Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,781 products)
- Apoptosis(6,260 products)
- Cell Cycle/Checkpoint(4,792 products)
- Chromatin/Epigenetics(2,440 products)
- Cytoskeletal Signaling(1,527 products)
- DNA Damage/DNA Repair(2,968 products)
- Endocrinology/Hormones(3,706 products)
- Enzyme(3,667 products)
- GPCR/G-Protein(9,005 products)
- Immunology and Inflammation(3,874 products)
- Influenza Virus(301 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,248 products)
- Membrane Transporter/Ion Channel(3,033 products)
- Metabolism(10,207 products)
- Microbiology/Virology(7,591 products)
- Neuroscience(10,382 products)
- Other Inhibitors(36,042 products)
- Oxidation-Reduction(42 products)
- PI3K/Akt/mTOR Signaling(1,444 products)
- Proteases/Proteasome(1,724 products)
- Stem Cell and Derivatives(825 products)
- Tyrosine Kinase/Adaptors(2,035 products)
- Ubiquitination(1,717 products)
Show 16 more subcategories
Found 66686 products of "Inhibitors"
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DDO-02001
CAS:DDO-02001 can be used in anti-arrhythmia research. DDO-02001 is a moderately potent inhibitor of Kv1.5 potassium channel with an IC50 value of 17.7 μM [1].Formula:C20H24N2O2Color and Shape:SolidMolecular weight:324.42Esreboxetine
CAS:Esreboxetine( PNU-165442, (S,S) -reboxetine) is a selective inhibitor of norepinephrine reuptake.Formula:C19H23NO3Color and Shape:SolidMolecular weight:313.39QW30
CAS:QW30 has a significant antitumour effect (IC50: 0.33 μM).Formula:C27H36N2O3Color and Shape:SolidMolecular weight:436.59FRG8701
CAS:FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.Formula:C22H30N2O4SPurity:98%Color and Shape:SolidMolecular weight:418.555,10-Dideazafolic acid
CAS:5,10-Dideazafolic acid is an antileukemic drug.Formula:C21H21N5O6Color and Shape:SolidMolecular weight:439.42L-Eflornithine
CAS:<p>L-Eflornithine: irreversible ODC inhibitor, KD 1.3±0.3 μM, Kinact 0.15±0.03 min-1, enantiomer of Eflornithine.</p>Formula:C6H12F2N2O2Purity:98%Color and Shape:SolidMolecular weight:182.17Nitroscanate
CAS:Nitroscanate is an anthelmintic found to be effective in certain strains of parasites in canines.Formula:C13H8N2O3SColor and Shape:SolidMolecular weight:272.28IACS-8968
CAS:IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and <5 for TDO).Formula:C17H18F3N5O2Purity:98%Color and Shape:SolidMolecular weight:381.35FR 64822
CAS:FR64822, a non-opioid pain reliever, is effective in rodent tests with an ED50 of 1.8 mg/kg orally.Formula:C11H14N4OColor and Shape:SolidMolecular weight:218.26SR 2640 hydrochloride
CAS:SR 2640 hydrochloride is a competitive antagonist of leukotriene D4 and E4 and can be used in studies about leukotrienes in human asthma.Formula:C23H19ClN2O3Purity:98.04%Color and Shape:SolidMolecular weight:406.86JNJ-40068782
CAS:JNJ-40068782 is a potent, selective and systemically active positive allosteric modulator of the mGlu2 receptor.Formula:C21H23N3OPurity:98%Color and Shape:SolidMolecular weight:333.43Lercanidipine. (R)-
CAS:(R)-Lercanidipine enantiomer: antihypertensive, blocks L-type Ca2+ channels, dilates blood vessels.Formula:C36H41N3O6Color and Shape:SolidMolecular weight:611.73CP 59430
CAS:CP 59430 is an azide analogue of prazosin. Prazosin is a highly selective α 1-adrenergic receptor antagonist.Formula:C21H22N8O3Color and Shape:SolidMolecular weight:434.45VU6010572
CAS:VU6010572: potent, selective mGlu3 modulator, IC50 245 nM, high CNS penetration.Formula:C20H18FNO3Color and Shape:SolidMolecular weight:339.36INO-1001 methanesulfonate
CAS:INO-1001 methanesulfonate is a strong PARP inhibitor with chemosensitization and radiosensitization effects.Formula:C24H29N3O7S2Color and Shape:SolidMolecular weight:535.63FGFR3-IN-5
CAS:FGFR3-IN-5: potent, selective FGFR3 inhibitor. IC50: 3 nM FGFR3, 44 nM FGFR2, 289 nM FGFR1. For cancer research.Formula:C24H24FN7O3Color and Shape:SolidMolecular weight:477.49OUN10989
CAS:OUN10989, an analog of LP-261, is a potent antimitotic inhibiting G2/M phase, first reported in J. Med. Chem 2011; no formal name yet.Formula:C19H15N3OColor and Shape:SolidMolecular weight:301.34Tameridone
CAS:Tameridone is a sedative used for cattle.Formula:C22H26N6O2Color and Shape:SolidMolecular weight:406.48Metabolex-36
CAS:Metabolex-36 is a selective GPR120 agonistFormula:C21H19ClF2N2O3Color and Shape:SolidMolecular weight:420.84TACC3 inhibitor 1
Potent TACC3 inhibitor 1 crosses the blood-brain barrier, induces apoptosis, G2/M arrest, ROS, and has anti-tumor effects.Formula:C20H21N5OSColor and Shape:SolidMolecular weight:379.48BuChE-IN-5
CAS:"BuChE-IN-5 is a potent inhibitor with an IC50 of 1.94 μM and shows promise for Alzheimer's research."Formula:C25H35N3Color and Shape:SolidMolecular weight:377.57SN-28049
CAS:SN-28049, a DNA intercalator, targets GC-rich DNA, impedes topo IIalpha/ topo I, and blocks SP-1 transcription, exhibiting anti-tumor effects in mice.Formula:C19H22N4O2Color and Shape:SolidMolecular weight:338.4ROCK-IN-(R)14f
CAS:ROCK-IN-(R)14f is a potent ROCK inhibitor.Formula:C18H18N4O2SColor and Shape:SolidMolecular weight:354.43AChE/Nrf2 modulator 1
CAS:AChE/Nrf2 modulator 1: oral, targets AChE/Nrf2, IC50s: 0.07 μM (eeAChE), 0.38 μM (hAChE); for Alzheimer's research.Formula:C27H27FN4O2Color and Shape:SolidMolecular weight:458.53RS 52367
CAS:RS 52367 is a beta-adrenergic antagonist.Formula:C18H34ClN3O3SColor and Shape:SolidMolecular weight:408Tarlox-TKI
CAS:Tarlox-TKI (Kinase inhibitor-1) is a pan-ErbB inhibitor, the active ingredient of Tarloxotinib, which has antitumor activity.Formula:C19H18BrClN6OPurity:97.03%Color and Shape:SolidMolecular weight:461.74Chinifur
CAS:Chinifur is a selective inhibitor and subversive substrate" for Trypanosoma congolense trypanothione reductase"Formula:C25H30N4O4Color and Shape:SolidMolecular weight:450.53HC102A
CAS:HC102A is an inhibitor of Mycobacterium tuberculosis DosRST signaling and persistence.Formula:C11H18N2O2Color and Shape:SolidMolecular weight:210.27Tubulin inhibitor 30
CAS:Tubulin Inhibitor 30, exhibiting an IC50 value of 0.52 μM, functions as an inhibitor of tubulin assembly. Additionally, it can induce ferroptosis.Formula:C22H19N3O5Color and Shape:SolidMolecular weight:405.4QA 241
CAS:QA 241 is a tricyclic quinolone.Formula:C19H21ClFN3O4Color and Shape:SolidMolecular weight:409.84SIRT2-IN-10
CAS:SIRT2-IN-10 (Compound 12) is a potent inhibitor of SIRT2 (IC50: 1.3 μM), which can be used in the study of cancer and neurodegenerative diseases.Formula:C28H21N5OSColor and Shape:SolidMolecular weight:475.56Polignate Sodium
CAS:Polignate Sodium is an Enzyme Inhibitor (Pepsin)Formula:C20H24Na2O10S2Color and Shape:SolidMolecular weight:534.5EXP-561 monohydrate
CAS:EXP-561 monohydrate is an investigational drug that acts as an inhibitor of the reuptake of serotonin, dopamine, and norepinephrine.Formula:C14H22ClNOColor and Shape:SolidMolecular weight:255.79AS1069562
CAS:AS1069562 inhibits 5-HT/NE reuptake, boosts IGF-1, FGF2 mRNA in dorsal root ganglia, spinal cord.Formula:C20H23NO5SPurity:98%Color and Shape:SolidMolecular weight:389.46GL-1001 disodium tetrahydrate
CAS:GL-1001 disodium tetrahydrate is an ACE2 inhibitor.Formula:C19H29Cl2N3Na2O8Color and Shape:SolidMolecular weight:544.33J-1063
CAS:J-1063 is a potent, selective ALK5 inhibitor with anti-fibrotic properties, useful for liver fibrosis research. (IC50: 0.039 μM).Formula:C24H19N5OSColor and Shape:SolidMolecular weight:425.51Variegatic acid
CAS:Variegatic acid inhibits β-hexosaminidase, TNF-α (IC50: 10.4, 16.8μM), and PKC β1 (IC50: 36.2μM) in RBL 2H3 cells.Formula:C18H12O9Color and Shape:SolidMolecular weight:372.28Acetryptine
CAS:Acetryptine is a biochemical.Formula:C12H14N2OColor and Shape:SolidMolecular weight:202.25Dabuzalgron HCl
CAS:Dabuzalgron, an adrenoceptor agonist, is used potentially for the treatment of urinary incontinence.Formula:C12H17Cl2N3O3SPurity:98%Color and Shape:SolidMolecular weight:354.25Keap1-Nrf2-IN-13
CAS:Keap1-Nrf2-IN-13 is a PPI inhibitor (IC50: 0.15 μM) that binds Keap1 strongly, useful for oxidative stress and inflammation research.Formula:C28H32N2O10S2Color and Shape:SolidMolecular weight:620.69C5aR-IN-2
CAS:C5aR-IN-2, a potent C5aR inhibitor, shows promise for researching inflammatory diseases.Formula:C36H40FN5O2Color and Shape:SolidMolecular weight:593.73Tubulin polymerization-IN-30
CAS:Compound 6e inhibits tubulin polymerization, disrupts microtubules, halts G2/M phase, and targets HeLa, SGC-7901, A549 with low IC50.Formula:C22H25N5O3Color and Shape:SolidMolecular weight:407.47TPN729MA
CAS:TPN729MA, a potent PDE5 inhibitor, IC50: 2.28 nM, targets erectile dysfunction research.Formula:C29H40N6O8SColor and Shape:SolidMolecular weight:632.73Alyssin
CAS:Alyssin: sulforaphane analog, antioxidant; boosts Nrf2 and phase II enzymes in cancer cells; lowers PAH metabolism, reducing cancer risk in vitro.Formula:C7H13NOS2Purity:98%Color and Shape:SolidMolecular weight:191.31Clitocine
CAS:Clitocine, an adenosine analogue derived from mushrooms, is a potent transcriptional transducer, an inhibitor of nonsense mutations, and has anticancer activityFormula:C9H13N5O6Purity:≥95.0%Color and Shape:SolidMolecular weight:287.23Antitubercular agent-14
CAS:Antitubercular agent-14 (Compound 1) shows antitubercular activity. The MIC value of Antitubercular agent-14 against M. tuberculosis is 0.3 μg/mL [1].Formula:C20H27ClN2Color and Shape:SolidMolecular weight:330.89UAWJ9-36-3
CAS:UAWJ9-36-3: Potent SARS-CoV-2 protease inhibitor, broad-spectrum antiviral, IC50=54 nM.Formula:C23H29N3O5Color and Shape:SolidMolecular weight:427.49SCH51048
CAS:SCH 51048 is a broad spectrum antifungal with oral activity.Formula:C37H42F2N8O3Color and Shape:SolidMolecular weight:684.78XR-5000
CAS:XR-5000 is a DNA topoisomerase I and II inhibitor.Formula:C18H19N3OPurity:98%Color and Shape:SolidMolecular weight:293.36NS5818
CAS:NS5818 inhibits ClC.Formula:C23H19Cl2N7O2Purity:98%Color and Shape:SolidMolecular weight:496.35
