Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,781 products)
- Apoptosis(6,260 products)
- Cell Cycle/Checkpoint(4,792 products)
- Chromatin/Epigenetics(2,440 products)
- Cytoskeletal Signaling(1,527 products)
- DNA Damage/DNA Repair(2,968 products)
- Endocrinology/Hormones(3,706 products)
- Enzyme(3,667 products)
- GPCR/G-Protein(9,005 products)
- Immunology and Inflammation(3,874 products)
- Influenza Virus(301 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,248 products)
- Membrane Transporter/Ion Channel(3,033 products)
- Metabolism(10,207 products)
- Microbiology/Virology(7,591 products)
- Neuroscience(10,382 products)
- Other Inhibitors(36,042 products)
- Oxidation-Reduction(42 products)
- PI3K/Akt/mTOR Signaling(1,444 products)
- Proteases/Proteasome(1,724 products)
- Stem Cell and Derivatives(825 products)
- Tyrosine Kinase/Adaptors(2,035 products)
- Ubiquitination(1,717 products)
Show 16 more subcategories
Found 66686 products of "Inhibitors"
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Inz-5
CAS:Inz-5 is a fungal-selective inhibitor of mitochondrial cytochrome bc1. Inz-5 impairs fungal virulence. It also prevents the evolution of drug resistance.Formula:C18H14F4N6Color and Shape:SolidMolecular weight:390.34Cindunistat HCl maleate
CAS:Cindunistat, a potent oral iNOS inhibitor for symptomatic knee osteoarthritis.Formula:C20H39ClN6O8S2Color and Shape:SolidMolecular weight:591.14JTT 551
CAS:JTT 551: Selective PTP1B inhibitor for type 2 diabetes research; Ki=0.22μM for PTP1B, 9.3μM for TCPTP.Formula:C34H43N3O3S2Purity:98%Color and Shape:SolidMolecular weight:605.85UCPH-102
CAS:UCPH-102: Selective EAAT1 inhibitor, IC50 0.43 μM, treats Alzheimer's, ALS, chronic pain, OCD; crosses blood-brain barrier, targets T-ALL cells.Formula:C21H18N2O2Color and Shape:SolidMolecular weight:330.38Triiodothyronine Sulfate
CAS:Triiodothyronine sulfate: Hypothyroidism prodrug, metabolizes into active thyroid hormone T3, binds and activates TRβ1.Formula:C15H11I3NNaO7SPurity:98%Color and Shape:SolidMolecular weight:753.02TRAP-6-IN-1
CAS:TRAP-6-IN-1 inhibits collagen/TRAP-6, IC50: 17.12/11.88 μM, blocks platelet aggregation.Formula:C18H20O3Color and Shape:SolidMolecular weight:284.35FWM-4
CAS:FWM-4 is a potent inhibitor of SARS-COV-2 NSP13 decapping enzyme.Formula:C24H18N4O4Color and Shape:SolidMolecular weight:426.42THR-β modulator-1
CAS:THR-β Modulator-1 (Compound 1a) is a potent modulator of the thyroid hormone receptor β, utilized in the study of thyroid hormone receptor-associated disordersFormula:C17H14Cl2N6O4Color and Shape:SolidMolecular weight:437.24Vinaxanthone
CAS:Vinaxanthone (SM-345431), an extract from Penicillium chrysogenum, is a semaphorin3A inhibitor with antimicrobial activity.Formula:C28H16O14Purity:82.56% - 97.8%Color and Shape:SolidMolecular weight:576.42Prenalterol hydrochloride
CAS:Prenalterol HCl: beta 1-specific agonist; treats acute cardiac failure, shock, low-output post-MI, Shy-Drager syndrome.Formula:C12H20ClNO3Color and Shape:SolidMolecular weight:261.75IDH1 Inhibitor 5
CAS:IDH1 Inhibitor 5 targets MOG cells (IC50: 64.4 nM) and R132H mutant IDH1 gliomas (IC50: 34.9 nM).Formula:C26H34N4O3Color and Shape:SolidMolecular weight:450.57Antifungal agent 50
CAS:Antifungal agent 50 exhibits minimum inhibitory concentrations (MICs) ranging from less than 0.063 to 1 μg/mL [1].Formula:C25H20ClN5O2SColor and Shape:SolidMolecular weight:489.98CDK7-IN-14
CAS:CDK7-IN-14, a potent CDK7 inhibitor from pyrimidines, may treat transcriptionally dysregulated cancers (CN114249712A).Formula:C22H24F3N6OPPurity:99.48%Color and Shape:SolidMolecular weight:476.43CP-113818
CAS:CP-113818 is a potent inhibitor of cholesterol acyltransferase (ACAT) and can be used to study Alzheimer's disease.Formula:C24H42N2OS3Color and Shape:SolidMolecular weight:470.8Mevociclib
CAS:Mevociclib (SY-1365) is a highly selective covalent inhibitor of CDK7. SY-1365 possesses therapeutic potential in both hematological and solid tumors.Formula:C31H35ClN8O2Purity:98.02% - 98.02%Color and Shape:SolidMolecular weight:587.11Edobacomab
CAS:Edobacomab (E5), a monoclonal IgM antibody targeting endotoxin, is utilized in the study of sepsis stemming from Gram-negative bacterial infections [1].Color and Shape:LiquidCIDD-0149897
CAS:<p>CIDD-0149897 is a potent, selective, and brain-penetrant agonist of ERβ that exhibits antitumor activity in glioblastoma [1].</p>Formula:C15H10FNO3Purity:98%Color and Shape:SolidMolecular weight:271.24NS5A-IN-2
CAS:NS5A-IN-2, a potent inhibitor, is highly effective against HCV 1b and shows increased activity for GT 3a with good metabolic stability.Formula:C46H45N7O7Purity:98%Color and Shape:SolidMolecular weight:807.89CYM50260
CAS:<p>CYM50260 is a potent and exquisitely selective agonist of sphingosine-1-phosphate 4 receptor (S1P4-R, EC50= nM) with no activity against S1P1-R, S1P2-R, S1P3-R</p>Formula:C14H11Cl3FNO2Purity:99.88%Color and Shape:SolidMolecular weight:350.6N-Demethyl Mifepristone
CAS:N-Demethyl Mifepristone (RU 42633), an active metabolite of Mifepristone, exhibits 61% of the affinity for the glucocorticoid receptor relative to Mifepristone'Formula:C28H33NO2Purity:98%Color and Shape:SolidMolecular weight:415.57MARK-IN-2
CAS:MARK-IN-2 is a potent microtubule affinity regulating kinase (MARK) inhibitor,(IC50:5 nM).Formula:C18H18ClF2N5OSPurity:98%Color and Shape:SolidMolecular weight:425.88Ilepatril
CAS:Ilepatril, also known as AVE-7688, is a vasopeptidase inhibitor for the treatment of hypertension.Formula:C22H28N2O5SColor and Shape:SolidMolecular weight:432.5322-(4′-py)-JA
CAS:<p>22-(4′-py)-JA, a semisynthetic derivative of junamycin A isolated from the Thai blue sponge (Xestospongia sp.), exhibits antimetastatic properties by inhibiting</p>Formula:C32H30N4O8Purity:98%Color and Shape:SolidMolecular weight:598.6CI 972 anhydrous
CAS:CI 972 anhydrous is an inhibitor of purine nucleoside phosphorylase (PNP) (Ki: 0.83 μM) used as a T cell-selective immunosuppressive agent.Formula:C11H12ClN5OSPurity:98%Color and Shape:SolidMolecular weight:297.76L-690488
CAS:L-690488 has more effective cell penetration than L-690330. L-690488 is a prodrug of L-690330 and is a selective inositol monophosphatase (IMPase) inhibitor.Formula:C32H52O16P2Purity:98%Color and Shape:SolidMolecular weight:754.69USP7-IN-1
CAS:USP7-IN-1 is a selective and reversible ubiquitin-specific protease 7 (USP7) inhibitor (IC50 = 77 μM).Formula:C23H24ClN3O3Purity:99.82%Color and Shape:SolidMolecular weight:425.91Ref: TM-T13268
1mg97.00€5mg188.00€10mg284.00€25mg452.00€50mg645.00€100mg867.00€200mg1,130.00€1mL*10mM (DMSO)217.00€BRD7-IN-1
CAS:BRD7-IN-1, a BI7273 derivative, forms PROTAC VZ185, targeting BRD7/9 with DC50s of 4.5/1.8 nM via VHL ligand linkage.Formula:C22H28Cl2N4O3Purity:98.95%Color and Shape:SolidMolecular weight:467.39Ref: TM-T17697
1mg99.00€2mg144.00€5mg235.00€10mg354.00€25mg635.00€50mg944.00€100mg1,311.00€200mgTo inquire1mL*10mM (DMSO)240.00€PPO-IN-2
CAS:PPO-IN-2 is a protoporphyrinogen IX oxidase inhibitor, exhibiting a Ki value of 16 nM [1].Formula:C17H15ClFN3O2S2Color and Shape:SolidMolecular weight:411.9β-Lactamase-IN-8
CAS:β-Lactamase-IN-8 (compound 20) is a potent and oral bioavailable broad-spectrum cyclic boronate β-lactamase inhibitor that can be used for researchingFormula:C10H14BNO4SColor and Shape:SolidMolecular weight:255.1KP496
CAS:KP496 is a selective, dual antagonist for Thromboxane A2 receptor and Leukotriene D4 receptor.Formula:C31H34ClN3O7S3Purity:98%Color and Shape:SolidMolecular weight:692.27TGFβ-IN-5
CAS:TGFβ-IN-5 (WAY-641966) is a potent TGFβ inhibitor with anti-prion activity for the study of fibroproliferative diseases associated with TGF-β signaling.Formula:C20H16N4Purity:99.29% - 99.62%Color and Shape:SolidMolecular weight:312.37TRPC5 modulator-1
CAS:TRPC5 modulator-1 (Compound 9) is a TRPC5 modulator (IC50<1 nM) that can be used to study neuropsychiatric disorders.Formula:C23H27FN2O4Color and Shape:SolidMolecular weight:414.47Perindopril acyl-β-D-glucuronide
CAS:Perindopril acyl-β-D-glucuronide is a metabolite of the ACE inhibitor perindopril [1].Formula:C25H40N2O11Purity:98%Color and Shape:SolidMolecular weight:544.59KMG-301AM
KMG-301AM, a fluorophore, allows for tracking mitochondrial changes over time with pseudo-colored imagery.Formula:C30H28N3O6Purity:98%Color and Shape:SolidMolecular weight:526.56ATI-22-107
CAS:ATI-22-107 is a positive cardiac inotropic agent which may affect myocyte calcium cycling and contractility.Formula:C31H32Cl2N4O8Color and Shape:SolidMolecular weight:659.51WRN inhibitor 2
CAS:WRN Inhibitor 2 (example 118), a potent inhibitor of the WRN (Werner Syndrome ATP-dependent helicase enzyme), exhibits a pIC50 value of 7.0 or greater [1].Formula:C15H11F3N2O5S2Purity:98%Color and Shape:SolidMolecular weight:420.38(R)-BDP9066
CAS:(R)-BDP9066 blocks MRCK to curb cancer cell spread, aiding research on diseases like cancer.Formula:C20H24N6Color and Shape:SolidMolecular weight:348.44Prohexadione calcium
CAS:Prohexadione calcium (BX-112) is a plant growth regulator that inhibits gibberellin biosynthesis in plants [1] [2].Formula:C10H11O5CaCaPurity:98%Color and Shape:SolidMolecular weight:251.27SQ 26655
CAS:SQ 26655 is an antagonist of thromboxane A2/prostaglandin H2.Formula:C21H34O4Purity:98%Color and Shape:SolidMolecular weight:350.49WAY-271999
CAS:WAY-271999 is an active molecule.Formula:C11H7ClN2O3Color and Shape:SolidMolecular weight:250.64dBRD4-BD1
CAS:dBRD4-BD1 selectively inhibits and degrades BRD4 (DC50=280nM), upregulates BRD2/3, and aids in creating BRD4-specific probes.Formula:C50H53F3N8O9Color and Shape:SolidMolecular weight:967A 56234
CAS:A 56234 is a high-ceiling diuretic.Formula:C16H9ClFKNO4Color and Shape:SolidMolecular weight:372.8T-0632
CAS:T-0632 is a potent and selective antagonist of CCKA receptor.Formula:C28H22FN3NaO5Purity:98%Color and Shape:SolidMolecular weight:522.488AXL-IN-14
CAS:AXL-IN-14: orally active, potent AXL inhibitor (IC50=0.8 nM); hinders Gas6/AXL migration, invasion; lowers p-AXL, p-AKT; anti-tumor.Formula:C32H24F2N4O4Purity:98%Color and Shape:SolidMolecular weight:566.55RORγt inverse agonist 14
CAS:RORγt inverse agonist 14 (8e) is a potent, selective, and orally active compound with an EC50 of 2.5 nM, exhibiting anti-inflammatory activity.Formula:C26H26F8N2O6S2Purity:98%Color and Shape:SolidMolecular weight:678.61RIP2 kinase inhibitor 1
CAS:Potent RIP2 kinase inhibitor with 0.03 μM IC50, selective for autoimmune disease treatment.Formula:C17H17N5O2SPurity:98%Color and Shape:SolidMolecular weight:355.41N-(2-Hydroxyphenyl)picolinamide
CAS:N-(2-Hydroxyphenyl)picolinamide is an active molecular compound.Formula:C12H10N2O2Color and Shape:SolidMolecular weight:214.22Elisartan
CAS:Elisartan is a non-peptide pro-drug of angiotensin II AT1 receptor antagonist HN-12206. It also shows anti-hypertension activities.Formula:C27H29ClN6O5Purity:98%Color and Shape:SolidMolecular weight:553.01TRPV2-selective blocker 1
CAS:TRPV2-selective blocker 1 (compound IV2-1) is a selective inhibitor of the TRPV2 channel, exhibiting an IC50 value of 6.3 μM.Formula:C15H18OS2Color and Shape:SolidMolecular weight:278.43Valtorcitabine dihydrochloride
CAS:Valtorcitabine dihydrochloride, a DNA polymerase inhibitor, is used potentially for the treatment of HBV infection.Formula:C14H24Cl2N4O5Color and Shape:SolidMolecular weight:399.27Tedizolid HCl (856866-72-3 free base)
Tedizolid HCl, a novel oxazolidinone antibiotic, IC50: MAO-A 8.7 uM, MAO-B 5.7 uM, approved post-linezolid, has a prodrug form tedizolid phosphate.Formula:C17H16ClFN6O3Purity:98%Color and Shape:SolidMolecular weight:406.8Satigrel
CAS:Satigrel is a new antiplatelet agent. It also inhibits platelet accumulation in prosthetic arterial grafts.Formula:C20H19NO4Purity:98%Color and Shape:SolidMolecular weight:337.37Pumaprazole
CAS:Pumaprazole (BY-841) is an antagonist of a reversible proton pump.Formula:C19H22N4O2Purity:99.91%Color and Shape:SolidMolecular weight:338.4Ref: TM-T16682
1mg92.00€5mg188.00€10mg311.00€25mg635.00€50mg1,017.00€100mg1,644.00€200mg2,213.00€1mL*10mM (DMSO)215.00€Pentabromopseudilin
CAS:Pentabromopseudilin (PBrP), a marine antibiotic derived from Pseudomonas bromoutilis and Alteromonas luteoviolaceus, demonstrates antimicrobial, antitumor, andFormula:C10H4Br5NOColor and Shape:SolidMolecular weight:553.66NB-506 Free Base
CAS:NB-506 Free Base is an indolocarbazole antitumor agent; a DNA topoisomerase I inhibitor.Formula:C27H22N4O10Color and Shape:SolidMolecular weight:562.48Eleven-Nineteen-Leukemia Protein IN-2
CAS:Eleven-Nineteen-Leukemia Protein IN-2 (compound 23), an ENL inhibitor, exhibits an IC50 of 10.7 nM and is utilized for leukemia research [1].Formula:C22H23N5O2Purity:98%Color and Shape:SolidMolecular weight:389.45WYE-132
CAS:WYE-125132: potent mTOR inhibitor, IC50 0.19 nM, selective over PI3Ks/hSMG1/ATR.Formula:C27H33N7O4Purity:99.16%Color and Shape:SolidMolecular weight:519.6INT-767
CAS:INT-767 is a highly potent farneson X receptor (FXR)/TGR5 dual agonist that prevents NASH and promotes visceral fat brown lipogenesis and mitochondrial functionFormula:C25H43NaO6SPurity:98%Color and Shape:SolidMolecular weight:494.66Glycosidase-IN-1
CAS:Glycosidase-IN-1, a D-mannose-derived inhibitor, has hypoglycemic effects and aids in creating immunosuppressants and β-glucosidase blockers.Formula:C13H23NO5Purity:98%Color and Shape:SolidMolecular weight:273.33Lepadin H
CAS:Lepadin H, a marine alkaloid and ferroptosis inducer, exhibits significant cytotoxicity by promoting p53 expression, escalating ROS production, and enhancingFormula:C26H45NO3Purity:98%Color and Shape:SolidMolecular weight:419.64Calicheamicin
CAS:Calicheamicin (Calicheamicin γ1) is an antitumor antibiotic and is a DNA synthesis inhibitor. It also is a cytotoxic agent that causes double-strand DNA breaks.Formula:C55H74IN3O21S4Purity:98.22% - 98.78%Color and Shape:SolidMolecular weight:1368.35O-Demethyl apixaban sulfate
CAS:O-Demethyl apixaban sulfate, a metabolite of the factor Xa inhibitor Apixaban, is in development for treating thrombotic diseases.Formula:C24H23N5O7SColor and Shape:SolidMolecular weight:525.53Abediterol
CAS:Abediterol (LAS100977): potent, long-acting beta-2 agonist for asthma and COPD treatment.Formula:C25H30F2N2O4Color and Shape:SolidMolecular weight:460.51CAXII-IN-1
CAS:CAXII-IN-1, antitumor, selectively inhibits CA XII with Ki of 3.8 nM for hCA XII and 56 nM for hCA IX.Formula:C13H7Cl2NO3SColor and Shape:SolidMolecular weight:328.17Cinsebrutinib
CAS:Cinsebrutinib, a Bruton's tyrosine kinase inhibitor, holds potential for research in cancer treatment.Formula:C22H26FN3O2Purity:98%Color and Shape:SolidMolecular weight:383.46A 77003
CAS:A 77003 is a HIV-1 protease inhibitor. A77003 impairs HIV-1 protease-mediated Gag processing.Formula:C44H58N8O6Color and Shape:SolidMolecular weight:794.98Ro 48-6791
CAS:Ro 48-6791, a GABA receptor agonist, is used potentially for anesthesia.Formula:C21H25FN6O2Color and Shape:SolidMolecular weight:412.46Therapeutic agent-1
CAS:Therapeutic Agent-1, a heteroaryl compound, serves as an enzyme replacement therapy to enhance glucocerebrosidase activity in the treatment of Gaucher disease [Formula:C18H20N6Color and Shape:SolidMolecular weight:320.39Altenusin
CAS:Altenusin is a natural nonsteroidal fungal metabolite, as a novel selective agonist of FXR with an EC50 value of 3.2 ± 0.2 μM.Formula:C15H14O6Purity:98.97% - 99.87%Color and Shape:SolidMolecular weight:290.27Tenalisib R Enantiomer
CAS:Tenalisib R Enantiomer is an R enantiomer of Tenalisib .Formula:C23H18FN5O2Purity:98%Color and Shape:SolidMolecular weight:415.42WAY-621924
CAS:<p>WAY-621924 is an active molecule.</p>Formula:C17H14N2O2SColor and Shape:SolidMolecular weight:310.37UFP-512
CAS:UFP-512 is a selective delta-opioid (DOP) receptor agonist.Formula:C31H33N5O5Purity:98%Color and Shape:SolidMolecular weight:555.62PQM130
CAS:PQM130 is a Feruloyl-Donepezil Hybrid compound against the neurotoxicity induced by Aβ1-42 oligomer (AβO) and shows anti-inflammatory activity.Formula:C23H27NO4Purity:98.73%Color and Shape:SolidMolecular weight:381.46MET kinase-IN-3
CAS:MET kinase-IN-3 is a potent, orally active MET inhibitor (IC50: 9.8 nM) that exhibits good broad-spectrum anti-proliferative effects on cancer cells.Formula:C25H16ClF2N5O2Color and Shape:SolidMolecular weight:491.88Antibacterial agent 159
CAS:Compound 6d (Antibacterial agent 159) is an antibiotic effective against impetigo and Clostridium difficile infection (CDI), with no observed recurrence for CDIFormula:C51H50N16O10S6Purity:98%Color and Shape:SolidMolecular weight:1239.4310β,17β-dihydroxyestra-1,4-dien-3-one
CAS:10β,17β-dihydroxyestra-1,4-dien-3-one (DHED) has neuroprotective effects, can improve cognitive dysfunction, and can be used to study brain injury.Formula:C18H24O3Color and Shape:SolidMolecular weight:288.38Raf inhibitor 3
CAS:Raf inhibitor 3 (Example 30), a potent inhibitor of both B-Raf and C-Raf, exhibits IC50 values below 15 nM. It is applicable in cancer research studies [1].Formula:C18H19FN8O2SPurity:98%Color and Shape:SolidMolecular weight:430.46Bocodepsin hydrochloride
CAS:Bocodepsin hydrochloride (OKI-179) is a selective HDAC inhibitor with antitumor properties, efficacious via oral administration.Formula:C26H40ClN5O6S2Purity:98%Color and Shape:SolidMolecular weight:618.21SOS1-IN-13
CAS:SOS1-IN-13 inhibits SOS1 (IC50: 6.5 nM) and pERK (327 nM); potential in cancer research.Formula:C21H22F3N3O2Color and Shape:SolidMolecular weight:405.41MS-444
CAS:MS-444 (BE-34776) is an MLCK and HuR inhibitor with antitumor activity that can be used to study triple-negative breast cancer and colorectal cancer.Formula:C13H10O4Purity:99.45% - 99.45%Color and Shape:SolidMolecular weight:230.22K-Ras G12C-IN-1
CAS:K-Ras G12C-IN-1 is a novel and irreversible inhibitor of mutant K-ras G12C.Formula:C22H23Cl2N3O3Color and Shape:SolidMolecular weight:448.34Colletofragarone A2
CAS:Colletofragarone A2 from Colletotrichum sp. blocks mutant p53 and HSP90, aiding cancer treatment.Formula:C22H26O6Color and Shape:SolidMolecular weight:386.44Oxicodegol trifluoroacetate
CAS:Oxicodegol trifluoroacetate is a mu-opioid agonist used in the treatment of Moderate to Severe Chronic Low Back PainFormula:C33H48F3NO11Color and Shape:SolidMolecular weight:691.74AEG40730 HCl
CAS:AEG40730: A potent, selective IAP inhibitor, induces cIAP1/2 degradation, reduces RIP1 ubiquitination, and depletes XIAP, c-IAP1.Formula:C52H70Cl2F6N8O8Color and Shape:SolidMolecular weight:1120.0704Hypusine
CAS:Hypusine is an N-terminal amino alcohol derivative of Lys occurring in bovine brain &Formula:C10H23N3O3Color and Shape:SolidMolecular weight:233.31CDD-1733
CAS:<p>CDD-1733 is a potent, non-covalent, and non-peptide inhibitor of the SARS-CoV-2 main protease (Mpro) with an inhibition constant (K i) of 12 nM.</p>Formula:C34H32F3N5O2Purity:98%Color and Shape:SolidMolecular weight:599.65Firuglipel
CAS:Firuglipel is an orally available and selective agonist of GPR119.Formula:C25H26FN3O5Purity:98%Color and Shape:SolidMolecular weight:467.49KRAS G12C inhibitor 28
CAS:KRAS G12C Inhibitor 28 is a compound that effectively inhibits the KRAS G12C mutation, exhibiting potent antitumor effects with an inhibitory concentration (Formula:C33H36F2N5O4PColor and Shape:SolidMolecular weight:635.64Bromodomain inhibitor-12 (edisylate)
CAS:Bromodomain Inhibitor-12 Edisylate (example 303) serves as a bromodomain inhibitor applicable to autoimmune and inflammatory disease research [1].Formula:C30H44N4O11S2Purity:98%Color and Shape:SolidMolecular weight:700.82AMOR
CAS:AMOR is unique to plant cell walls and enhances plant fertilization efficiency and capacityFormula:C13H22O12Color and Shape:SolidMolecular weight:370.31Methyl 12-methyltridecanoate
CAS:<p>Methyl 12-methyltridecanoate ((R)-betaxolol hydrochloride), a biosurfactant derived from Brevibacterium casei LS14, enhances the biocompatibility of</p>Formula:C15H30O2Purity:98%Color and Shape:SolidMolecular weight:242.4RNA polymerase II-IN-1
CAS:RNA polymerase II-IN-1 (19iv), an amatoxin, inhibits Pol II at 36.66 nM IC50, is more toxic to cancer cells, less to normal cells than α-Amanitin.Formula:C38H53N11O12SPurity:98%Color and Shape:SolidMolecular weight:887.96JYL-1511
CAS:JYL-1511 is the TRPV1 channel partial agonist.Formula:C21H29N3O3S2Purity:98%Color and Shape:SolidMolecular weight:435.6CI-949
CAS:CI-949 inhibits LTC4/D4, histamine, TXB2 release (IC50: 0.5, 11.4, 0.1 μM).Formula:C20H20N6O3Purity:98%Color and Shape:SolidMolecular weight:392.41Amebucort
CAS:Amebucort is a synthetic glucocorticoid corticosteroid. It may used for the research of inflammatory disorders.Formula:C28H40O7Purity:98%Color and Shape:SolidMolecular weight:488.61Dasolampanel etibutil
CAS:Dasolampanel etibutil is a novel selective antagonist of ionotropic glutamate receptor 5 (iGluR5).Formula:C23H32ClN5O3Color and Shape:SolidMolecular weight:461.98RK-0133114
RK-0133114, R-enantiomer of RK-701, is a G9a inhibitor (IC50 = 3.7 μM) for SCD research.Formula:C26H30N4O3Color and Shape:SolidMolecular weight:446.54IMD-biphenylC
CAS:IMD-biphenylC: New, dual-action imidazoquinolinone dimer; inhibits tumor growth, low inflammation/toxicity.Formula:C35H33N5O3Purity:98%Color and Shape:SolidMolecular weight:571.67FLT3-IN-14
CAS:FLT3-IN-14: FLT3 inhibitor; FLT3-WT IC50=5.6nM, FLT3-ITD IC50=1.4nM; blocks Y591 phosphorylation; G1 arrest; pro-apoptotic.Formula:C25H24N6O2SColor and Shape:SolidMolecular weight:472.56Pazelliptine
CAS:Pazelliptine is a DNA topoisomerase inhibitor and antitumor drug.Formula:C22H27N5Color and Shape:SolidMolecular weight:361.48E235
CAS:<p>E235, an activator of the transcription factor 4 (ATF4), enhances the integrated stress response (ISR) and DNA damage response, thereby reducing cell viability</p>Formula:C28H25FN4OSPurity:98.85%Color and Shape:SolidMolecular weight:484.59MC-Val-Cit-PAB-NH-C2-NH-Boc
CAS:MC-Val-Cit-PAB-NH-C2-NH-Boc is a cathepsin-cleavable ADC linker utilized in constructing antibody-drug conjugates (ADCs) [1].Formula:C36H54N8O10Color and Shape:SolidMolecular weight:758.86ICMT-IN-18
CAS:ICMT-IN-18 (compound 35) serves as an ICMT inhibitor with an IC50 value of 0.066 μM [1].Formula:C22H26N2OColor and Shape:SolidMolecular weight:334.45JT002
CAS:JT002 is an orally active NLRP3 inflammasome inhibitor that decreases the production of NLRP3-dependent proinflammatory cytokines (such as IL-1β, IL-1α, IL-18)Formula:C20H24N4O5SPurity:98%Color and Shape:SolidMolecular weight:432.49Biotin-PEG7-Maleimide
CAS:Biotin-PEG7-Maleimide is a biotinylation agent that selectively binds to thiol (SH) groups and is utilized in the synthesis of Drug-Linker Conjugates forFormula:C33H55N5O12SPurity:98.76%Color and Shape:SolidMolecular weight:745.88HSP90/mTOR-IN-1
"HSP90/mTOR-IN-1 is a dual Hsp90/mTOR inhibitor (IC50: 69/29 nM), halting SW780 cell growth and inducing apoptosis/autophagy in cancer research."Formula:C36H34ClFN6O5SColor and Shape:SolidMolecular weight:717.21L 743310
CAS:L 743310 is an antagonist of the neurokinin-1 receptor.Formula:C30H33BrF6N4O2Purity:98%Color and Shape:SolidMolecular weight:675.5CM-10-18
CAS:CM-10-18: potent ER α-glucosidase inhibitor, strong antiviral against hemorrhagic fever viruses, protects mice from dengue fatality.Formula:C17H35NO5Color and Shape:SolidMolecular weight:333.46Cladosporin
CAS:Cladosporin, from Cladosporium cladosporioid fungus, halts dermatophyte growth on agar at 75 μg/mL.Formula:C16H20O5Color and Shape:SolidMolecular weight:292.33GABA-IN-2
CAS:GABA-IN-2 (Compound 5), a GABA inhibitor, exhibits both larvicidal and insecticidal properties, achieving an 87% mortality rate at a concentration of 50 mg/L [1Formula:C12H4Cl2F6N4SeColor and Shape:SolidMolecular weight:468.0415(S)-HEDE
CAS:15(S)-HEDE is produced from 11Z,14Z-eicosadienoic acid by 15-LO. 15(S)-HEDE is an inhibitor of RBL-1 cell 5-LO with an IC50 value of 26 μM.Formula:C20H36O3Color and Shape:SolidMolecular weight:324.5KRIBB3
CAS:KRIBB3: novel anticancer microtubule inhibitor; halts MDA-MB-231 cell migration/invasion by targeting Hsp27 phosphorylation.Formula:C19H19NO4Color and Shape:SolidMolecular weight:325.36Brivudine monophosphate
CAS:Brivudine monophosphate, a phosphate ester, inhibits DNA repair, induces apoptosis, and may downregulate STAT3 and chemoresistance genes.Formula:C11H14BrN2O8PColor and Shape:SolidMolecular weight:413.12Bcl-2-IN-11
CAS:Bcl-2-IN-11 (compound 6) is a potent and selective inhibitor of Bcl-2 activity, exhibiting an IC50 of 0.9 nM, and demonstrates minimal inhibition against Bcl-xlFormula:C45H49ClFN7O8SColor and Shape:SolidMolecular weight:902.43Glycolithocholic acid
CAS:Glycolithocholic acid (Lithocholic acid glycine conjugate) is a glycine conjugate of lithocholic acid.Formula:C26H43NO4Purity:99.75% - 99.83%Color and Shape:SolidMolecular weight:433.62ICI-M247496
CAS:ICI-M247496 is a non-polyglutamated analog of CB3717 and quinazoline-based inhibitor of thymidylate synthase.Formula:C19H16N4O3Color and Shape:SolidMolecular weight:348.36IDO1/2-IN-1
CAS:First potent oral dual IDO1/IDO2 inhibitor with antitumor properties; IC50: 28 nM (IDO1), 144 nM (IDO2).Formula:C16H18BrFN8O4Color and Shape:SolidMolecular weight:485.27PPARδ agonist 9
CAS:PPARδ agonist 9 (compound 21), with an EC50 of 3.6 nM, is effective in vivo, decreasing serum MCP-1 concentrations in mice and markedly reducing atheroscleroticFormula:C26H28ClF3N4O3SPurity:98%Color and Shape:SolidMolecular weight:569.04PR-104A
CAS:PR-104A is a hypoxia-targeted anticancer agent.Formula:C14H19BrN4O9SColor and Shape:SolidMolecular weight:499.29TCS 46b
CAS:TCS 46b is a NR1A/NR2B NMDA receptor antagonist with oral activity.Formula:C22H23N3OPurity:99.78% - 99.78%Color and Shape:SolidMolecular weight:345.44(Iso)-MS4322
CAS:(Iso)-MS4322 ((Iso)-YS43-22) is a protein arginine methyltransferase 5 (PRMT5 ) degrader with potential anticancer activity.Formula:C55H76N10O12SPurity:99.05% - 99.79%Color and Shape:SolidMolecular weight:1101.32Cgp 6809
CAS:CGP 6809: a methylnitrosoureido-sugar derivative active against various mice/rat tumors; promising for bowel/lung cancer trials.Formula:C12H23N3O7Color and Shape:SolidMolecular weight:321.33ZLN024
CAS:ZLN024 is an activator of AMPK allosteric.Formula:C13H13BrN2OSPurity:99.751%Color and Shape:SolidMolecular weight:325.22Ref: TM-T13411
1mg87.00€5mg187.00€10mg284.00€25mg452.00€50mg645.00€100mg867.00€200mg1,130.00€1mL*10mM (DMSO)188.00€Aminoguanidine hemisulfate
CAS:Aminoguanidine hemisulfate, an inhibitor of nitric oxide synthases (NOS) and reactive oxygen species (ROS), effectively suppresses ANE-induced ROS production inFormula:CH6N4H2SO4Purity:98%Color and Shape:SolidMolecular weight:123.115JA-ACC
CAS:Jasmonyl-ACC (JA-ACC), a derivative of 1-aminocyclopropane-1-carboxylic acid (ACC)—the direct precursor to ethylene—impedes root growth in Arabidopsis, withFormula:C16H23NO4Color and Shape:SolidMolecular weight:293.36ML-090
CAS:ML-090 is NOX1-specific inhibitor(IC50 = 90 nM) which is >100 selectivity for NOX1 over NOX2, NOX3, NOX4 (all IC50s >10 μM).Formula:C14H10N4Purity:98.55%Color and Shape:SolidMolecular weight:234.26h-NTPDase-IN-5
CAS:h-NTPDase-IN-5 (compound 3b) serves as a pan-inhibitor of NTPDase, exhibiting inhibitory concentration 50 (IC50) values of 1.10 μM (h-NTPDase1), 44.73 μM (h-Formula:C23H21N3O2SPurity:98%Color and Shape:SolidMolecular weight:403.5CDK9-IN-29
CAS:<p>CDK9-IN-29 (compound Z11) is a potent inhibitor of CDK9, exhibiting high kinase selectivity and an IC50 value of 3.20 nM.</p>Formula:C29H33F2N5O4Purity:98%Color and Shape:SolidMolecular weight:553.6Axl/Mer/CSF1R-IN-1
CAS:Axl/Mer-IN-1 is a compound that functions as an inhibitor for Axl/Mer receptor tyrosine kinase (Axl/Mer RTK) and CSF1R, exhibiting dissociation constants (Kds)Formula:C25H24F3N5O5Color and Shape:SolidMolecular weight:531.48PD 168368
CAS:PD 168368 is a mixed neuromodulin B receptor (NMB-R) antagonist and potent FPR1/FPR2/FPR3 agonist that inhibits the gastrin-releasing peptide receptor.Formula:C31H34N6O4Purity:98.11% - 99.87%Color and Shape:SolidMolecular weight:554.64Ref: TM-T8691
1mg88.00€5mg170.00€10mgTo inquire25mg518.00€50mgTo inquire100mgTo inquire1mL*10mM (DMSO)To inquireNBI-35965
CAS:<p>NBI-35965 is a CRF1 receptor antagonist.</p>Formula:C21H22Cl2N4Color and Shape:SolidMolecular weight:401.33CD235
CAS:CD235 is a structurally similar analog of CD161. CD161 is an orally bioavailable inhibitor of BET bromodomain.Formula:C26H20FN5O2Purity:98%Color and Shape:SolidMolecular weight:453.47SARS-CoV-2/MERS Mpro-IN-1
SARS-CoV-2/MERS Mpro-IN-1 is a potent inhibitor of the main proteases in SARS-CoV-2 and MERS, exhibiting IC50 values of 0.10 and 0.06 µM, respectively.Formula:C30H36N4O7Color and Shape:SolidMolecular weight:564.63Leucettinib-92
CAS:Leucettinib-92 (compound 92) is a kinase inhibitor selective for DYRK/CLK families, displaying IC50 values of 147 nM (CLK1), 39 nM (CLK2), 5.2 nM (CLK4), 0.8 μMFormula:C21H22N4OSPurity:98%Color and Shape:SolidMolecular weight:378.49SOMG-833 HCl
CAS:SOMG-833 HCl is a selective inhibitor of c-MET. It acts by blocking c-MET dependent neoplastic effects and exerting antitumor activity.Formula:C22H22F3N5O2Purity:98%Color and Shape:SolidMolecular weight:445.44CP 375
CAS:CP 375 is a Fe3+ chelating agent (log K1: 14.50).Formula:C11H17NO3Purity:98%Color and Shape:SolidMolecular weight:211.26ICMT-IN-34
CAS:ICMT-IN-34 (compound 39) serves as an effective inhibitor of ICMT, exhibiting an IC50 value of 0.17 μM [1].Formula:C21H25Cl2NOColor and Shape:SolidMolecular weight:378.34Zaurategrast
CAS:Zaurategrast is an effective and oral-effective inhibitor of the α4-integrin.Formula:C26H25BrN4O3Purity:98%Color and Shape:SolidMolecular weight:521.41PF-02575799
CAS:PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).Formula:C42H37FN4O4Purity:98%Color and Shape:SolidMolecular weight:680.77SKF-86002 dihydrochloride
CAS:p38 MAP kinase inhibitorFormula:C16H14Cl2FN3SPurity:98%Color and Shape:SolidMolecular weight:370.27ZIKV-IN-1
CAS:ZIKV-IN-1 blocks Zika virus effectively (EC50: 2.8 μM, EC90: 6.8 μM), targets the RdRp domain, and is low-toxic.Formula:C21H18BrF2N3O3Color and Shape:SolidMolecular weight:478.29ISPA-28
CAS:ISPA-28: reversible PSAC antagonist via direct CLAG3 binding.Formula:C21H24N6O3Color and Shape:SolidMolecular weight:408.45Z-YVAD-CMK
CAS:Z-YVAD-CMK is an inhibitor of both caspase-1 and caspase-3, as referenced in [1].Formula:C30H37ClN4O9Purity:98%Color and Shape:SolidMolecular weight:633.09DU-34569 Maleate
CAS:DU-34569 Maleate, an antiviral agent, acts against influenza A, parainfluenza Sendai, coxsackie A21, and rhinovirus.Formula:C18H27NO4Purity:98%Color and Shape:SolidMolecular weight:321.41MK-8666
CAS:MK-8666, a partial GPCR agonist targeting GPR40, may treat type 2 diabetes by enhancing insulin secretion and lowering glucose safely.Formula:C29H31NO6SColor and Shape:SolidMolecular weight:521.62IKK-IN-1
CAS:IKK-IN-1 is an inhibitor of IKK.Formula:C22H26ClN3O4Purity:98%Color and Shape:SolidMolecular weight:431.913-Hydroxycarbofuran
CAS:3-Hydroxycarbofuran, a principal metabolite of Carbofuran, acts as a reversible inhibitor of acetylcholinesterase (AChE) [1].Formula:C12H15NO4Purity:98%Color and Shape:SolidMolecular weight:237.25DMP 323
CAS:DMP 323 is a potent inhibitor of HIV-1 protease.Formula:C35H38N2O5Purity:98%Color and Shape:SolidMolecular weight:566.69Activated C Subunit
CAS:Activated C Subunit is utilized in synthesizing exon jumping oligomer conjugates that complement specific target sites within the human anti-muscular atrophyFormula:C37H37ClN5O5PColor and Shape:SolidMolecular weight:698.15BN 50739
CAS:BN 50739 is a PAF antagonist that inhibits cardiac arrhythmias and may prevent ischaemia-induced VF.Formula:C28H26ClN5O2S3Color and Shape:SolidMolecular weight:596.19ROCK2-IN-7
CAS:<p>ROCK2 inhibitor is a chemical compound associated with the therapeutic management of psoriasis.</p>Formula:C26H28FN5OPurity:98%Color and Shape:SolidMolecular weight:445.53Leteprinim
CAS:Leteprinim (AIT 082 acid) is an hypoxanthine derivative that stimulates in vitro neurite outgrowth and the production of adenosine and neurotrophins fromFormula:C15H13N5O4Purity:99.08%Color and Shape:SolidMolecular weight:327.29Ref: TM-T32658L
1mg87.00€2mg124.00€5mg187.00€10mg284.00€25mg452.00€50mg645.00€100mg867.00€200mg1,159.00€Pentixafor
CAS:<p>Pentixafor is a peptide that selectively targets the CXCR4 receptor and can be labeled with Gallium-68 (68Ga) for visualization using positron emission</p>Formula:C60H80N14O14Purity:98%Color and Shape:SolidMolecular weight:1221.36HPK1-IN-37
CAS:HPK1-IN-37 (compound A85), with an IC50 value of 3.7 nM, is a potent inhibitor of HPK1.Formula:C27H35N7O4Color and Shape:SolidMolecular weight:521.61LY303336
CAS:LY303336 is an antagonist of AT1 receptor.Formula:C30H37N4O11PSPurity:98%Color and Shape:SolidMolecular weight:692.67BMS-189664
CAS:BMS-189664 is an inhibitor of thrombin.Formula:C22H34N6O4SPurity:98%Color and Shape:SolidMolecular weight:478.61PBI-1393
CAS:PBI-1393 can be used as an enhancer for Th1 type cytokine production and primary T cell activation.Formula:C19H31N9O4Color and Shape:SolidMolecular weight:449.51TMX-2164
CAS:TMX-2164: strong, irreversible BCL6 inhibitor, IC50=152 nM, long-lasting action, inhibits cell proliferation.Formula:C25H24ClFN6O6SColor and Shape:SolidMolecular weight:591.01AS100
CAS:AS100 is a bioactive chemical.Formula:C23H24Cl3N7O4Color and Shape:SolidMolecular weight:568.84β-catenin-IN-4
CAS:β-Catenin-IN-4 is a β-catenin inhibitor characterized by a K_i value of 0.64 μM.Formula:C38H33ClF3N5O9Color and Shape:SolidMolecular weight:796.14EGFR-IN-61
CAS:EGFR-IN-61 inhibits EGFR kinase (IC50: 42 nM L858R/T790M, 137 nM L858R/T790M/C797S, 743 nM WT) and slows A549 & H1975 cell growth (IC50: 2.14 & 1.82 μM).Formula:C33H37ClN8O3Purity:98%Color and Shape:SolidMolecular weight:629.15ICMT-IN-1
CAS:ICMT-IN-1 (compound 75) is a potent ICMT inhibitor with an IC50 value of 0.0013 μM.Formula:C24H33NO2Color and Shape:SolidMolecular weight:367.52WQ 2743
CAS:WQ 2743 is a potent agent of antimicrobial.Formula:C19H15BrF3N5O3Purity:98%Color and Shape:SolidMolecular weight:498.25PF-06807656
PF-06807656 remains effective against ROMK with N171D mutation, unlike other inhibitors; it has an IC50 of 160 nM for Tl+ flux.Formula:C19H20ClN5O4SPurity:98%Color and Shape:SolidMolecular weight:449.91KDM5-IN-1
CAS:KDM5-IN-1 is an effective and selective inhibitor of KDM5 with an IC50 of 15.1 nM.Formula:C17H20N6OPurity:99.50%Color and Shape:SolidMolecular weight:324.38Ref: TM-T15649
1mg64.00€5mg187.00€10mg284.00€25mg452.00€50mg645.00€100mg867.00€500mgTo inquire1mL*10mM (DMSO)137.00€S1P1 agonist 6 hemicalcium
CAS:<p>Compound I (S1P1 agonist 6 hemicalcium) is an S1P1 agonist that diminishes autoimmune activity by inhibiting lymphocyte trafficking, and serves as an</p>Formula:C25H26F3NO3CaPurity:98%Color and Shape:SolidMolecular weight:465.51RSV L-protein-IN-3
CAS:RSV L-protein-IN-3 is an inhibitor of the wild-type RSV polymerase, exhibiting an IC50 of 10.4 μM and an EC50 of 2.1 μM (against RSV), and possesses lowerFormula:C31H34N4O4Purity:98%Color and Shape:SolidMolecular weight:526.63Roslin 2 bromide
CAS:Roslin 2 bromide (Benzylhexamethylenetetramine bromide) is a p53 reactivator that disrupts the binding of FAK and p5.Formula:C13H19BrN4Purity:99.34%Color and Shape:SolidMolecular weight:311.22Ref: TM-T24730
2mg44.00€5mg65.00€10mg87.00€25mg148.00€50mg213.00€100mg314.00€200mg452.00€1mL*10mM (DMSO)71.00€Iomazenil
CAS:Iomazenil is an antagonist and partial inverse agonist of benzodiazepine and potential therapy for alcohol abuse.Formula:C15H14IN3O3Purity:98%Color and Shape:SolidMolecular weight:411.19IKK-IN-4
CAS:IKK-IN-4 is a potent and selective inhibitor of IkappaB kinase 2 with IC 50 values of 45 and 650 nM against IKKβ and IKKα, respectively [1].Formula:C18H19N5SColor and Shape:SolidMolecular weight:337.44Robalzotan
CAS:Robalzotan is a selective 5-HT1A receptor antagonist.Formula:C18H23FN2O2Purity:98%Color and Shape:SolidMolecular weight:318.39MurA-IN-4
CAS:MurA-IN-4 exhibits antibacterial properties as a MurA inhibitor, impeding the synthesis of bacterial cell walls [1].Formula:C8H12ClNO3Color and Shape:SolidMolecular weight:205.64SQ 32970
CAS:SQ 32970 is a potent Endothia aspartic proteinase inhibitor.Formula:C33H51N5O4SColor and Shape:SolidMolecular weight:613.85AU1235
CAS:AU1235 is a Mycobacterium tuberculosis inhibitor.Formula:C17H19F3N2OPurity:99.54% - 99.87%Color and Shape:SolidMolecular weight:324.34Ref: TM-T10411
1mg74.00€2mg97.00€5mg188.00€10mg293.00€25mg494.00€50mg715.00€100mg1,008.00€500mg2,015.00€1mL*10mM (DMSO)To inquireVipoglanstat
CAS:Vipoglanstat: inhibits prostaglandin E synthase, anti-inflammatory, reduces leukocyte infiltration and lung injury from endotoxin/sepsis.Formula:C30H34Cl2F5N5O3Color and Shape:SolidMolecular weight:678.52GSK-2245035 maleate
CAS:GSK-2245035 maleate is a selective Toll-like receptor 7 (TLR7) agonist with preferential Type-1 interferon (IFN)-stimulating properties.Formula:C24H38N6O6Color and Shape:SolidMolecular weight:506.6MK-8666 Tris
CAS:MK-8666, a partial GPCR agonist, targets GPR40 to enhance insulin secretion, potentially treating type 2 diabetes without adverse effects.Formula:C33H42N2O9SColor and Shape:SolidMolecular weight:642.764WEHI-345 analog
CAS:WEHI-345 analog is an Src inhibitor.Formula:C23H25N7OPurity:98%Color and Shape:SolidMolecular weight:415.49Casein Kinase II Inhibitor IV
CAS:Casein kinase II inhibitor IV is an effective small molecule inducer, which can be used to induce epidermal keratinocyte differentiation.Formula:C24H23N5O3Purity:99.65% - 99.75%Color and Shape:SolidMolecular weight:429.47Ref: TM-T10687
1mg87.00€5mg170.00€10mg259.00€25mg429.00€50mg605.00€100mg815.00€500mg1,624.00€1mL*10mM (DMSO)180.00€SLLN-15
CAS:SLLN-15: oral, potent autophagy enhancer; targets macroautophagy in TNBC.Formula:C19H23N7Se2Purity:98%Color and Shape:SolidMolecular weight:507.35Du011
CAS:Du011 is a biogenesis inhibitor of the E.Formula:C20H15F2NO4SColor and Shape:SolidMolecular weight:403.4Tomicorat
CAS:Tomicorat is an anti-inflammatory agent.Formula:C32H30FNO5Color and Shape:SolidMolecular weight:527.58CCT365623 hydrochloride
CAS:CCT365623 hydrochloride is an orally active inhibitor of lysyl oxidase (LOX) (IC50: 0.89 μM). It suppresses EGFR (pY1068) and AKT phosphorylation driven by EGF.Formula:C18H18ClNO4S3Purity:98%Color and Shape:SolidMolecular weight:443.99L-736380
CAS:<p>L-736380, a CCK-B antagonist, reduces gastric acid (ID50: 0.064mg/kg) and blocks [(125)I]CCK-8S in mouse brains (ED50: 1.7mg/kg).</p>Formula:C25H29N9O2Color and Shape:SolidMolecular weight:487.56TMDJ-035
CAS:TMDJ-035 is a selective inhibitor of the RyR2 (ryanodine receptor 2).Formula:C16H12F3N5OPurity:98%Color and Shape:SolidMolecular weight:347.293-Methylhistamine dihydrochloride
CAS:N tau-methylhistamine, a histamine metabolite, indicates histamine release in plasma/urine with fewer artifacts.Formula:C6H13Cl2N3Purity:90% - 99.83%Color and Shape:Off-White To Pale Yellow SolidMolecular weight:198.094Arginase inhibitor 1
CAS:Arginase inhibitor 1 is a potent inhibitor of human arginases I and II (IC50s: 223 and 509 nM).Formula:C13H27BN2O4Color and Shape:SolidMolecular weight:286.18Pecavaptan
CAS:Pecavaptan is a vasopressin receptor antagonist.Formula:C22H19Cl2F3N6O3Color and Shape:SolidMolecular weight:543.33Zevotrelvir
CAS:Zevotrelvir (Compound 52) serves as an inhibitor of coronavirus, demonstrating IC50 values below 0.1 μM for 229E hCoV protease and below 0.1 mM for SARS-CoV-3C-Formula:C28H26F3N5O3Purity:98%Color and Shape:SolidMolecular weight:537.53AC-4
CAS:AC-4 is a blocker of photoswitchable TRPV1 channel.Formula:C26H25F3N4O2SColor and Shape:SolidMolecular weight:514.56CcpA-IN-1
CAS:<p>CcpA-IN-1 is a Staphylococcus aureus antibiotic exhibiting significant bactericidal activity (MICs=460 nM) [1].</p>Formula:C77H82F12N8OP3RuPurity:98%Color and Shape:SolidMolecular weight:1557.5GNE-490
CAS:GNE-490 is an effective inhibitor of pan-PI3K with IC50s of 3.5 nM, 25 nM, 5.2 nM, 15 nM for PI3Kα, PI3Kβ, PI3Kδ and PI3Kγ, respectively.Formula:C18H22N6O2SPurity:99.77%Color and Shape:SolidMolecular weight:386.47Ref: TM-T22339
1mg85.00€2mg115.00€5mg188.00€10mg321.00€25mg509.00€50mg702.00€100mg932.00€200mg1,283.00€1mL*10mM (DMSO)205.00€ROCK2-IN-6 hydrochloride
CAS:ROCK2-IN-6 hydrochloride (Comp A)为一种选择性ROCK2抑制剂，适用于研究ROCK介导的疾病、自身免疫性病症与炎症。Formula:C26H22ClF2N7OPurity:98%Color and Shape:SolidMolecular weight:521.95Org 33201
CAS:Org 33201 is a potent aromatase inhibitor.Formula:C21H28N2SColor and Shape:SolidMolecular weight:340.53Cgp 57813
CAS:CGP 57813 is a lipophilic compound, which can be used as an inhibitor of HIV-1 protease.Formula:C43H58N4O8Color and Shape:SolidMolecular weight:758.94Cipralisant
CAS:Cipralisant: H3 receptor antagonist (in vivo), agonist (in vitro, pKi 9.9), Ki 0.47 nM in rats, may treat ADHD.Formula:C14H20N2Purity:98%Color and Shape:SolidMolecular weight:216.32Dagrocorat
CAS:Dagrocorat is a novel and dissociated agonist of glucocorticoid receptor.Formula:C29H29F3N2O2Purity:98%Color and Shape:SolidMolecular weight:494.55PARPYnD
CAS:PARPYnD: Photoaffinity PARP probe; inhibits PARP2, PARP1, PARP6 (IC50: 6, 38, 230 nM); tags PARP1/2 with N3 fluorescent probe.Formula:C34H31N9O3Color and Shape:SolidMolecular weight:613.67GNE-3476
CAS:GNE-3476 is an NMDA PAM with low GluN2A efficacy, AMPAR activity, and weak at GluN2B receptors.Formula:C18H22N4OSColor and Shape:SolidMolecular weight:342.46CDD-1845
CAS:<p>CDD-1845, a non-covalent, non-peptide inhibitor, exhibits potent inhibition of SARS-CoV-2 M^pro with a K_i value of 3 nM.</p>Formula:C34H31N5O2Purity:98%Color and Shape:SolidMolecular weight:541.64
