Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,524 products)
- Apoptosis(5,793 products)
- Cell Cycle/Checkpoint(4,452 products)
- Chromatin/Epigenetics(2,242 products)
- Cytoskeletal Signaling(1,382 products)
- DNA Damage/DNA Repair(2,826 products)
- Endocrinology/Hormones(3,507 products)
- Enzyme(3,640 products)
- GPCR/G-Protein(8,333 products)
- Immunology and Inflammation(3,527 products)
- Influenza Virus(296 products)
- JAK/STAT signaling(404 products)
- MAPK Signaling(1,203 products)
- Membrane Transporter/Ion Channel(2,792 products)
- Metabolism(9,449 products)
- Microbiology/Virology(6,981 products)
- Neuroscience(9,926 products)
- Other Inhibitors(37,921 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,400 products)
- Proteases/Proteasome(1,597 products)
- Stem Cell and Derivatives(830 products)
- Tyrosine Kinase/Adaptors(2,015 products)
- Ubiquitination(1,650 products)
Show 16 more subcategories
Found 66639 products of "Inhibitors"
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SPR-00305
CAS:<p>SPR-00305 is a novel potent inhibitor of the mvfr pathway</p>Formula:C24H19ClN2O3Color and Shape:SolidMolecular weight:418.87TRPC4/5-IN-1
<p>TRPC4/5-IN-1, a TRPC5/4 inhibitor with IC50s 0.54 μM/2.06 μM, targets skin inflammation and proteinuric kidney diseases.</p>Formula:C21H21N3OColor and Shape:SolidMolecular weight:331.41YKL-05-093
CAS:<p>YKL-05-093 is a alt inducible kinase (SIK) inhibitor. YKL-05-093 increases bone formation and bone mass.</p>Formula:C35H40N6O4Color and Shape:SolidMolecular weight:608.73NVP-CFC218
CAS:<p>NVP-CFC218 is a novel potent and selective p53-HDM2 inhibitor.</p>Formula:C37H45ClN4O4Color and Shape:SolidMolecular weight:645.23KMH-233
CAS:<p>KMH-233 effectively blocks LAT1, inhibiting L-leucine uptake and cell growth, boosting betastatin and cisplatin efficacy at 25 μM.</p>Formula:C32H25N7O5Color and Shape:SolidMolecular weight:587.58Carmegliptin dihydrochloride
CAS:<p>Carmegliptin dihydrochloride (RG-1579, RO4876904) is a salt of Camegliptin, a DPP-4 inhibitor for type 2 diabetes.</p>Formula:C20H30Cl2FN3O3Color and Shape:SolidMolecular weight:450.38GSK268
<p>GSK268 is a BET inhibitor.</p>Formula:C26H27N5O3Color and Shape:SolidMolecular weight:457.53Zetomipzomib
CAS:<p>KZR-616: Immunoproteasome inhibitor targeting LMP7 (IC50: 39/57 nM) & LMP2 (IC50: 131/179 nM), potential in autoimmune disease research.</p>Formula:C30H42N4O8Color and Shape:SolidMolecular weight:586.68Merigolix
CAS:<p>Merigolix is a potent gonadotrophin releasing hormone (GnRH) antagonist .</p>Formula:C36H35F7N4O6Color and Shape:SolidMolecular weight:752.68Protopine hydrochloride
CAS:<p>Protopine inhibits thromboxane, lowers intracellular calcium, and reduces cell adhesion by altering adhesive factors.</p>Formula:C20H20ClNO5Purity:98%Color and Shape:Prisms From Alc SolidMolecular weight:389.83AHR antagonist 5 hemimaleate
<p>Potent oral AHR antagonist with IC50 < 0.5 μM, hinders tumor growth with anti-PD-1.</p>Formula:C29H28FN7O4Color and Shape:SolidMolecular weight:499.55Massarilactone H
CAS:<p>Massarilactone H, a polyketide, is a neuraminidase inhibitor, with an IC 50 of 8.18 µM .</p>Formula:C11H12O5Color and Shape:SolidMolecular weight:224.21PCSK9-IN-16
CAS:<p>PCSK9-IN-16, holds potential for research into hypercholesterolemia and other cardiovascular diseases [1].</p>Formula:C16H20N6O2S3Color and Shape:SolidMolecular weight:424.56MK-7445
CAS:<p>MK-7445 is a conformationally constrained inhibitor of non-nucleoside reverse transcriptase.</p>Formula:C21H13Cl2N7OColor and Shape:SolidMolecular weight:450.28PNU-248686A
CAS:<p>PNU-248686A is an inhibitor of matrix metalloproteinase (MMP).</p>Formula:C22H18ClNaO5S2Purity:98%Color and Shape:SolidMolecular weight:484.95Demethoxyviridin
CAS:<p>Demethoxyviridin inhibits mammalian Ptdlns 3-kinase (p110) and is antifungal.</p>Formula:C19H14O5Purity:98%Color and Shape:SolidMolecular weight:322.31Arterolane maleate
CAS:<p>Arterolane, an adenosine triphosphatase inhibitor, is used potentially for the treatment of malaria.</p>Formula:C26H40N2O8Purity:98%Color and Shape:SolidMolecular weight:508.612Kinamycin B
CAS:<p>Kinamycin B is an antibacterial agent with anticancer activity.</p>Formula:C20H16N2O8Purity:98%Color and Shape:SolidMolecular weight:412.35O-GlcNAcase-IN-1
<p>O-GlcNAcase-IN-1 is a potent and novel inhibitor of O-GlcNAcase(OGA) with an IC 50 value of 46 nM.</p>Formula:C15H22N6Color and Shape:SolidMolecular weight:286.38Isobetanin
CAS:<p>Isobetanin is a betacyanin that has been shown to enhance vitexin-2-O-xyloside mediated inhibition of proliferation of T24 bladder cancer cells.</p>Formula:C24H26N2O13Color and Shape:SolidMolecular weight:550.47Anti-inflammatory agent 9
<p>Benzimidazothiazole-derived Compound 28 from tilomisole targets COX-2, has potent anti-inflammatory effects & is orally bioavailable.</p>Formula:C18H15N5O2SColor and Shape:SolidMolecular weight:365.41HDAC-IN-33
<p>HDAC-IN-33 inhibits HDAC1/2/6 (IC50: 24/46/47 nM), exhibits potent antitumor activity in vitro and in vivo, and activates antitumor immunity.</p>Formula:C21H25N3O3Color and Shape:SolidMolecular weight:367.44PAD2-IN-1 hydrochloride
<p>PAD2-IN-1 hydrochloride: potent, selective PAD2 inhibitor; 95x less on PAD4, 79x less on PAD3; benzimidazole derivative.</p>Formula:C25H30ClFN6O3Color and Shape:SolidMolecular weight:517BMS-986118
CAS:<p>BMS-986118 is a GPR40 full agonist targeting type II diabetes, prompting insulin release without hypoglycemia risk.</p>Formula:C25H28ClF3N4O4Purity:98%Color and Shape:SolidMolecular weight:540.96Lycopodine
CAS:<p>Lycopodine, a bioactive compound derived from Lycopodium clavatum spores, effectively inhibits the proliferation of HeLa cells through the induction of</p>Formula:C16H25NOPurity:98%Color and Shape:SolidMolecular weight:247.38FTI 276 TFA
CAS:<p>FTI 276 TFA targets plasmodium falciparum & humans, inhibits PFT with IC50s: 0.9 nM (parasite) & 0.5 nM (human).</p>Formula:C23H28F3N3O5S2Color and Shape:SolidMolecular weight:547.61JAK3-IN-7
CAS:<p>JAK3-IN-7 is a potent and selective JAK3 inhibitor (IC50<0.01 μM) for the treatment of rejection in organ transplantation, graft-versus-host reaction after</p>Formula:C17H20N6OPurity:98.81%Color and Shape:SolidMolecular weight:324.38Pociredir
CAS:<p>Pociredir (FTX-6058), a potent EED inhibitor (KD=0.163 nM), may help in SCD research.</p>Formula:C22H18FN5O2Color and Shape:SolidMolecular weight:403.41NVP-CGM097 sulfate
CAS:<p>NVP-CGM097 sulfate is a potent and selective inhibitor of MDM2 (hMDM2, IC50 of 1.7±0.1 nM).</p>Formula:C38H49ClN4O8SPurity:98%Color and Shape:SolidMolecular weight:757.34Coleon-U-quinone
CAS:<p>Coleon-U-quinone, a P-gp inhibitor, reduces cancer cell viability and enhances Doxorubicin sensitivity in resistant cells.</p>Formula:C20H24O5Color and Shape:SolidMolecular weight:344.4HDAC6-IN-12
<p>HDAC6-IN-12 is a potent inhibitor of HDAC6 that binds in the DNA chain, causing DNA damage and exhibiting anticancer effects that can be used in cancer research</p>Formula:C24H39F2N3O5Color and Shape:SolidMolecular weight:487.58MEIS-IN-1
CAS:<p>MEIS-IN-1 is a potent MEIS inhibitor that induces the expansion of hematopoietic stem cells in mice and humans.</p>Formula:C24H21F3N2O4Color and Shape:SolidMolecular weight:458.43Isoleucyl tRNA synthetase-IN-2
CAS:<p>Isoleucyl tRNA synthetase-IN-2 is a selective and potent inhibitor (Ki: 114 nM) that targets isoleucyl tRNA synthetase (IleRS).</p>Formula:C22H33N5O8SColor and Shape:SolidMolecular weight:527.59HIF-1/2α-IN-1
<p>HIF-1/2α-IN-1, an orally active compound, functions as an inhibitor of HIF-2α.</p>Formula:C17H16N6O4Color and Shape:SolidMolecular weight:368.35Antileishmanial agent-4
<p>Antileishmanial agent-4, a ribonucleoside analogue, functions as an antileishmanial agent [1].</p>Formula:C17H18N4O4Color and Shape:SolidMolecular weight:342.35LasR-IN-3
<p>LasR-IN-3 inhibits LasR in Pseudomonas, disrupting its dimer, causing loss of function.</p>Formula:C22H19N3O2Color and Shape:SolidMolecular weight:357.41Musettamycin
CAS:<p>Musettamycin triggers erythroid differentiation in blood cells, acts like anthracycline antibiotics, but only inhibits gram-positive bacteria.</p>Formula:C36H45NO14Color and Shape:SolidMolecular weight:715.74BI-44370
CAS:<p>BI-44370, a CGRP (calcitonin gene-related peptide) receptor antagonist, can be used to treat migraines and other chronic pain.</p>Formula:C35H47N5O6Color and Shape:SolidMolecular weight:633.78PF-06372222
CAS:<p>PF-06372222: a small-molecule that modulates GCGR and antagonizes GLP-1R, affecting insulin and glucagon.</p>Formula:C26H28F3N5O3Purity:98%Color and Shape:SolidMolecular weight:515.53Rodatristat
CAS:<p>Rodatristat is an effective tryptophan hydroxylase 1 and TPH2 inhibitor (IC50s: 33 nM and 7 nM, respectively).</p>Formula:C27H27ClF3N5O3Purity:98%Color and Shape:SolidMolecular weight:561.98PI3K-IN-23
<p>PI3K-IN-23 is a (E)-9-oxooctadec-10-en-12-ynoic acid analogue that promotes glucose uptake (EC50: 7.00 μM).</p>Formula:C24H33NO4SColor and Shape:SolidMolecular weight:431.59ONO-5334
CAS:<p>ONO-5334: selective cathepsin K inhibitor, potential for osteoporosis study; Ki: 0.10 nM (human), 0.049 nM (rabbit), 0.85 nM (rat).</p>Formula:C21H34N4O4SPurity:98.22% - 99.60%Color and Shape:SolidMolecular weight:438.58TDI-11861
CAS:<p>TDI-11861 is a second-gen sAC (ADCY10) inhibitor with an IC50 of 5.5 nM and slow dissociation.</p>Formula:C22H25ClF2N6O3Color and Shape:SolidMolecular weight:494.92Aurora inhibitor 1
CAS:<p>Aurora inhibitor 1 is a potent Aurora inhibitor (IC50: ≤ 4 nM and ≤13 nM for Aurora A and Aurora B kinase).</p>Formula:C23H25N9SPurity:98%Color and Shape:SolidMolecular weight:459.57Py-MPB-amino-C3-PBD
CAS:<p>Py-MPB-amino-C3-PBD is a cytotoxic agent comprised non-alkylating group,with antimicrobial activity.</p>Formula:C41H44N8O6Purity:98%Color and Shape:SolidMolecular weight:744.84NTPDase-IN-3
CAS:<p>NTPDase-IN-3 inhibits NTPDase1/2/3/8 (IC50: 0.21/1.07/0.38/0.05 μM), useful for cancer and thrombosis research.</p>Formula:C22H24ClN3OS2Color and Shape:SolidMolecular weight:446.03Factor B-IN-3
CAS:<p>Factor B-IN-3 is a potent inhibitor of complement factor B. Factor B-IN-3 can be used to study inflammatory and immune-related diseases.</p>Formula:C24H29N3O4Color and Shape:SolidMolecular weight:423.5Gepotidacin hydrochloride
CAS:<p>Gepotidacin (GSK-2140944) is a potent DNA topoisomerase inhibitor, a novel antibacterial efficacious against various anaerobes.</p>Formula:C24H29ClN6O3Color and Shape:SolidMolecular weight:484.98Galidesivir
CAS:<p>Galidesivir (BCX4430) is an antiviral compound that inhibits viral RNA-dependent RNA polymerase (RdRp) activity and reduces lung infections in infected animals.</p>Formula:C11H15N5O3Purity:96.73% - 99.13%Color and Shape:SolidMolecular weight:265.27GRPR antagonist-2
<p>GRPR antagonist-2 blocks GRPR, kills some cancer cells, effective on HGC-27 (IC50: 0.77 μM) & Pan02 (IC50: 2.5 μM).</p>Formula:C28H32F3N5O4Color and Shape:SolidMolecular weight:559.58SB 243213 hydrochloride
CAS:<p>SB 243213 hydrochloride is an orally active, selective and high-affinity antagonist of 5-hydroxytryptamine (5-HT)2C receptor(pKi of 9.37 and a pKb of 9.8).It</p>Formula:C22H20ClF3N4O2Purity:98%Color and Shape:SolidMolecular weight:464.87HOE-288
CAS:<p>HOE-288 is a converting enzyme (CE) inhibitor.</p>Formula:C27H38N2O5Color and Shape:SolidMolecular weight:470.60Terguride
CAS:<p>Terguride: treats hyperprolactinemia, blocks 5-HT2A/B, activates dopamine receptors, studied for PAH.</p>Formula:C20H28N4OColor and Shape:SolidMolecular weight:340.46Artemisiane E
CAS:<p>Artemisiane E is a potent PI3K/AKT pathway inhibitor with an IC 50 of 8.9 μM .</p>Formula:C20H22O5Color and Shape:SolidMolecular weight:342.39Dictyostatin
CAS:<p>Dictyostatin: potent microtubule stabilizer & anticancer agent with antiproliferative effects; researched for tauopathies.</p>Formula:C32H52O6Color and Shape:SolidMolecular weight:532.75DFBTA
<p>DFBTA inhibits ANO1 with IC50 of 24 nM, effectively treating inflammatory pain orally.</p>Formula:C18H10ClF2NO3SColor and Shape:SolidMolecular weight:393.79HS-731
CAS:<p>HS-731 is a μ-Opioid Receptor Agonist.</p>Formula:C20H26N2O5Color and Shape:SolidMolecular weight:374.43Antibacterial agent 110
<p>Compound 4e, an antibacterial against P. aeruginosa, disrupts cell membranes (MIC: 1 μg/ml).</p>Formula:C22H21N5O4SColor and Shape:SolidMolecular weight:451.5Imolamine hydrochloride
CAS:<p>Imolamine hydrochloride is a blood platelet aggregation antagonist.</p>Formula:C14H21ClN4OColor and Shape:SolidMolecular weight:296.80AB 5046A
CAS:<p>AB 5046A is a chlorosis inducing substance isolated from Nodulisporium SP.</p>Formula:C10H14O4Color and Shape:SolidMolecular weight:198.22CDK4-IN-1
CAS:<p>CDK4 inhibitor is a novel and specific CDK4/Cyclin D1 inhibitor with an IC50 of 10 nM; 1500 and 500 fold than CDK1/Cyclin B (IC50>15 uM) and CDK2/Cyclin A (IC50</p>Formula:C22H29ClN8Purity:98%Color and Shape:SolidMolecular weight:440.97ATM Inhibitor-2
<p>ATM Inhibitor -2 is a potent and selective inhibitor of ATM (IC50<1 nM).</p>Formula:C26H31N7O3Color and Shape:SolidMolecular weight:489.57SOS1-IN-10
<p>SOS1-IN-10 is a potent inhibitor of SOS1 that acts on KRAS G12C-SOS1 (IC50: 13 nM).</p>Formula:C22H19F5N4OColor and Shape:SolidMolecular weight:450.4sEH inhibitor-4
<p>Compound B15: potent sEH inhibitor (0.03 nm), reduces inflammation & pain.</p>Formula:C27H28Cl2N4O3Color and Shape:SolidMolecular weight:527.44Nepaprazole sodium
CAS:<p>Nepaprazole Na (TY-11345), a proton pump inhibitor, may treat gastric ulcers; it reduces H+/K(+)-ATPase activity, with IC50 of 5.8-9.9 microM.</p>Formula:C18H18N3NaO2SColor and Shape:SolidMolecular weight:363.41PPARα agonist 1
<p>PPARα agonist 1 is a complete and potent PPARα agonist.</p>Formula:C27H34O4Color and Shape:SolidMolecular weight:422.56PAIR2
CAS:<p>PAIR2 is a selective IRE1α RNase partial antagonist, blocking its ATP site and preventing KIRA from hindering XBP1 splicing.</p>Formula:C27H26F4N6O3SColor and Shape:SolidMolecular weight:590.59AFP-07
CAS:<p>AFP-07 is a highly selective and potent agonist. It was used for the prostacyclin receptor.</p>Formula:C22H29F2NaO5Purity:98%Color and Shape:SolidMolecular weight:434.45DNA crosslinker 3 dihydrochloride
CAS:<p>Compound 1: a DNA minor groove binder with 1.4°C ΔTm; useful in cancer research.</p>Formula:C15H22Cl2N8OColor and Shape:SolidMolecular weight:401.29NPR-C activator 1
CAS:<p>NPR-C activator 1 is an activator of the natriuretic peptide receptor C (NPR-C), which can be used to study cardiovascular diseases.</p>Formula:C18H24N6O3Purity:98.74%Color and Shape:SolidMolecular weight:372.42Antibacterial agent 82
<p>Antibacterial agent 82 (compound 7p) is an antibacterial agent [1].</p>Formula:C22H18N2O2Color and Shape:SolidMolecular weight:342.39Carbonic anhydrase inhibitor 4
<p>CA inhibitor 4, photoprobe; targets hCA I-XIV; Ki: 640-1166 nM.</p>Formula:C21H18N2O4SColor and Shape:SolidMolecular weight:394.44COX-2/NO-IN-1
<p>COX-2/NO-IN-1: oral iNOS & NO blocker (IC50=3.52μM), COX-2 supressor, anti-inflammatory, protects kidneys.</p>Formula:C15H15NO3Color and Shape:SolidMolecular weight:257.28L5-DA
<p>L5-DA, a G-quadruplex ligand, stabilizes G4s in HeLa cells, induces apoptosis, and is cytotoxic with an IC50 of 4.3 μM.</p>Formula:C32H34N6O2Color and Shape:SolidMolecular weight:534.65Anti-Aβ agent 1A
<p>Anti-Aβ agent 1A is a potent anti-amyloid-β agent.</p>Formula:C35H49NO4Color and Shape:SolidMolecular weight:547.77HPK1-IN-3
<p>HPK1-IN-3: Selective HPK1 inhibitor, ATP-competitive, IC50=0.25nM; boosts IL-2 in PBMCs, EC50=108nM.</p>Formula:C23H22F4N6O2Color and Shape:SolidMolecular weight:490.45GW-597901 cinnamate
CAS:<p>GW-597901 cinnamate is a long-acting beta(2)-agonist.</p>Formula:C34H46N2O8SColor and Shape:SolidMolecular weight:642.80AMG-222 tosylate
CAS:<p>AMG-222 tosylate is a DPP-IV inhibitor in clinical development for type II diabetes.</p>Formula:C39H47N9O6SColor and Shape:SolidMolecular weight:769.91Macbecin I
CAS:<p>Hsp90 inhibitor</p>Formula:C30H42N2O8Purity:98%Color and Shape:SolidMolecular weight:558.66EBI-1051
CAS:<p>EBI-1051 is a highly potent and orally efficacious inhibitor of MEK (IC50: 3.9 nM).</p>Formula:C18H15F2IN2O5Purity:98%Color and Shape:SolidMolecular weight:504.22IRAK4-IN-19
<p>IRAK4-IN-19, an IRAK4 inhibitor (IC50: 4.3 nM), hampers IL23 synthesis and arthritis progression.</p>Formula:C25H26F2N8OColor and Shape:SolidMolecular weight:492.52Antiviral agent 6
<p>Antiviral agent 6 showed excellent anti-TSWV effects in vivo (EC50: 188 mg/L).</p>Formula:C23H27BrN2O3S2Color and Shape:SolidMolecular weight:523.51CXCR4 antagonist 3
<p>CXCR4 antagonist 3, aka compound 12a, has 11 nM IC50, shares TIQ15 traits, and is promising in HIV research.</p>Formula:C22H31N5Color and Shape:SolidMolecular weight:365.52Carbonic anhydrase inhibitor 8
<p>R-13, a carbonic anhydrase inhibitor, has Ki of 60.7 nM (hCA I), 320.7 nM (hCA II), and 2298 nM (hCA IV).</p>Formula:C20H25N3O4SColor and Shape:SolidMolecular weight:403.5EGFR-IN-47
<p>EGFR-IN-47: strong oral EGFRL858R/T790M/C797S blocker, induces cell death; promising for NSCLC research. IC50: 0.01 μM.</p>Formula:C29H35N7Color and Shape:SolidMolecular weight:481.64Anticancer agent 78
<p>Anticancer agent 78: anti-aromatase (IC50=0.9 μM), cytotoxic, potential in breast cancer research.</p>Formula:C19H14BrNO4Color and Shape:SolidMolecular weight:400.22UNC7467
CAS:<p>UNC7467, potent IP6K2/1/6 inhibitor (4.9/8.9/1320 nM); lowers inositol pyrophosphates, minimal impact on other inositol phosphates; for obesity research.</p>Formula:C20H13NO3Purity:98.28% - 98.64%Color and Shape:SoildMolecular weight:315.32EP4 receptor antagonist 2
CAS:<p>EP4 receptor antagonist 2 (compound 2-13) is a potent agonist of the EP4 receptor (IC50: 7.8 nM) and has antitumour effects.</p>Formula:C27H29N3O5Color and Shape:SolidMolecular weight:475.54Ambuic acid
CAS:<p>Ambuic acid: cyclohexanone with antifungal, quorum-inhibiting, antibacterial properties, blocks cyclic peptides; reduces MRSA abscesses in mice.</p>Formula:C19H26O6Color and Shape:SolidMolecular weight:350.41HDAC-IN-35
<p>HDAC-IN-35 (Compound 14) is an effective and selective inhibitor of VEGFR-2 and HDAC, with IC50 values of 13.2 and 0.166 μM for VEGFR-2 and HDAC6, respectively.</p>Formula:C17H13ClF3N3O3Color and Shape:SolidMolecular weight:399.75Bometolol Hydrochloride
CAS:<p>Bometolol Hydrochloride is a beta-adrenergic blocking compound used for the treatment of cardiovascular disease.</p>Formula:C25H33ClN2O7Purity:98%Color and Shape:SolidMolecular weight:508.99PF-5177624
CAS:<p>PF-5177624 is a selective and potent PDK1 inhibitor inducing anti-tumor activity in breast cancer cells.</p>Formula:C25H25FN8O2Color and Shape:SolidMolecular weight:488.52TRK-IN-12
CAS:<p>TRK-IN-12 (9e), a macrocyclic TRK inhibitor (G595R IC50=13.1 nM), outperforms LOXO-101 in Ba/F3-NTRK1 cells.</p>Formula:C18H19ClFN5O3SColor and Shape:SolidMolecular weight:439.89PARP1-IN-5
<p>PARP1-IN-5 is a potent, selective, orally active, low-toxicity PARP-1 inhibitor with an IC50 value of 14.7 nM. PARP1-IN-5 can be used in cancer research.</p>Formula:C25H24N2O5SColor and Shape:SolidMolecular weight:464.53GNE-203
CAS:<p>GNE-203 is a Met inhibitor.</p>Formula:C30H29Cl2F3N8O3Color and Shape:SolidMolecular weight:677.50MM-589
CAS:<p>MM-589 is a potent WD repeat domain 5 (WDR5) inhibitor and mixed lineage leukemia (MLL) protein-protein interaction.</p>Formula:C28H44N8O5Purity:98%Color and Shape:SolidMolecular weight:572.70Cimpuciclib tosylate
CAS:<p>Cimpuciclib tosylate, a selective CDK4 inhibitor (IC50: 0.49 nM), exhibits anti-tumor activity.</p>Formula:C37H43FN8O4SColor and Shape:SolidMolecular weight:714.85Cap-dependent endonuclease-IN-2
<p>Cap-dependent endonuclease-IN-2 strongly blocks influenza A virus RNA polymerase; it's a CEN inhibitor.</p>Formula:C30H24FN3O7SColor and Shape:SolidMolecular weight:589.59OMDM169
CAS:<p>OMDM169: potent/selective MAGL inhibitor, raises 2-AG, analgesic via cannabinoid receptors, IC50: 0.13-0.41μM in rat/COS-7, inactive at CB1/CB2.</p>Formula:C25H45NO5Purity:98%Color and Shape:SolidMolecular weight:439.63RAD51-IN-6
CAS:<p>RAD51-IN-6, a potent RAD51 gene inhibitor, may help research mitochondrial disorders. (WO2021164746A1, cmpd 23)</p>Formula:C27H40N3O5PSColor and Shape:SolidMolecular weight:549.66RSV-IN-5
CAS:<p>RSV-IN-5: Dual inhibitor for RSV fusion proteins, effective on wild-type A2 and D486N mutant with EC50s of 2.0 nM & 8.1 nM. Potent anti-RSV.</p>Formula:C28H37N7O2Color and Shape:SolidMolecular weight:503.64Antitumor agent-75
<p>Antitumor agent-75 is a novel and potent antitumor agent.</p>Formula:C26H23FN6Color and Shape:SolidMolecular weight:438.5CFT8634
CAS:<p>CFT8634 degrades BRD9, for synovial sarcoma and SMARCB1 tumor research, from patent WO2021178920A1.</p>Formula:C37H45F3N6O5Color and Shape:SolidMolecular weight:710.79VEGFR-2-IN-26
CAS:<p>VEGFR-2-IN-26 inhibits VEGFR-2 (IC50: 15.5 nM), combating various cancers' cell growth.</p>Formula:C24H19F3N6O2Color and Shape:SolidMolecular weight:480.44NSD2-IN-1
CAS:<p>NSD2-IN-1: potent, selective NSD2-PWWP1 inhibitor, IC50 0.11 μM, induces gene expression changes, apoptosis, cell cycle arrest.</p>Formula:C29H31N5Color and Shape:SolidMolecular weight:449.59FXIa-IN-9
CAS:<p>FXIa-IN-9, a potent FXIa inhibitor (K i : human 0.17 nM, rabbit 0.5 nM), forms hydrogen bonds and has anticoagulant properties.</p>Formula:C23H18Cl2F3N9O2Color and Shape:SolidMolecular weight:580.35Casuarinin
CAS:<p>Casuarinin, an ellagitannin found in pomegranates and certain Casuarina/Stachyurus plants, is a carbonic anhydrase inhibitor and astringent.</p>Formula:C41H28O26Color and Shape:SolidMolecular weight:936.65NMDA receptor antagonist-3
<p>NMDA antagonist-3: recovery rate 40% at 100 μM, low toxicity in SH-SY5Y, human stem cells.</p>Formula:C13H19N3O6Color and Shape:SolidMolecular weight:313.31Rivenprost
CAS:<p>Rivenprost, selective EP4 agonist (Ki: 0.7 nM), promotes bone growth, osteoblast differentiation, and aids wound healing.</p>Formula:C24H34O6SColor and Shape:SolidMolecular weight:450.59LolCDE-IN-2
CAS:<p>LolCDE-IN-2 is a potent Lol protein (LolCDE) inhibitor. LolCDE-IN-2 shows antibacterial activity with a MIC of 2 μg/ml against E. coli MG1655 [1].</p>Formula:C22H17N5OPurity:98%Color and Shape:SolidMolecular weight:367.40Dyrk1A-IN-2
<p>Dyrk1A-IN-2 is a DYRK1A inhibitor (EC50: 37 nM). dyrk1A-IN-2 exhibits efficient promotion of human β-cell replication, as well as low cytotoxicity.</p>Formula:C27H32N6O4Color and Shape:SolidMolecular weight:504.58APJ receptor agonist 3
CAS:<p>APJ receptor agonist 3 is a highly effective and orally administerable agonist of the APJ receptor, demonstrating a potent EC50 value of 0.027 nM.</p>Formula:C26H29ClN4O5Color and Shape:SolidMolecular weight:512.98Dexnebivolol
CAS:<p>Dexnebivolol (R67138), a ß-adrenergic antagonist, is Nebivolol's enantiomer with β1 blocking and vasodilation properties.</p>Formula:C22H25F2NO4Color and Shape:SolidMolecular weight:405.43PptT-IN-3
<p>PptT-IN-3 (5p), an inhibitor of PptT in Mycobacterium tuberculosis, IC50=3.5μM, is key for TB research.</p>Formula:C16H27N5O3SColor and Shape:SolidMolecular weight:369.48Danavorexton
CAS:<p>Danavorexton is an orexin receptor agonist.</p>Formula:C21H32N2O5SColor and Shape:SolidMolecular weight:424.55Anticancer agent 54
<p>Anticancer agent 54 blocks cell cycle in G0/G1, induces apoptosis, and fights cancer via DNA embedding and ROS.</p>Formula:C33H36N6Color and Shape:SolidMolecular weight:516.68GRPR antagonist-1
<p>GRPR antagonist-1 targets GRPR, kills specific cancer cells (e.g., PC3, Pan02, HGC-27), and promotes apoptosis by modulating Bcl-2 and Bax.</p>Formula:C29H33F3N4O4Color and Shape:SolidMolecular weight:558.59Tribenuron
CAS:<p>Tribenuron, a slow acting sulfonylurea herbicide, controls broadleaf weed.</p>Formula:C14H15N5O6SColor and Shape:SolidMolecular weight:381.36Agosterol A
CAS:<p>Agosterol A is isolated from marine sponge Spongia.</p>Formula:C33H52O8Color and Shape:SolidMolecular weight:576.76TCMDC-136230
<p>TCMDC-136230 is a novel inhibitor of Plasmodium calcium kinetics with minimal inhibition of haemoglobin crystallisation.</p>Formula:C24H34N4O2SColor and Shape:SolidMolecular weight:442.62Wikstrol A
CAS:<p>Wikstrol A: antifungal, anti-mitotic, anti-HIV agent with various IC50/MDC values (67.8-131 µM) and deforms P. oryzae mycelia.</p>Formula:C30H22O10Color and Shape:SolidMolecular weight:542.49(Rac)-Plevitrexed
CAS:<p>(Rac)-Plevitrexed is a racemate of Plevitrexed. Plevitrexed is an orally active and potent inhibitor of thymidylate synthase (TS).</p>Formula:C26H25FN8O4Purity:98%Color and Shape:SolidMolecular weight:532.53PCTR1
CAS:<p>PCTR1, derived from DHA, hastens inflammation resolution and boosts macrophage function, reducing PGE2, PGD2, and TXB2 in mice.</p>Formula:C32H47N3O9SColor and Shape:SolidMolecular weight:649.8NAZ2329
CAS:<p>NAZ2329: Cell-permeable, targets R5 RPTPs, inhibits hPTPRZ1 (IC50=7.5 μM) & hPTPRG (IC50=4.8 μM), hampers glioblastoma growth, affects stem cell traits.</p>Formula:C21H18F3NO4S3Color and Shape:SoildMolecular weight:501.56VEGFR-2-IN-13
<p>VEGFR-2-IN-13 (Compound 19a) is a potent VEGFR-2 inhibitor (IC50: 3.4 nM). vEGFR-2-IN-13 arrests the HepG2 cell cycle in G2/M phase and induces apoptosis.</p>Formula:C24H18N6O2SColor and Shape:SolidMolecular weight:454.5Tauro-ω-muricholic acid sodium
<p>Tauro-ω-muricholic acid sodium (TωMCA sodium) is an analogue of tauro-α-muricholic acid, a bile acid of hepatic origin.</p>Formula:C26H44NNaO7SColor and Shape:SolidMolecular weight:537.68HER2-IN-8
CAS:<p>HER2-IN-8 is an inhibitor of HER-2 that can be used in the study of cancer and inflammation-related diseases.</p>Formula:C26H25F2N9O3Color and Shape:SolidMolecular weight:549.53Antidepressant agent 2
<p>Antidepressant agent 2 showed significant antidepressant effects with a MED value of 0.1 mg/kg.</p>Formula:C21H22ClFN2O3SColor and Shape:SolidMolecular weight:436.93Lentiginosine
CAS:<p>Lentiginosine is a selective amyloglucosidase inhibitor.</p>Formula:C8H15NO2Color and Shape:SolidMolecular weight:157.21HPK1-IN-16
CAS:<p>HPK1-IN-16, a potent HPK1 inhibitor, useful for cancer research and treatment.</p>Formula:C28H27FN4OColor and Shape:SolidMolecular weight:454.54HBV-IN-24
<p>HBV-IN-24 inhibits HBV DNA, HBsAg, HBeAg (EC50: 0.6, 0.6, 4.6 nM), and has antiviral properties with neurotoxicity mitigation.</p>Formula:C23H27NO6Color and Shape:SolidMolecular weight:413.46Carbodine
CAS:<p>Carbodine is an antiviral targeting CTP synthetase, effective against influenza A0/PR-8/34 and A2/Aichi/2/68.</p>Formula:C10H15N3O4Purity:98%Color and Shape:SolidMolecular weight:241.24PF1070A
CAS:<p>PF1070A is a natural cyclic tetrapeptide HDAC Inhibitor through the inhibition of PfHDAC1 catalytic activity, potently inducing the synthesis of metallothionein</p>Formula:C31H44N4O6Color and Shape:SolidMolecular weight:568.7NLRP3-IN-6
<p>NLRP3-IN-6 (Compound 34) is a selective inhibitor of the NLRP3 inflammasome.</p>Formula:C18H15ClN2O4S3Color and Shape:SolidMolecular weight:454.97JAK-IN-19
<p>JAK-IN-19 inhibits JAK (pIC50: 7.2, 7.7), less so for VEGFR2 (7.0) and Aurora B (5.8).</p>Formula:C26H36FN5O2Color and Shape:SolidMolecular weight:469.59GSK-3β inhibitor 7
<p>GSK-3β inhibitor 7 is a GSK-3β inhibitor (IC50: 5.25 μM).</p>Formula:C27H23BrN4O2SColor and Shape:SolidMolecular weight:547.47DJT06001
CAS:<p>DJT06001 is a selective Factor Xa inhibitor, reducing thrombus formation with low risk of bleeding.</p>Formula:C21H20ClN3O5SColor and Shape:SolidMolecular weight:461.92Pim-1 kinase inhibitor 2
CAS:<p>Compound 13, a potent Pim-1 inhibitor, induces apoptosis with potential for cancer research.</p>Formula:C24H14N4O3Color and Shape:SolidMolecular weight:406.39OP-5244
CAS:<p>OP-5244 has comparable potency to bisphosphonic acid series and targets CD73.</p>Formula:C19H29ClN5O9PPurity:98%Color and Shape:SolidMolecular weight:537.89NBTIs-IN-5
CAS:<p>NBTIs-IN-5 inhibits Mycobacterium abscessus DNA with IC50 1.5μM, halts growth at MIC90 0.4μM.</p>Formula:C24H25F3N4O2Color and Shape:SolidMolecular weight:458.48RhlR antagonist 1
<p>RhlR antagonist 1: IC50 of 26 μM, selective for RhlR, inhibits P. aeruginosa biofilm and virulence factors.</p>Formula:C12H10F2OColor and Shape:SolidMolecular weight:208.2CB-7646
CAS:<p>CB-7646 is a stable trimelamol (TM) analogue, which is an antitumor agent.</p>Formula:C8H16N6O2Color and Shape:SolidMolecular weight:228.25Agarospirol
CAS:<p>Agarospirol has partial anti-inflammatory activity.</p>Formula:C15H26OPurity:98%Color and Shape:SolidMolecular weight:222.37BMS-248360
CAS:<p>BMS-248360: Oral dual hAT1/hETA antagonist with Kis of 10nM & 1.9nM, respectively; treats hypertension.</p>Formula:C36H45N5O5SPurity:98%Color and Shape:SolidMolecular weight:659.84YM-202074
CAS:<p>YM-202074: Selective mGlu1 antagonist, binds allosteric site (Ki=4.8 nM), inhibits mGlu1 (IC50=8.6 nM).</p>Formula:C22H30N4O2SColor and Shape:SolidMolecular weight:414.56(rel)-AR234960
CAS:(rel)-AR234960 is an active relative configuration of AR234960. AR234960 is a non-peptide agonist of MAS.Formula:C27H30FN5O5SColor and Shape:SolidMolecular weight:555.63Heme Oxygenase-2-IN-1
<p>Heme Oxygenase-2-IN-1 is a selective HO-2 inhibitor with IC50s: 14.9 μM (HO-1), 0.9 μM (HO-2).</p>Formula:C19H17N3O2Color and Shape:SolidMolecular weight:319.36PI3K-IN-37
CAS:<p>PI3K-IN-37 inhibits PI3K α/β/δ (IC50: 6/8/4 nM) and mTOR (IC50: 4 nM).</p>Formula:C25H26N6O2Color and Shape:SolidMolecular weight:442.51AVE-1330A free acid
CAS:<p>AVE-1330A free acid is a broad-spectrum non-beta-lactam beta-lactamase inhibitor.</p>Formula:C7H11N3O6SColor and Shape:SolidMolecular weight:265.24BI 224436
CAS:<p>BI 224436 is an inhibitor of HIV-1 noncatalytic site integrase. With EC50 values of less than 15 nM against different HIV-1 laboratory strains.</p>Formula:C27H26N2O4Color and Shape:SolidMolecular weight:442.51Chitin synthase inhibitor 1
<p>Potent, selective CHS inhibitor with 0.12 mM IC50; effective against drug-resistant fungi.</p>Formula:C22H20ClN3O3Color and Shape:SolidMolecular weight:409.87BIIE-0246 HCl
CAS:<p>BIIE-0246: A potent, non-peptide Y2 receptor antagonist; >650-fold more selective than Y1, Y4, Y5.</p>Formula:C49H59Cl2N11O6Color and Shape:SolidMolecular weight:968.97Pareptide monohydrochloride
CAS:<p>Pareptide monohydrochloride is a metabolically stable analog of melatonin inhibitor (MIF).</p>Formula:C14H27ClN4O3Purity:98%Color and Shape:SolidMolecular weight:334.84ACHN-975 TFA
CAS:<p>ACHN-975 TFA is a selective LpxC inhibitor with a subnanomolar inhibitory. It is against a wide range of gram-negative bacterias with low MIC values (≤1 μg/mL).</p>Formula:C22H24F3N3O6Purity:98%Color and Shape:SolidMolecular weight:483.4377MEK4 inhibitor-2
CAS:<p>MEK4 Inhibitor-2, a novel MEK4 inhibitor, demonstrates efficacy against pancreatic adenocarcinoma, exhibiting an IC50 value of 83 nM.</p>Formula:C20H15FN4O3SColor and Shape:SolidMolecular weight:410.42MAO-B-IN-5
CAS:<p>MAO-B-IN-5: potent, selective oral MAO-B inhibitor, IC50=0.204μM, potential for Parkinson's research.</p>Formula:C19H21FN2O2Purity:97.68%Color and Shape:SolidMolecular weight:328.38Antitumor agent-47
<p>Antitumor agent-47, a silibinin derivative, shows cytotoxicity in NCI-H1299 (IC50: 8.07µM) and HT29 (IC50: 6.27µM) cells.</p>Formula:C30H27NO11Color and Shape:SolidMolecular weight:577.54LXR antagonist 2
<p>LXR antagonist 2 inhibits adipogenesis, downregulates LXR genes, and reduces lipids in hyperlipidemic mice (LXRβ IC50: 0.36μM, LXRα IC50: 2.25μM).</p>Formula:C34H40N2O5SColor and Shape:SolidMolecular weight:588.76Antitubercular agent-29
<p>Compound 6xa inhibits drug-resistant tuberculosis with MICs 0.03 μg/mL for DS-Mtb and 0.03-0.06 for DR-Mtb, SI>40 for Vero cells.</p>Formula:C20H12ClN3O5Color and Shape:SolidMolecular weight:409.78Omaciclovir
CAS:<p>Omaciclovir (ABT-091) is a herpesvirus herpesvirus replication inhibitor with antiviral activity that is used in the study of herpesvirus infections.</p>Formula:C10H15N5O3Purity:99.46% - 99.46%Color and Shape:SolidMolecular weight:253.26THR-β agonist 5
CAS:<p>THR-β agonist 5 (compound 54) is a potent THR-β agonist, with an EC 50 of <50 nM [1].</p>Formula:C22H23N5O2Color and Shape:SolidMolecular weight:389.45Fipravirimat
CAS:<p>Fipravirimat is a potent inhibitor of HIV-1 with potential applications in HIV and AIDS research.</p>Formula:C43H67FN2O4SColor and Shape:SolidMolecular weight:727.07ATR-IN-11
<p>ATR-IN-11, a potent ATR kinase inhibitor, shows promise as a lead for DNA damage response-targeted cancer drugs.</p>Formula:C25H30N6O2Color and Shape:SolidMolecular weight:446.54Pefcalcitol
CAS:<p>Pefcalcitol is a novel antipsoriatic prodrug candidate containing a 16-en-22-oxa-vitamin D3 structure.</p>Formula:C26H34F5NO4Color and Shape:SolidMolecular weight:519.54JH-XVII-10
<p>JH-XVII-10: potent, oral DYRK1A/B inhibitor (IC50: 3/5 nM), shows antitumor activity in HNSCC.</p>Formula:C21H16F4N8OColor and Shape:SolidMolecular weight:472.4Monoamine Oxidase B inhibitor 1
<p>Potent, selective MAO-B inhibitor; reversible; oral; crosses BBB; IC50=0.02 nM; potential for Parkinson's research.</p>Formula:C18H15FO3Color and Shape:SolidMolecular weight:298.31Estrogen receptor antagonist 4
CAS:<p>Estrogen receptor antagonist 4 blocks ER, impacting cell growth and cancer research potential.</p>Formula:C23H29BF4N4O2Color and Shape:SolidMolecular weight:480.31HIV-1 inhibitor-40
<p>HIV-1 inhibitor-40 (4ab) is a potent NNRTI (EC50: 1.9 nM), non-toxic in vivo, and a sensitive CYP inhibitor.</p>Formula:C25H18N6O2Color and Shape:SolidMolecular weight:434.45CYP121A1-IN-1
<p>CYP121A1-IN-1: Strong inhibitor for CYP121A1, hinders Mycobacterium tuberculosis growth (MIC 90 ~6.25 μM), reduces mycocyclosin synthesis.</p>Formula:C22H20N4OColor and Shape:SolidMolecular weight:356.42Saphenamycin
CAS:<p>Saphenamycin is an antibiotic from a strain of Streptomyces.</p>Formula:C23H18N2O5Purity:98%Color and Shape:SolidMolecular weight:402.40BW A868C
CAS:BW A868C is a potent, selective PGD2 antagonist and a BW245C analogue, inert to other prostaglandin receptors.Formula:C25H37N3O5Color and Shape:SolidMolecular weight:459.58ZLWT-37
<p>ZLWT-37: Oral CDK inhibitor, CDK9 IC50=0.002 µM, CDK2 IC50=0.054 µM; halts HCT116 cells at G2/M, induces apoptosis.</p>Formula:C26H30ClN5OColor and Shape:SolidMolecular weight:464TP-6076
CAS:<p>TP-6076 is a fluorocycline antibiotic, inhibiting bacterial protein synthesis, exhibiting great antimicrobial activity against carbapenem-resistant A.</p>Formula:C28H32F3N3O7Color and Shape:SolidMolecular weight:579.56Lamivudine, (+/-)-trans-
CAS:<p>Lamivudine, a drug for HIV-1 and HBV, inhibits reverse transcriptase and resembles zalcitabine.</p>Formula:C8H11N3O3SPurity:98%Color and Shape:SolidMolecular weight:229.26SD-2590 HCl
CAS:<p>SD-2590 HCl is an MMP-2,-3, -9, -8, 13, and -14 inhibitor.</p>Formula:C22H26ClF3N2O7SPurity:98%Color and Shape:SolidMolecular weight:554.96MEN-10354
CAS:<p>MEN-10354 is a less potent and less selective NK-2 tachykinin receptor antagonist compared to the linear analog, R 396.</p>Formula:C37H46N8O9Color and Shape:SolidMolecular weight:746.81Nedocromil sodium
CAS:<p>Nedocromil sodium is a pharmacologic stabilizer of mast cells, has been shown to normalize cytokine levels and attenuate cardiac remodeling.</p>Formula:C19H17NNaO7Purity:98%Color and Shape:SolidMolecular weight:394.335RORγt inhibitor 2
CAS:<p>RORγt Inhibitor 2, a potent inhibitor of RORγt, exhibits an IC50 of 9.2 nM and is utilized in the study of cancer, inflammation, or autoimmune diseases that are</p>Formula:C31H33F5N2O7SColor and Shape:SolidMolecular weight:672.663-IN-PP1
CAS:<p>3-IN-PP1: PKD inhibitor (IC50: 94-108 nM for PKD1/2/3), broad anticancer agent for research.</p>Formula:C17H18N6Color and Shape:SolidMolecular weight:306.36GLS-1-IN-1
<p>GLS-1-IN-1 (compound 1d) is a GLS-1 inhibitor that inhibits Hep G2, MCF 7 and MCF 10A cells.</p>Formula:C26H25FN4OSColor and Shape:SolidMolecular weight:460.5716,16-Dimethyl prostaglandin E2
CAS:<p>16,16-Dimethyl prostaglandin E2 regulates hematopoietic stem cells via EP2/EP4 and Wnt, taken orally.</p>Formula:C22H36O5Purity:98%Color and Shape:SolidMolecular weight:380.52BRD5631
CAS:<p>BRD5631 is an autophagy enhancer, enhances autophagy through an mTOR-independent pathway.</p>Formula:C30H35N3O4Purity:98%Color and Shape:SolidMolecular weight:501.62Resolvin E4
CAS:<p>RvE4, a bioactive lipid from eicosapentaenoic acid and synthesized by 15-LO, is anti-inflammatory and boosts efferocytosis in human macrophages.</p>Formula:C20H30O4Color and Shape:SolidMolecular weight:334.45JTP-117968
CAS:<p>JTP-117968: Non-steroidal SGRM, glucocorticoid receptor modulator, IC50 = 6.8 nM, offers better inhibitory/activatory balance.</p>Formula:C31H31F3N2O2Color and Shape:SolidMolecular weight:520.59Lu 26-046
CAS:<p>Lu 26-046 is a muscarinic receptor agonist.</p>Formula:C10H12N2OSColor and Shape:SolidMolecular weight:208.28FGFR4-IN-10
<p>FGFR4-IN-10 (compound 5a) is a potent, selective FGFR4 inhibitor with IC50 of 70.7 nM, sparing FGFR1-3.</p>Formula:C20H19F3N6O3Color and Shape:SolidMolecular weight:448.4Spicamycin
CAS:<p>Spicamycin can be used as a potent inducer of differentiation of human myeloid leukemia cells (HL-60) and murine myeloid leukemia cells (M1).</p>Formula:C30H51N7O7Color and Shape:SolidMolecular weight:621.77β-N-Acetyl-D-hexosaminidase-IN-1
<p>β-N-Acetyl-D-hexosaminidase-IN-1 is a newly discovered chemical compound that acts as an inhibitor for β-N-acetyl-D-hexosaminidase.</p>Formula:C18H13F2NO2SColor and Shape:SolidMolecular weight:345.36Keap1-Nrf2-IN-4
<p>Keap1-Nrf2-IN-4 hinders MGC-803 cell growth (IC50=2.55μM), migration, and induces apoptosis with low toxicity.</p>Formula:C26H34N2OColor and Shape:SolidMolecular weight:390.56XIAP degrader-1
<p>XIAP degrader-1 is a small primary amine molecule that promotes the degradation of X-linked apoptosis inhibitory protein (XIAP).</p>Formula:C34H45N5O4Color and Shape:SolidMolecular weight:587.75LPA5 antagonist 1
<p>LPA5 antagonist 1: selective, potent (IC50=32 nM), high brain permeability, studies inflammatory/neuropathic pain.</p>Formula:C28H26N2O4SColor and Shape:SolidMolecular weight:486.58LSD1/2-IN-4
<p>LSD1/2-IN-4, a PCPA derivative, inhibits LSD1 (Ki 0.11 μM) & LSD2 (Ki 130 μM), potentially useful in T-cell leukemia research.</p>Formula:C9H8BrF2NColor and Shape:SolidMolecular weight:248.07Etamicastat
CAS:<p>Etamicastat can be used in the research of cardiovascular diseases.</p>Formula:C14H15F2N3OSPurity:98%Color and Shape:SolidMolecular weight:311.35(E)-10-Hydroxynortriptyline maleate
CAS:<p>(E)-10-Hydroxy Nortriptyline maleate, a derivative of antidepressant Nortriptyline, eases depression symptoms.</p>Formula:C23H25NO5Purity:98%Color and Shape:SolidMolecular weight:395.4555-Ph-IAA-AM
<p>5-Ph-IAA-AM, eggshell-permeable analog of 5-Ph-IAA, boosts protein degradation in embryos, useful for studying proteins in C. elegans.</p>Formula:C19H17NO4Color and Shape:SolidMolecular weight:323.34hCA IX-IN-1
<p>hCA IX-IN-1 inhibits human carbonic anhydrases I, II, IX, and XII with Ki values of 331.4, 28.4, 9.4, 17.8 nM and exhibits anticancer properties.</p>Formula:C19H18N2O3SColor and Shape:SolidMolecular weight:354.42SphK1-IN-2
<p>SphK1-IN-2: SphK1 inhibitor, IC50: 19.81 nM; less effective on SphK2. Induces apoptosis, hinders cancer cell growth.</p>Formula:C27H30BrNO4SColor and Shape:SolidMolecular weight:544.5LY503430
CAS:<p>LY503430: Oral AMPA enhancer with nootropic, neuroprotective properties, mitigates 6-OHDA/MPTP brain damage.</p>Formula:C20H25FN2O3SPurity:98%Color and Shape:SolidMolecular weight:392.49VEGFR-IN-3
CAS:<p>VEGFR-IN-3 inhibits cancer cell growth (OVCAR-4, MDA-MB-468) with IC50s: 0.29, 0.35μM. Used in cancer research.</p>Formula:C27H28N2O6Color and Shape:SolidMolecular weight:476.52O4
CAS:<p>O4 is a novel stabilizer of amyloid- fibrils. O4 used for accelerating the formation of end-stage mature fibrils.</p>Formula:C24H15NO7Purity:98%Color and Shape:SolidMolecular weight:429.38
