Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,833 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,875 products)
- Chromatin/Epigenetics(2,613 products)
- Cytoskeletal Signaling(1,567 products)
- DNA Damage/DNA Repair(2,872 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,019 products)
- Immunology and Inflammation(3,904 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,257 products)
- Membrane Transporter/Ion Channel(3,155 products)
- Metabolism(10,137 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,446 products)
- Other Inhibitors(35,847 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,429 products)
- Proteases/Proteasome(1,691 products)
- Stem Cell and Derivatives(732 products)
- Tyrosine Kinase/Adaptors(1,982 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66515 products of "Inhibitors"
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Ascofuranone
CAS:Ascofuranone is an inhibitor of the ubiquinol oxidase activity of Trypanosoma brucei mitochondrial alternative oxidase (TAO), as well as an inhibitor of HsDHODHFormula:C23H29ClO5Color and Shape:SolidMolecular weight:420.93SB 224289
CAS:SB 224289: selective 5-HT1B antagonist, pKi 8.2, 60x selectivity, effective orally.Formula:C32H32N4O3Purity:98%Color and Shape:SolidMolecular weight:520.62Cdc7-IN-10
CAS:Cdc7-IN-10 is a potent inhibitor of Cdc7 (IC50 ≤ 1 nM) and can be used in studies of proliferative diseases.Formula:C20H22F2N4O2SColor and Shape:SolidMolecular weight:420.48Thiomuscimol hydrobromide
CAS:Thiomuscimol hydrobromide is an agonist of GABAA receptor.Formula:C4H6N2OSPurity:98%Color and Shape:SolidMolecular weight:130.17Iloprost
CAS:Iloprost (Ciloprost) is an inhibitor of platelet aggregation and vasodilatation used in the study of cardiovascular disease.Formula:C22H32O4Color and Shape:Colorless OilMolecular weight:360.49SP-471
SP-471 is a potent inhibitor of dengue virus (DENV) protease (IC50: 18 μM) and inhibits the inter- and intramolecular protease processes of DENV.Formula:C33H26BrN5Color and Shape:SolidMolecular weight:572.5MEIS-IN-3
MEIS-IN-3 is a potent inhibitor of MEIS.Formula:C25H26N2O4Color and Shape:SolidMolecular weight:418.48AAK1-IN-3 TFA
AAK1-IN-3 TFA, an AAK1 inhibitor with IC50 of 11 nM, crosses the blood-brain barrier, is a quinoline analogue, and may aid neuropathic pain research.Formula:C24H22F6N4O4Color and Shape:SolidMolecular weight:544.45FAK-IN-3
FAK-IN-3 inhibits FAK, reduces PA-1 cell migration/invasion, and tumor growth, with no major side effects.Formula:C28H28N6O4Color and Shape:SolidMolecular weight:512.56LAS195319
CAS:LAS195319 is a potent and selective inhaled PI3Kδ Inhibitor (IC50 = 0.5 nM) for the Treatment of Respiratory Diseases.Formula:C29H26N10O3SColor and Shape:SolidMolecular weight:594.65VGD071
CAS:VGD071, a compound that targets sortilin, presents a promising avenue for forthcoming research utilizing mouse models of breast cancer.Formula:C32H41N3O4S2Color and Shape:SolidMolecular weight:595.82BRD0418
CAS:BRD0418 acts as an upregulator of TRIB1 expression by leading to reprogramming of hepatic lipoprotein metabolism from adipogenesis to clearance it.Formula:C29H32N2O5Purity:99.57%Color and Shape:SolidMolecular weight:488.57Org-6906
CAS:DCB-3503, a tylophorine analog, may treat cancer and suppress immunity by blocking protein synthesis and modulating HSC70's ATPase activity.Formula:C13H16ClNPurity:98%Color and Shape:SolidMolecular weight:221.73Pociredir
CAS:Pociredir (FTX-6058), a potent EED inhibitor (KD=0.163 nM), may help in SCD research.Formula:C22H18FN5O2Color and Shape:SolidMolecular weight:403.41Human enteropeptidase-IN-2
Human enteropeptidase-IN-2 is a potent inhibitor of enteropeptidase (enteropeptidase) and can be used in anti-obesity studies.Formula:C20H19F3N4O7Color and Shape:SolidMolecular weight:484.38SARS-CoV-2-IN-23
SARS-CoV-2-IN-23 (compound GRL-0617) is an inhibitor of SARS-COV-2 papain-like protease (PLpro) (IC 50 = 2.3 μM) [1].Formula:C21H22N2OColor and Shape:SolidMolecular weight:318.41FXIa-IN-10
FXIa-IN-10 is a potent, orally bioavailable inhibitor of Activator XI (FXIa) (Ki: 0.17 nM).Formula:C23H18Cl2F3N9O2Color and Shape:SolidMolecular weight:580.35CVT-5440
CAS:CVT-5440 is a selective, high-affinity (2B) adenosine receptor antagonist with good selectivity.Formula:C27H28N6O5Color and Shape:SolidMolecular weight:516.55NRX-2663
CAS:NRX-2663 boosts β-catenin binding to E3 ligase SCFβ-TrCP (Kd: 54.8 nM, EC50: 22.9 nM).Formula:C20H13F3N2O5Color and Shape:SolidMolecular weight:418.32Anticancer agent 62
CAS:Anticancer agent 62 inhibits HepG2, Bel-7402, MCF-7 growth with IC50: 0.019, 0.060, 0.016 μM respectively, and halts tumors.Formula:C20H19ClN3Na2O8PSColor and Shape:SolidMolecular weight:573.85GL0388
GL0388, a Bax activator, induces apoptosis, hinders breast cancer growth, and has IC50 of 0.299-1.57 μM.Formula:C21H17FN2OColor and Shape:SolidMolecular weight:332.37Pelecopan
CAS:Pelecopan (BCX9930), an oral complement factor D inhibitor, prevents hemolysis in PNH (IC50=14.3 nM).Formula:C23H19FN2O4Color and Shape:SolidMolecular weight:406.41HR-546
CAS:HR-546 is a prostaglandin E2 and prostaglandin F2alpha antagonist.Formula:C26H44O6Color and Shape:SolidMolecular weight:452.62OUN58101
CAS:OUN58101, also MDK-8101/BI-D, is an RSV L-protein inhibitor with no formal name, first reported in patent WO 2005042530.Formula:C32H36N6O6Color and Shape:SolidMolecular weight:600.66THR-β agonist 5
CAS:THR-β agonist 5 (compound 54) is a potent THR-β agonist, with an EC 50 of <50 nM [1].Formula:C22H23N5O2Color and Shape:SolidMolecular weight:389.45SH498
CAS:SH498 is a novel Bmi-1-mediated anti-tumor agent with significant anti-proliferative effects.Formula:C27H25F3N2O4Color and Shape:SolidMolecular weight:498.49Mf 268
CAS:Mf 268 is a pseudo-reversible carbamate-type inhibitor which interacts with the catalytic and regulatory anionic site of the enzyme.Formula:C28H46N4O3Color and Shape:SolidMolecular weight:486.69RXR antagonist 1
RXR antagonist 1 is a Retinoid X Receptor (RXR) modulator that exhibits high RXR antagonism (pA2: 8.06). RXR antagonist 1 can be used to study type 2 diabetes.Formula:C28H33F3N2O3Color and Shape:SolidMolecular weight:502.57TD-0212
CAS:TD-0212: Oral dual antagonist for AT1 (pKi 8.9) & NEP inhibitor (pIC50 9.2).Formula:C28H34FN3O4SPurity:98%Color and Shape:SolidMolecular weight:527.65Anti-inflammatory agent 13
Pentacyclic triterpene, Anti-inflammatory 13 inhibits DAMP/PAMP inflammation models.Formula:C30H48O4Color and Shape:SolidMolecular weight:472.7PD-149163
CAS:PD-149163: brain-penetrating, selective NTR1 agonist; shows pro-cognitive, anti-psychotic, anxiolytic effects.Formula:C42H71N9O6Color and Shape:SolidMolecular weight:798.07DC41SMe
CAS:DC41SMe, a DC1 derivative and CC-1065 analogue, targets cancer with 18-25 pM IC50 against Ramos, Namalwa, HL60/s cells.Formula:C38H36ClN5O4S2Purity:98%Color and Shape:SolidMolecular weight:726.31SHR0687
CAS:SHR0687: potent KOR agonist, selective, favorable PK, effective in rat pain model, minimal BBB penetration, less CNS side effects.Formula:C39H60N8O5Color and Shape:SolidMolecular weight:720.94PGDM
CAS:PGD2 is involved in allergy, asthma, sleep, temperature regulation, inhibits clotting, and relaxes blood vessels; PGDM, its metabolite, is a biomarker.Formula:C16H24O7Color and Shape:SolidMolecular weight:328.36FPR2 agonist 2
Potent FPR2 agonist, crosses blood-brain barrier, EC50: 0.13 nM; reduces inflammation and mitochondrial dysfunction, inhibits caspase-3.Formula:C25H20F2N4O2Color and Shape:SolidMolecular weight:446.45Topoisomerase I/II inhibitor 4
Topoisomerase I/II inhibitor 4 halts cell growth and spread, induces apoptosis, and is used in liver cancer research.Formula:C27H21N5O6Color and Shape:SolidMolecular weight:511.49HER2-IN-8
CAS:HER2-IN-8 is an inhibitor of HER-2 that can be used in the study of cancer and inflammation-related diseases.Formula:C26H25F2N9O3Color and Shape:SolidMolecular weight:549.53MDL-27088
CAS:MDL-27088 is an angiotensin-covering enzyme inhibitor.Formula:C25H28N2O5Color and Shape:SolidMolecular weight:436.50Sapintoxin D
CAS:Sapintoxin D is a fluorescent phorbol ester and selective activator of protein kinase C.Formula:C30H37NO8Color and Shape:SolidMolecular weight:539.62Dual FAAH/sEH-IN-1
CAS:Dual FAAH/sEH-IN-1 inhibits both sEH (IC50: 9.6 nM) and FAAH (IC50: 7 nM), offering potent anti-inflammatory effects.
Formula:C25H22ClN3O3S2Purity:99.89%Color and Shape:SolidMolecular weight:512.04Pocenbrodib
CAS:Pocenbrodib (FT-7051) is a potent inhibitor of the bromodomain of the CBP/p300 family with potential antitumour activity and is palatable for cancer research.Formula:C28H32FN3O6Purity:98.48% - 99.54%Color and Shape:SolidMolecular weight:525.57AZD 3147
CAS:AZD 3147 inhibits mTORC1 (40.7 nM), mTORC2 (5.75 nM), and PI3Kα/β/δ/γ (912/5495/9333/6310 nM IC50s).
Formula:C24H31N5O4S2Purity:99.99%Color and Shape:SolidMolecular weight:517.66NDI-034858
CAS:NDI-034858 (TAK-279) is a tyrosine kinase 2 (TYK2) inhibitor (Kd<200 pM) that targets the JH2 structural domain of Tyk2 for the treatment of autoimmune diseasesFormula:C23H24N8O3Purity:>99.99%Color and Shape:SolidMolecular weight:460.49Suzetrigine
CAS:Suzetrigine (VX-548) is an oral NaV1.8 inhibitor with analgesic properties for acute pain research.Formula:C21H20F5N3O4Purity:98.08% - 99.27%Color and Shape:SolidMolecular weight:473.39Ref: TM-T69552
1mg55.00€5mg108.00€10mg161.00€25mg253.00€300g129,112.00€50mg434.00€100mg707.00€200mg973.00€1mL*10mM (DMSO)112.00€Eravacycline dihydrochloride
CAS:Eravacycline dihydrochloride (TP-434-046) is a potent and broad-spectrum antibacterial agent against six E. coli (MICs: 0.125-0.25 mg/L).Formula:C27H33Cl2FN4O8Purity:95% - 99.68%Color and Shape:SolidMolecular weight:631.48MAO-B-IN-17
CAS:MAO-B-IN-17 is a selective and potent monoamine oxidase B (MAO-B) inhibitor (IC50: 5.08 μM) for the study of central nervous system disorders like Parkinson's.Formula:C17H17F2NO2Purity:99.41%Color and Shape:SoildMolecular weight:305.32GLPG0974
CAS:GLPG0974 is an antagonist of FFA2/GPR43 with IC50 of 9 nM.Formula:C25H25ClN2O4SPurity:99.8%Color and Shape:SolidMolecular weight:484.99PREP inhibitor-1
CAS:PREP inhibitor-1 is a prolyl oligopeptidase (PREP) inhibitor for the study of Alzheimer's disease.Formula:C22H28N4O2Purity:98.78%Color and Shape:SoildMolecular weight:380.48Gepotidacin mesylate dihydrate
CAS:Gepotidacin mesylate dihydrate (GSK2140944 mesylate dihydrate) is an antibiotic and an inhibitor of bacterial type II topoisomerase.Formula:C25H36N6O8SPurity:99.85%Color and Shape:SolidMolecular weight:580.65BMS453
CAS:BMS453 (BMS-189453), a synthetic retinoid, is a potent and selective agonist of RARβ and a potent testicular toxin.Formula:C27H24O2Purity:99.93%Color and Shape:SolidMolecular weight:380.48BMS-986141
CAS:BMS-986141(UDM-003183) is a selective and potent protease-activated receptor-4 (PAR-4) antagonist with oral activity and an IC50 value of 0.4 nM.BMS-98614Formula:C27H23N5O5S2Purity:98.43% - 99.26%Color and Shape:SolidMolecular weight:561.63MIV-247
CAS:MIV-247 is a cathepsin S inhibitor that attenuates mechanically abnormal pain in preclinical neuropathic pain models and can be used to study myocardial injury.Formula:C17H24F3N3O4Purity:99.27%Color and Shape:SolidMolecular weight:391.39Vofopitant dihydrochloride
CAS:Vofopitant dihydrochloride (GR 205171A) is a tachykinin NK1 receptor antagonist and a potential compound for the treatment of pathologic vomiting.Formula:C21H25Cl2F3N6OPurity:98.99%Color and Shape:SolidMolecular weight:505.36Ref: TM-T13329L
1mg94.00€5mg222.00€10mg356.00€25mg675.00€50mg1,009.00€100mg1,378.00€500mg2,673.00€1mL*10mM (DMSO)248.00€Treprostinil diethanolamine
CAS:Treprostinil diethanolamine (UT-15C) is a potent agonist of EP2, DP1 and IP, with values of 3.6, 4.4, 32.1, 212, 826, 2505 and 4680 nM for EP2, DP1, IP, EP1,Formula:C27H45NO7Purity:99.86%Color and Shape:SolidMolecular weight:495.65L-371,257
CAS:L-371,257 is a competitive antagonist of oxytocin receptor with pA2 of 8.4 and Ki of 19 nM. L-371,257 shows a Ki of 3.7 nM for vasopressin receptor 1a.Formula:C28H33N3O6Purity:99.79%Color and Shape:SolidMolecular weight:507.58ELOVL1-IN-2
CAS:ELOVL1-IN-2 weakly inhibits ELOVL1 enzyme (IC50: 21 μM) and shows moderate potency in HEK293 cells (IC50: 6.7 μM).Formula:C18H15FN2OPurity:99.94%Color and Shape:SolidMolecular weight:294.32Dersimelagon
CAS:Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist.Cost-effective and quality-assured.Formula:C36H45F4N3O5Purity:97.35% - 98.23%Color and Shape:SolidMolecular weight:675.75USP15-IN-1
CAS:USP15-IN-1 is a potent USP15 inhibitor (IC50 is 3.76 μM).Formula:C22H23N3O3Purity:99.509% - 99.81%Color and Shape:SolidMolecular weight:377.44GSK3368715 dihydrochloride
CAS:GSK3368715 dihydrochloride (EPZ019997 dihydrochloride) is a PRMTs inhibitor , with anticancer activity, for the study of advanced solid tumors.Formula:C20H40Cl2N4O2Purity:99.66% - 99.66%Color and Shape:SolidMolecular weight:439.46JTK-109
CAS:JTK-109 is an inhibitor of hepatitis C virus NS5B RNA-dependent RNA polymerase inhibitor and inhibits G1b and G3a subgenomic replicons and recombinant enzymes.Formula:C37H33ClFN3O4Purity:98.48% - 99.68%Color and Shape:SolidMolecular weight:638.13Ref: TM-T27696
1mg296.00€5mg718.00€10mg982.00€25mg1,485.00€50mg2,008.00€100mg2,637.00€1mL*10mM (DMSO)1,108.00€AZ12601011
CAS:AZ12601011 is a TGFBR1 kinase inhibitor that inhibits the growth of breast tumors.Formula:C19H15N5Purity:98.81%Color and Shape:SolidMolecular weight:313.36Ref: TM-T10426
1mg99.00€5mg235.00€10mg376.00€25mg728.00€50mg1,093.00€100mg1,510.00€1mL*10mM (DMSO)259.00€ALOX15-IN-2
CAS:ALOX15-IN-2: Potent ALOX15 inhibitor. IC50: 1.55 μM for LA; 2.79 μM for AA. Stops linoleic/arachidonic acid oxidation.Formula:C23H29N3O4SPurity:99.98%Color and Shape:SolidMolecular weight:443.56Ref: TM-T62606
1mg46.00€5mg90.00€10mg160.00€25mg313.00€50mg537.00€100mg767.00€500mg1,558.00€1mL*10mM (DMSO)100.00€Evixapodlin
CAS:Evixapodlin (PD-1/PD-L1-IN 7) is a human PD-1/PD-L1 protein/protein interaction inhibitor (IC50: 0.213).Evixapodlin has anticancer and antiviral activities.Formula:C34H36Cl2N8O4Purity:97.02%Color and Shape:SolidMolecular weight:691.61Ref: TM-T36487
1mg111.00€5mg264.00€10mg424.00€25mg747.00€50mg1,008.00€100mg1,359.00€200mg1,833.00€1mL*10mM (DMSO)405.00€AZD5462
CAS:AZD5462 is a potent orally available relaxin receptor RXFP1 agonist for the study of heart failure and cancer.Formula:C30H41FN2O6Purity:98.32% - 99.63%Color and Shape:SolidMolecular weight:544.65IDX184
CAS:IDX184 is a potent, orally active, targeted HCV polymerase inhibitor and nucleoside polymerase.IDX184 effectively inhibits HCV polymerase (IC50=0.31 μM, Ki=52.3Formula:C25H35N6O9PSPurity:97.15%Color and Shape:SolidMolecular weight:626.62Aleglitazar
CAS:Aleglitazar (R1439) (R1439) is a potent dual PPARα/γ agonist, with IC50s of 38 nM and 19 nM for human PPARa and PPARγ, respectively.Formula:C24H23NO5SPurity:99.03%Color and Shape:SolidMolecular weight:437.51Ref: TM-T14176
1mg233.00€5mg532.00€10mg718.00€25mg1,099.00€50mg1,485.00€100mg1,998.00€1mL*10mM (DMSO)538.00€HOIPIN-8 sodium
CAS:HOIPIN-8 sodium is a LUBAC inhibitor for the study of inflammatory and immune diseases.Formula:C23H15F2N4NaO3Purity:97.34%Color and Shape:SolidMolecular weight:456.38Ref: TM-T62826
1mg66.00€5mg145.00€10mg224.00€25mg358.00€50mg512.00€100mg707.00€200mg973.00€1mL*10mM (DMSO)146.00€LSN3318839
CAS:LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled signaling and canFormula:C26H23Cl2N3O2Purity:99.70%Color and Shape:SolidMolecular weight:480.39Obicetrapib
CAS:Obicetrapib (AMG-899) is an inhibitor of cholesteryl ester transfer protein.Formula:C32H31F9N4O5Purity:99.26% - >99.99%Color and Shape:SolidMolecular weight:722.6D75-4590
CAS:D75-4590, a β-1,6-Glucan synthetase inhibitor, combats fungal infections by targeting cell walls.Formula:C21H27N5Purity:98.56% - 98.85%Color and Shape:SolidMolecular weight:349.47Ref: TM-T61194
5mg39.00€10mg62.00€25mg122.00€50mg187.00€100mg269.00€200mg358.00€1mL*10mM (DMSO)46.00€DRF-1042
CAS:DRF-1042 is a camptothecin analog with anticancer and insecticidal activity and is used to study solid tumors such as prostate and colon cancer.Formula:C22H20N2O6Purity:98.34%Color and Shape:SolidMolecular weight:408.4Simmitecan hydrochloride
CAS:Simmitecan hydrochloride is a camptothecin derivative, a topoisomerase I inhibitor with anticancer activity, which can be used to study is solid tumors.Formula:C34H39ClN4O6Purity:98.20% - 98.93%Color and Shape:SolidMolecular weight:635.15VX-984
CAS:VX-984 (M9831) is an oral DNA-PK inhibitor, crossing the blood-brain barrier, targeting GBM and NSC-LC.Formula:C23H21D2N7OPurity:97.65% - 99.98%Color and Shape:SolidMolecular weight:415.49Ref: TM-T11067
1mg117.00€5mg248.00€10mg369.00€25mg575.00€50mg863.00€100mg1,305.00€200mg1,755.00€1mL*10mM (DMSO)271.00€WAY-213613 hydrochloride
CAS:WAY-213613 hydrochloride: potent, selective GLT-1/EAAT2 inhibitor (IC50 85 nM); weaker for EAAT1/3; inactive at glutamate receptors; research tool for CNS.Formula:C16H13BrF2N2O4Purity:99.14% - 99.37%Color and Shape:SoildMolecular weight:415.19Ref: TM-T13330
1mg35.00€5mg80.00€10mg92.00€25mg215.00€50mg359.00€100mg610.00€200mg827.00€1mL*10mM (DMSO)89.00€BCL6-IN-3
CAS:BCL6-IN-3: potent BCL6 inhibitor, 70 nM GI50 in SU-DHL4, affects cell functions, antitumor.Formula:C24H31ClF2N6O2Purity:98.17%Color and Shape:SolidMolecular weight:508.99Ref: TM-T10487
1mg109.00€5mg241.00€10mg355.00€25mg532.00€50mg745.00€100mg1,018.00€500mgTo inquire1mL*10mM (DMSO)370.00€NB-360
CAS:NB-360: potent, brain-penetrant BACE1/2 inhibitor; IC50s: 5-6 nM; high selectivity vs pepsin, cathepsin E/D.Formula:C21H19F4N5O2Purity:99.72%Color and Shape:SolidMolecular weight:449.4Ref: TM-T12188
1mg104.00€5mg215.00€10mg318.00€25mg510.00€50mg692.00€100mg888.00€500mg1,783.00€1mL*10mM (DMSO)235.00€INCB054329
CAS:INCB054329 is a BET inhibitor targeting BRD2/3/4 and BRDT with IC50s ranging from 1-119 nM.Formula:C19H16N4O3Purity:99.52%Color and Shape:SolidMolecular weight:348.36NRX-252114
CAS:NRX-252114 promotes mutant β-catenin degradation, binding it to E3 ligase SCFβ-TrCP (EC50: 6.5 nM; Kd: 0.4 nM).Formula:C22H12Cl2F3N3O2SPurity:99.70%Color and Shape:SolidMolecular weight:510.32Umibecestat
CAS:Umibecestat inhibits human and mouse BACE-1 (IC50: 11 nM & 10 nM), potentially for Alzheimer's research.Formula:C19H15ClF7N5O2Purity:99.88%Color and Shape:SolidMolecular weight:513.8Ref: TM-T13253
1mg163.00€5mg334.00€10mg485.00€25mg807.00€50mg1,099.00€100mg1,485.00€1mL*10mM (DMSO)376.00€Darizmetinib
CAS:Darizmetinib (HRX215) is an MKK4 inhibitor.Formula:C21H17F2N5O3SPurity:98.03% - 99.57%Color and Shape:SolidMolecular weight:457.45Ref: TM-T72956
1mg69.00€2mg89.00€5mg147.00€10mg224.00€25mg324.00€50mg400.00€100mg587.00€1mL*10mM (DMSO)148.00€Dazostinag disodium
CAS:Dazostinag disodium (TAK-676) is a synthetic novel interferon gene (STING) agonist.Cost-effective and quality-assured.Formula:C21H20F2N8Na2O10P2S2Purity:98.84% - 99.96%Color and Shape:SolidMolecular weight:754.48Zelasudil
CAS:Zelasudil (RXC007) is a Rho-related (ROCK) kinase inhibitor for the study of idiopathic pulmonary fibrosis and inflammation.Formula:C22H21F2N7OPurity:99.15%Color and Shape:SolidMolecular weight:437.445Ref: TM-T69665
1mg92.00€5mg168.00€10mg248.00€25mg421.00€50mg587.00€100mg820.00€1mL*10mM (DMSO)170.00€SB-224289 hydrochloride
CAS:SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.Formula:C32H33ClN4O3Purity:98.99% - 99.96%Color and Shape:SolidMolecular weight:557.08Tigemonam
CAS:Tigemonam is a monobactam, a novel orally administered monobactam that protects against gram-negative aerobic bacterial pathogens. Cost-effective and quality-assured.Formula:C12H15N5O9S2Purity:97.71% - >99.99%Color and Shape:SolidMolecular weight:437.41BQ-788
CAS:BQ-788 is an ETB receptor antagonist with potential hypertensive activity that inhibits exogenous ET-1-induced elevation of coronary perfusion pressure.Formula:C34H51N5O7Purity:98.81%Color and Shape:SolidMolecular weight:641.8Ref: TM-T10595
1mg130.00€2mg178.00€5mg313.00€10mg447.00€25mg713.00€50mg964.00€100mg1,305.00€500mg2,592.00€1mL*10mM (DMSO)341.00€USP5-IN-1
USP5-IN-1, a powerful USP5 deubiquitinase inhibitor, selectively binds with 2.8 μM affinity, blocking USP5's di-ubiquitin cleavage.
Formula:C19H20ClN3O5SPurity:99.76%Color and Shape:SoildMolecular weight:437.9SYM2206
CAS:SYM2206 is a low affinity non-competitive AMPA receptor antagonist with an IC50 value of 1.6 μM.SYM2206 exhibits anticancer activity by blocking Nav1.6-mediatedFormula:C20H22N4O3Purity:99.8%Color and Shape:SolidMolecular weight:366.41FABPs ligand 6
CAS:FABPs ligand 6 (MF6) is an inhibitor of FABP5 and FABP7.Formula:C28H27FN2O3Purity:97.45%Color and Shape:SolidMolecular weight:458.52AChE/BChE-IN-10
CAS:AChE/BChE-IN-10 inhibits AChE/BChE (IC50: 0.176/0.47 μM), crosses the blood-brain barrier, and prevents Aβ-aggregation.
Formula:C26H30N2O2Purity:99.55% - 99.88%Color and Shape:SoildMolecular weight:402.53CP-642931
CAS:CP-642931 (Sorbitol dehydrogenase-IN-1) is a sorbitol dehydrogenase inhibitor used in the study of diabetes mellitus and cardiovascular disease.Formula:C17H25N7OPurity:99.67% - >99.99%Color and Shape:SolidMolecular weight:343.43Elacytarabine
CAS:Elacytarabine (M7594 0037), a lipid-conjugated derivative of the nucleoside analog cytarabine, is an antineoplastic drug. It has cytotoxicity in solid tumors.Formula:C27H45N3O6Purity:97.69%Color and Shape:SolidMolecular weight:507.66AChE-IN-26
CAS:AChE-IN-26 (compound 4a) is an AChE (acetylcholinesterase) inhibitor (IC50: 0.42 μM).
Formula:C21H21BrN2O3Purity:99.24% - 99.85%Color and Shape:SoildMolecular weight:429.31DN02
DN02: a potent, selective BRD8(1) bromodomain probe; Ki=32 nM; 30x more affine than BRD8(2).Formula:C22H24FN3O3Purity:98.22% - 99.74%Color and Shape:SolidMolecular weight:397.44AM103
CAS:AM103 is an effective and selective inhibitor of FLAP (IC50 = 4.2 nM).Formula:C36H38N3NaO4SPurity:99.75%Color and Shape:SolidMolecular weight:631.76JNJ-6204
CAS:JNJ-6204 is a deuterated compound that efficiently inhibits CSNK1D and CSNK1E.Formula:C19H11D6FN6OPurity:97.42% - 99.87%Color and Shape:SolidMolecular weight:370.41Etamicastat hydrochloride
CAS:Etamicastat hydrochloride (BIA 5-453 hydrochloride) is a peripherally selective dopamine beta-hydroxylase inhibitor that reduces hypertension.Formula:C14H16ClF2N3OSPurity:98.54%Color and Shape:SolidMolecular weight:347.81Ref: TM-T11238L
1mg80.00€5mg173.00€10mg259.00€25mg423.00€50mg577.00€100mg827.00€1mL*10mM (DMSO)190.00€Vofopitant
CAS:Vofopitant (GR 205171) is a potent NK1 receptor antagonist with anxiolytic and antiemetic activity for the study of post-traumatic stress disorder (PTSD).Formula:C21H23F3N6OPurity:97.86%Color and Shape:SolidMolecular weight:432.44BODIPY FL prazosin
CAS:BODIPY FL prazosin is an α1-adrenergic antagonist that inhibits α1a-AR and α1b-AR.
Formula:C28H32BF2N7O3Purity:97.27%Color and Shape:SolidMolecular weight:563.41Moiramide B
CAS:Moiramide B is an acetyl coenzyme A carboxylase inhibitor with antimicrobial activity, strongly inhibiting Gram-positive bacteria.Formula:C25H31N3O5Purity:98.53% - 99.90%Color and Shape:SolidMolecular weight:453.53Enbezotinib
CAS:Enbezotinib is an inhibitor of RET autophosphorylation and can be used in cancer research.Formula:C21H21FN6O3Purity:99.84%Color and Shape:SolidMolecular weight:424.43Ref: TM-T62285
1mg77.00€5mg166.00€10mg253.00€25mg414.00€50mg567.00€100mg745.00€1mL*10mM (DMSO)182.00€
