Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,832 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,875 products)
- Chromatin/Epigenetics(2,611 products)
- Cytoskeletal Signaling(1,563 products)
- DNA Damage/DNA Repair(2,873 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,014 products)
- Immunology and Inflammation(3,900 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,256 products)
- Membrane Transporter/Ion Channel(3,154 products)
- Metabolism(10,141 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,369 products)
- Other Inhibitors(35,851 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,429 products)
- Proteases/Proteasome(1,690 products)
- Stem Cell and Derivatives(735 products)
- Tyrosine Kinase/Adaptors(1,982 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66522 products of "Inhibitors"
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OT antagonist 1
CAS:OT antagonist 1 is a potent and selective antagonist of Oxytocin(Ki of 50 nM)Formula:C22H22N4O3Purity:98%Color and Shape:SolidMolecular weight:390.44Antitrypanosomal agent 4
CAS:Compound 19: potent, blood-brain penetrant antitrypanosomal; IC50: T. cruzi 1.2 μM, T.b. brucei 70 nM.Formula:C18H14ClN3O5SColor and Shape:SolidMolecular weight:419.84Boxidine
CAS:Boxidine inhibits the transformation of 7-dehydrocholesterol to cholesterol & also inhibits sterol absorption.Formula:C19H20F3NOColor and Shape:SolidMolecular weight:335.36SGX393
CAS:SGX393 is an inhibitor of the CML mutant Bcr-AblT315I, thereby preempting in vitro resistance when combined with nilotinib or dasatinib.Formula:C21H22N6OColor and Shape:SolidMolecular weight:374.44O-2093
CAS:anandamide uptake inhibitorFormula:C34H43Cl2NO3Purity:98%Color and Shape:SolidMolecular weight:584.62Indantadol HCl
CAS:Indantadol HCl (CHF-3381) is a NMDA antagonist and nonselective MAO inhibitor.Formula:C11H15ClN2OPurity:99.56%Color and Shape:SolidMolecular weight:226.7PBOX-15
CAS:PBOX-15 induces apoptosis, regulates death receptors, enhances TRAIL effects, and inhibits T cell migration in myeloma cells.Formula:C28H19NO3Color and Shape:SolidMolecular weight:417.46Tyrosinase-IN-12
CAS:Tyrosinase-IN-12(Non-competitive tyrosinase inhibitor) is a potent non-competitive tyrosinase inhibitor with an IC50 of 49.33 ± 2.64 µM and a Ki of 31.25 ± 0.25Formula:C16H12ClN3SPurity:99.2%Color and Shape:SoildMolecular weight:313.8RU 45144
CAS:RU 45144 is an estradiol derivative with antiestrogenic activity.Formula:C28H37NO3Purity:98%Color and Shape:SolidMolecular weight:435.6Perzinfotel
CAS:Perzinfotel, a neuroprotective NMDA antagonist with high affinity (IC50=30 nM), is selective and competitive.Formula:C9H13N2O5PColor and Shape:SolidMolecular weight:260.18Dexlofexidine Free Base
CAS:Dexlofexidine Free Base is a less potent (+) isomer of lofexidine and an alpha-2 adrenoceptor agonist, 10x weaker than levlofexidine.Formula:C11H12Cl2N2OColor and Shape:SolidMolecular weight:259.13Ipsalazide
CAS:Ipsalazide is a novel salicylazosulfapyridine analog for the treatment of inflammatory bowel disease.
Formula:C16H11N3Na2O6Purity:99.43%Color and Shape:SolidMolecular weight:387.25Anabasine hydrochloride
CAS:neuronal nicotinic ACh receptor partial agonistFormula:C10H15ClN2Purity:98%Color and Shape:White To Off-White SolidMolecular weight:198.693McN5691
CAS:McN5691 is a voltage sensitive calcium channel blocker.Formula:C30H35NO3Purity:98.93% - 99.38%Color and Shape:SolidMolecular weight:457.6Kelletinin I
CAS:Kelletinin I inhibit preferentially DNA polymerase alpha.Formula:C32H26O12Purity:98%Color and Shape:SolidMolecular weight:602.54JR-AB2-011
CAS:JR-AB2-011: selective mTORC2 inhibitor, IC50 = 0.36μM, blocks Rictor-mTOR, Ki = 0.19μM, cytotoxic in glioblastoma.Formula:C17H14Cl2FN3OSPurity:98.33% - 99.41%Color and Shape:SolidMolecular weight:398.28Ref: TM-T11728
1mg90.00€5mg192.00€10mg326.00€25mg597.00€50mg895.00€100mg1,198.00€1mL*10mM (DMSO)212.00€L-NMMA acetate
CAS:L-NMMA acetate inhibits all NOS types (nNOS, eNOS, iNOS); Ki: 0.18, 0.4, 6 µM respectively.Formula:C9H20N4O4Purity:99.72% - 99.80%Color and Shape:White To Off-White SolidMolecular weight:248.28Antiparasitic agent-10
CAS:Antiparasitic agent-10 (Compound 94) targets Schistosoma mansoni, shows promise for treating Schistosomiasis.Formula:C13H17N3O4S3Color and Shape:SolidMolecular weight:375.49N-Monoacetylcystine
CAS:N-Monoacetylcystine is a paracetamol poisoning antidote. It is used in the treatment of influenza A virus pandemic.Formula:C8H14N2O5S2Purity:98%Color and Shape:SolidMolecular weight:282.34Texasin
CAS:Texasin is a selective inhibitor of human leukocyte 5-lipoxygenase.Formula:C16H12O5Purity:98%Color and Shape:SolidMolecular weight:284.26ABT-100
CAS:ABT-100 is a potent, highly selective, and orally active farnesyl transferase inhibitor with broad-spectrum antitumor activity.Formula:C27H19F3N4O3Purity:98%Color and Shape:SolidMolecular weight:504.46Flutroline
CAS:Flutroline is a gamma-carboline antipsychotic agent.Formula:C27H25F3N2OColor and Shape:SolidMolecular weight:450.5P2Y1-IN-16
CAS:P2Y1-IN-16 is a novel antagonist of P2Y1.Formula:C23H22F3N3O2Color and Shape:SolidMolecular weight:429.43J 2931
CAS:J 2931 is an inhibitor of mosquito larvae growth.Formula:C23H32O2Color and Shape:SolidMolecular weight:340.5Ambrein
CAS:Ambrein, main in ambergris and sperm whale secretion, may enhance aphrodisiac effects; serves as a precursor for scent derivatives and acts as an analgesic.Formula:C30H52OColor and Shape:SolidMolecular weight:428.73Anti-inflammatory agent 54
CAS:Anti-inflammatory agent 54 (compound 9c), a Coixol derivative, exhibits anti-inflammatory properties by inhibiting the NF-κB pathway and reducing the expressionFormula:C17H16N2O5Color and Shape:SolidMolecular weight:328.32NEP-28
CAS:NEP-28, a novel SARM, is a highly selective AR agonist with superior tissue-selective effects and boosts neprilysin activity.Formula:C10H10BrF3N2SColor and Shape:SolidMolecular weight:327.16IRC-083927 HCl
CAS:IRC-083927 HCl, a novel anticancer agent, blocks microtubule assembly, hinders cancer cell growth, and is effective against drug-resistant tumors.Formula:C22H19FN4O4SColor and Shape:SolidMolecular weight:454.47Pulrodemstat Methylbenzenesulfonate
CAS:LSD1-IN-7 Methylbenzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.Formula:C31H31F2N5O5SPurity:98%Color and Shape:SolidMolecular weight:623.67NL-103
CAS:NL-103, a dual-targeting compound, inhibits HDACs & Hh pathway, countering vismodegib-resistant Smo mutations.Formula:C26H27Cl2N5O4Color and Shape:SolidMolecular weight:544.43FR-7534
CAS:FR-7534 is a calcium antagonist structurally similar to nifedipine.Formula:C19H22N2O7Color and Shape:SolidMolecular weight:390.39NC-2100
CAS:NC-2100 is an aperoxisome proliferator-activated receptor-gamma (PPARgamma) activator.Formula:C20H16N2O3SColor and Shape:SolidMolecular weight:364.42Darinaparsin
CAS:Darinaparsin, a dimethylated arsenic-glutathione compound, is cytotoxic to various cancer cells with diverse IC50 values and inhibits tumor growth in mice.Formula:C12H22AsN3O6SColor and Shape:SolidMolecular weight:411.31SKF 86466 hydrochloride
CAS:SKF 86466 hydrochloride is an α2-adrenoceptor antagonist.Formula:C11H15Cl2NPurity:98%Color and Shape:SolidMolecular weight:232.15CGI560
CAS:CGI560 is a potent BTK inhibitor with IC50 = 400 nM for BTK.Formula:C29H27N5OColor and Shape:SolidMolecular weight:461.56ARUK3001185
CAS:ARUK3001185 (8l): potent, selective Notum inhibitor; oral, brain-penetrant; IC50=6.7 nM; for rodent disease models.Formula:C9H4Cl2F3N3Color and Shape:SolidMolecular weight:282.05HIV-1 inhibitor-45
CAS:HIV-1 inhibitor-45 is a potent inhibitor of HIV-1 RNase H (IC50: 0.067 μM) and has antiviral effects.Formula:C23H24N4O8SColor and Shape:SolidMolecular weight:516.52RyRs activator 3
CAS:RyRs activator 3 (compound A4) serves as an insecticide highly effective against both the diamondback moths, M.Formula:C23H19BrCl2N6O3Purity:98%Color and Shape:SolidMolecular weight:578.25HCV-IN-3
CAS:HCV-IN-3 is a hepatitis C virus (HCV) NS3/4a protein inhibitor (IC50: 20 μM; Kd: 29 μM).Formula:C13H11F2NOPurity:98%Color and Shape:SolidMolecular weight:235.23AZD5213
CAS:AZD5213: selective human H3 receptor antagonist, pKi 9.3, for sleep/cognition research.Formula:C19H25N3O2Color and Shape:SolidMolecular weight:327.42CGS 24891
CAS:CGS 24891 is a 5-lipoxygenase inhibitor.Formula:C18H17FN2O4Color and Shape:SolidMolecular weight:344.34APX2009
CAS:APX2009, a 2nd-gen APE1/Ref-1 inhibitor, curbs NFkB activity, survivin, and prostate cancer cell growth; induces cell cycle arrest.Formula:C21H25NO4Color and Shape:SolidMolecular weight:355.43AHR antagonist 5
CAS:Potent, oral AHR blocker from WO2018195397; IC50 < 0.5μM; hinders tumor growth with anti-PD-1.Formula:C25H27Cl3FN7Purity:98%Color and Shape:SolidMolecular weight:550.89BAY-707 acetate
CAS:BAY-707: potent, selective MTH1 inhibitor with excellent engagement and pharmacokinetics but no anticancer efficacy alone or combined.Formula:C17H24N4O4Color and Shape:SolidMolecular weight:348.18Momelotinib Mesylate
CAS:Momelotinib Mesylate is an ATP-competitive JAK1/JAK2 inhibitor (IC50: 11 nM/18 nM). It has 10-fold selectivity versus JAK3.Formula:C24H26N6O5SPurity:98%Color and Shape:SolidMolecular weight:510.57α-Lipoic Acid Choline Ester
CAS:Alpha-Lipoic Acid Choline Ester is used potentially to treat presbyopia.Formula:C13H26ClNO2S2Purity:98%Color and Shape:SolidMolecular weight:327.93ICSN3250
CAS:ICSN3250 is a novel specific mTOR inhibitor via a unique mechanism which is distinct from previous mTOR inhibitors.Formula:C31H40N4O8Color and Shape:SolidMolecular weight:596.67LCAHA
CAS:LCAHA is a USP2a inhibitor. LCAHA inhibits growth of cyclin D1-dependent cells.Formula:C24H41NO3Color and Shape:SolidMolecular weight:391.59LC-1028
CAS:LC-1028 is a novel potent selective, covalent and irreversible inhibitor of p97 (valosin-containing protein) with IC50 =33 nM.Formula:C28H27N5OColor and Shape:SolidMolecular weight:449.55Cyanabactin
CAS:Cyanabactin is a novel ABA receptor agonist. It preferentially activates Pyrabactin Resistance 1 (PYR1) with low nanomolar potency.Formula:C18H18N2O2SColor and Shape:SolidMolecular weight:326.41
