CymitQuimica logo
Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

Show 16 more subcategories

Found 66513 products of "Inhibitors"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • ChE/Aβ1-42-IN-1


    ChE/Aβ1-42-IN-1 (compound 28) is a potent aggregation inhibitor of ChE and Aβ 1-42 with excellent BBB permeability.
    Formula:C19H24N2O3
    Color and Shape:Solid
    Molecular weight:328.41

    Ref: TM-T60940

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Samuraciclib hydrochloride hydrate


    Samuraciclib (CT7001) is a potent oral CDK7 inhibitor (IC50: 41 nM) with anti-breast cancer properties.
    Formula:C22H35ClN6O3
    Color and Shape:Solid
    Molecular weight:521.7

    Ref: TM-T63650

    25mg
    938.00€
    50mg
    1,254.00€
    100mg
    1,890.00€
  • Rodatristat

    CAS:
    Rodatristat is an effective tryptophan hydroxylase 1 and TPH2 inhibitor (IC50s: 33 nM and 7 nM, respectively).
    Formula:C27H27ClF3N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:561.98

    Ref: TM-T16780

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • U 75875

    CAS:
    U 75875 is a protease inhibitor.
    Formula:C45H61N7O7
    Color and Shape:Solid
    Molecular weight:812.01

    Ref: TM-T34976

    25mg
    2,583.00€
    50mg
    3,402.00€
    100mg
    4,680.00€
  • GYKI-53784

    CAS:
    GYKI-53784 (LY 303070) is an effective selective AMPA receptor antagonist.
    Formula:C19H20N4O3
    Color and Shape:Solid
    Molecular weight:352.39

    Ref: TM-T32035

    5mg
    2,512.00€
    10mg
    3,412.00€
    25mg
    5,068.00€
    50mg
    6,839.00€
  • GENZ-882706

    CAS:
    GENZ-882706 is a potent colony stimulating factor-1 receptor (CSF-1R) Inhibitor.
    Formula:C26H25N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:455.51

    Ref: TM-T11390

    25mg
    2,808.00€
    50mg
    3,492.00€
    100mg
    4,500.00€
  • 5-HT1A antagonist 1


    Compound 6f is a potent, selective 5-HT1A receptor blocker (Ki: 35 nM), useful in CNS disorder research.
    Formula:C23H29ClN6O2
    Color and Shape:Solid
    Molecular weight:456.97

    Ref: TM-T62843

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • TTA-P1

    CAS:
    TTA-P1: potent T-type calcium channel inhibitor; impacts neuron firing, hormone secretion, cell growth; potential in absence epilepsy research.
    Formula:C19H27Cl2FN2O
    Color and Shape:Solid
    Molecular weight:389.33

    Ref: TM-T61747

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • ATX inhibitor 22


    ATX inhibitor 22 is a novel inhibitor of ATX (autotaxin) (IC50: 218.9 μM) that lacks inhibitory activity against LPAR1.
    Formula:C19H17Cl3F2N2O4S
    Color and Shape:Solid
    Molecular weight:513.77

    Ref: TM-T63564

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Antileishmanial agent-4


    Antileishmanial agent-4, a ribonucleoside analogue, functions as an antileishmanial agent [1].
    Formula:C17H18N4O4
    Color and Shape:Solid
    Molecular weight:342.35

    Ref: TM-T61100

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Resolvin E2

    CAS:
    RvE2, a bioactive lipid from the SPM family, is made from EPA and reduces inflammatory neutrophil infiltration and helps treat NAFLD and other diseases.
    Formula:C20H30O4
    Color and Shape:Solid
    Molecular weight:334.45

    Ref: TM-T35881

    10µg
    386.00€
    25µg
    892.00€
    50µg
    1,665.00€
    100µg
    2,935.00€
  • Rodatristat ethyl

    CAS:
    Rodatristat ethyl is an oral TPH1 inhibitor reducing 5-HT levels & lowering PAH at low doses.
    Formula:C29H31ClF3N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:590.04

    Ref: TM-T16779

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Tubulin polymerization-IN-3


    Tubulin polymerization-IN-3 is a potent inhibitor of microtubulin polymerization (IC50: 3.84 μM) and induces apoptosis in colon cancer cells.
    Formula:C20H20ClN5O3
    Color and Shape:Solid
    Molecular weight:413.86

    Ref: TM-T62121

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • K-14585

    CAS:
    K-14585 blocks PAR(2), reduces NFkappaB activity, and IL-8 response, but alone can boost IL-8.
    Formula:C51H56Cl2N8O4
    Color and Shape:Solid
    Molecular weight:915.95

    Ref: TM-T27708

    5mg
    3,931.00€
  • IDO1-IN-14


    IDO1-IN-14 is an IDO1 enzyme inhibitor with an IC50 of 396.9 nM and suppresses HeLa cell activity with an EC50 of 3393 nM.
    Formula:C18H12Cl2FN3O2
    Color and Shape:Solid
    Molecular weight:392.21

    Ref: TM-T61789

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • YM-355179

    CAS:
    YM-355179 is a novel, selective antagonist of CC chemokine receptor 3 with oral activity.
    Formula:C33H34FN4O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:617.64

    Ref: TM-T29181

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • AMPK Activator SC4

    CAS:
    SC4 is a potent, direct AMPK activator. SC4 preferentially activates α2 complexes and stimulates skeletal muscle glucose uptake.
    Formula:C26H18ClN3O4
    Color and Shape:Solid
    Molecular weight:471.89

    Ref: TM-T70862

    25mg
    2,178.00€
    50mg
    2,862.00€
    100mg
    3,870.00€
  • GNTI TFA

    CAS:
    GNTI TFA is a selective kappa opioid receptor antagonist.
    Formula:C31H31F6N5O7
    Color and Shape:Solid
    Molecular weight:699.60

    Ref: TM-T69818

    25mg
    2,178.00€
    50mg
    2,862.00€
    100mg
    3,870.00€
  • TP003

    CAS:

    TP003 is a novel non-selective GABAA receptor benzodiazepine site agonist with affinity for α1β2gam2, α2β3gam2, α3β3gam2, α5β2gam2, EC50 of 20.3, 10.6, 3.24, 5.

    Formula:C23H16F3N3O
    Purity:99.17%
    Color and Shape:Solid
    Molecular weight:407.39

    Ref: TM-T23466

    2mg
    39.00€
    5mg
    58.00€
    10mg
    96.00€
    25mg
    168.00€
    50mg
    251.00€
    100mg
    364.00€
  • USP7-IN-6

    CAS:
    USP7-IN-6 is a potent inhibitor of ubiquitin-specific protease 7 (USP7, IC50: 6.8 nM).
    Formula:C41H43N7O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:729.89

    Ref: TM-T13271

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • HSP90-IN-10


    HSP90-IN-10 is a potent HSP90 inhibitor, targeting HCC1954 cells (IC50: 6 μM) and inducing apoptosis, sparing normal cells.
    Formula:C30H26FN3O6
    Color and Shape:Solid
    Molecular weight:543.54

    Ref: TM-T63827

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • DDCPPB-Glu

    CAS:
    DDCPPB-Glu is a 6-5 fused ring heterocycle antifolate that shows antitumor activity.
    Formula:C22H27N5O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:441.48

    Ref: TM-T25296

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Tenellin

    CAS:
    Tenellin is a fungal metabolite that inhibits Mg2+-, Ca2+-, and Na+/K+-ATPase activities in erythrocytes. Tenellin is cytotoxic to Sf9 and Sf21 insect cells.
    Formula:C21H23NO5
    Color and Shape:Solid
    Molecular weight:369.41

    Ref: TM-T71806

    1mg
    883.00€
  • iNOS/PGE2-IN-1


    iNOS/PGE2-IN-1: iNOS/PGE2 inhibitor, reduces LPS-induced NO, low ulcer risk, anti-inflammatory.
    Formula:C26H22ClN3O4
    Color and Shape:Solid
    Molecular weight:475.92

    Ref: TM-T63104

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MI-1851

    CAS:
    MI-1851 is a potent peptidomimetic inhibitor. MI-1851could prevent proteolytic processing of the S protein from SARSCoV-2 by endogenous furin in HEK293 cells.
    Formula:C34H53N15O6
    Color and Shape:Solid
    Molecular weight:767.88

    Ref: TM-T69640

    25mg
    2,718.00€
    50mg
    3,582.00€
    100mg
    4,950.00€
  • PptT-IN-2


    PptT-IN-2 inhibits PptT enzyme crucial in tuberculosis, with 2.5 μM IC50, showing potential in TB research.
    Formula:C22H29N5O2
    Color and Shape:Solid
    Molecular weight:395.5

    Ref: TM-T61847

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • IACS-8779

    CAS:
    IACS-8779 is a potent STING agonist that efficiently stimulates interferon gene activity and exhibits strong systemic antitumor effects.
    Formula:C21H25N9O10P2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:689.55

    Ref: TM-T11595

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Teoprolol

    CAS:
    Teoprolol is a blocker of β-adrenergic receptor.
    Formula:C23H30N6O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:454.52

    Ref: TM-T13124

    25mg
    1,783.00€
    50mg
    2,440.00€
    100mg
    3,087.00€
  • AS2521780

    CAS:
    AS2521780 is an inhibitor of PKCθ (IC50: 0.48 nM).
    Formula:C30H41N7OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:547.76

    Ref: TM-T14328

    25mg
    2,718.00€
    50mg
    3,582.00€
    100mg
    4,950.00€
  • Mepixetil


    Mepixetil is a potent angiotensin II receptor antagonist[1].
    Formula:C12H18N2O3
    Color and Shape:Solid
    Molecular weight:238.28

    Ref: TM-T60329

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Complex III-IN-2


    Complex III-IN-2 inhibits complex III, with antifungal EC50: 29.31 mg/L vs R. solani, 29.98 mg/L vs S. sclerotiorum.
    Formula:C15H21ClN2O2S
    Color and Shape:Solid
    Molecular weight:328.86

    Ref: TM-T60949

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Carmegliptin dihydrochloride

    CAS:
    Carmegliptin dihydrochloride (RG-1579, RO4876904) is a salt of Camegliptin, a DPP-4 inhibitor for type 2 diabetes.
    Formula:C20H30Cl2FN3O3
    Color and Shape:Solid
    Molecular weight:450.38

    Ref: TM-T68652

    25mg
    2,178.00€
    50mg
    2,862.00€
    100mg
    3,870.00€
  • Sacibertinib

    CAS:
    Sacibertinib inhibits Trk, targeting EGFR-TK (EC50 110 nM) & HER2 (EC50 244 nM), with anticancer properties.
    Formula:C32H31ClN6O4
    Color and Shape:Solid
    Molecular weight:599.08

    Ref: TM-T64225

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • CBP/p300-IN-16


    CBP/p300-IN-16 (compound 1) is a potent inhibitor of EP300/CBP HAT, acting on HAT EP300 (IC50: 0.61 μM) and LK2 H3K27 (IC50: 2.24 μM).
    Formula:C26H31N3O4
    Color and Shape:Solid
    Molecular weight:449.54

    Ref: TM-T62700

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Suloctidil HCl

    CAS:
    Suloctidil HCl is a peripheral vascular dilator.
    Formula:C20H36ClNOS
    Color and Shape:Solid
    Molecular weight:374.02

    Ref: TM-T0712L

    25mg
    1,998.00€
    50mg
    2,412.00€
    100mg
    2,880.00€
  • Pan-Trk-IN-3


    Pan-Trk-IN-3: potent Trk inhibitor (IC50: 2-26 nM), effective against drug-resistant mutants, induces apoptosis, anti-tumor effects.
    Formula:C29H31ClN8O3
    Color and Shape:Solid
    Molecular weight:575.06

    Ref: TM-T64070

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SSTR5 antagonist 2 TFA

    CAS:
    Potent, oral SSTR5 antagonist 2 TFA may treat type 2 diabetes.
    Formula:C34H36F4N2O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:660.65

    Ref: TM-T13022L

    25mg
    1,639.00€
    50mg
    2,142.00€
    100mg
    2,790.00€
  • Antimalarial agent 2


    Antimalarial agent 2 is an orally active, novel antimalarial agent that exhibits rapid in vitro killing effects.
    Formula:C27H25N3O5
    Color and Shape:Solid
    Molecular weight:471.5

    Ref: TM-T63043

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • J-104118

    CAS:
    J-104118 potentially inhibits squalene synthase.
    Formula:C28H26Cl2FNO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:546.41

    Ref: TM-T27646

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Tubulin polymerization-IN-8

    CAS:
    Compound IIc inhibits tubulin polymerization, arrests cell cycle at G2/M in HCT116 cells, IC50 12.7 μM, potential for cancer research.
    Formula:C21H24N4O4S
    Color and Shape:Solid
    Molecular weight:428.5

    Ref: TM-T62349

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Azaphilone-9

    CAS:
    AZA-9 inhibits cancer growth by blocking HuR-ARE RNA binding; IC50=1.2μM.
    Formula:C21H23BrO5
    Color and Shape:Solid
    Molecular weight:435.31

    Ref: TM-T72920

    25mg
    2,583.00€
    50mg
    3,402.00€
    100mg
    4,680.00€
  • α5β1 integrin agonist-1

    CAS:
    α5β1 integrin agonist-1 is an α5β1 integrin agonist that selectively delivers 5-FU to tumour cells and induces tumour cell death.
    Formula:C24H26FN5O9
    Color and Shape:Solid
    Molecular weight:547.49

    Ref: TM-T63868

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • RIP1 kinase inhibitor 1

    CAS:
    RIP1 kinase inhibitor 1 is an orally available and brain-penetrating inhibitor of RIP1 kinase with pKi of 9.04.
    Formula:C24H20ClN5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:461.9

    Ref: TM-T12725

    25mg
    1,080.00€
    50mg
    1,414.00€
    100mg
    2,152.00€
  • BMS-986034

    CAS:
    BMS-986034 is a GPR119 agonist.
    Formula:C24H24Cl2N6O4
    Color and Shape:Solid
    Molecular weight:531.39

    Ref: TM-T70550

    25mg
    2,043.00€
    50mg
    2,682.00€
    100mg
    3,600.00€
  • Antitumor agent-78


    Antitumor agent-78 blocks GPx-4, raises COX2, triggers apoptosis, halts EMT, and stifles cancer cell growth and migration.
    Color and Shape:Soild

    Ref: TM-T63768

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Lp-PLA2-IN-6

    CAS:
    Lp-PLA2-IN-6: Potent tetracyclic inhibitor of rhLp-PLA2, with pIC50 of 10.0, and potential in neurodegenerative research.
    Formula:C25H21F5N4O3
    Color and Shape:Solid
    Molecular weight:520.45

    Ref: TM-T63633

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • GLS1 Inhibitor-5


    GLS1 Inhibitor-5 (24y): Selective, oral glutaminase 1 inhibitor; IC50 68 nM; induces apoptosis; anti-tumor.
    Color and Shape:Solid

    Ref: TM-T64259

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • NBTIs-IN-4


    NBTIs-IN-4, a broad-spectrum Gram-positive antibacterial, inhibits DNA rotamases/topoisomerase IV, with low resistance.
    Formula:C22H24FN5O5S
    Color and Shape:Solid
    Molecular weight:489.52

    Ref: TM-T63275

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BM635 hydrochloride


    BM635 hydrochloride, an MmpL3 inhibitor, strongly blocks Divergent bacteriophage H37Rv (MIC50: 0.08 μM), with doubled in vivo potency.
    Formula:C25H30ClFN2O
    Color and Shape:Solid
    Molecular weight:428.97

    Ref: TM-T62358

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Adafosbuvir

    CAS:
    Adafosbuvir has antiviral activity.
    Formula:C22H29FN3O10P
    Color and Shape:Solid
    Molecular weight:545.457

    Ref: TM-T26560

    25mg
    1,773.00€
    50mg
    2,322.00€
    100mg
    3,060.00€
  • LX2761

    CAS:
    LX2761 is a stable inhibitor for SGLT1/2 with IC50s of 2.2/2.7 nM; it targets SGLT1 in the GI tract.
    Formula:C32H47N3O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:601.80

    Ref: TM-T15797

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • LSD1/2-IN-3


    LSD1/2-IN-3 selectively inhibits LSD1 (Ki 11 nM) over LSD2 (Ki 7 μM), and hinders tumor stem cell proliferation.
    Formula:C9H8BrF2N
    Color and Shape:Solid
    Molecular weight:248.07

    Ref: TM-T60360

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GABAA receptor agonist 1


    Compound 3e, a potent GABAA agonist, targets GABA sites and has potential anti-depressive effects in mice.
    Formula:C20H30O3
    Color and Shape:Solid
    Molecular weight:318.45

    Ref: TM-T60842

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • L-690330 hydrate


    L-690330 hydrate inhibits IMPase; Ki: 0.30 μM (human), 0.42 μM (bovine cortex); 0.27 μM (recom. human), 0.19 μM (bovine).
    Formula:C8H14O9P2
    Color and Shape:Solid
    Molecular weight:316.14

    Ref: TM-T60820

    100mg
    1,296.00€
  • FGFR-IN-6

    CAS:
    FGFR-IN-6 (Compound 5) is an FGFR inhibitor.
    Formula:C23H22N6O3
    Color and Shape:Solid
    Molecular weight:430.46

    Ref: TM-T62391

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • SGLT inhibitor-1

    CAS:
    SGLT inhibitor-1 is a potentsodium glucose co-transporter proteins (SGLTs) dual inhibitor(hSGLT1 and hSGLT2 with IC50s of 43 nM and 9 nM, respectively).
    Formula:C24H27FO8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:462.46

    Ref: TM-T12893

    25mg
    2,313.00€
    50mg
    3,042.00€
    100mg
    4,140.00€
  • Antibiotic MA 144M1

    CAS:
    Antibiotic MA 144M1, an anthracycline, targets gram-positive bacteria and animal tumors; derived from Streptomyces fermentation or aclacinomycin A conversion.
    Formula:C42H55NO15
    Color and Shape:Solid
    Molecular weight:813.88

    Ref: TM-T68946

    25mg
    8,388.00€
    50mg
    11,142.00€
    100mg
    16,290.00€
  • WS-898


    WS-898 boosts paclitaxel efficacy in resistant cells by inhibiting ABCB1; IC50: SW620/Ad300 - 5.0 nM, KB-C2 - 3.67 nM, HEK293/ABCB1 - 3.68 nM.
    Formula:C33H25N7OS
    Color and Shape:Solid
    Molecular weight:567.66

    Ref: TM-T64016

    25mg
    1,269.00€
    50mg
    1,659.00€
    100mg
    2,490.00€
  • Methyl 5-thia-6,8,11,14-eicosatetraenoate

    CAS:
    Methyl 5-thia-6,8,11,14-eicosatetraenoate is a bioactive chemical.
    Formula:C20H32O2S
    Color and Shape:Solid
    Molecular weight:336.53

    Ref: TM-T33332

    25mg
    1,908.00€
    50mg
    2,502.00€
    100mg
    3,330.00€
  • PDHK-IN-3


    PDHK-IN-3 (compound 7) is a potent inhibitor of pyruvate dehydrogenase kinase(PDHK) with IC50s of 0.21 and 1.54 μM for PDHK2 and PDHK4, respectively [1].
    Formula:C17H16N2O2
    Color and Shape:Solid
    Molecular weight:280.32

    Ref: TM-T60527

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AZ14145845


    AZ14145845 is an in vivo potent and highly selective type I1/2 Mer/Axl bispecific kinase inhibitor.
    Formula:C32H35N9O
    Color and Shape:Solid
    Molecular weight:561.68

    Ref: TM-T63968

    25mg
    1,054.00€
    50mg
    1,378.00€
    100mg
    2,197.00€
  • HDAC6-IN-12


    HDAC6-IN-12 is a potent inhibitor of HDAC6 that binds in the DNA chain, causing DNA damage and exhibiting anticancer effects that can be used in cancer research
    Formula:C24H39F2N3O5
    Color and Shape:Solid
    Molecular weight:487.58

    Ref: TM-T63247

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • KRAS G12D inhibitor 3

    CAS:
    KRAS G12D Inhibitor 3, a compound targeting the KRAS G12D mutation, demonstrates potent antitumor efficacy with an inhibitory concentration (IC50) of less than
    Formula:C34H31ClF3N5O2
    Color and Shape:Solid
    Molecular weight:634.09

    Ref: TM-T72394

    25mg
    2,988.00€
    50mg
    3,943.00€
    100mg
    5,490.00€
  • MEIS-IN-1

    CAS:
    MEIS-IN-1 is a potent MEIS inhibitor that induces the expansion of hematopoietic stem cells in mice and humans.
    Formula:C24H21F3N2O4
    Color and Shape:Solid
    Molecular weight:458.43

    Ref: TM-T62859

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GSD-11


    GSD-11: Potent, selective anti-austerity agent; blocks Akt/mTOR pathway, hinders PANC-1 cell migration & colony growth. Promising for pancreatic cancer study.
    Formula:C20H28O2
    Color and Shape:Solid
    Molecular weight:300.44

    Ref: TM-T60672

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LY503430

    CAS:
    LY503430: Oral AMPA enhancer with nootropic, neuroprotective properties, mitigates 6-OHDA/MPTP brain damage.
    Formula:C20H25FN2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:392.49

    Ref: TM-T27959

    25mg
    2,853.00€
    50mg
    3,763.00€
    100mg
    5,220.00€
  • Anti-Influenza agent 3


    Compound 11h: Potent, low-toxicity anti-influenza, inhibits M2 ion channels. EC50: 3.29μM (H3N2), 2.45μM (H1N1).
    Formula:C16H22ClNOS
    Color and Shape:Solid
    Molecular weight:311.87

    Ref: TM-T60778

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • XR8-69


    XR8-69 is a SARS-CoV-2 PLpro inhibitor. XR8-69 has a low micromolar antiviral effect in SARS-CoV-2 infected human cells.
    Formula:C26H30N4O2S
    Color and Shape:Solid
    Molecular weight:462.61

    Ref: TM-T62928

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • DNA-PK-IN-9


    DNA-PK-IN-9 (YK6) is a potent DNA-PK inhibitor with an IC50 of 10.47 nM, important in cancer research.
    Formula:C21H21N5O2
    Color and Shape:Solid
    Molecular weight:375.42

    Ref: TM-T61533

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • O-GlcNAcase-IN-1


    O-GlcNAcase-IN-1 is a potent and novel inhibitor of O-GlcNAcase(OGA) with an IC 50 value of 46 nM.
    Formula:C15H22N6
    Color and Shape:Solid
    Molecular weight:286.38

    Ref: TM-T60571

    2mg
    63.00€
  • Oral antiplatelet agent 1

    CAS:
    Oral antiplatelet agent 1 is a potent antiplatelet agent with an IC50 of 2.94 μM in vitro.
    Formula:C23H24N4O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:468.53

    Ref: TM-T12316

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Org-31710

    CAS:
    Org-31710 is a progesterone receptor antagonist potentially for contraception.
    Formula:C30H39NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:445.64

    Ref: TM-T28263

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • (E)-10-Hydroxynortriptyline maleate

    CAS:
    (E)-10-Hydroxy Nortriptyline maleate, a derivative of antidepressant Nortriptyline, eases depression symptoms.
    Formula:C23H25NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:395.455

    Ref: TM-T11135

    25mg
    1,639.00€
    50mg
    2,142.00€
    100mg
    2,790.00€
  • hMAO-B/MB-COMT-IN-2


    Dual inhibitor hMAO-B/MB-COMT-IN-2 targets hMAO-B (IC50: 4.27μM) & MB-COMT (IC50: 2.69μM), aids in neurodegenerative research.
    Formula:C17H18N2O3
    Color and Shape:Solid
    Molecular weight:298.34

    Ref: TM-T60658

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CVS-1578

    CAS:
    CVS-1578 is a potent serine protease inhibitor, targeting the S2S3 thrombin and FXa subsites.
    Formula:C20H30N6O5S
    Color and Shape:Solid
    Molecular weight:466.55

    Ref: TM-T70110

    25mg
    2,313.00€
    50mg
    3,042.00€
    100mg
    4,140.00€
  • 4,5'-Dimethylangelicin-NHS


    NHS-modified coumarin, 4,5'-Dimethylangelicin-NHS, shows photochemical activity & photosensitivity.
    Formula:C21H19NO7S
    Color and Shape:Solid
    Molecular weight:429.44

    Ref: TM-T62365

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PI3Kβ-IN-1

    CAS:
    PI3Kβ-IN-1 is a selective, orally active PI3Kβ inhibitor (IC50: 2 nM).
    Formula:C25H14F2N8
    Color and Shape:Solid
    Molecular weight:464.43

    Ref: TM-T62948

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Antibacterial agent 78


    Antibacterial agent 78 (compound 30) is an antibacterial agent with improved cytotoxicity profile[1].
    Formula:C16H23N3S2
    Color and Shape:Solid
    Molecular weight:321.5

    Ref: TM-T60865

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PROTAC CDK12/13 Degrader-1


    PROTAC CDK12/13 Degrader-1 (7f) selectively degrades CDK12/13 at nanomolar potency, targeting breast cancer.
    Color and Shape:Solid

    Ref: TM-T64284

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Glucosylceramide synthase-IN-3


    Glucosylceramide synthase-IN-3 (BZ1) is a potent, brain-accessible, oral GCS inhibitor with a 16 nM IC50, relevant for Gaucher's disease study.
    Formula:C21H20FN3O3
    Color and Shape:Solid
    Molecular weight:381.4

    Ref: TM-T61632

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Sekdel sequence

    CAS:
    Sekdel sequence, as a signal, leads to retention of at least two proteins in the endoplasmic reticulum of animal cells.
    Formula:C29H49N7O14
    Color and Shape:Solid
    Molecular weight:719.74

    Ref: TM-T34601

    25mg
    2,043.00€
    50mg
    2,682.00€
    100mg
    3,600.00€
  • Dazucorilant

    CAS:
    Dazucorilant (CORT113176), a selective non-steroidal GR modulator, has high affinity with a K i <1 nM, useful for neurological research.
    Formula:C29H22F4N4O3S
    Color and Shape:Solid
    Molecular weight:582.57

    Ref: TM-T38983

    25mg
    4,834.00€
  • ARG1-IN-1

    CAS:
    ARG1-IN-1 is a human arginase 1 inhibitor with an IC 50 of 29 nM.
    Formula:C11H21BN2O4
    Color and Shape:Solid
    Molecular weight:256.11

    Ref: TM-T39932

    5mg
    6,353.00€
  • FLT3/TrKA-IN-1


    FLT3/TrKA-IN-1: Potent dual kinase inhibitor for FLT3 & TrKA, promising for AML research.
    Formula:C28H30N4O2
    Color and Shape:Solid
    Molecular weight:454.56

    Ref: TM-T62801

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • L 668411

    CAS:
    L 668411, the 2,3-ditritiated methyl ester of L 659699, inhibits HMG-CoA synthase.
    Formula:C19H30O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:338.44

    Ref: TM-T24320

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • FTO-IN-6

    CAS:
    FTO-IN-6 is a selective inhibitor of fat mass and obesity associated protein (FTO).
    Formula:C14H12N4O6
    Color and Shape:Solid
    Molecular weight:332.27

    Ref: TM-T60994

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • DNA crosslinker 2 dihydrochloride

    CAS:
    Potent DNA crosslinker 2 binds minor groove, increases Tm by 1.2°C, and inhibits NCI-H460, A2780, MCF-7 cancer cells.
    Formula:C15H22Cl2N8O
    Color and Shape:Solid
    Molecular weight:401.29

    Ref: TM-T74338

    25mg
    1,773.00€
    50mg
    2,322.00€
    100mg
    3,060.00€
  • Antibacterial agent 110


    Compound 4e, an antibacterial against P. aeruginosa, disrupts cell membranes (MIC: 1 μg/ml).
    Formula:C22H21N5O4S
    Color and Shape:Solid
    Molecular weight:451.5

    Ref: TM-T62740

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AAK1-IN-2 TFA


    AAK1-IN-2 TFA (compound (S)-31) is a selective and potent AAK1 inhibitor (IC50: 5.8 nM) that can cross the blood-brain barrier.
    Formula:C24H22F6N4O4
    Color and Shape:Solid
    Molecular weight:544.45

    Ref: TM-T63833

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • HBV-IN-19 TFA

    CAS:
    HBV-IN19 TFA suppresses HBsAg, hampers HBV infection, and aids in HBV research.
    Formula:C26H31F3N2O8
    Color and Shape:Solid
    Molecular weight:556.53

    Ref: TM-T63937

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • AChE-IN-10


    AChE-IN-10 (24r) inhibits AChE (IC50=2.4 nM), reducing amyloid buildup, tau phosphorylation, and promotes neuron health.
    Formula:C23H27F2NO4S
    Color and Shape:Solid
    Molecular weight:451.53

    Ref: TM-T62743

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ONO-8809

    CAS:
    ONO-8809: Thromboxane A2 antagonist, reduces airway hyperresponse, macrophage accumulation, and MMP-9 in SHRSP brains.
    Formula:C30H46BrNO4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:596.66

    Ref: TM-T28251

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • hCAIX/XII-IN-5


    Coumarin 9a: Selective inhibitor of hCA IX/XII (Ki 93.3/85.7 nM), blocks cancer cell growth, and induces apoptosis.
    Formula:C18H13NO3
    Color and Shape:Solid
    Molecular weight:291.3

    Ref: TM-T60602

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CB2 receptor antagonist 1

    CAS:
    Compound 29 is a potent, CB2-selective antagonist/reverse agonist. Derivatives 23 & 24 offer antinociception; 24 activates cannabinoid/TRPV1 receptors.
    Formula:C28H47NO3
    Color and Shape:Solid
    Molecular weight:445.68

    Ref: TM-T62631

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MAP3K14-IN-173

    CAS:
    MAP3K14-IN-173 is a potent MAP3K14 kinase inhibitor.
    Formula:C29H31N7O2
    Color and Shape:Solid
    Molecular weight:509.60

    Ref: TM-T69894

    25mg
    2,583.00€
    50mg
    3,402.00€
    100mg
    4,680.00€
  • LAF-153

    CAS:
    LAF-153 is a reversible Methionine Aminopeptidase‑2 (MetAP-2) Inhibitor.
    Formula:C18H32N2O7
    Color and Shape:Solid
    Molecular weight:388.46

    Ref: TM-T68911

    25mg
    3,258.00€
    50mg
    4,303.00€
    100mg
    6,030.00€
  • 5(S),6(R)-DiHETE

    CAS:
    5(S),6(R)-DiHETE is a dihydroxy fatty acid from LTA4 hydrolysis and weak LTD4 agonist with ED50 of 1.3 μM for guinea pig ileum contraction.
    Formula:C20H32O4
    Color and Shape:Solid
    Molecular weight:336.47

    Ref: TM-T37652

    25mg
    2,313.00€
    50mg
    3,042.00€
    100mg
    4,140.00€
  • Annonin VI

    CAS:
    Annonin VI is a natural inhibitor of NADH:ubiquinone oxidoreductase.
    Formula:C37H66O7
    Color and Shape:Solid
    Molecular weight:622.92

    Ref: TM-T71047

    25mg
    4,609.00€
    50mg
    6,103.00€
    100mg
    8,730.00€
  • SARS 3CLpro-IN-1

    CAS:
    SARS 3CLpro-IN-1: stereospecific SARS 3CL protease inhibitor, octahydroisochromene class, IC50 = 95 μM.
    Formula:C22H38N4O2
    Color and Shape:Solid
    Molecular weight:390.56

    Ref: TM-T61774

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LSD1-IN-16


    LSD1-IN-16 (4b) inhibits LSD1, MAO-A/B; IC50: 0.015-0.366 μM. Halts prostate cancer cell growth; IC50: 15.2 μM.
    Formula:C20H18N2OS
    Color and Shape:Solid
    Molecular weight:334.43

    Ref: TM-T61021

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€