Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,523 products)
- Apoptosis(5,792 products)
- Cell Cycle/Checkpoint(4,449 products)
- Chromatin/Epigenetics(2,238 products)
- Cytoskeletal Signaling(1,383 products)
- DNA Damage/DNA Repair(2,825 products)
- Endocrinology/Hormones(3,507 products)
- Enzyme(3,640 products)
- GPCR/G-Protein(8,333 products)
- Immunology and Inflammation(3,526 products)
- Influenza Virus(296 products)
- JAK/STAT signaling(404 products)
- MAPK Signaling(1,202 products)
- Membrane Transporter/Ion Channel(2,790 products)
- Metabolism(9,448 products)
- Microbiology/Virology(6,981 products)
- Neuroscience(9,926 products)
- Other Inhibitors(37,926 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,400 products)
- Proteases/Proteasome(1,597 products)
- Stem Cell and Derivatives(831 products)
- Tyrosine Kinase/Adaptors(2,016 products)
- Ubiquitination(1,650 products)
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Found 66641 products of "Inhibitors"
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MtTMPK-IN-3
CAS:<p>MtTMPK-IN-3 inhibits Mycobacterium tuberculosis kinase with IC50 0.12μM, MIC 12.5μM on Mtb, cytotoxic EC50 12.5μM on MRC-5 cells.</p>Formula:C23H23Cl2N3O3Color and Shape:SolidMolecular weight:460.35Gallinamide A
CAS:<p>Gallinamide A is a potent inhibitor of cathepsin L with an IC 50 value of 17.6 pM.</p>Formula:C31H52N4O7Color and Shape:SolidMolecular weight:592.77Antitumor agent-77
<p>Antitumor agent-77 suppresses cancer cell growth, migration, induces apoptosis, and hinders EMT.</p>Formula:C7H11F3N2O5PtColor and Shape:SolidMolecular weight:455.25CYP121A1-IN-1
<p>CYP121A1-IN-1: Strong inhibitor for CYP121A1, hinders Mycobacterium tuberculosis growth (MIC 90 ~6.25 μM), reduces mycocyclosin synthesis.</p>Formula:C22H20N4OColor and Shape:SolidMolecular weight:356.42CXCR4 antagonist 3
<p>CXCR4 antagonist 3, aka compound 12a, has 11 nM IC50, shares TIQ15 traits, and is promising in HIV research.</p>Formula:C22H31N5Color and Shape:SolidMolecular weight:365.52U 75875
CAS:<p>U 75875 is a protease inhibitor.</p>Formula:C45H61N7O7Color and Shape:SolidMolecular weight:812.01MtTMPK-IN-7
<p>MtTMPK-IN-7 inhibits MtbTMPK (IC50: 47 μM), active against M. brevis (MIC: 2.3-4.7 μM), useful for tuberculosis research.</p>Formula:C27H29ClN6O3Color and Shape:SolidMolecular weight:521.01DS-9300
CAS:<p>DS-9300, an orally administered potent and selective inhibitor of EP300/CBP HAT, exhibits a significant inhibitory activity with an IC50 value of 28 nM.</p>Formula:C25H26F3N5O3Color and Shape:SolidMolecular weight:501.50ABL-001-Amide-PEG3-acid
ABL-001-Amide-PEG3-acid, an analogue to ABL-001, primarily serves as a labeled chemical or fluorescent probe.Formula:C29H33ClF2N6O9Purity:98%Color and Shape:SolidMolecular weight:683.06Aristoforin
CAS:<p>Aristoforin is a SIRT1 and SIRT2 inhibitor that induces cell cycle arrest, shows potent antitumor effects, and inhibits lymphangiogenesis in vivo.</p>Formula:C37H54O6Color and Shape:SolidMolecular weight:594.82BAY-693
CAS:<p>BAY-693 is a ERK5 negative control agent with IC50 (ERK5) = 6400 nM. Its analog, BAY-885, is a potent and selective ERK5 (MAPK7) inhibitor with IC50 of 40 nM</p>Formula:C26H30F3N7O2Color and Shape:SolidMolecular weight:529.56Neuraminidase-IN-4
<p>Neuraminidase-IN-4 inhibits neuraminidase (EC50: 1.59 μM) and has strong anti-H5N1 activity.</p>Formula:C21H20N2O6SColor and Shape:SolidMolecular weight:428.46U75302
CAS:<p>U75302 is an antagonist of thymosin beta-4 (TB4) receptor with a Ki value of 159 nM on guinea pig lung membranes.</p>Formula:C22H35NO3Purity:98%Color and Shape:Light Yellow OilMolecular weight:361.52(S)-3-Hydroxy Midostaurin
CAS:<p>(S)-3-Hydroxy Midostaurin is a potent inhibitor of kinases(IC50 of <400 nM for 13 kinases (VEGFR-2, TRK-A, FLT3, et)).</p>Formula:C35H30N4O5Purity:98%Color and Shape:SolidMolecular weight:586.64Complex III-IN-2
<p>Complex III-IN-2 inhibits complex III, with antifungal EC50: 29.31 mg/L vs R. solani, 29.98 mg/L vs S. sclerotiorum.</p>Formula:C15H21ClN2O2SColor and Shape:SolidMolecular weight:328.86TAK-915
CAS:<p>TAK-915: potent, brain-ready PDE2A inhibitor, 0.61 nM IC50, 4100x selectivity over PDE1A.</p>Formula:C19H18F4N4O5Purity:98%Color and Shape:SolidMolecular weight:458.36Antibacterial agent 110
<p>Compound 4e, an antibacterial against P. aeruginosa, disrupts cell membranes (MIC: 1 μg/ml).</p>Formula:C22H21N5O4SColor and Shape:SolidMolecular weight:451.5IRE1α kinase-IN-5
<p>IRE1α kinase-IN-5 (compound 7) is a potent inhibitor of IRE1α (Ki: 98 nM) and is an ATP-competitive ligand for IRE1α.</p>Formula:C28H30N6O3SColor and Shape:SolidMolecular weight:530.64SG3199
CAS:<p>SG3199, a PBD dimer, binds DNA's minor groove, forms covalent cross-links, and is cytotoxic to various human cancer cells.</p>Formula:C33H36N4O6Color and Shape:SolidMolecular weight:584.66Dictyostatin
CAS:<p>Dictyostatin: potent microtubule stabilizer & anticancer agent with antiproliferative effects; researched for tauopathies.</p>Formula:C32H52O6Color and Shape:SolidMolecular weight:532.75BILA 1906 BS
CAS:<p>BILA 1906 BS is an inhibitor of substrate analog protease.</p>Formula:C41H52N6O4SPurity:98%Color and Shape:SolidMolecular weight:724.95EGFR-IN-47
<p>EGFR-IN-47: strong oral EGFRL858R/T790M/C797S blocker, induces cell death; promising for NSCLC research. IC50: 0.01 μM.</p>Formula:C29H35N7Color and Shape:SolidMolecular weight:481.64Terguride
CAS:<p>Terguride: treats hyperprolactinemia, blocks 5-HT2A/B, activates dopamine receptors, studied for PAH.</p>Formula:C20H28N4OColor and Shape:SolidMolecular weight:340.46VEGFR-2-IN-10
<p>VEGFR-2-IN-10 has enhanced antiangiogenic potency against VEGFR2 phosphorylation induced by VEGF with an IC50 value of 0.7 μM and no cytotoxic effects.</p>Formula:C20H21N3O2Color and Shape:SolidMolecular weight:335.4Chitin synthase inhibitor 7
<p>Compound 9c, a chitin synthase inhibitor, has an IC50 of 0.37 nM and is useful for studying fungal infections.</p>Formula:C24H25N3O5Color and Shape:SolidMolecular weight:435.47XR8-89
CAS:<p>XR8-89, a potent PLpro inhibitor (IC50=0.1μM), blocks SARS-CoV-2 replication; useful for research.</p>Formula:C29H36N4O2SColor and Shape:SolidMolecular weight:504.69TLR7/8 antagonist 2
<p>TLR7/8 antagonist 2: potent, orally active, IC50: 4.9 nM (TLR7), 0.6 nM (TLR8); potential for lupus therapy research.</p>Formula:C22H26FN5Color and Shape:SolidMolecular weight:379.47Gusperimus
CAS:<p>Gusperimus was synthesized by chemical modification of spergualin and in combination with cyclosporine A to prevent diabetes in susceptible NOD mice.</p>Formula:C17H37N7O3Color and Shape:SolidMolecular weight:387.52Protectin D1
CAS:<p>Protectin D1 (Neuroprotectin D1) is a neuroprotectin produced by nerve cells and is a potential cardioprotective agent.</p>Formula:C22H32O4Purity:99.72% - 99.79%Color and Shape:SolidMolecular weight:360.49PPARγ agonist 1
<p>PPARγ agonist 1 is a potent agonist of PPARγ that efficiently activates hPPARγ without causing full agonism, thereby avoiding adverse effects.</p>Formula:C34H39NO3Color and Shape:SolidMolecular weight:509.68Keap1-Nrf2-IN-4
<p>Keap1-Nrf2-IN-4 hinders MGC-803 cell growth (IC50=2.55μM), migration, and induces apoptosis with low toxicity.</p>Formula:C26H34N2OColor and Shape:SolidMolecular weight:390.56NTPDase-IN-3
CAS:<p>NTPDase-IN-3 inhibits NTPDase1/2/3/8 (IC50: 0.21/1.07/0.38/0.05 μM), useful for cancer and thrombosis research.</p>Formula:C22H24ClN3OS2Color and Shape:SolidMolecular weight:446.03(S)-Seco-Duocarmycin SA
CAS:<p>(S)-Seco-Duocarmycin SA is a DNA alkylating agent and antibiotic with potent antitumor activity that can be used to synthesize ADC compounds.</p>Formula:C25H24ClN3O7Purity:98%Color and Shape:SolidMolecular weight:513.93JH-XVII-10
<p>JH-XVII-10: potent, oral DYRK1A/B inhibitor (IC50: 3/5 nM), shows antitumor activity in HNSCC.</p>Formula:C21H16F4N8OColor and Shape:SolidMolecular weight:472.4Alentemol hydrobromide
CAS:<p>Alentemol hydrobromide is a Dopamine agonist.</p>Formula:C19H26BrNOPurity:98%Color and Shape:SolidMolecular weight:364.32Antiangiogenic agent 2
<p>Antiangiogenic agent 2 (compound 3b) is a potent inhibitor of thymidine phosphorylase (IC50: 39.71 μM) and exhibits anti-angiogenic effects.</p>Formula:C26H26FN3O4Color and Shape:SolidMolecular weight:463.5Tubulin inhibitor 16
<p>Tubulin inhibitor 16 is a potent tubulin inhibitor with antiproliferative activity. Tubulin inhibitor 16 exhibits cytotoxicity in HepG2 cells [1].</p>Formula:C16H12FNO2Color and Shape:SolidMolecular weight:269.27GSK 366
CAS:<p>GSK 366 is a potent kynurenine-3-monooxygenase (KMO) inhibitor (IC50s: 0.7 nM and 2.3 nM for P. fluorescens-KMO and human KMO).</p>Formula:C17H16ClN3O4Purity:98%Color and Shape:SolidMolecular weight:361.78Tenellin
CAS:<p>Tenellin is a fungal metabolite that inhibits Mg2+-, Ca2+-, and Na+/K+-ATPase activities in erythrocytes. Tenellin is cytotoxic to Sf9 and Sf21 insect cells.</p>Formula:C21H23NO5Color and Shape:SolidMolecular weight:369.41AChE-IN-10
<p>AChE-IN-10 (24r) inhibits AChE (IC50=2.4 nM), reducing amyloid buildup, tau phosphorylation, and promotes neuron health.</p>Formula:C23H27F2NO4SColor and Shape:SolidMolecular weight:451.53CHK-IN-1
CAS:<p>CHK-IN-1 is a dual inhibitor of CHK1 and CHK2 with antiproliferative activity.</p>Formula:C18H19ClFN5OSPurity:>99.99%Color and Shape:SolidMolecular weight:407.89Spicamycin
CAS:<p>Spicamycin can be used as a potent inducer of differentiation of human myeloid leukemia cells (HL-60) and murine myeloid leukemia cells (M1).</p>Formula:C30H51N7O7Color and Shape:SolidMolecular weight:621.77FGFR4-IN-10
<p>FGFR4-IN-10 (compound 5a) is a potent, selective FGFR4 inhibitor with IC50 of 70.7 nM, sparing FGFR1-3.</p>Formula:C20H19F3N6O3Color and Shape:SolidMolecular weight:448.4KR-67607
CAS:<p>KR-67607, or NTX-101, is a novel 11β-HSD1 inhibitor that protects against eye injury by reducing cortisol and preserving eye structures.</p>Formula:C24H29Cl2F3N4O4SColor and Shape:SolidMolecular weight:597.48HER2-IN-9
<p>HER2-IN-9, an oral HER2 inhibitor (IC50: 0.03 μM), hinders growth and spread of HER2+ breast cancer.</p>Formula:C19H14BrF3N2OColor and Shape:SolidMolecular weight:423.23GSK2578999A
CAS:<p>GSK2578999A is a betulin derivative with antitumor activity.</p>Formula:C46H62ClNO7Purity:98%Color and Shape:SolidMolecular weight:776.44Quinagolide hydrochloride
CAS:<p>Quinagolide hydrochloride is a selective agonist of dopamine D2 receptor.</p>Formula:C20H34ClN3O3SPurity:98%Color and Shape:SolidMolecular weight:432.02ICA-105665
CAS:<p>ICA-105665 is an orally active Kv7.2/7.3/7.5 channel opener, CNS-penetrant with antiseizure effects, and low hepatocyte cytotoxicity.</p>Formula:C19H15F2N3O2Purity:98%Color and Shape:SolidMolecular weight:355.34Cenicriviroc Sulfone
CAS:<p>Cenicriviroc Sulfone, a Cenicriviroc derivative, inhibits CCR2/CCR5 to block HIV entry into cells.</p>Formula:C41H52N4O5SColor and Shape:SolidMolecular weight:712.94264W94
CAS:<p>264W94 robustly inhibits IBAT, induces CYP7A1, and significantly reduces cholesterol.</p>Formula:C23H31NO4SPurity:98%Color and Shape:SolidMolecular weight:417.56BM635 hydrochloride
<p>BM635 hydrochloride, an MmpL3 inhibitor, strongly blocks Divergent bacteriophage H37Rv (MIC50: 0.08 μM), with doubled in vivo potency.</p>Formula:C25H30ClFN2OColor and Shape:SolidMolecular weight:428.97Adafosbuvir
CAS:<p>Adafosbuvir has antiviral activity.</p>Formula:C22H29FN3O10PColor and Shape:SolidMolecular weight:545.457IACS-8779 disodium
CAS:<p>IACS-8779 disodium: potent STING agonist, strong systemic anti-tumor effects, effective in melanoma model.</p>Formula:C21H23N9Na2O10P2S2Color and Shape:SolidMolecular weight:733.52Isoleucyl tRNA synthetase-IN-1
CAS:<p>Isoleucyl tRNA synthetase-IN-1 is a selective and potent inhibitor (Ki: 88 nM) that targets isoleucyl tRNA synthetase (IleRS).</p>Formula:C23H35N5O7SColor and Shape:SolidMolecular weight:525.62MCTR2
CAS:<p>MCTR2, synthesized from DHA in macrophages, aids in tissue repair and reduces inflammation by promoting eicosanoid PGD2 and PGF2α decrease.</p>Formula:C27H40N2O6SColor and Shape:SolidMolecular weight:520.68GSK852
<p>GSK852 is a potent, second bromodomain (BD2)-selective, bromo and extra-terminal domain (BET) inhibitor with pIC50 of 7.9.</p>Formula:C24H26N2O4Color and Shape:SolidMolecular weight:406.47Cilazaprilat
CAS:<p>Cilazaprilat is the active metabolite of cilazapril, a pyridazine angiotensin-converting enzyme (ACE) inhibitor with antihypertensive activity.</p>Formula:C20H27N3O5Color and Shape:SolidMolecular weight:389.45Chitin synthase inhibitor 1
<p>Potent, selective CHS inhibitor with 0.12 mM IC50; effective against drug-resistant fungi.</p>Formula:C22H20ClN3O3Color and Shape:SolidMolecular weight:409.87GSK8814
CAS:<p>GSK8814 is a selective and ATAD2/2B bromodomain chemical probe and inhibitor (binding constant pKd=8.1 and a pKi=8.9 in BROMOscan).</p>Formula:C28H35F2N5O3Purity:98%Color and Shape:SolidMolecular weight:527.61BRD-7880
CAS:<p>BRD-7880 is a potent and highly specific inhibitor of aurora kinases B and C.</p>Formula:C32H38N4O7Color and Shape:SolidMolecular weight:590.67Carbonic anhydrase inhibitor 3
<p>Carbonic anhydrase inhibitor 3 (compound 11g) is an inhibitor of carbonic anhydrase II that reduces the intraocular pressure in glaucomatous rabbits [1].</p>Formula:C15H17N3O3SColor and Shape:SolidMolecular weight:319.38AY-22,252
CAS:<p>AY-22,252 is an inhibitor of beef heart & rat brain nucleoside-3',5'- monophosphate phosphodiesterase.</p>Formula:C27H37NaO7Color and Shape:SolidMolecular weight:496.57Sekdel sequence
CAS:<p>Sekdel sequence, as a signal, leads to retention of at least two proteins in the endoplasmic reticulum of animal cells.</p>Formula:C29H49N7O14Color and Shape:SolidMolecular weight:719.74MtTMPK-IN-2
CAS:<p>MtTMPK-IN-2 inhibits M. tuberculosis TMPK (IC50: 1.1 μM), Mtb H37Rv (MIC: 12.5 μM), and is cytotoxic in MRC-5 cells (EC50: 6.1 μM).</p>Formula:C23H24ClN3O3Color and Shape:SolidMolecular weight:425.91NR1H4 activator 1
CAS:<p>NR1H4 activator 1 is a potent and selective agonist of Famesoid X Receptor (FXR).</p>Formula:C34H53NO7SPurity:98%Color and Shape:SolidMolecular weight:619.85Equisetin
CAS:<p>Equisetin: a QSI from Fusarium equiseti, curbs P. aeruginosa virulence, fights Gram-positive bacteria & HIV-1 integrase; not antibacterial to Gram-negative.</p>Formula:C22H31NO4Purity:98%Color and Shape:SolidMolecular weight:373.49CK2 inhibitor 3
<p>CK2 inhibitor 3: potent CK2 blocker, IC50 of 280 nM, suppresses tumor cell growth, highly selective among 320 kinases.</p>Formula:C13H9BrN4O3SColor and Shape:SolidMolecular weight:381.2MsbA-IN-5
<p>MsbA-IN-5 (compound 40) is a potent and highly selective inhibitor of MsbA (IC50: 2 nM). MsbA-IN-5 can be used in Gram-negative studies.</p>Formula:C23H19Cl2N5OColor and Shape:SolidMolecular weight:452.34Tubulin inhibitor 14
<p>Tubulin inhibitor 14 blocks NQO2 and microtubule formation, disrupts blood vessels, and may target tumors; IC50 of 1.0 μM.</p>Formula:C15H9F2NOColor and Shape:SolidMolecular weight:257.23Oiligodendrocyte differentiation promoter 1
CAS:<p>Oiligodendrocyte differentiation promoter 1 is a promoter of oiligodendrocyte differentiation .</p>Formula:C25H25Cl2NO5Purity:98%Color and Shape:SolidMolecular weight:490.38URAT1 inhibitor 2
<p>URAT1 inhibitor 2: oral URAT1/CYP blocker, IC50 of 1.36μM (URAT1), 16.97μM (CYP1A2), 5.22μM (CYP2C9); potential gout treatment.</p>Formula:C21H18BrN3O2SColor and Shape:SolidMolecular weight:456.36SARS-CoV-2 nsp14-IN-2
<p>SARS-CoV-2 nsp14-IN-2: Strong Nsp14 methyltransferase inhibitor (IC50: 0.09 μM), potential for COVID-19 research.</p>Formula:C21H21N5O5SColor and Shape:SolidMolecular weight:455.49Antibiotic MA 144M1
CAS:<p>Antibiotic MA 144M1, an anthracycline, targets gram-positive bacteria and animal tumors; derived from Streptomyces fermentation or aclacinomycin A conversion.</p>Formula:C42H55NO15Color and Shape:SolidMolecular weight:813.88Antibacterial agent 62
<p>Novel anti-TB agent 62 is a redox compound with bactericidal activity against active and dormant bacteria.</p>Formula:C24H33BrN2O2Color and Shape:SolidMolecular weight:461.44MK-7128
CAS:<p>MK-7128 is a CB1 receptor inverse agonist.</p>Formula:C29H25ClF2N4O2Color and Shape:SolidMolecular weight:534.98ER272
CAS:<p>ER272 is a natural PKC activator, inducing hippocampal neurogenesis.</p>Formula:C24H34O6Color and Shape:SolidMolecular weight:418.52Pyruvate Carboxylase-IN-2
CAS:<p>Pyruvate Carboxylase-IN-2, erianin analog, inhibits PC with IC50s of 0.065/0.097 μM in lysate/cell assays, targets HCC.</p>Formula:C21H22O8Color and Shape:SolidMolecular weight:402.39NVP-CGM097 sulfate
CAS:<p>NVP-CGM097 sulfate is a potent and selective inhibitor of MDM2 (hMDM2, IC50 of 1.7±0.1 nM).</p>Formula:C38H49ClN4O8SPurity:98%Color and Shape:SolidMolecular weight:757.34KRAS G12D inhibitor 16
CAS:<p>KRAS G12D inhibitor 16 targets KRAS G12D with IC50 of 0.7 nM and mutant form at 0.35 μM, useful in various cancer studies.</p>Formula:C32H39IN6O3Color and Shape:SolidMolecular weight:682.59GDC-0339
CAS:<p>GDC-0339: oral Pim kinase inhibitor for multiple myeloma (Kis: Pim1 - 0.03 nM, Pim2 - 0.1 nM, Pim3 - 0.02 nM), well-tolerated.</p>Formula:C20H22F3N7OSColor and Shape:SolidMolecular weight:465.5VEGFR-2-IN-18
<p>VEGFR-2-IN-18 is a potent VEGFR-2 inhibitor with a 60 nM IC50, promoting cell apoptosis and anticancer effects.</p>Formula:C20H13ClN4O2Color and Shape:SolidMolecular weight:376.8JBIR-22
CAS:<p>JBIR-22 is a natural inhibitor for protein−protein interaction of the homodimer of proteasome assembly factor 3.</p>Formula:C23H33NO6Color and Shape:SolidMolecular weight:419.51Falecalcitriol
CAS:<p>Falecalcitriol is an analog of calcitriol. It has a higher potency both in vivo and in vitro systems, which is longer duration of action in vivo.</p>Formula:C27H38F6O3Purity:98%Color and Shape:SolidMolecular weight:524.58OMDM169
CAS:<p>OMDM169: potent/selective MAGL inhibitor, raises 2-AG, analgesic via cannabinoid receptors, IC50: 0.13-0.41μM in rat/COS-7, inactive at CB1/CB2.</p>Formula:C25H45NO5Purity:98%Color and Shape:SolidMolecular weight:439.63HDAC-IN-33
<p>HDAC-IN-33 inhibits HDAC1/2/6 (IC50: 24/46/47 nM), exhibits potent antitumor activity in vitro and in vivo, and activates antitumor immunity.</p>Formula:C21H25N3O3Color and Shape:SolidMolecular weight:367.44IDH1 Inhibitor 1
CAS:<p>Oral, brain-penetrant mutant IDH1 inhibitor targeting R132H/C with IC50: 0.021/0.045μM; 2.52μM for IDH1WT.</p>Formula:C20H18F4N6O2Purity:98%Color and Shape:SolidMolecular weight:450.39NDT-30805
<p>NDT-30805, a triazolopyridine, blocks IL-1β in PBMC (IC50: 0.013μM) & NLRP3 inflammasome, for inflammation research.</p>Formula:C23H22N6SColor and Shape:SolidMolecular weight:414.53BACE1-IN-2
CAS:<p>BACE1-IN-2 is a BACE1 inhibitor (IC50: 22 nM).</p>Formula:C19H15F4N5O2Purity:98%Color and Shape:SolidMolecular weight:421.35AFP-07 free acid
CAS:<p>AFP 07 free acid is a 7,7-difluoroprostacyclin derivative. It also acts as a selective and highly potent agonist for the IP receptor.</p>Formula:C22H30F2O5Purity:98%Color and Shape:SolidMolecular weight:412.47L 734217
CAS:<p>L 734217 is an antagonist of the fibrinogen receptor.</p>Formula:C18H31N3O4Purity:98%Color and Shape:SolidMolecular weight:353.46CDK1-IN-3
<p>CDK1-IN-3 is a selective inhibitor targeting CDK1 (36.8 nM), CDK2 (305.17 nM), CDK5 (369.37 nM); used in cancer research.</p>Formula:C28H25ClF3N5O2Color and Shape:SolidMolecular weight:555.98D1R antagonist 1
CAS:<p>Compound 12a (D1R antagonist 1) is a D1R antagonist that participates in both G-protein-coupled and β-arrestin-mediated signaling pathways [1].</p>Formula:C22H26BrNO4Purity:98%Color and Shape:SolidMolecular weight:448.35T-3861174
CAS:<p>T-3861174 is a prolyl tRNA synthetase (PRS) inhibitor, exhibiting significant in vitro anti-tumor activity with GCN2-ATF4 pathway activation.</p>Formula:C26H25FN6O2Color and Shape:SolidMolecular weight:472.51PD-1/PD-L1-IN-13
<p>PD-1/PD-L1-IN-13 is a potent immune checkpoint PD-1/PD-L1 inhibitor with an IC50 value of 10.2 nM for PD-1/PD- L1 interaction.PD-1/PD-L1-IN-13 promotes CD8+ T-</p>Formula:C36H34ClF2N3O9Color and Shape:SolidMolecular weight:726.12ABT 491 Hydrochloride
CAS:<p>ABT-491 hydrochloride is an active platelet activator receptor (PAF-R) antagonist with good selectivity and oral administration.</p>Formula:C28H23ClFN5O2Color and Shape:SolidMolecular weight:515.97Tilpisertib fosmecarbil
CAS:<p>Tilpisertib fosmecarbil is a potent inhibitor of serine/threonine kinases with anti-inflammatory properties.</p>Formula:C35H36ClN8O7PColor and Shape:SolidMolecular weight:747.14CD73-IN-13
<p>CD73-IN-13, a potent CD73 inhibitor, may be developed for tumor-related disease treatment.</p>Formula:C13H11F3N4O2Color and Shape:SolidMolecular weight:312.25HER2-IN-7
CAS:<p>HER2-IN-7 is a potent HER2 inhibitor with potential for researching ErbB-related diseases, especially cancer.</p>Formula:C28H26F3N7O3Color and Shape:SolidMolecular weight:565.55GSK340
<p>GSK340 is a BET inhibitor.</p>Formula:C26H31N3O2Color and Shape:SolidMolecular weight:417.55PF1070A
CAS:<p>PF1070A is a natural cyclic tetrapeptide HDAC Inhibitor through the inhibition of PfHDAC1 catalytic activity, potently inducing the synthesis of metallothionein</p>Formula:C31H44N4O6Color and Shape:SolidMolecular weight:568.7
