Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,787 products)
- Apoptosis(6,265 products)
- Cell Cycle/Checkpoint(4,800 products)
- Chromatin/Epigenetics(2,446 products)
- Cytoskeletal Signaling(1,530 products)
- DNA Damage/DNA Repair(2,964 products)
- Endocrinology/Hormones(3,708 products)
- Enzyme(3,669 products)
- GPCR/G-Protein(9,019 products)
- Immunology and Inflammation(3,883 products)
- Influenza Virus(301 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,248 products)
- Membrane Transporter/Ion Channel(3,038 products)
- Metabolism(10,216 products)
- Microbiology/Virology(7,607 products)
- Neuroscience(10,383 products)
- Other Inhibitors(36,019 products)
- Oxidation-Reduction(42 products)
- PI3K/Akt/mTOR Signaling(1,442 products)
- Proteases/Proteasome(1,726 products)
- Stem Cell and Derivatives(823 products)
- Tyrosine Kinase/Adaptors(2,039 products)
- Ubiquitination(1,718 products)
Show 16 more subcategories
Found 66684 products of "Inhibitors"
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GDC-0349
CAS:<p>GDC-0349 (RG-7603) is a potent and selective ATP-competitive inhibitor of mTOR, 790-fold inhibitory effect against PI3Kα and other 266 kinases. Phase 1.</p>Formula:C24H32N6O3Purity:96.00% - 98.17%Color and Shape:SolidMolecular weight:452.55PF-04979064
CAS:<p>PF-04979064 is a potent and selective PI3K and mTOR dual kinase inhibitor(Ki of 0.13 nM and 1.42 nM,respectively).</p>Formula:C24H26N6O3Purity:98.20% - ≥98%Color and Shape:SolidMolecular weight:446.5PXS-5153A
CAS:PXS-5153A rapidly inhibits lysyl oxidase 2/3 enzymes, blocks activity in 15 mins, and reduces fibrosis.Formula:C20H25Cl2FN4O2SPurity:99.58%Color and Shape:SolidMolecular weight:475.41AMG 837 calcium hydrate
CAS:AMG 837 calcium hydrate is a potent GPR40 agonist with an EC50 of 13 nM.Formula:C52H44CaF6O8Purity:98.07%Color and Shape:SolidMolecular weight:950.97CeMMEC1
CAS:CeMMEC1 is an inhibitor of BRD4, and also has a great affinity for TAF1(IC50=0.9 μM).Formula:C19H16N2O4Purity:98.9% - 99.92%Color and Shape:SolidMolecular weight:336.34Pan-RAS-IN-1
CAS:Pan-RAS-IN-1 is an inhibitor of pan-Ras. It disrupts the interaction of Ras proteins and their effectors.Formula:C36H41Cl2F3N6O2Purity:99.77%Color and Shape:SolidMolecular weight:717.65Ref: TM-T16432
1mg80.00€2mg97.00€5mg144.00€10mg216.00€25mg439.00€50mg660.00€100mg938.00€500mg1,882.00€1mL*10mM (DMSO)221.00€PXS-5120A
CAS:PXS-5120A is an irreversible fluoroallylamine Lysyl Oxidase-like 2/3 (LOXL2/3) inhibitor with anti-fibrotic activity.Formula:C22H25ClFN3O4SPurity:97.02%Color and Shape:SolidMolecular weight:481.97Ref: TM-T12584
1mg216.00€2mg309.00€5mg487.00€10mg645.00€25mg944.00€50mg1,293.00€100mg1,730.00€1mL*10mM (DMSO)530.00€PKC-IN-1
CAS:PKC-IN-1 is an ATP-competitive and reversible conventional PKC enzymes inhibitor (PKCα, PKCβI, PKCβII, PKCθ, PKCγ, PKC mu and PKCε with IC50s of 2.3, 8.1, 7.6,Formula:C25H37FN8O2Purity:98% - 98.79%Color and Shape:SolidMolecular weight:500.61Sorivudine
CAS:Sorivudine (BV-araU) is an antiviral blocking DNA synthesis in viruses like varicella, HSV-1, and Epstein-Barr.Formula:C11H13BrN2O6Purity:99.74%Color and Shape:SolidMolecular weight:349.13HM43239
CAS:HM43239: oral FLT3 inhibitor; IC50: FLT3 WT 1.1nM, ITD 1.8nM, D835Y 1.0nM; blocks p-STAT5/p-ERK; affects SYK, JAK1/2, TAK1; halts leukemia cell growth.Formula:C29H33ClN6Purity:99.7%Color and Shape:SolidMolecular weight:501.07Ref: TM-T9428
1mg49.00€5mg104.00€10mg166.00€25mg325.00€50mg490.00€100mg682.00€200mg903.00€1mL*10mM (DMSO)115.00€Src Inhibitor 3
CAS:Src Inhibitor 3 blocks c-Src kinase (IC50 <3 nM CSK HTRF, <4 nM Caliper), boosting T cell growth from receptor signals.Formula:C34H32ClFN8O4Purity:98.35%Color and Shape:SolidMolecular weight:671.12Ref: TM-T13000
1mg92.00€5mg187.00€10mg320.00€25mg507.00€50mg702.00€100mgTo inquire1mL*10mM (DMSO)279.00€BMS-986176
CAS:<p>AAK1-IN-1 is a highly selective and potent inhibitor of adaptor associated kinase 1 (AAK1, IC50 = 2 nM).</p>Formula:C19H23F4N3OPurity:98.58% - 98.7%Color and Shape:SolidMolecular weight:385.4Lumateperone
CAS:<p>Lumateperone (ITI 722) is a 5HT2A receptor antagonist and a dopamine receptor phosphoprotein modulator (DPPM).</p>Formula:C24H28FN3OPurity:99.68% - 99.91%Color and Shape:SolidMolecular weight:393.5CAY10781
CAS:CAY10781 inhibits NRP-1/VEGF-A binding by 43% at 12.5μM and blocks VEGFR2 phosphorylation in CAD cells.Formula:C11H9N3O3Purity:99.49%Color and Shape:SolidMolecular weight:231.21Ref: TM-T37424
2mg42.00€5mg57.00€10mg81.00€25mg131.00€50mg180.00€100mg334.00€200mg467.00€1mL*10mM (DMSO)84.00€PKI-402
CAS:PKI-402 is a potent PI3K and mTOR inhibitor. PKI-402 inhibits PI3Kα, mTOR, PI3Kβ, PI3Kδ and PI3Kγ with IC50s of 2, 3, 7, 14 and 16 nM, respectively.Formula:C29H34N10O3Purity:99.94%Color and Shape:SolidMolecular weight:570.65MK-8353
CAS:MK-8353 (SCH900353) is a potent, selective and orally available inhibitor of ERK1/2 (IC50s of 23.0 nM and 8.8 nM, respectively)Formula:C37H41N9O3SPurity:96.15% - 97.19%Color and Shape:SolidMolecular weight:691.84Ref: TM-T12069
1mg81.00€2mg97.00€5mg156.00€10mg271.00€25mg588.00€50mg938.00€100mg1,415.00€1mL*10mM (DMSO)230.00€INCB3344
CAS:INCB3344 is an effective, specific and orally bioavailable CCR2 antagonist with IC50 values of 9.5 nM (mCCR2) and 5.1 nM (hCCR2) in binding antagonism and 7.8Formula:C29H34F3N3O6Purity:98% - 98.2%Color and Shape:SolidMolecular weight:577.59Ref: TM-TQ0103
1mg70.00€5mg153.00€10mg243.00€25mg378.00€50mg540.00€100mg747.00€200mg1,026.00€1mL*10mM (DMSO)188.00€SB-616234-A
CAS:SB-616234-A is a selective and orally bioavailable antagonist of 5-HT1B receptor, with anxiolytic and antidepressant activity.Formula:C32H36ClN5O3Purity:99.72%Color and Shape:SolidMolecular weight:574.11GSK-F1
CAS:GSK-F1 (PI4KA inhibitor-F1) is a novel potent PI4KA inhibitor.Formula:C27H18F5N5O4SPurity:97.03%Color and Shape:SolidMolecular weight:603.52Ref: TM-T19840
1mg110.00€5mg226.00€10mg335.00€25mg538.00€50mg730.00€100mg938.00€200mg1,320.00€1mL*10mM (DMSO)320.00€Y06137
CAS:<p>Y06137, selective BET inhibitor, Kd 81 nM for BRD4(1), researched for castration-resistant prostate cancer treatment.</p>Formula:C27H32N4O2Purity:99.85%Color and Shape:SolidMolecular weight:444.57
