Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,849 products)
- Apoptosis(6,366 products)
- Cell Cycle/Checkpoint(4,907 products)
- Chromatin/Epigenetics(2,623 products)
- Cytoskeletal Signaling(1,585 products)
- DNA Damage/DNA Repair(2,872 products)
- Endocrinology/Hormones(3,759 products)
- Enzyme(3,673 products)
- GPCR/G-Protein(9,051 products)
- Immunology and Inflammation(3,945 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(417 products)
- MAPK Signaling(1,259 products)
- Membrane Transporter/Ion Channel(3,162 products)
- Metabolism(10,149 products)
- Microbiology/Virology(7,672 products)
- Neuroscience(10,549 products)
- Other Inhibitors(35,857 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,435 products)
- Proteases/Proteasome(1,693 products)
- Stem Cell and Derivatives(734 products)
- Tyrosine Kinase/Adaptors(1,991 products)
- Ubiquitination(1,743 products)
Show 16 more subcategories
Found 66517 products of "Inhibitors"
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FM26
CAS:FM26, an isoxazole-based RORγt inverse agonist, cuts EL4 IL-17a mRNA; potent with 264 nM IC50.Formula:C22H15ClF3N3O3Purity:98%Color and Shape:SolidMolecular weight:461.82CBP-IN-1
CAS:CBP-IN-1 (compound 12) acts as a potent CBP inhibitor exhibiting an IC50 of 1.5 nM and additionally suppresses CBP BRET and BRD4(1) with IC50 values of 690 nMFormula:C27H33F2N7OPurity:98%Color and Shape:SolidMolecular weight:509.59Siramesine Fumarate
CAS:Siramesine Fumarate, a sigma receptor agonist, is used potentially for the treatment of generalized anxiety disorder.Formula:C34H35FN2O5Purity:98%Color and Shape:SolidMolecular weight:570.65KD-026
CAS:KD-026 (SLx 4090), a microsomal triglyceride transfer protein (MTP) inhibitor(IC50 = 8.0 nM), is used in type 2 diabetes studies.Formula:C31H25F3N2O4Purity:99.74%Color and Shape:SolidMolecular weight:546.54Ref: TM-T27719
1mg81.00€2mg104.00€5mg170.00€1mL*10mM (DMSO)210.00€10mg259.00€25mg444.00€50mg562.00€100mg775.00€200mg1,026.00€(R)-tert-OMe-byakangelicin
CAS:(R)-tert-OMe-byakangelicin, a furanocoumarin, exhibits inhibitory effects on liver drug metabolizing enzyme (DME) activity and can be isolated from the immatureFormula:C18H20O7Purity:98%Color and Shape:SolidMolecular weight:348.35KNI 174
CAS:KNI 174 is a new type of anti‐AIDS drug used as an HIV‐1 protease inhibitorFormula:C36H45N5O7SColor and Shape:SolidMolecular weight:691.84MMV009085
CAS:MMV009085 is a potent inhibitor of the Plasmodium falciparum hexose transporter (Pf HT1), with potential as an anti-malarial agent.Formula:C22H22N2O6Color and Shape:SolidMolecular weight:410.42DosatiLink-2
CAS:DosatiLink-2 is an inhibitor of the Abelson murine leukemia (ABL) enzyme [1].Formula:C65H85Cl2F2N13O15SColor and Shape:SolidMolecular weight:1429.42Anticancer agent 93
CAS:Anticancer Agent 93, a 4-Hydroxycoumarin derivative, inhibits the invasion and migration of lung cancer cells through modulation of epithelial-mesenchymalFormula:C16H10ClNO4Color and Shape:SolidMolecular weight:315.71Butriptyline
CAS:Butriptyline (Butriptylene), a tricyclic antidepressant, is effective when administered orally [1].Formula:C21H27NColor and Shape:SolidMolecular weight:293.45ICMT-IN-37
CAS:ICMT-IN-37 (compound 41) serves as an inhibitor of ICMT with an IC50 value of 0.308 μM [1].Formula:C22H28ClNOColor and Shape:SolidMolecular weight:357.92E6130
CAS:E6130 may be effective in the treatment of inflammatory bowel disease and is a highly selective CX3CR1 regulator for oral administration.Formula:C28H37ClF3N3O3Color and Shape:SolidMolecular weight:556.06SB-649701
CAS:SB-649701 is a potent antagonist of the human CCR8 receptor, exhibiting a pIC50 value of 7.7, and is utilized in asthma research [1].Formula:C27H28N4O3Purity:98%Color and Shape:SolidMolecular weight:456.54USP1-IN-3
CAS:USP1-IN-3 is a selective inhibitor of USPI that inhibits USPI-UAFI (IC50<30 nM). USP1-IN-3 can be used to study cancer.Formula:C27H24F3N7OColor and Shape:SolidMolecular weight:519.52KB-R7785
CAS:KB-R7785 is a novel ADAM12/MMP inhibitor improving heart function and insulin sensitivity by blocking HB-EGF and TNF-alpha.Formula:C18H27N3O4Color and Shape:SolidMolecular weight:349.42iso-TRAP-6
CAS:iso-TRAP-6 (iso-SFLLRN), a hexapeptide made from isoserine instead of serine, is a PAR1 agonist that activates platelets via PAR-1.Formula:C34H56N10O9Purity:98.55%Color and Shape:SolidMolecular weight:748.87Flurofamide
CAS:Flurofamide is an effective bacterial urease inhibitor and has potential in the treatment of infected urinary calculi.Formula:C7H9FN3O2PPurity:96.01% - 98%Color and Shape:SolidMolecular weight:217.14DC_AC50
CAS:"DC_AC50 inhibits Atox1/CCS to reduce cancer cell growth and prevent chemotherapy resistance."Formula:C17H12BrF2N3OSPurity:99.84% - 99.9%Color and Shape:SolidMolecular weight:424.26LY 106737
CAS:LY 106737 is opioid antagonist in the class of phenylpiperidine.Formula:C21H27NOPurity:98%Color and Shape:SolidMolecular weight:309.45Omiloxetine
CAS:Omiloxetine, an SSRI developed by Ferrer Internacional, was shelved in 2005 after preclinical trials.Formula:C27H25F2NO4Color and Shape:SolidMolecular weight:465.49TG2-179-1
CAS:Nalmefene (ORF 11676) is a μ-opioid antagonist and partial κ agonist used to study opioid overdose and alcohol dependence.Formula:C22H14ClFN4O2S2Color and Shape:SolidMolecular weight:484.95L-Allooctopine
CAS:L-Allooctopine competitively inhibits D-octopine [1].Formula:C9H18N4O4Color and Shape:SolidMolecular weight:246.26HBF-0259
CAS:HBF-0259 is an inhibitors of hepatitis B virus surface antigen (HBsAg) secretion with an EC50 of 11.3 μM and a CC50 value of >50 μM in HepG2.2.15 cells.Formula:C16H12Cl2FN5Purity:98.07% - 99.42%Color and Shape:SolidMolecular weight:364.2Ref: TM-T27527
2mg34.00€5mg49.00€1mL*10mM (DMSO)50.00€10mg71.00€25mg114.00€50mg172.00€100mg249.00€200mg349.00€CCT241533
CAS:CCT241533 is an effective and selective ATP competitive inhibitor of CHK2 (Ki: 1.16 nM; IC50: 3 nM).Formula:C23H27FN4O4Purity:98%Color and Shape:SolidMolecular weight:442.48VU0364739
CAS:VU0364739, a selective phospholipase D2 (PLD2) inhibitor with an IC50 of 22 nM, effectively reduces cancer cell proliferation [1].Formula:C26H27FN4O2Purity:98%Color and Shape:SolidMolecular weight:446.52PAN12314
CAS:PAN12314 (Compound 5a) is a 5-HT4R partial agonist with cognition-enhancing effects in animals, lacking a formal name.Formula:C21H30N4O2Color and Shape:SolidMolecular weight:370.49MCC
CAS:MCC, a non-cleavable linker utilized in the production of antibody-drug conjugates (ADCs), is exemplified by MCC-DM1 [1].Formula:C12H16N2O3Color and Shape:SolidMolecular weight:236.27δ-Tocotrienol
CAS:δ-Tocotrienol (Delta-Tocotrienol) is a potential angiogenic inhibitor.Formula:C27H40O2Purity:99.86%Color and Shape:SolidMolecular weight:396.61Ref: TM-TMA2474
1mg46.00€5mg92.00€1mL*10mM (DMSO)101.00€10mg145.00€25mg281.00€50mg423.00€100mg625.00€RXFP1 receptor agonist-1
CAS:RXFP1 receptor agonist-1 (Example 2), an agonist of the RXFP1 receptor, suppresses cAMP production in HEK293 cells that constitutively express the human RXFP1,Formula:C31H29F7N2O4Color and Shape:SolidMolecular weight:626.56Zoxamide
CAS:Zoxamide (RH-7281) is an oomycete-specific fungicide that impedes nuclear division in Phytophthora capsici germlings and disrupts the microtubule cytoskeleton [Formula:C14H16Cl3NO2Color and Shape:SolidMolecular weight:336.64Lithium citrate
CAS:Lithium citrate decreases elevated intracerebral N-acetyl aspartate levels in Canavan disease [1].Formula:C6H5Li3O7Color and Shape:SolidMolecular weight:209.92Quizalofop-P
CAS:Quizalofop-P, a selective herbicide, is absorbed by weed stems and leaves before translocating both upward and downward within the plant, concentrating inFormula:C17H13ClN2O4Purity:98%Color and Shape:SolidMolecular weight:344.75Myristoyl tetrapeptide-12
CAS:Myristoyl Tetrapeptide-12 activates SMAD2 and facilitates the association of SMAD3 with DNA, promoting eyelash hair growth [1] [2].Formula:C32H63N7O5Purity:98%Color and Shape:SolidMolecular weight:625.89Pentiapine
CAS:Pentiapine (CGS 10746) is a novel inhibitor of dopamine release.Formula:C15H17N5SPurity:99.35%Color and Shape:SolidMolecular weight:299.39Ref: TM-T12405
1mg487.00€5mg753.00€1mL*10mM (DMSO)938.00€10mg1,216.00€25mg1,691.00€50mg2,262.00€100mg3,068.00€Osivelotor
CAS:Osivelotor is an allosteric modulator of hemoglobin S (HbS) [1].Formula:C20H22N2O6Purity:98%Color and Shape:SolidMolecular weight:386.4Laxifloran
CAS:Laxifloran possesses antibacterial and antifungal properties.Formula:C17H18O5Color and Shape:SolidMolecular weight:302.32Dim16
CAS:Dim16, a dual inhibitor of PCSK9/HMG-CoAR, demonstrates potent activity with an IC50 of 19 nM against PCSK9 and significantly impedes PCSK9-LDLR interactionFormula:C29H38IN5Color and Shape:SolidMolecular weight:583.5520-HETE inhibitor-1
CAS:20-HETE Inhibitor-1 (Comp 83) serves as an inhibitor of 20-HETE formation [1].Formula:C19H24N4OColor and Shape:SolidMolecular weight:324.42AAK1-IN-2
CAS:AAK1-IN-2, a potent (IC50=5.8 nM) AAK1 inhibitor, selective & brain-penetrant, is used for neuropathic pain studies.Formula:C20H20N4Color and Shape:SolidMolecular weight:316.4DI-591
CAS:DI-591: High-affinity DCN1-UBC12 inhibitor; permeates cells; Ki: DCN1 - 12 nM, DCN2 - 10.4 nM; doesn't bind DCN3-5.Formula:C31H47N5O4SColor and Shape:SolidMolecular weight:585.8L-Biotin
CAS:L-Biotin, or simply biotin, is a water-soluble vitamin crucial for carboxylation reactions in various enzymes.Formula:C10H16N2O3SColor and Shape:SolidMolecular weight:244.31WT IDH1 Inhibitor 2
CAS:WT IDH1 Inhibitor 2 blocks wild-type and R132H mutant IDH1 (IC50: 120 nM); related to GSK321.Formula:C28H28FN5O3Color and Shape:SolidMolecular weight:501.55M190S
CAS:M109S is a novel small molecule that shields cells from mitochondria-dependent apoptosis, demonstrating effectiveness both in vitro and in vivo.Formula:C21H21N5O2Purity:98%Color and Shape:SolidMolecular weight:375.42N-type calcium channel blocker-1
CAS:N-type calcium channel blocker-1 is an orally active analgesic agent,shows high affinity to functionally block N-type calcium channels.Formula:C31H47N3Purity:98%Color and Shape:SolidMolecular weight:461.73EGFR-IN-32
CAS:EGFR-IN-32, a potent EGFR blocker, shows promise for EGFR-mutated illnesses. (Patent WO2021185297A1, compound 2)Formula:C31H34N6O3Color and Shape:SolidMolecular weight:538.64WAY-215718
CAS:WAY-215718 is an active molecule.Formula:C18H12ClN3OS2Color and Shape:SolidMolecular weight:385.89ASN90
CAS:ASN90 is a specific, orally active inhibitor of the O-GlcNAcase (OGA) enzyme, demonstrating an IC50 of 10.2 nM.Formula:C17H21N5O3SColor and Shape:SolidMolecular weight:375.45SAD-448
CAS:SAD-448 is a cannabinoid receptor type 1 (CB1) agonist. SAD-448 controls spasticity via action on the peripheral nerve CB1 receptor.Formula:C24H28N4O8SColor and Shape:SolidMolecular weight:532.57Antiproliferative agent-41
CAS:Antiproliferative Agent-41 (Compound 14), classified as indanorine [1], functions as an antiproliferative compound.Formula:C20H20O4Color and Shape:SolidMolecular weight:324.37S-(N-Methylsulfinylbutylthiocarbamoyl)-L-cysteine
CAS:S-(N-Methylsulfinylbutylthiocarbamoyl)-L-cysteine (SFN-Cys) is an isothiocyanate derivative, functioning as an active metabolite of sulforaphane, a class I andFormula:C9H18N2O3S3Color and Shape:SolidMolecular weight:298.45
