Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,782 products)
- Apoptosis(6,263 products)
- Cell Cycle/Checkpoint(4,792 products)
- Chromatin/Epigenetics(2,441 products)
- Cytoskeletal Signaling(1,528 products)
- DNA Damage/DNA Repair(2,965 products)
- Endocrinology/Hormones(3,707 products)
- Enzyme(3,667 products)
- GPCR/G-Protein(9,009 products)
- Immunology and Inflammation(3,875 products)
- Influenza Virus(301 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,248 products)
- Membrane Transporter/Ion Channel(3,033 products)
- Metabolism(10,209 products)
- Microbiology/Virology(7,592 products)
- Neuroscience(10,381 products)
- Other Inhibitors(36,040 products)
- Oxidation-Reduction(42 products)
- PI3K/Akt/mTOR Signaling(1,442 products)
- Proteases/Proteasome(1,724 products)
- Stem Cell and Derivatives(826 products)
- Tyrosine Kinase/Adaptors(2,035 products)
- Ubiquitination(1,717 products)
Show 16 more subcategories
Found 66683 products of "Inhibitors"
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JTT-552
CAS:JTT-552, a uric acid transporter 1 (URAT1) inhibitor, is used potentially for the treatment of hyperuricemia.Formula:C15H12ClNO3Purity:98%Color and Shape:SolidMolecular weight:289.71Thiochrome
CAS:Thiochrome is a selective enhancer of M4 muscarinic receptor of acetylcholine (ACh) affinity.Formula:C12H14N4OSPurity:98%Color and Shape:SolidMolecular weight:262.33KRAS inhibitor-7
CAS:KRAS inhibitor-7 is a potent KRAS G12C inhibitor.Formula:C26H27ClF2N6O2Purity:98%Color and Shape:SolidMolecular weight:528.98ACDPP hydrochloride
CAS:mGlu5 receptor antagonistFormula:C12H13ClN6OPurity:98%Color and Shape:SolidMolecular weight:292.72PA-9
CAS:PA-9 is the first small-molecule PAC1 receptor antagonist.Formula:C17H18N6O2Purity:98%Color and Shape:SolidMolecular weight:338.36IFN α-IFNAR-IN-1
CAS:Nonpeptidic IFN-α/IFNAR blocker, halts MVA-triggered BM-pDC IFN-α response; IC50: 2-8 μM.Formula:C18H17NSPurity:98%Color and Shape:SolidMolecular weight:279.4Besifloxacin
CAS:Besifloxacin is the fourth generation of fluoroquinolones, which can be used to treat bacterial conjunctivitisFormula:C19H21ClFN3O3Purity:98%Color and Shape:SolidMolecular weight:393.84NSC-658497
CAS:NSC-658497 is a SOS1-Ras interaction inhibitor that acts by dose-dependently inhibiting SOS1 GEF activity.Formula:C20H10N2O6S2Purity:98%Color and Shape:SolidMolecular weight:438.43A-123189
CAS:A-123189 is a potent, alpha1D-selective antagonist.Formula:C26H28N4O3SPurity:98%Color and Shape:SolidMolecular weight:476.59GRL-0820
CAS:GRL-0820 is a SARS-CoV-2 Protease inhibitor (IC50 = 73 nM). GRL-0820 blocked SARS-CoV-2 infection but viral breakthrough occurred.Formula:C17H13ClN2O2Purity:98.27%Color and Shape:SolidMolecular weight:312.75Ref: TM-T69535
1mg99.00€5mg235.00€10mg376.00€25mg747.00€50mg1,121.00€100mg1,768.00€1mL*10mM (DMSO)259.00€K00135
CAS:K00135 (IMIDAZOPYRIDAZIN 1) is a selective inhibitor of Pim kinases and can be used in studies about gastric cancer and antileukemic therapeutics.Formula:C18H18N4OPurity:98.16%Color and Shape:SolidMolecular weight:306.36BI-4924
CAS:BI-4924 is a PHGDH inhibitor that disrupts serine biosynthesis by intracellular trapping and can be used to study metabolic disorders.Formula:C21H20Cl2N2O6SPurity:99.55%Color and Shape:SolidMolecular weight:499.36Tulopafant
CAS:Tulopafant (RP 59227) is a potent platelet-activating factor (PAF) antagonist that increases capillary patency and prolongs allograft heart survival.Formula:C25H19N3O2SPurity:99.38%Color and Shape:SolidMolecular weight:425.5AMG 487 (S-enantiomer)
CAS:AMG 487 S-enantiomer is the S enantiomer of AMG 487. AMG 487 is an CXCR3 antagonist.Formula:C32H28F3N5O4Purity:98%Color and Shape:SolidMolecular weight:603.59TRPC6-IN-1
CAS:TRPC6-IN-1 is an inhibitor of the Transient Receptor Potential Canonical 6 Channel (TRPC6) (EC50: 4.66 μM).Formula:C21H23FN4O3Purity:98%Color and Shape:SolidMolecular weight:398.43NF-κB-IN-11
CAS:NF-κB-IN-11 (Compound 3i) is an inhibitor of NF-κB, effectively blocking TNF-α-induced NF-κB pathway activation and the nuclear translocation of NF-κB.Formula:C19H18O5Purity:98%Color and Shape:SolidMolecular weight:326.345-Methylurapidil
CAS:5-Methylurapidil is an alpha1A-adrenoceptor antagonist.Formula:C21H31N5O3Purity:98%Color and Shape:SolidMolecular weight:401.5RAC 109
CAS:RAC 109 is a chiral antiarrhythmic agent.Formula:C20H28N2O2Purity:98%Color and Shape:SolidMolecular weight:328.45Sp-Cyclic AMPS (sodium salt)
CAS:Sp-cAMPS Na salt activates PKA I/II and competitively inhibits PDE3A (Ki: 47.6 μM), also binds PDE10 GAF (EC50: 40 μM).Formula:C10H12N5NaO5PSColor and Shape:SolidMolecular weight:367.25VPC 23019
CAS:<p>VPC 23019 is a competitive antagonist at the S1P1 and S1P3 receptors (pKi= 7.86 and 5.93, respectively).</p>Formula:C17H29N2O5PPurity:98%Color and Shape:SolidMolecular weight:372.4Retaspimycin
CAS:Retaspimycin is a potent and water-soluble Hsp90 inhibitor(EC50s of 119 nM for both Hsp90 and Grp9).Formula:C31H45N3O8Purity:98%Color and Shape:SolidMolecular weight:587.7Seviteronel R enantiomer
CAS:Seviteronel R enantiomer (VT-464 R enantiomer) is a Seviteronel isomer produced during the manufacturing process.Formula:C18H17F4N3O3Purity:97.97% - >99.99%Color and Shape:SolidMolecular weight:399.34Ref: TM-T13312
1mg111.00€5mg259.00€10mg378.00€25mg643.00€50mg914.00€100mg1,216.00€1mL*10mM (DMSO)283.00€MI-192
CAS:MI-192: Selective HDAC2/3 inhibitor, IC50=30/16 nM, induces apoptosis in myeloid leukemia, potential in leukemia/anti-stroke treatment.Formula:C24H21N3O2Color and Shape:SolidMolecular weight:383.442-PMDQ
CAS:2-PMDQ is an α1-adrenoceptor antagonist.Formula:C21H23N5OPurity:98%Color and Shape:SolidMolecular weight:361.44SNT-207858
CAS:SNT-207858: selective, BBB-penetrating, oral MC-4 receptor antagonist with 22 nM IC50 (binding), 11 nM (function).Formula:C32H45Cl4N5O3Purity:98%Color and Shape:SolidMolecular weight:689.54DA 5018
CAS:DA 5018 is a capsaicin derivative and is also a new non-narcotic analgesic. It has an antipruritic effect.Formula:C22H31ClN2O3Purity:98%Color and Shape:SolidMolecular weight:406.95Lascufloxacin
CAS:Lascufloxacin: potent, oral fluoroquinolone antibiotic for respiratory infections, effective against quinolone-resistant strains.Formula:C21H24F3N3O4Purity:98%Color and Shape:SolidMolecular weight:439.43TTT-28
CAS:TTT-28, a thiazole-valine peptidomimetic, selectively inhibits ABCB1 to reverse MDR with low toxicity.Formula:C31H31N3O6SPurity:98%Color and Shape:SolidMolecular weight:573.66Razaxaban hydrochloride
CAS:Razaxaban hydrochloride is a highly potent, selective and orally active inhibitor of factor Xa(Ki of 0.19 nM),has strongly antithrombotic activity.Formula:C24H21ClF4N8O2Purity:98%Color and Shape:SolidMolecular weight:564.92LUF 6283
CAS:partial agonist of hydroxycarboxylic acid receptor 2 (HCA2)Formula:C8H12N2O2Color and Shape:SolidMolecular weight:168.19Ebselen oxide
CAS:Ebselen oxide (EB-2) is a HER2 inhibitor with antibacterial and antifungal activity and has shown cytoprotective effects against HN2 in vitro.Formula:C13H9NO2SePurity:98%Color and Shape:SolidMolecular weight:290.18Azelastine
CAS:<p>Azelastine (Azelastinum) is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.</p>Formula:C22H24ClN3OPurity:99.35%Color and Shape:White Crystal PowderMolecular weight:381.90BMS270394
CAS:BMS270394 is a RARγ agonist used in the study of breast cancer and skin diseases.Formula:C23H26FNO4Color and Shape:SolidMolecular weight:399.46VU0410425
CAS:VU0410425 is a metabotropic glutamate receptor subtype 1 negative allosteric modulator.Formula:C19H16ClN3O3Purity:98%Color and Shape:SolidMolecular weight:369.84-Acetylsimvastatin
CAS:4-Acetylsimvastatin is acetylated simvastatin. Simvastatin is a competitive inhibitor of HMG-CoA reductase (Ki: 0.2 nM).Formula:C27H40O6Purity:98%Color and Shape:SolidMolecular weight:460.6AGI-41998
CAS:<p>AGI-41998: a potent MAT2A inhibitor that crosses the blood-brain barrier, targeting SAM enzymes for cancer therapy and CNS research.</p>Formula:C22H16BrF3N4O2Color and Shape:SolidMolecular weight:505.29L 368935
CAS:L 368935 is an antagonist of the cholecystokinin receptor.Formula:C27H26N8O2Purity:98%Color and Shape:SolidMolecular weight:494.55Nevanimibe
CAS:Nevanimibe is an orally active and selective inhibitor of acyl-coenzyme A:cholesterol O-acyltransferase 1 (ACAT1) (EC50 of 9 nM).Formula:C27H39N3OPurity:98%Color and Shape:SolidMolecular weight:421.62N20C hydrochloride
CAS:N20C hydrochloride (2-((3,3-diphenylpropyl)amino)acetamide hydrochloride) is a non-competitive NMDA receptor open-channel blocker.Formula:C17H21ClN2OPurity:99.9%Color and Shape:SolidMolecular weight:304.81Plantainoside C
CAS:Plantainoside C is a useful organic compound for research related to life sciences. The catalog number is T125990 and the CAS number is 136083-86-8.Formula:C30H38O15Color and Shape:SolidMolecular weight:638.619TH-Z835
CAS:TH-Z835 is a selective inhibitor for the KRAS (G12D) mutation, demonstrating an inhibitory concentration (IC50) of 1.6 μM.Formula:C30H38N6OPurity:98%Color and Shape:SolidMolecular weight:498.66Lubeluzole
CAS:Lubeluzole, a well-known neuroprotective agent, is recently proved useful to potentiate the activity of anti-cancer drugs.Formula:C22H25F2N3O2SPurity:98%Color and Shape:SolidMolecular weight:433.51IHVR-19029
CAS:IHVR-19029: ER α-glucosidases I/II inhibitor, IC50 0.48μM; halts Ebola, Dengue, Rift Valley fever virus replication.Formula:C23H45N3O5Color and Shape:SolidMolecular weight:443.62Rolapitant
CAS:Rolapitant Hydrochloride is an oral NK1-receptor blocker that prevents nausea and has a fast onset and long half-life.Formula:C25H26F6N2O2Purity:99.86%Color and Shape:SolidMolecular weight:500.48Ref: TM-T3716
1mg50.00€2mg66.00€5mg93.00€10mg124.00€25mg188.00€50mg311.00€100mg465.00€500mg1,035.00€1mL*10mM (DMSO)92.00€WS-383 free base
CAS:WS-383 free base is a selective and reversible DCN1-UBC12 interaction inhibitor(IC50 of 11 nM).Formula:C18H20ClN9S2Purity:98%Color and Shape:SolidMolecular weight:461.99NBC 6
CAS:NLRP3-IN-NBC6: potent NLRP3 inflammasome inhibitor, IC50 574 nM, Ca2+ independent, inhibits inflammasome in THP-1 cells/BMDMs.Formula:C18H16BCl3N2O2Color and Shape:SolidMolecular weight:409.5TWIK-1/TREK-1-IN-2
CAS:TWIK-1/TREK-1-IN-2 (Compound 2g) serves as an inhibitor of both TWIK-1 and TREK-1, targeting the TREK-1 homodimer and TWIK-1/TREK-1 heterodimer with IC50 valuesFormula:C20H29F3N2O2Purity:98%Color and Shape:SolidMolecular weight:386.45Galidesivir triphosphate
CAS:Galidesivir triphosphate halts viral RNA replication by inhibiting RDRP and NS5B, and combats Ebola in mice; derived from prodrug Galidesivir.Formula:C11H18N5O12P3Purity:98%Color and Shape:SolidMolecular weight:505.21Beaucage reagent
CAS:Beaucage reagent, which is found to be effective in causing DNA cleavage.Formula:C7H4O3S2Purity:98.50%Color and Shape:White To Off-White PowderMolecular weight:200.23ICI 162,846
CAS:ICI 162,846 is an orally active and potent H2 receptor antagonist that inhibits gastric secretion and may be used in the study of duodenal ulcers.Formula:C11H17F3N6OPurity:97.45%Color and Shape:SolidMolecular weight:306.29
