Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,832 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,875 products)
- Chromatin/Epigenetics(2,611 products)
- Cytoskeletal Signaling(1,564 products)
- DNA Damage/DNA Repair(2,873 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,014 products)
- Immunology and Inflammation(3,900 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,256 products)
- Membrane Transporter/Ion Channel(3,154 products)
- Metabolism(10,139 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,369 products)
- Other Inhibitors(35,851 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,429 products)
- Proteases/Proteasome(1,690 products)
- Stem Cell and Derivatives(734 products)
- Tyrosine Kinase/Adaptors(1,982 products)
- Ubiquitination(1,725 products)
Show 16 more subcategories
Found 66522 products of "Inhibitors"
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K00135
CAS:K00135 (IMIDAZOPYRIDAZIN 1) is a selective inhibitor of Pim kinases and can be used in studies about gastric cancer and antileukemic therapeutics.Formula:C18H18N4OPurity:98.16%Color and Shape:SolidMolecular weight:306.36BI-4924
CAS:BI-4924 is a PHGDH inhibitor that disrupts serine biosynthesis by intracellular trapping and can be used to study metabolic disorders.Formula:C21H20Cl2N2O6SPurity:99.55%Color and Shape:SolidMolecular weight:499.36Tulopafant
CAS:Tulopafant (RP 59227) is a potent platelet-activating factor (PAF) antagonist that increases capillary patency and prolongs allograft heart survival.Formula:C25H19N3O2SPurity:99.38%Color and Shape:SolidMolecular weight:425.5LKM38
CAS:LKM38, a cholesterol probe, mimics cholesterol, supports resistant cell growth, and regulates homeostasis, aiding in cholesterol protein studies.Formula:C28H44N2OPurity:97.75%Color and Shape:SolidMolecular weight:424.66FAAH-IN-1
CAS:FAAH-IN-1 is a fatty acid amide hydrolase (FAAH) inhibitor, with IC50s of 145 nM and 650 nM for rat and human FAAH, respectively.Formula:C20H19ClN4OSPurity:98%Color and Shape:SolidMolecular weight:398.91NF-κB-IN-11
CAS:NF-κB-IN-11 (Compound 3i) is an inhibitor of NF-κB, effectively blocking TNF-α-induced NF-κB pathway activation and the nuclear translocation of NF-κB.Formula:C19H18O5Purity:98%Color and Shape:SolidMolecular weight:326.34Aftobetin
CAS:Aftobetin is a biochemical.Formula:C26H32N2O5Color and Shape:SolidMolecular weight:452.545-Methylurapidil
CAS:5-Methylurapidil is an alpha1A-adrenoceptor antagonist.Formula:C21H31N5O3Purity:98%Color and Shape:SolidMolecular weight:401.5(Rac)-Etavopivat
CAS:(Rac)-Etavopivat, an oral PKR activator, targets sickle cell disease and haemoglobinopathies.Formula:C22H23N3O6SColor and Shape:SolidMolecular weight:457.5RAC 109
CAS:RAC 109 is a chiral antiarrhythmic agent.Formula:C20H28N2O2Purity:98%Color and Shape:SolidMolecular weight:328.45Sisapronil
CAS:Sisapronil is a member of the phenylpyrazole class of antiparasitics.
Formula:C15H6Cl2F8N4Color and Shape:SolidMolecular weight:465.13Retaspimycin
CAS:Retaspimycin is a potent and water-soluble Hsp90 inhibitor(EC50s of 119 nM for both Hsp90 and Grp9).Formula:C31H45N3O8Purity:98%Color and Shape:SolidMolecular weight:587.7Seviteronel R enantiomer
CAS:Seviteronel R enantiomer (VT-464 R enantiomer) is a Seviteronel isomer produced during the manufacturing process.Formula:C18H17F4N3O3Purity:97.97% - >99.99%Color and Shape:SolidMolecular weight:399.34Ref: TM-T13312
1mg105.00€5mg245.00€10mg358.00€25mg610.00€50mg867.00€100mg1,153.00€1mL*10mM (DMSO)268.00€SNT-207858
CAS:SNT-207858: selective, BBB-penetrating, oral MC-4 receptor antagonist with 22 nM IC50 (binding), 11 nM (function).Formula:C32H45Cl4N5O3Purity:98%Color and Shape:SolidMolecular weight:689.54DA 5018
CAS:DA 5018 is a capsaicin derivative and is also a new non-narcotic analgesic. It has an antipruritic effect.Formula:C22H31ClN2O3Purity:98%Color and Shape:SolidMolecular weight:406.95TTT-28
CAS:TTT-28, a thiazole-valine peptidomimetic, selectively inhibits ABCB1 to reverse MDR with low toxicity.Formula:C31H31N3O6SPurity:98%Color and Shape:SolidMolecular weight:573.66Razaxaban hydrochloride
CAS:Razaxaban hydrochloride is a highly potent, selective and orally active inhibitor of factor Xa(Ki of 0.19 nM),has strongly antithrombotic activity.Formula:C24H21ClF4N8O2Purity:98%Color and Shape:SolidMolecular weight:564.92LUF 6283
CAS:partial agonist of hydroxycarboxylic acid receptor 2 (HCA2)Formula:C8H12N2O2Purity:99.41%Color and Shape:SolidMolecular weight:168.19Ref: TM-T22938
1mg35.00€5mg75.00€10mg92.00€25mg158.00€50mg227.00€100mg339.00€1mL*10mM (DMSO)To inquireEbselen oxide
CAS:Ebselen oxide (EB-2) is a HER2 inhibitor with antibacterial and antifungal activity and has shown cytoprotective effects against HN2 in vitro.Formula:C13H9NO2SePurity:98%Color and Shape:SolidMolecular weight:290.18Azelastine
CAS:Azelastine (Azelastinum) is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.Formula:C22H24ClN3OPurity:99.35% - 99.99%Color and Shape:White Crystal PowderMolecular weight:381.90BMS270394
CAS:BMS270394 is a RARγ agonist used in the study of breast cancer and skin diseases.Formula:C23H26FNO4Color and Shape:SolidMolecular weight:399.46VU0410425
CAS:VU0410425 is a metabotropic glutamate receptor subtype 1 negative allosteric modulator.Formula:C19H16ClN3O3Purity:98%Color and Shape:SolidMolecular weight:369.84-Acetylsimvastatin
CAS:4-Acetylsimvastatin is acetylated simvastatin. Simvastatin is a competitive inhibitor of HMG-CoA reductase (Ki: 0.2 nM).Formula:C27H40O6Purity:98%Color and Shape:SolidMolecular weight:460.6L 368935
CAS:L 368935 is an antagonist of the cholecystokinin receptor.Formula:C27H26N8O2Purity:98%Color and Shape:SolidMolecular weight:494.55Nevanimibe
CAS:Nevanimibe is an orally active and selective inhibitor of acyl-coenzyme A:cholesterol O-acyltransferase 1 (ACAT1) (EC50 of 9 nM).Formula:C27H39N3OPurity:98%Color and Shape:SolidMolecular weight:421.62SPV106
CAS:SPV106 is a ligand of lysine acetyltransferases (KATs).Formula:C22H40O4Purity:98%Color and Shape:SolidMolecular weight:368.55N20C hydrochloride
CAS:N20C hydrochloride (2-((3,3-diphenylpropyl)amino)acetamide hydrochloride) is a non-competitive NMDA receptor open-channel blocker.Formula:C17H21ClN2OPurity:99.9%Color and Shape:SolidMolecular weight:304.81TH-Z835
CAS:TH-Z835 is a selective inhibitor for the KRAS (G12D) mutation, demonstrating an inhibitory concentration (IC50) of 1.6 μM.Formula:C30H38N6OPurity:98%Color and Shape:SolidMolecular weight:498.66Lubeluzole
CAS:Lubeluzole, a well-known neuroprotective agent, is recently proved useful to potentiate the activity of anti-cancer drugs.Formula:C22H25F2N3O2SPurity:98%Color and Shape:SolidMolecular weight:433.51IHVR-19029
CAS:IHVR-19029: ER α-glucosidases I/II inhibitor, IC50 0.48μM; halts Ebola, Dengue, Rift Valley fever virus replication.Formula:C23H45N3O5Color and Shape:SolidMolecular weight:443.62Droxicainide
CAS:Droxicainide is an antiarrhythmic agent.Formula:C16H24N2O2Purity:99.86%Color and Shape:SolidMolecular weight:276.37Ref: TM-T11099
1mg94.00€5mg167.00€10mg235.00€25mg366.00€50mg492.00€100mg637.00€200mg863.00€1mL*10mM (DMSO)167.00€Sp-Cyclic AMPS (sodium salt)
CAS:Sp-cAMPS Na salt activates PKA I/II and competitively inhibits PDE3A (Ki: 47.6 μM), also binds PDE10 GAF (EC50: 40 μM).Formula:C10H12N5NaO5PSColor and Shape:SolidMolecular weight:367.25Rolapitant
CAS:Rolapitant Hydrochloride is an oral NK1-receptor blocker that prevents nausea and has a fast onset and long half-life.Formula:C25H26F6N2O2Purity:99.86%Color and Shape:SolidMolecular weight:500.48Ref: TM-T3716
1mg48.00€2mg63.00€5mg88.00€10mg117.00€25mg178.00€50mg295.00€100mg442.00€500mg982.00€1mL*10mM (DMSO)96.00€2,5-Dihydroxybiphenyl
CAS:2,5-Dihydroxybiphenyl: a small molecule that induces trichothiodystrophy A protein dimerization, modulating TFIIH activity.
Formula:C12H10O2Purity:99.66%Color and Shape:White To Grey-Brownish PowderMolecular weight:186.21WS-383 free base
CAS:WS-383 free base is a selective and reversible DCN1-UBC12 interaction inhibitor(IC50 of 11 nM).Formula:C18H20ClN9S2Purity:98%Color and Shape:SolidMolecular weight:461.99MI-192
CAS:MI-192: Selective HDAC2/3 inhibitor, IC50=30/16 nM, induces apoptosis in myeloid leukemia, potential in leukemia/anti-stroke treatment.Formula:C24H21N3O2Color and Shape:SolidMolecular weight:383.44TWIK-1/TREK-1-IN-2
CAS:TWIK-1/TREK-1-IN-2 (Compound 2g) serves as an inhibitor of both TWIK-1 and TREK-1, targeting the TREK-1 homodimer and TWIK-1/TREK-1 heterodimer with IC50 valuesFormula:C20H29F3N2O2Purity:98%Color and Shape:SolidMolecular weight:386.45Galidesivir triphosphate
CAS:Galidesivir triphosphate halts viral RNA replication by inhibiting RDRP and NS5B, and combats Ebola in mice; derived from prodrug Galidesivir.Formula:C11H18N5O12P3Purity:98%Color and Shape:SolidMolecular weight:505.21(R)-Praziquantel
CAS:(R)-Praziquantel is an active enantiomer of praziquantel.Formula:C19H24N2O2Purity:98%Color and Shape:SolidMolecular weight:312.41Beaucage reagent
CAS:Beaucage reagent, which is found to be effective in causing DNA cleavage.Formula:C7H4O3S2Purity:98.50%Color and Shape:White To Off-White PowderMolecular weight:200.23ICI 162,846
CAS:ICI 162,846 is an orally active and potent H2 receptor antagonist that inhibits gastric secretion and may be used in the study of duodenal ulcers.Formula:C11H17F3N6OPurity:97.45%Color and Shape:SolidMolecular weight:306.29Clitocine
CAS:Clitocine, an adenosine analogue derived from mushrooms, is a potent transcriptional transducer, an inhibitor of nonsense mutations, and has anticancer activityFormula:C9H13N5O6Purity:≥95.0%Color and Shape:SolidMolecular weight:287.23Nicotinoyl cyclandelate
CAS:Nicotinoyl cyclandelate can effectively reduce blood pressure in the femoral artery and perfusion pressure in cerebral blood vessels.Formula:C23H27NO4Purity:98%Color and Shape:SolidMolecular weight:381.46SKLB70326
CAS:SKLB70326 is a cell-cycle progression inhibitor that acts by inducing G0/G1 phase arrest and apoptosis in human hepatic carcinoma cells.Formula:C15H13N3O2SPurity:98%Color and Shape:SolidMolecular weight:299.35ML089
CAS:ML089 (CID-22416235) is a phosphomannose isomerase (PMI) inhibitor.ML089 is a probe for the study of congenital dysglycosylation type Ia (CDG-Ia).Formula:C13H8FNOSPurity:99.86% - >99.99%Color and Shape:SolidMolecular weight:245.27AL-9
CAS:AL-9 is a GT-1b and GT-2a replication inhibitor.Formula:C23H22N4O3Purity:98%Color and Shape:SolidMolecular weight:402.45ERK1/2 inhibitor 1
CAS:ERK1/2 inhibitor 1 is a potent, orally bioavailable ERK1/2 inhibitor, showing 60% inhibition at 1 nM and an IC50 of 3.0 nM against ERK1 and ERK2, respectively.
Formula:C29H32ClN5O4Purity:98.81%Color and Shape:SolidMolecular weight:550.05Amcinafal
CAS:Amcinafal is an active diol,and used against virus replication and interferon production.Formula:C26H35FO6Purity:98%Color and Shape:SolidMolecular weight:462.557α,25-Dihydroxycholesterol
CAS:7α, 25-dihydroxycholesterol (7α,25-OHC) is a potent and selective agonist and endogenous ligand of the orphan GPCR receptor EBI2 (GPR183).Formula:C27H46O3Purity:98%Color and Shape:SolidMolecular weight:418.65(RS)-Eflucimibe
CAS:Eflucimibe is an ACAT inhibitor.Formula:C29H43NO2SPurity:98%Color and Shape:SolidMolecular weight:469.72
