Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,832 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,875 products)
- Chromatin/Epigenetics(2,611 products)
- Cytoskeletal Signaling(1,564 products)
- DNA Damage/DNA Repair(2,873 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,014 products)
- Immunology and Inflammation(3,900 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,256 products)
- Membrane Transporter/Ion Channel(3,154 products)
- Metabolism(10,139 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,369 products)
- Other Inhibitors(35,851 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,429 products)
- Proteases/Proteasome(1,690 products)
- Stem Cell and Derivatives(734 products)
- Tyrosine Kinase/Adaptors(1,982 products)
- Ubiquitination(1,725 products)
Show 16 more subcategories
Found 66522 products of "Inhibitors"
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Mercaptomerin sodium
CAS:Mercaptomerin sodium can be used to treat cardiac edema.Formula:C16H25HgNNaO6SColor and Shape:SolidMolecular weight:583.02SDZ-285604
CAS:SDZ-285604 is a novel sterol 14a-demethylases (CYP51) inhibitor.Formula:C24H20ClN3OColor and Shape:SolidMolecular weight:401.89Dexetimide HCl
CAS:Dexetimide HCl is a muscarinic antagonist that has been used to treat neuroleptic-induced parkinsonism. Benzetimide is the (-)-enantimorph of dexetimide.Formula:C23H27ClN2O2Color and Shape:SolidMolecular weight:398.93HL271
CAS:HL271, a derivative of metformin, is a potent AMPK activator that increases AMPK phosphorylation. HL271 attenuates aging-associated cognitive impairment.Formula:C13H17ClF3N5OPurity:98%Color and Shape:SolidMolecular weight:351.76Ibodutant
CAS:Ibodutant is an effective and selective tachykinin NK2 receptor antagonist (pKi: 10.1).Formula:C37H48N4O4SPurity:98%Color and Shape:SolidMolecular weight:644.87CJ-14897
CAS:CJ-14897 is the (7R,8S)-isomer; a cytokine production inhibitor.Formula:C12H15NO5Color and Shape:SolidMolecular weight:253.25CTPB
CAS:CTPB is a potent p300 histone acetyltransferase (HAT) activator that can be used in the preparation of hair growth promoters and/or hair loss treatments.Formula:C31H43ClF3NO2Purity:99.51%Color and Shape:SolidMolecular weight:554.13RSK2-IN-2
CAS:RSK2-IN-2 (Compound 25) is a reversible covalent inhibitor of the RPS6KA3 ( RSK2 ) kinase which also inhibits MSK1, MSK2, and RSK3 [1].Formula:C16H11N5OColor and Shape:SolidMolecular weight:289.29Tinlorafenib
CAS:Tinlorafenib (PF-07284890), a BRAFV600E/K inhibitor, is oral & CNS-permeable, used for BRAF-linked CNS tumors. IC50: 4.25/2.7 nM.Formula:C19H19ClF2N4O3SColor and Shape:SolidMolecular weight:456.89INF55
CAS:INF55 inhibits NorA efflux pump.Formula:C14H10N2O2Purity:98%Color and Shape:SolidMolecular weight:238.24EGFR-IN-46
CAS:EGFR-IN-46: Potent EGFR/FAK inhibitor (IC50: 20.17 & 14.25 nM), curbs cancer cell growth, triggers apoptosis.Formula:C27H32F3N3O3Color and Shape:SolidMolecular weight:503.561E7-03
CAS:1E7-03 is an inhibitor of HIV-1 transcription, by targeting host Protein Phosphatase-1 (PP1).Formula:C28H29N3O6Color and Shape:SolidMolecular weight:503.55(+/-)-PPCC oxalate
CAS:Sigma receptor ligand with high sigma-1 affinity; binds sigma-2 as well (Ki = 1.5 & 50.8 nM). Selective over dopaminergic, muscarinic receptors, DAT, SERT.Formula:C50H60N2O10Color and Shape:SolidMolecular weight:849.0345-trans-Prostaglandin E2
CAS:5-trans-PGE2 speeds up fibrinolysis, boosts tissue-PA mediated plasminogen activation, and blocks platelet clumping in human PRP.Formula:C20H32O5Color and Shape:SolidMolecular weight:352.47Pirifibrate
CAS:Pirifibrate (EL-466) can be used in the hyperlipoproteinemias research that is a hypolipemic substance [1].
Formula:C17H18ClNO4Color and Shape:SolidMolecular weight:335.78SIB-1553A hydrochloride
CAS:SIB-1553A hydrochloride is a nicotinic acetylcholine receptor agonist and a selective neuronal nAChR ligandFormula:C13H20ClNOSPurity:99.56% - 99.73%Color and Shape:SolidMolecular weight:273.82Acetyltrialanine
CAS:Acetyltrialanine is a dipeptide compound that binds at two sites on the Tb+3-pancreatic elastase complex and can be used as a nitrogen source.Formula:C11H19N3O5Purity:97.03%Color and Shape:White PowderMolecular weight:273.29AG-205
CAS:(rac)-AG-205 inhibits Pgrmc1, affects sterol gene INSIG1, and hinder NF-kB/BDNF/PI3K/AKT in neuronal hypoxic resistance.Formula:C22H23ClN6OSColor and Shape:SolidMolecular weight:454.98Perimetazine
CAS:Perimetazine has effects on central nervous system depressent such as sedative and muscle relaxant effects.Formula:C22H28N2O2SColor and Shape:SolidMolecular weight:384.53NSC109131
CAS:NSC109131 is an inhibitor of human tyrosyl-DNA phosphodiesterase 1 (TDP1).Formula:C27H34N4O2SColor and Shape:SolidMolecular weight:478.65ONO-1603
CAS:ONO-1603, a prolyl endopeptidase inhibitor, is used potentially for the treatment of Alzheimer's disease.Formula:C16H19ClN2O3Purity:98%Color and Shape:SolidMolecular weight:322.79N-Boc-15-aminopentadecanoic acid
CAS:N-Boc-15-aminopentadecanoic acid, an alkane with carboxylic end and Boc-protected amine, useful as a PROTAC linker.Formula:C20H39NO4Color and Shape:SolidMolecular weight:357.53PDE5-IN-3
CAS:PDE5-IN-3: Inhibits PDE5 (1.57 nM), EGFR (5.827 μM), Wnt pathway (1286.96 ng/mL), induces apoptosis, and has antitumor effects.Formula:C21H14BrN5O2Color and Shape:SolidMolecular weight:448.27Exifone
CAS:Exifone (NSC-680919) is a mixed, nonessential activator of HDAC1 that is capable of binding to both free and substrate-bound enzyme, resulting in an increasedFormula:C13H10O7Purity:99.77% - 99.95%Color and Shape:Yellow SolidMolecular weight:278.21Dexnafenodone Hydrochloride
CAS:Dexnafenodone Hydrochloride is an adrenergic receptor antagonist and serotonin uptake inhibitor.Formula:C20H24ClNOColor and Shape:SolidMolecular weight:329.86MRS2603
CAS:MRS2603 is an antagonist of P2Y1 and P2Y13 receptors in 1321N1 human astrocytoma cells.Formula:C14H12ClN4O8PPurity:98%Color and Shape:SolidMolecular weight:430.69CAY10506
CAS:CAY10506, a hybrid lipoic acid-TZD, activates PPARγ to control glucose and lipid levels with an EC50 of 10 μM.Formula:C20H26N2O4S3Color and Shape:SolidMolecular weight:454.63Darexaban glucuronide
CAS:Darexaban glucuronide is the major component in plasma after oral administration of darexaban to humans. Darexaban (YM150) is a direct inhibitor of factor Xa.Formula:C33H38N4O10Color and Shape:SolidMolecular weight:650.68Hexamide
CAS:Hexamide is a protein inhibitor.Formula:C13H17NOColor and Shape:SolidMolecular weight:203.28Naftidrofuryl
CAS:Naftidrofuryl treats peripheral and cerebral vascular issues, boosts cell oxidation, and relaxes muscles.Formula:C24H33NO3Color and Shape:SolidMolecular weight:383.52MDH1-IN-2
CAS:MDH1-IN-2 is a potent MDH1 inhibitor with potential anticancer activity for the study of diseases related to the immune system.Formula:C25H33NO5Purity:99.21%Color and Shape:SolidMolecular weight:427.53Rimiterol
CAS:Rimiterol, a beta 2 stimulant, therefore affects the cardiovascular system less than isoproterenol.Formula:C12H17NO3Color and Shape:SolidMolecular weight:223.27GSK575594A
CAS:GSK575594A is a selective agonist of GPR55.Formula:C24H23F2N3O3SColor and Shape:SolidMolecular weight:471.52GTS467
CAS:GTS467 is a EAAT2 Activator.Formula:C22H28N4O3Color and Shape:SolidMolecular weight:396.48DHODH-IN-20
CAS:Dhodh-in-20 (Compound 133), a potent DHODH inhibitor, may help study acute myeloid leukemia and inhibit tumor growth.Formula:C24H25F4N3O3Color and Shape:SolidMolecular weight:479.47BIPM
CAS:BIPM inhibits ROCK2, alters SH-SY5Y cell migration, actin fibers, neurite length, and reduces cofilin phosphorylation.Formula:C23H22N2O3Color and Shape:SolidMolecular weight:374.43R 151885
CAS:R 151885 delays ovulation in rats.Formula:C16H13F2N3OColor and Shape:SolidMolecular weight:301.29K812
CAS:K812 is an ASK1-specific inhibitor discovered to prolong survival in a mouse model of amyotrophic lateral sclerosis.Formula:C30H27N3O5Color and Shape:SolidMolecular weight:509.55AChE-IN-21
CAS:AChE-IN-21 (I-8), potent, selective AChE inhibitor, IC50: 2.66 nM, good BBB permeability.Formula:C24H29NO4Color and Shape:SolidMolecular weight:395.49BI-831266
CAS:BI-831266 is a potent and selective Aurora kinase B inhibitor.Formula:C27H38ClN7O2Color and Shape:SolidMolecular weight:528.09Blancoxanthone
CAS:Blancoxanthone, a plant-derived molecule, may inhibit COVID-19, influenza, SARS, and MERS-CoV.Formula:C23H22O5Color and Shape:SolidMolecular weight:378.42TC-G 1000
CAS:α2D-adrenoceptor agonistFormula:C17H18N2O4SPurity:98%Color and Shape:SolidMolecular weight:346.4ML 1035
CAS:ML 1035 is a benzamide that elicits contractions from guinea-pig non-stimulated ileum.Formula:C18H19ClN4O6Color and Shape:SolidMolecular weight:422.82A-1048400
CAS:A-1048400 is a potent and selective N-type and T-type calcium channel blocker.Formula:C36H37N3O2Color and Shape:SolidMolecular weight:543.7ZLD2218
CAS:ZLD2218, a potent inhibitor of BRD4 with an IC50 value of 107 nM, has been demonstrated to mitigate kidney injury and fibrosis through extensive studies.Formula:C22H18N4OColor and Shape:SolidMolecular weight:354.4Bicisate dihydrochloride
CAS:Bicisate dihydrochloride is usually complex with technetium Tc99m to measure cerebral blood flow with single-photon emission computed tomography (SPECT).Formula:C12H26Cl2N2O4S2Color and Shape:SolidMolecular weight:397.38Butacaine sulfate
CAS:Butacaine sulfate is applied to mucous membranes as a local anesthetic.Formula:C18H30N2O2H2O4SColor and Shape:Off-White SolidMolecular weight:355.48Helenalin Acetate
CAS:Helenalin Acetate: anti-inflammatory, anti-cancer, hinders C/EBPß and p300 cooperation.Formula:C17H20O5Purity:98%Color and Shape:SolidMolecular weight:304.34U 84569
CAS:U-84569 blocks human platelet clustering by reducing cAMP phosphodiesterase activity and platelet PLC activity.Formula:C25H23NO4Color and Shape:SolidMolecular weight:401.45Ro 363
CAS:RO 363: Potent β1-adrenoceptor agonist, boosts heart contractility, lowers diastolic pressure.Formula:C19H25NO6Purity:98%Color and Shape:SolidMolecular weight:363.4
