits human and rat CYP11B1 (IC50: 9/25 nM) orally to research cortisol-related diseases.</p>Color and Shape:SolidONO-5334
CAS:<p>ONO-5334: selective cathepsin K inhibitor, potential for osteoporosis study; Ki: 0.10 nM (human), 0.049 nM (rabbit), 0.85 nM (rat).</p>Formula:C21H34N4O4SPurity:98.22% - 99.60%Color and Shape:SolidMolecular weight:438.58J-104132
CAS:<p>J-104132: potent human ETA/B antagonist; Ki: ETA=0.034nM, ETB=0.104nM; prevents ET-1 effects, ED50 i.v.=0.045mg/kg, p.o.=0.35mg/kg.</p>Formula:C31H33NO7Purity:98%Color and Shape:SolidMolecular weight:531.60Ranakinin
CAS:<p>Ranakinin is a novel tachykinin receptor agonist; from the brain of frog, Rana ridibunda.</p>Formula:C62H95N17O15SColor and Shape:SolidMolecular weight:1350.59AS2521780
CAS:AS2521780 is an inhibitor of PKCθ (IC50: 0.48 nM).Formula:C30H41N7OSPurity:98%Color and Shape:SolidMolecular weight:547.76HER2-IN-10
<p>HER2-IN-10 is a psoralen derivative that induces apoptosis. HER2-IN-10 shows anti-breast cancer activity and light-activated cytotoxicity [1].</p>Formula:C15H13NO5Color and Shape:SolidMolecular weight:287.27PD-L1-IN-1
<p>PD-L1-IN-1, potent PD-L1 inhibitor with 115 nM IC50, suppresses tumors, boosts immune response, and spares healthy cells.</p>Formula:C21H23N5O2Color and Shape:SolidMolecular weight:377.44
