Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,853 products)
- Apoptosis(6,368 products)
- Cell Cycle/Checkpoint(4,909 products)
- Chromatin/Epigenetics(2,633 products)
- Cytoskeletal Signaling(1,587 products)
- DNA Damage/DNA Repair(2,868 products)
- Endocrinology/Hormones(3,765 products)
- Enzyme(3,673 products)
- GPCR/G-Protein(9,054 products)
- Immunology and Inflammation(3,952 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(417 products)
- MAPK Signaling(1,259 products)
- Membrane Transporter/Ion Channel(3,163 products)
- Metabolism(10,156 products)
- Microbiology/Virology(7,674 products)
- Neuroscience(10,550 products)
- Other Inhibitors(35,855 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,437 products)
- Proteases/Proteasome(1,692 products)
- Stem Cell and Derivatives(733 products)
- Tyrosine Kinase/Adaptors(1,992 products)
- Ubiquitination(1,744 products)
Show 16 more subcategories
Found 66513 products of "Inhibitors"
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Totrombopag choline
CAS:Eltrombopag (LGD-4665, GSK2285921, SB559448) is an oral TPO receptor agonist for thrombocytopenia treatment.Formula:C30H35N9O3Color and Shape:SolidMolecular weight:569.67SDH-IN-3
CAS:SDH-IN-3 is a succinate dehydrogenase (SDH) inhibitor, demonstrating potent antifungal activity with an inhibition concentration (IC50) of 7.2 μg/mL and anFormula:C15H11F2N3OSPurity:98%Color and Shape:SolidMolecular weight:319.33Amb123203
CAS:Amb123203 is an inhibitor of the budding of mVP40 and eVP40 VLPs that acts by blocking mVP40-795 Nedd4 protein-protein interaction.Formula:C25H27N5OSColor and Shape:SolidMolecular weight:445.58PK68
CAS:PK68 selectively inhibits RIPK1 (IC50=90nM), potentially useful in inflammation and cancer metastasis studies.Formula:C22H24N4O3SPurity:98.09% - 99.64%Color and Shape:SolidMolecular weight:424.52Ref: TM-T12493
1mg77.00€5mg166.00€1mL*10mM (DMSO)178.00€10mg260.00€25mg492.00€50mg708.00€100mg888.00€AChE-IN-19
CAS:AChE-IN-19: strong AChE blocker (IC50: 0.56 μM), hinders Aβ clumps, neuro-protective, non-toxic to SH-SY5Y, for Alzheimer's research.Formula:C30H33NO7Color and Shape:SolidMolecular weight:519.59ABT-255
CAS:ABT-255: novel 2-pyridone antimicrobial for tuberculosis, effective against drug-sensitive/resistant Mycobacterium tuberculosis in vitro/in vivo.
Formula:C21H24FN3O3Color and Shape:SolidMolecular weight:385.43RXFP1 receptor agonist-6
CAS:RXFP1 receptor agonist-6 (Example 7) serves as an agonist for the RXFP1 receptor and effectively suppresses cAMP production in HEK293 cells that stably expressFormula:C38H32F5N3O7Color and Shape:SolidMolecular weight:737.67D-Ala-Lys-AMCA
CAS:D-Ala-Lys-AMCA, a PEPT1 substrate, transports into Caco-2/liver cancer cells with blue fluorescence.Formula:C21H28N4O6Purity:98%Color and Shape:SolidMolecular weight:432.47Tyrphostin AG1433
CAS:Tyrphostin AG1433 (AG1433) is an inhibitor of tyrosine kinases and also a dual inhibitor of PDGFRβ(IC50s = 5.0 μM) and VEGFR-2 (Flk-1/KDR)(IC50s = 9.3 μM).Formula:C16H14N2O2Purity:98.47%Color and Shape:SolidMolecular weight:266.29TMC-649128
CAS:TMC-649128, a RNA polymerase NS5B inhibitor, is used for the treatment of HCV infection.Formula:C18H26N6O6Color and Shape:SolidMolecular weight:422.44ROCK-IN-9
CAS:ROCK-IN-9 (Compound T345), a ROCK inhibitor, exhibits cytotoxicity in HepG2 cells with an IC50 of 40.8 μM.Formula:C20H20FN5O2Purity:98%Color and Shape:SolidMolecular weight:381.4PF-4778574
CAS:PF-4778574 is a positive AMPA receptor allosteric modulation (EC50: 45 to 919 nM in different cells).Formula:C19H22N2O3S2Purity:98%Color and Shape:SolidMolecular weight:390.52EGFR/CSC-IN-1
CAS:EGFR/CSC-IN-1 is a dual inhibitor targeting both the epidermal growth factor receptor (EGFR [IC50 10.52 nM]) and cancer stem cells (CSC), with potentialFormula:C54H54Cl2FN7O7S2Purity:98%Color and Shape:SolidMolecular weight:1067.08JNJ-28583867
CAS:JNJ-28583867 is an inhibitor of histamine H(3) receptor antagonist and serotonin reuptake.Formula:C24H32N2O2SColor and Shape:SolidMolecular weight:412.59NAS-181
CAS:NAS-181 is a potent and selective rat 5-hydroxytryptamine 1B (r5-HT1B) antagonist (Ki: 47 nM).NAS-181 enhances the accumulation of 5-HTP in rat brain regions.Formula:C20H30N2O7SColor and Shape:SolidMolecular weight:442.53Pentiapine
CAS:Pentiapine (CGS 10746) is a novel inhibitor of dopamine release.Formula:C15H17N5SPurity:99.35%Color and Shape:SolidMolecular weight:299.39Ref: TM-T12405
1mg487.00€5mg753.00€1mL*10mM (DMSO)938.00€10mg1,216.00€25mg1,691.00€50mg2,262.00€100mg3,068.00€CV1808
CAS:CV-1808 is a coronary vasodilator, antihypertensive, and antipsychotic following systemic administration in vivo. CV-1808 is an adenosine A2 receptor agonist.Formula:C16H18N6O4Color and Shape:Off-White To Pale Yellow SolidMolecular weight:358.35Cerivastatin
CAS:Cerivastatin is an HMG-CoA reductase inhibitor with anticancer and lipid-lowering effects and can be used to study primary hyperlipidemia.Formula:C26H34FNO5Purity:97.80% - 99.56%Color and Shape:SolidMolecular weight:459.55ICMT-IN-37
CAS:ICMT-IN-37 (compound 41) serves as an inhibitor of ICMT with an IC50 value of 0.308 μM [1].Formula:C22H28ClNOColor and Shape:SolidMolecular weight:357.92ONO 4817
CAS:ONO-4817 suppresses MMPs, limiting plaque progression and aortic hyperplasia in hyperlipidemic rabbits.Formula:C22H28N2O6Color and Shape:SolidMolecular weight:416.47TA-1887
CAS:TA-1887: Selective SGLT2 inhibitor, treats type 2 diabetes, lowers glucose in high-fat diet mice, boosts UGE, has good pharmacokinetics.Formula:C24H26FNO5Color and Shape:SolidMolecular weight:427.47GT-2394
CAS:GT-2394 is a histamine H3 receptor agonist.Formula:C14H21N3O2Color and Shape:SolidMolecular weight:263.34Amebucort
CAS:Amebucort is a synthetic glucocorticoid corticosteroid. It may used for the research of inflammatory disorders.Formula:C28H40O7Purity:98%Color and Shape:SolidMolecular weight:488.61YM49598
CAS:YM49598 is a tachykinin receptor antagonist with high affinity for NK(1) and NK(2). It inhibits rat bladder contraction induced by NK(1) agonists.Formula:C36H45Cl2N2O2Purity:98%Color and Shape:SolidMolecular weight:608.66IIIM-8
CAS:IIIM-8 is a melanogenesis inhibitor that suppresses pigment production in both in vitro and in vivo settings, exhibiting no cytotoxic effects on Human AdultFormula:C14H17NO4Purity:98%Color and Shape:SolidMolecular weight:263.29RSV L-protein-IN-4
CAS:RSV L-protein-IN-4 (Compound C) is a noncompetitive inhibitor of the RSV polymerase with an IC50 of 0.88 μM.Formula:C32H35N5O6Purity:98%Color and Shape:SolidMolecular weight:585.65MP7
CAS:MP7 (PDK1 inhibitor) is a inhibitor of phosphoinositide-dependent kinase-1 (PDK1).Formula:C28H22F2N4O4Purity:99.89%Color and Shape:SolidMolecular weight:516.5AY 31906
CAS:AY 31906: High ceiling diuretic, boosts sodium/chloride excretion without affecting potassium, GFR, or renal flow in dogs.Formula:C15H24N6O3SColor and Shape:SolidMolecular weight:368.45FEN1-IN-5
CAS:FEN1-IN-5 (compound 12A) is a potent Flap endonuclease-1 (FEN1) inhibitor with an IC50 value of 12 nM, playing a role in DNA repair mechanisms [1].Formula:C21H17N3O4SPurity:98%Color and Shape:SolidMolecular weight:407.44Adaprolol
CAS:Adaprolol is a beta-adrenergic antagonist. Enantiomers of Adaprolol may be used in the treatment of Glaucoma or other ailments of the eye.Formula:C26H39NO4Color and Shape:SolidMolecular weight:429.59Cyclopentenyl uracil
CAS:Cyclopentenyl uracil 是一种无细胞毒性的尿苷激酶 (uridine kinase) 抑制剂，可有效阻断完整小鼠体内宿主和肿瘤组织对循环尿苷的回收。Formula:C10H12N2O5Color and Shape:SolidMolecular weight:240.21Proteasome-IN-4
Proteasome-IN-4, a potent non-covalent inhibitor (IC50=8.39nM), halts cancer cell growth, useful for oncology studies.Formula:C44H58N6O5Color and Shape:SolidMolecular weight:750.97AChE-IN-44
CAS:AChE-IN-44 (Compound Tap4), an AChE inhibitor, is convertible into its thiazole salt form known as Tat2 [1].Formula:C31H38ClN3OS2Color and Shape:SolidMolecular weight:568.24KRAS G12C mutant protein inhibitor A-1
CAS:KRAS G12C mutant protein inhibitor A-1 can be used in studies about Ras.Formula:C31H26ClF4N7O2Color and Shape:SolidMolecular weight:640.03RORγt inverse agonist 14
CAS:RORγt inverse agonist 14 (8e) is a potent, selective, and orally active compound with an EC50 of 2.5 nM, exhibiting anti-inflammatory activity.Formula:C26H26F8N2O6S2Purity:98%Color and Shape:SolidMolecular weight:678.61PD-1/PD-L1-IN-27
CAS:PD-1/PD-L1-IN-27: potent anti-cancer, IC50 134nM, minimal T cell harm, boosts CD8+ T cells, reduces fatigue.Formula:C44H35NO6Purity:98%Color and Shape:SolidMolecular weight:673.75Pazelliptine
CAS:Pazelliptine is a DNA topoisomerase inhibitor and antitumor drug.Formula:C22H27N5Color and Shape:SolidMolecular weight:361.48RASP-IN-1
CAS:RASP-IN-1 (Compound A), a lipophilic compound, serves as an inhibitor for macular degeneration and exhibits biological activity within the rabbit retina.Formula:C16H16N2O2Color and Shape:SolidMolecular weight:268.31NVS-SM2
CAS:NVS-SM2 boosts SMN2 splicing, enhances exon 7 inclusion, and raises SMN protein levels orally.Formula:C23H30N6OColor and Shape:SolidMolecular weight:406.52ZINC03129319
CAS:ZINC03129319 is an inhibitor of dengue virus (DENV) NS2B-NS3 protease.Formula:C24H14N2O6S2Purity:90%Color and Shape:SolidMolecular weight:490.51TRβ agonist 3
CAS:TRβ agonist 3 (Compound 3) is a potent TRβ agonist that is a new potential TRβ-selective thyromimetics.Formula:C20H25NO3Color and Shape:SolidMolecular weight:327.42AGN 194310
CAS:AGN 194310 (VTP-194310) is retinioic acid receptors (RARs) pan-antagonist. The Kd values of 3 nM, 2 nM, 5 nM for RARα, RARβ, RARγ, respectively[1][2].Formula:C28H24O2SColor and Shape:SolidMolecular weight:424.55CP-24879 hydrochloride
CAS:CP-24879 HCl, a Δ5D/Δ6D dual-inhibitor, reduces liver lipid buildup and inflammation.
Formula:C11H18ClNOPurity:98.08%Color and Shape:SolidMolecular weight:215.72TMV-IN-3
CAS:TMV-IN-3 is a chalcone derivative that inhibits TMV with a 120.3 μg/mL EC50, used in research on infection and cancer.Formula:C28H26O4Color and Shape:SolidMolecular weight:426.5Fosfluridine tidoxil
CAS:Fosfluridine tidoxil, a thymidylate synthase inhibitor, is used potentially for the treatment of colorectal cancer, and breast cancer.Formula:C34H62FN2O10PSColor and Shape:SolidMolecular weight:740.9KRAS G12C inhibitor 59
CAS:KRAS G12C Inhibitor 59 is a compound with anticancer properties.Formula:C32H39F6N7O5Purity:98%Color and Shape:SolidMolecular weight:715.69Antitumor agent-114
CAS:Antitumor Agent-114, a potent STING (stimulator of interferon genes) agonist, activates immune responses and diminishes tumor size in mouse breast cancer modelsFormula:C39H50F2N10O13P2Purity:98%Color and Shape:SolidMolecular weight:966.82RR-RJW100
RR-RJW100: potent LRH-1 & SF-1 agonist; studies metabolic disorders, diabetes, liver disease, IBD.Formula:C28H34OColor and Shape:SolidMolecular weight:386.57MDL-19744A
CAS:MDL-19744A is an alpha 1-adrenergic receptor antagonist and renal vasodilator.Formula:C21H25NO3SColor and Shape:SolidMolecular weight:371.49SREBP/SCAP-IN-2
CAS:SREBP/SCAP-IN-2 (compound 13) acts as a selective inhibitor of SREBP/SCAP [1].Formula:C27H37ClF2N4OColor and Shape:SolidMolecular weight:507.06
