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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66626 products of "Inhibitors"

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  • SBI-581


    <p>SBI-581: oral, potent TAO3 inhibitor, IC50=42nM, alters TKS5α at RAB11+ vesicles, blocks invadopodia, good mouse pharmacokinetics, anti-tumor.</p>
    Formula:C24H21N3O2
    Color and Shape:Solid
    Molecular weight:383.44
  • EF1502 free base

    CAS:
    <p>EF1502 is a potent and selective GABA transporter inhibitor.</p>
    Formula:C22H26N2O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:414.58
  • L-690330 hydrate


    <p>L-690330 hydrate inhibits IMPase; Ki: 0.30 μM (human), 0.42 μM (bovine cortex); 0.27 μM (recom. human), 0.19 μM (bovine).</p>
    Formula:C8H14O9P2
    Color and Shape:Solid
    Molecular weight:316.14
  • DNA Gyrase-IN-1


    <p>DNA Gyrase-IN-1: potent, selective promoter inhibitor. IC50: 2.6 μM, inhibits Mtb, MIC: 0.49 μM. Useful for tuberculosis research.</p>
    Formula:C24H24FN7O6
    Color and Shape:Solid
    Molecular weight:525.49
  • Foroxymithine

    CAS:
    <p>Foroxymithine is an inhibitor of angiotensin-converting enzyme.</p>
    Formula:C22H37N7O11
    Purity:98%
    Color and Shape:Solid
    Molecular weight:575.57
  • Antifungal agent 25


    <p>Antifungal agent 25: broad-spectrum, stable in vivo, effective against Candida albicans, including fluconazole-resistant strains.</p>
    Color and Shape:Solid
  • Ketomethylenebestatin

    CAS:
    <p>Ketomethylenebestatin, a weaker carba-analog of aminopeptidase inhibitor bestatin, is 10x less potent.</p>
    Formula:C17H25NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:307.38
  • Anti-TSWV agent 1


    <p>Anti-TSWV agent 1 is a highly effective inactivator (EC50:144 μg/mL) of tomato spotted wilt virus (TSWV).</p>
    Formula:C22H27ClN4OS3
    Color and Shape:Solid
    Molecular weight:495.12
  • Dictyostatin

    CAS:
    <p>Dictyostatin: potent microtubule stabilizer &amp; anticancer agent with antiproliferative effects; researched for tauopathies.</p>
    Formula:C32H52O6
    Color and Shape:Solid
    Molecular weight:532.75
  • GSK5852


    <p>GSK5852, an HCV NS5B inhibitor, has IC50 of 50 nM; potently fights HCV with EC50 of 3.0 nM for GT1a and 1.7 nM for GT1b.</p>
    Formula:C27H27BF2N2O6S
    Color and Shape:Solid
    Molecular weight:556.39
  • SARS-CoV-2-IN-24


    <p>SARS-CoV-2-IN-24 blocks PLpro, altering its shape and stopping virus replication—useful for SARS-CoV-2 research.</p>
    Formula:C27H30N4O5
    Color and Shape:Solid
    Molecular weight:490.55
  • C.I. Pigment Red 60

    CAS:
    <p>C.I. Pigment Red 60 is a bright, scarlet, semi-transparent red pigment.</p>
    Formula:C17H9N2Na3O9S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:518.35
  • Terguride

    CAS:
    <p>Terguride: treats hyperprolactinemia, blocks 5-HT2A/B, activates dopamine receptors, studied for PAH.</p>
    Formula:C20H28N4O
    Color and Shape:Solid
    Molecular weight:340.46
  • Minnelide

    CAS:
    <p>Minnelide is a prodrug of triptolide,and shows potent antitumor activity in a number of tumor types.</p>
    Formula:C21H25Na2O10P
    Purity:98.49% - 99.59%
    Color and Shape:Solid
    Molecular weight:514.37
  • DSP-6952

    CAS:
    <p>DSP-6952 is a 5-HT4 receptor partial agonist, inhibiting visceral hypersensitivity and ameliorating gastrointestinal dysfunction.</p>
    Formula:C21H32BrClN4O5
    Color and Shape:Solid
    Molecular weight:535.86
  • Tuberculosis inhibitor 5


    <p>Compound 11i: potent, non-toxic anti-tuberculosis biphenyl analogue.</p>
    Formula:C25H18N2O2S
    Color and Shape:Solid
    Molecular weight:410.49
  • Samuraciclib

    CAS:
    <p>Samuraciclib (CT7001) is an oral CDK7 inhibitor with 41 nM IC50, notable for its high selectivity and potency against breast cancer cells.</p>
    Formula:C22H30N6O
    Color and Shape:Solid
    Molecular weight:394.51
  • G-9791

    CAS:
    <p>G-9791 is an effective and selective inhibitor of group-I PAK.</p>
    Formula:C26H26ClFN6O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:508.98
  • AGN-795

    CAS:
    <p>AGN-795 is a biochemical.</p>
    Formula:C14H20N2
    Color and Shape:Solid
    Molecular weight:216.328
  • U91356

    CAS:
    <p>U91356 is an agonist of the dopamine receptors.</p>
    Formula:C13H17N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:231.29
  • Allosucrose

    CAS:
    <p>Allosucrose is a biochemical.</p>
    Formula:C12H22O11
    Color and Shape:Solid
    Molecular weight:342.30
  • A4B17


    <p>A4B17 is an inhibitor of androgen receptor N-terminal with potential for androgen-responsive prostate cancer treatment.</p>
    Formula:C14H7F4NS
    Color and Shape:Solid
    Molecular weight:297.27
  • 9(S),10(S),13(S)-TriHOME

    CAS:
    <p>9(S),10(S),13(S)-TriHOME is an oxylipin derived from linoleic acid. It has been detected in beer and in bronchoalveolar lavage fluid (BALF) from female smokers.</p>
    Formula:C18H34O5
    Color and Shape:Solid
    Molecular weight:330.46
  • IRAK4-IN-9

    CAS:
    <p>IRAK4-IN-9 is a potent IRAK4 inhibitor with an IC50 of 1.5 nM, promising for inflammatory, autoimmune diseases, and cancer research.</p>
    Formula:C22H25N7
    Color and Shape:Solid
    Molecular weight:387.48
  • Ep vinyl quinidine

    CAS:
    <p>3-Epiquinine is a Quinidine stereoisomer, used in malaria, antiarrhythmic, inhibits P450db, and blocks K+ channels, IC50: 19.9 μM.</p>
    Formula:C20H24N2O2
    Color and Shape:Solid
    Molecular weight:324.42
  • Saussureamine C

    CAS:
    <p>Saussureamine C is an inhibitor of H274Y and N294S mutants.</p>
    Formula:C19H26N2O5
    Color and Shape:Solid
    Molecular weight:362.42
  • AVE-1330A free acid

    CAS:
    <p>AVE-1330A free acid is a broad-spectrum non-beta-lactam beta-lactamase inhibitor.</p>
    Formula:C7H11N3O6S
    Color and Shape:Solid
    Molecular weight:265.24
  • Vanin-1-IN-3


    <p>Vanin-1-IN-3 (OMP-7) is a vanin-1 inhibitor with an IC 50 of 0.038 μM [1].</p>
    Formula:C17H22F3NO5
    Color and Shape:Solid
    Molecular weight:377.36
  • RSV-IN-5

    CAS:
    <p>RSV-IN-5: Dual inhibitor for RSV fusion proteins, effective on wild-type A2 and D486N mutant with EC50s of 2.0 nM &amp; 8.1 nM. Potent anti-RSV.</p>
    Formula:C28H37N7O2
    Color and Shape:Solid
    Molecular weight:503.64
  • Carbonic anhydrase inhibitor 9


    <p>Carbonic anhydrase inhibitor 9 targets hCA II and IX with Ki of 56.4 and 56.9 nM respectively; shows antiproliferative activity.</p>
    Formula:C22H20BrN5O4S
    Color and Shape:Solid
    Molecular weight:530.39
  • Domitroban

    CAS:
    <p>Domitroban, also known as S-145, is a thromboxane (Tx) A2-receptor antagonist with partial agonistic activity in vascular smooth muscle.</p>
    Formula:C20H27NO4S
    Color and Shape:Solid
    Molecular weight:377.5
  • FTI-2628

    CAS:
    <p>FTI-2628 is a novel inhibitor of protein farnesyltransferase (FT), inhibiting the growth of P. falciparum in red blood cells and suppressing parasitemia.</p>
    Formula:C31H34N4O3S
    Color and Shape:Solid
    Molecular weight:542.69
  • IRAK4-IN-11


    <p>IRAK4-IN-11 (compound 6) is a potent inhibitor of IRAK4 with an IC 50 of 0.008 μM. IRAK4-IN-11 exhibits cell pIRAK4 potencies with an IC 50 of 0.19 μM [1].</p>
    Formula:C16H19N7O
    Color and Shape:Solid
    Molecular weight:325.37
  • NTPDase-IN-3

    CAS:
    <p>NTPDase-IN-3 inhibits NTPDase1/2/3/8 (IC50: 0.21/1.07/0.38/0.05 μM), useful for cancer and thrombosis research.</p>
    Formula:C22H24ClN3OS2
    Color and Shape:Solid
    Molecular weight:446.03
  • K027


    <p>K027 is a potent organophosphate (OP) inhibitor of acetylcholinesterase (AChE) reactivation. k027 can be used to study Alzheimer's disease.</p>
    Formula:C15H18Br2N4O2
    Color and Shape:Solid
    Molecular weight:446.14
  • KRAS G12D inhibitor 12


    <p>KRAS G12D inhibitor 12 targets Ras protein for cancer research. (Patent WO2021108683A1, Compound 134)</p>
    Formula:C23H21ClFN5O3
    Color and Shape:Solid
    Molecular weight:469.9
  • Carbonic anhydrase inhibitor 8


    <p>R-13, a carbonic anhydrase inhibitor, has Ki of 60.7 nM (hCA I), 320.7 nM (hCA II), and 2298 nM (hCA IV).</p>
    Formula:C20H25N3O4S
    Color and Shape:Solid
    Molecular weight:403.5
  • CS-0777

    CAS:
    <p>CS-0777 is a potent, selective, and orally active S1P1 agonist (sphingosine 1-phosphate receptor modulator).</p>
    Formula:C21H31N2O5P
    Color and Shape:Solid
    Molecular weight:422.45
  • CXCR2 antagonist 6


    <p>CXCR2 antagonist 6: strong CXCR2 affinity (IC50=0.044 μM), hinders calcium mobilization (IC50=0.66 μM).</p>
    Formula:C17H16F2N4OS
    Color and Shape:Solid
    Molecular weight:362.4
  • 12(S)-HETE

    CAS:
    <p>Enpatoran hydrochloride (M5049 hydrochloride) is a TLR7/8 inhibitor with antiviral activity that is used in the study of autoimmune diseases.</p>
    Formula:C20H32O3
    Color and Shape:Solid
    Molecular weight:320.47
  • DC41SMe

    CAS:
    <p>DC41SMe, a DC1 derivative and CC-1065 analogue, targets cancer with 18-25 pM IC50 against Ramos, Namalwa, HL60/s cells.</p>
    Formula:C38H36ClN5O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:726.31
  • TAK-637

    CAS:
    <p>TAK-637 is a tachykinin 1 (NK1) receptor antagonist.</p>
    Formula:C30H25F6N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:573.53
  • CAII-IN-3


    <p>CAII-IN-3, a thiosemicarbazone, potently inhibits CA-II with an IC50 of 13.4 μM.</p>
    Formula:C18H18F2N4S
    Color and Shape:Solid
    Molecular weight:360.42
  • RS 12254

    CAS:
    <p>RS 12254 is a dopamine agonist and antihypertensive agent.</p>
    Formula:C28H40N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:468.63
  • Deldeprevir Na

    CAS:
    <p>Deldeprevir Na is an Antiviral Polyprotein cleavage inhibitor. HCV NS3/4A inhibitor.</p>
    Formula:C45H55F2N6NaO8S2
    Color and Shape:Solid
    Molecular weight:933.08
  • 22-HDHA

    CAS:
    <p>22-HDHA is an oxidation product of docosahexaenoic acid .</p>
    Formula:C22H32O3
    Color and Shape:Solid
    Molecular weight:344.49
  • AY-22,252

    CAS:
    <p>AY-22,252 is an inhibitor of beef heart &amp; rat brain nucleoside-3',5'- monophosphate phosphodiesterase.</p>
    Formula:C27H37NaO7
    Color and Shape:Solid
    Molecular weight:496.57
  • VU0463271 quarterhydrate


    <p>VU0463271 quarterhydrate is a potent KCC2 antagonist, with an IC 50 of 61 nM [1].</p>
    Formula:C19H20N4O2S2
    Color and Shape:Solid
    Molecular weight:387
  • CXCR4 antagonist 3


    <p>CXCR4 antagonist 3, aka compound 12a, has 11 nM IC50, shares TIQ15 traits, and is promising in HIV research.</p>
    Formula:C22H31N5
    Color and Shape:Solid
    Molecular weight:365.52
  • OP-5244 sodium


    <p>OP-5244 sodium: potent oral CD73 inhibitor (IC50: 0.25 nM), potential in cancer research by hindering adenosine, reversing immunosuppression.</p>
    Formula:C19H28ClN5NaO9P
    Color and Shape:Solid
    Molecular weight:559.87
  • PIM-1/HDAC-IN-1


    <p>PIM-1/HDAC-IN-1 (4d): inhibits PIM-1 (IC50: 343.87nM), HDAC1 (63.65nM), HDAC6 (62.39nM); induces apoptosis in MCF-7 cells.</p>
    Formula:C22H19N3O3
    Color and Shape:Solid
    Molecular weight:373.4
  • PF-06648671

    CAS:
    <p>PF-06648671 is a γ-secretase modulator for the treatment of neurodegenerative and/or neurological disorders.</p>
    Formula:C25H23ClF4N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:538.92
  • Trypanothione synthetase-IN-4


    <p>Trypanothione synthetase-IN-4, an L. infantum inhibitor, has potent anti-leishmanicidal properties (EC50: 0.6 μM).</p>
    Formula:C29H52INO2
    Color and Shape:Solid
    Molecular weight:573.63
  • MEK4 inhibitor-2

    CAS:
    <p>MEK4 Inhibitor-2, a novel MEK4 inhibitor, demonstrates efficacy against pancreatic adenocarcinoma, exhibiting an IC50 value of 83 nM.</p>
    Formula:C20H15FN4O3S
    Color and Shape:Solid
    Molecular weight:410.42
  • JH-XVII-10


    <p>JH-XVII-10: potent, oral DYRK1A/B inhibitor (IC50: 3/5 nM), shows antitumor activity in HNSCC.</p>
    Formula:C21H16F4N8O
    Color and Shape:Solid
    Molecular weight:472.4
  • EGFR-IN-47


    <p>EGFR-IN-47: strong oral EGFRL858R/T790M/C797S blocker, induces cell death; promising for NSCLC research. IC50: 0.01 μM.</p>
    Formula:C29H35N7
    Color and Shape:Solid
    Molecular weight:481.64
  • MrgprX2 antagonist-7


    <p>MrgprX2 antagonist-7 is an anti-allergic agent with significant anti-allergic effects and inhibits mast cell degranulation.</p>
    Formula:C24H22ClF3N6O3
    Color and Shape:Solid
    Molecular weight:534.92
  • Dyrk1A-IN-4

    CAS:
    <p>Dyrk1A-IN-4, compound 48, is an oral DYRK1A/DYRK2 inhibitor with IC50s: 2 nM (DYRK1A), 6 nM (DYRK2), anticancer properties.</p>
    Formula:C14H13F3N6
    Color and Shape:Solid
    Molecular weight:322.29
  • Anticancer agent 78


    <p>Anticancer agent 78: anti-aromatase (IC50=0.9 μM), cytotoxic, potential in breast cancer research.</p>
    Formula:C19H14BrNO4
    Color and Shape:Solid
    Molecular weight:400.22
  • Naltalimide

    CAS:
    <p>Naltalimide: µ-opioid receptor partial agonist, improves bladder storage by affecting spinal cord reflex.</p>
    Formula:C28H28N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:472.53
  • Nafarelin acetate hydrate

    CAS:
    <p>Nafarelin: a GnRH agonist used to treat endometriosis, precocious puberty, and control IVF. Delivered as a nasal spray. Marketed as Synarel by Pfizer.</p>
    Formula:C66H83N17O13·xC2H4O2·xH2O
    Color and Shape:Solid
    Molecular weight:1400.563
  • EBI-907

    CAS:
    <p>EBI-907 is a potent, oral B-RafV600E inhibitor with an IC50 of 4.9 nM, over 10x stronger than Vemurafenib, and effective against key cancer kinases.</p>
    Formula:C23H21ClF2N4O3S
    Color and Shape:Solid
    Molecular weight:506.95
  • TY 11345

    CAS:
    <p>TY 11345 is a proton pump inhibitor.</p>
    Formula:C18H18N3NaO2S
    Color and Shape:Solid
    Molecular weight:363.41
  • HER2-IN-7

    CAS:
    <p>HER2-IN-7 is a potent HER2 inhibitor with potential for researching ErbB-related diseases, especially cancer.</p>
    Formula:C28H26F3N7O3
    Color and Shape:Solid
    Molecular weight:565.55
  • NA 0346

    CAS:
    <p>NA 0346 is a derivative of SF 2370 that shows long lasting antihypertensive action as well as potent protein kinases inhibitory activity.</p>
    Formula:C26H22N4O3
    Color and Shape:Solid
    Molecular weight:438.48
  • Sovesudil hydrochloride


    <p>Sovesudil (PHP-201) HCl: potent local ROCK inhibitor; targets ROCK I/II (IC50: 3.7/2.3 nM); lowers IOP, non-congesting.</p>
    Formula:C23H23ClFN3O3
    Color and Shape:Solid
    Molecular weight:443.9
  • Dyrk1A/B-IN-1


    <p>Dyrk1A/B-IN-1 (3n) is a potent DYRK1A/B inhibitor, cell-permeable, with Ki values of 67.8 nM (1A) and 237.9 nM (1B), IC50s of 1.1 and 0.8 μM.</p>
    Formula:C21H17N3O2S2
    Color and Shape:Solid
    Molecular weight:407.51
  • Gusperimus

    CAS:
    <p>Gusperimus was synthesized by chemical modification of spergualin and in combination with cyclosporine A to prevent diabetes in susceptible NOD mice.</p>
    Formula:C17H37N7O3
    Color and Shape:Solid
    Molecular weight:387.52
  • Canosimibe

    CAS:
    <p>Canosimibe is a cholesterol absorption inhibitor</p>
    Formula:C44H60FN3O10
    Color and Shape:Solid
    Molecular weight:809.96
  • Teoprolol

    CAS:
    <p>Teoprolol is a blocker of β-adrenergic receptor.</p>
    Formula:C23H30N6O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:454.52
  • Equisetin

    CAS:
    <p>Equisetin: a QSI from Fusarium equiseti, curbs P. aeruginosa virulence, fights Gram-positive bacteria &amp; HIV-1 integrase; not antibacterial to Gram-negative.</p>
    Formula:C22H31NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:373.49
  • JAK2/FLT3-IN-1 TFA


    <p>JAK2/FLT3-IN-1 (TFA), an oral JAK2/FLT3 inhibitor, shows anticancer properties; IC50: JAK2 (0.7 nM), FLT3 (4 nM), JAK1 (26 nM), JAK3 (39 nM).</p>
    Formula:C27H35F4N7O3
    Color and Shape:Solid
    Molecular weight:581.61
  • PDE4B-IN-3


    <p>PDE4B-IN-3 is a potent inhibitor of PDE4B (IC50: 0.94 μM) and exhibits anti-inflammatory effects.</p>
    Formula:C30H35N3O4S2
    Color and Shape:Solid
    Molecular weight:565.75
  • VEGFR-2-IN-17


    <p>VEGFR-2-IN-17 (15a) is a potent VEGFR-2 inhibitor with an IC50 of 67.25 nM, showing significant antitumor effects.</p>
    Formula:C21H14ClN3O2
    Color and Shape:Solid
    Molecular weight:375.81
  • MK-8318

    CAS:
    <p>MK-8318 is an effective and selective antagonist of the CRTh2 receptor (Ki: 5.0 nM).</p>
    Formula:C27H26F4N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:534.5
  • Antileishmanial agent-4


    <p>Antileishmanial agent-4, a ribonucleoside analogue, functions as an antileishmanial agent [1].</p>
    Formula:C17H18N4O4
    Color and Shape:Solid
    Molecular weight:342.35
  • Ibafloxacine

    CAS:
    <p>Ibafloxacine (R835) is a fluoroquinolone antibiotic that is used exclusively in veterinary applications and shows zero good bacteriostatic effect against</p>
    Formula:C15H14FNO3
    Purity:97.67%
    Color and Shape:Solid
    Molecular weight:275.27
  • Idraparinux Na

    CAS:
    <p>Idraparinux Na is an Antithrombotic, Indirect, Selective, Synthetic Factor Xa Inhibitor</p>
    Formula:C38H55Na9O49S7
    Color and Shape:Solid
    Molecular weight:1727.14
  • iMDK quarterhydrate


    <p>iMDK quarterhydrate, PI3K inhibitor, blocks MDK growth; suppresses NSCLC safely with MEK inhibitor.</p>
    Formula:C21H15FN2O3S
    Color and Shape:Solid
    Molecular weight:380.91
  • TEI-9063

    CAS:
    <p>TEI-9063 is a stable and highly specific prostacyclin analogue of prostacyclin receptor in mast cell tumor p-815 cells.</p>
    Formula:C23H38O4
    Color and Shape:Solid
    Molecular weight:378.55
  • L 731735

    CAS:
    <p>L 731735 is a farnesyltransferase inhibitor.</p>
    Formula:C19H40N4O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:420.61
  • SCH-900822

    CAS:
    <p>SCH-900822 is a potent and selective glucagon receptor antagonist.</p>
    Formula:C34H43Cl2N7O2
    Color and Shape:Solid
    Molecular weight:652.66
  • AZD-3409

    CAS:
    <p>AZD-3409 is a more potent prenyl transferase inhibitor than lonafarnib with varied IC(50) in cells, acting on gefitinib-resistant breast cancer.</p>
    Formula:C34H41FN4O4S2
    Color and Shape:Solid
    Molecular weight:652.84
  • CYP2C9/CYP2C19-IN-1


    <p>CYP2C9/CYP2C19-IN-1 is a potent inhibitor of CYP2C9/CYP2C19 without liver toxicity or genotoxicity and can be used to study Zika virus (ZIKV) infection.</p>
    Formula:C27H28N2O6S
    Color and Shape:Solid
    Molecular weight:508.59
  • Protease-Activated Receptor-1 antagonist 3


    <p>PAR-1 antagonist 3: potent (IC50: 7 nM), binds hERG K+ channels (IC50: 9 μM).</p>
    Formula:C30H34N4O3
    Color and Shape:Solid
    Molecular weight:498.62
  • RdRP-IN-4


    <p>RdRP-IN-4, an oral arylbenzohydrazide, inhibits influenza A/B by targeting PB1 of RdRP, with EC50s of 53 nM (H1N1) and 20 nM (Flu B), and aids infected mice.</p>
    Formula:C17H17Br2N3O2
    Color and Shape:Solid
    Molecular weight:455.14
  • (rel)-AR234960

    CAS:
    <p>(rel)-AR234960 is an active relative configuration of AR234960. AR234960 is a non-peptide agonist of MAS.</p>
    Formula:C27H30FN5O5S
    Color and Shape:Solid
    Molecular weight:555.63
  • NA 382

    CAS:
    <p>NA 382 is a staurosporine derivative that inhibits multidrug resistance.</p>
    Formula:C31H28N4O6
    Color and Shape:Solid
    Molecular weight:552.58
  • MAP855

    CAS:
    <p>MAP855: potent, selective, oral MEK1/2 inhibitor; IC50=3 nM, pERKEC50=5 nM; effective on wild-type/mutant MEK1/2.</p>
    Formula:C28H23ClF2N6O3
    Color and Shape:Solid
    Molecular weight:564.97
  • Valopicitabine dihydrochloride

    CAS:
    <p>Valopicitabine, a NS5B inhibitor, is used potentially for the treatment of HCV infection.</p>
    Formula:C15H25ClN4O6
    Color and Shape:Solid
    Molecular weight:392.84
  • COX-2-IN-8


    <p>COX-2-IN-8 (Compound 6a) is a potent, selective, orally active COX-2 inhibitor (IC50: 6.585 μM) with a higher COX-2 selectivity than Celecoxib.</p>
    Formula:C19H19N3O4S2
    Color and Shape:Solid
    Molecular weight:417.5
  • Notch inhibitor 1

    CAS:
    <p>Notch inhibitor 1 blocks Notch 1/3 (IC50: 7.8/8.5 nM) and aids cancer research.</p>
    Formula:C26H25F7N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:574.49
  • Coleon-U-quinone

    CAS:
    <p>Coleon-U-quinone, a P-gp inhibitor, reduces cancer cell viability and enhances Doxorubicin sensitivity in resistant cells.</p>
    Formula:C20H24O5
    Color and Shape:Solid
    Molecular weight:344.4
  • BAY-091

    CAS:
    <p>BAY-091 is a novel potent and highly selective PIP4K2A kinase inhibitor.</p>
    Formula:C26H21FN4O2
    Purity:97.66% - 99.23%
    Color and Shape:Soild
    Molecular weight:440.47
  • Anticancer agent 79


    <p>Anticancer agent 79 (3d) has potent activity against breast cancer, with cytotoxic effects on T47-D, IC50=13.64±0.26μM.</p>
    Formula:C20H12F3NO5
    Color and Shape:Solid
    Molecular weight:403.31
  • MSX-3

    CAS:
    <p>MSX-3 is an antagonist of the A2A adenosine receptor and a prodrug of MSX-2.</p>
    Formula:C21H23N4Na2O7P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:520.389
  • c-Met/HDAC-IN-2

    CAS:
    <p>Potent dual c-Met/HDAC inhibitor, IC50: HDAC1 5.4 nM, c-Met 18.49 nM; anti-cancer, induces apoptosis, G2/M arrest in HCT-116.</p>
    Formula:C34H33N5O7
    Color and Shape:Solid
    Molecular weight:623.66
  • NS2B/NS3-IN-5


    <p>Compound 25b inhibits DENV2/ZIKV NS2B/NS3 proteases; IC50: ZIKV 0.67μM, DENV2 4.38μM.</p>
    Formula:C14H9IN2O3S
    Color and Shape:Solid
    Molecular weight:412.2
  • RSV-IN-7

    CAS:
    <p>RSV-IN-7 (example 253) is a RSV inhibitor ( EC 50 : &lt; 0.4 μΜ) .</p>
    Formula:C27H22F3N7O3
    Color and Shape:Solid
    Molecular weight:549.50
  • CD33 splicing modulator 1


    <p>Compound 1 modulates CD33, affects microglial cells, and may aid in neurodegenerative disease research.</p>
    Formula:C25H25FN6O
    Color and Shape:Solid
    Molecular weight:444.5