Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,781 products)
- Apoptosis(6,260 products)
- Cell Cycle/Checkpoint(4,789 products)
- Chromatin/Epigenetics(2,437 products)
- Cytoskeletal Signaling(1,525 products)
- DNA Damage/DNA Repair(2,967 products)
- Endocrinology/Hormones(3,706 products)
- Enzyme(3,667 products)
- GPCR/G-Protein(9,000 products)
- Immunology and Inflammation(3,869 products)
- Influenza Virus(301 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,249 products)
- Membrane Transporter/Ion Channel(3,029 products)
- Metabolism(10,207 products)
- Microbiology/Virology(7,583 products)
- Neuroscience(10,380 products)
- Other Inhibitors(36,059 products)
- Oxidation-Reduction(43 products)
- PI3K/Akt/mTOR Signaling(1,445 products)
- Proteases/Proteasome(1,725 products)
- Stem Cell and Derivatives(825 products)
- Tyrosine Kinase/Adaptors(2,037 products)
- Ubiquitination(1,716 products)
Show 16 more subcategories
Found 66687 products of "Inhibitors"
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Lubabegron fumarate
CAS:Lubabegron (LY591281, LY488756 fumarate) is a beta-agonist approved in 2018 to lower ammonia in cattle waste, aiding environment and health.Formula:C29H29N3O3SC4H4O4Color and Shape:SolidMolecular weight:557.66COX-2-IN-18
CAS:COX-2-IN-18 is a potent COX-2 inhibitor similar to Celecoxib, showing promise in cancer research. IC50=0.775μM.Formula:C18H19N3O3S2Color and Shape:SolidMolecular weight:389.49SA 2572
CAS:SA 2572 is a newly synthesized Ca2+ antagonist having a inhibitory effect on the fast Na+ inward channel.Formula:C32H41ClN2O6SColor and Shape:SolidMolecular weight:617.2Rho-Kinase-IN-2
CAS:Rho-Kinase-IN-2, an oral ROCK inhibitor (IC50=3nM), penetrates the CNS; potential in Huntington's research.Formula:C20H25FN4O2Color and Shape:SolidMolecular weight:372.44Enpp-1-IN-6
CAS:Enpp-1-IN-6, a potent enpp-1 inhibitor, may aid cancer and infectious disease studies (WO2021203772A1, compound 51).Formula:C22H28N4O5SColor and Shape:SolidMolecular weight:460.55Antileishmanial agent-9
CAS:Compound 16c: potent anti-Leishmania agent, IC50=4.01 μM, low toxicity in L-6 cells, IC50=40.1 μM.Formula:C23H26O4Color and Shape:SolidMolecular weight:366.45Anti-Trypanosoma cruzi agent-4
CAS:Anti-Trypanosoma cruzi Agent-4 is a Trypanosoma cruzi inhibitor utilized for the investigation of infections caused by this parasite.Formula:C17H16N2O3Color and Shape:SolidMolecular weight:296.32FLT3/ITD-IN-3
CAS:FLT3/ITD-IN-3 (Compound 19) is a potent FLT3-ITD inhibitor with IC50 values: FLT3D835Y (0.3 nM), FLT3 (0.4 nM), inhibits AML cell proliferation.Formula:C22H26ClN7O2Color and Shape:SolidMolecular weight:455.94GW2433
CAS:GW2433 is an agonist of PPAR receptor.Formula:C28H28Cl3FN2O4Color and Shape:SolidMolecular weight:581.89URAT1 inhibitor 4
CAS:URAT1 inhibitor 4 is a potent, orally active Lesinurad derivative with a 7.56 μM IC50, showing greater in vivo efficacy.Formula:C27H20BrN3O4S3Color and Shape:SolidMolecular weight:626.56Influenza virus-IN-3
CAS:Influenza virus-IN-3 inhibits H5N1, H5N2, H5N6, H5N8 with low toxicity; targets neuraminidase.Formula:C25H32N2O4SColor and Shape:SolidMolecular weight:456.6NVP018
CAS:<p>NVP018 (BC 556) inhibits HBV, HCV, HIV-1 replication, barely affects drug transporters, and resists HCV/HIV-1 resistance development.</p>Formula:C45H62FN5O11Color and Shape:SolidMolecular weight:868MRGPRX4 modulator-1
CAS:MRGPRX4 modulator-1 (compound 31-2), potent MRGPR X4 antagonist, IC50 < 100nM, for itch, pain, autoimmune research.Formula:C16H13ClF3NO3Color and Shape:SolidMolecular weight:359.73Modimelanotide
CAS:Modimelanotide: melanocortin peptide from α-MSH, developed for acute kidney injury, non-selective receptor agonist.Formula:C113H181N33O25SColor and Shape:SolidMolecular weight:2433.92VS-II-173
CAS:VS-II-173 is a novel potent Pim1 and Pim3 inhibitor, selectively inducing AML cell death.Formula:C14H8N4O2Color and Shape:SolidMolecular weight:264.24Neuroinflammatory-IN-2
CAS:Neuroinflammatory-IN-2: anti-neuroinflammatory, inhibits MAO-B (IC50: 10.30µM), 96.33% Aβ1-42 aggregation reduction, neuroprotective in PC-12 cells.Formula:C25H27FN2O3Color and Shape:SolidMolecular weight:422.49HC103A
CAS:<p>HC103A is an inhibitor of Mycobacterium tuberculosis DosRST signaling and persistence.</p>Formula:C18H14N2O3SColor and Shape:SolidMolecular weight:338.38Nilotinib N-oxide
CAS:Nilotinib N-oxide is a small-molecule tyrosine kinase inhibitor approved for the treatment of imatinib-resistant chronic myelogenous leukemia.Formula:C28H22F3N7O2Color and Shape:SolidMolecular weight:545.52SARS-CoV-2 nsp13-IN-4
CAS:Potent SARS-CoV-2 nsp13-IN-4 selectively inhibits nsp13 helicase with 57 μM IC50, offering antiviral effects.Formula:C20H15BrN4OColor and Shape:SolidMolecular weight:407.26RO-57-Bpyne
CAS:RO-57-Bpyne: a γ-secretase modulator photoaffinity probe that targets presenilin's allosteric sites to lower Aβ pathology.Formula:C32H27N5O4Purity:98%Color and Shape:SolidMolecular weight:545.59HSP90-IN-12
CAS:VAC, a potent anti-cancer vibsanin A analog, inhibits cell proliferation and affects HSP90 protein levels.Formula:C25H36O4Color and Shape:SolidMolecular weight:400.55BPIC
CAS:BPIC is an agent of anti-tumor that acts by inhibiting inflammation and scavenging free radicals.Formula:C27H20N2O5Color and Shape:SolidMolecular weight:452.465-Hexadecyl methotrexate
CAS:5-Hexadecyl methotrexate is a amphipathic analog of methotrexate.Formula:C36H54N8O5Color and Shape:SolidMolecular weight:678.879Rostaporfin
CAS:Rostaporfin, a synthetic photosensitizer, accumulates in tumor cells and produces cytotoxic singlet oxygen upon light exposure.Formula:C37H42Cl2N4O2SnColor and Shape:SolidMolecular weight:764.37RS-30199
CAS:RS-30199 is a 5-HT1A receptor.Formula:C14H18ClNColor and Shape:SolidMolecular weight:235.75V11294A
CAS:V11294A, a PDE4 inhibitor, maintains anti-inflammatory effects for 24h+ with a 300mg dose in humans, sans side effects.Formula:C23H31N5O2Color and Shape:SolidMolecular weight:409.52(R)-FTY720-OMe
CAS:(R)-FTY720-OMe, an FTY720 analogue, selectively inhibits SK2 without affecting SK1.Formula:C20H35NO2Color and Shape:SolidMolecular weight:321.5BChE-IN-15
BChE-IN-15 is a compound characterized as a pseudo-irreversible, covalent inhibitor of butyrylcholinesterase (BChE), demonstrating potent activity with anFormula:C22H33N3O2Color and Shape:SolidMolecular weight:371.52Hydroflumethiazide
CAS:Hydroflumethiazide is a thiazide diuretic. It has also shown the activity of anti-hypertensive.Formula:C8H8F3N3O4S2Color and Shape:Crystals SolidMolecular weight:331.29Org 24461
CAS:Org 24461 is a synaptic and nonsynaptic glycine transporter type-1 inhibitor.Formula:C19H20F3NO3Color and Shape:SolidMolecular weight:367.36PDE5-IN-6c
CAS:<p>PDE5-IN-6c is a potent and selective inhibitor of PDE5A1.</p>Formula:C23H21ClN4O2Purity:98%Color and Shape:SolidMolecular weight:420.89BIIL 260
CAS:BIIL 260 is a leukotriene B4 (BLT1) receptor antagonist with anti-inflammatory activity.Formula:C30H30N2O3Color and Shape:SolidMolecular weight:466.57DW532
CAS:DW532, a simplified hematoxylin analogue, inhibits tyrosine kinases, has anti-cancer effects, disrupts cell division, and suppresses angiogenesis.Formula:C16H12O6Color and Shape:SolidMolecular weight:300.26DM-01
CAS:<p>DM-01 is a potent and selective inhibitor of EZH2.</p>Formula:C23H24F3N3O2Color and Shape:SolidMolecular weight:431.45JMI-105
CAS:JMI-105, a potent antimalarial, inhibits PfFP-2; IC50: 8.8/14.3 μM for CQ S/R strains; reduces murine P. berghei parasitemia, extends survival.Formula:C20H23N3O2Color and Shape:SolidMolecular weight:337.42PIM1-IN-6
CAS:PIM1-IN-6 (5h) inhibits PIM-1 (IC50: 0.60 μM) and is cytotoxic to HCT-116 (IC50: 1.51 μM) and MCF-7 cells (IC50: 15.2 μM).Formula:C21H18N6O4Color and Shape:SolidMolecular weight:418.41Laurinterol
CAS:Laurinterol is an antimicrobial from the marine alga Laurencia okamurai.Formula:C15H19BrOColor and Shape:SolidMolecular weight:295.21TDRL-X80
CAS:TDRL-X80 inhibits XPA DNA binding; effective on single, double, and cisplatin-damaged DNA; IC50: 18-29 μM (FP), 21-39 μM (ELISA).Formula:C23H15ClN2O6Color and Shape:SolidMolecular weight:450.83FabH-IN-1
CAS:FabH-IN-1, a broad-spectrum antibiotic and antioxidant, inhibits bacterial FabH enzyme.Formula:C17H16N2OSColor and Shape:SolidMolecular weight:296.39CG500354
CAS:<p>CG500354 suppresses tumors, induces neural differentiation, and stops growth in human GBM cells via cAMP/CREB pathway.</p>Formula:C20H18F2N2O3SColor and Shape:SolidMolecular weight:404.43DA 3003-2
CAS:DA 3003-2: Potent Cdc25 inhibitor, halts cell division, may aid prostate cancer research.Formula:C15H16ClN3O3Color and Shape:SolidMolecular weight:321.76Perillic acid
CAS:Perillic acid, a perillyl alcohol metabolite, induces lung cancer cell arrest, apoptosis, and has anti-HSV-1 and immune-modulating effects.Formula:C10H14O2Color and Shape:SolidMolecular weight:166.22MDL-72274 HCl
CAS:MDL-72274 HCl is a selective and effective inhibitor of SSAO for the treatment of Parkinson's disease.Formula:C9H11Cl2NColor and Shape:SolidMolecular weight:204.1LUF7346
CAS:LUF7346 is an allosteric modulator of hERG.Formula:C20H15BrN2O3Color and Shape:SolidMolecular weight:411.25MS2126
CAS:MS2126 is a Human p53 and CREB Binding Protein interaction inhibitor.Formula:C12H15NOColor and Shape:SolidMolecular weight:189.25(S)-PI3Kα-IN-4
CAS:(S)-PI3Kα-IN-4 is a potent inhibitor of PI3Kα, with an IC50 of 2.3 nM.Formula:C25H23ClFN5O5SColor and Shape:SolidMolecular weight:560G-573
CAS:G-573, a potent MEK inhibitor, has an IC50 of 0.406µM for pERK and inhibits HCT116/H2122 tumor growth with IC50s of 3.43/2.56µM.Formula:C13H9ClN2Color and Shape:SolidMolecular weight:228.68MK771
CAS:MK771, a TRH analog, potentially eases opiate withdrawal symptoms.Formula:C16H22N6O4SColor and Shape:SolidMolecular weight:394.45Ro 63-0563
CAS:Ro 63-0563 is a potent, 5-HT6 receptors selective antagonist.Formula:C13H17N5O2SPurity:98%Color and Shape:SolidMolecular weight:307.37CXCR3 Antagonist 6c
CAS:CXCR3 antagonist 6c blocks CXCR3 and inhibits Ca2+ movement and T-cell migration (IC50: 0.06 µM & 100 nM) with selectivity over 14 other GPCRs.Formula:C30H32Cl3N5O3Color and Shape:SolidMolecular weight:616.97
