Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,849 products)
- Apoptosis(6,366 products)
- Cell Cycle/Checkpoint(4,907 products)
- Chromatin/Epigenetics(2,623 products)
- Cytoskeletal Signaling(1,585 products)
- DNA Damage/DNA Repair(2,872 products)
- Endocrinology/Hormones(3,759 products)
- Enzyme(3,673 products)
- GPCR/G-Protein(9,051 products)
- Immunology and Inflammation(3,945 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(417 products)
- MAPK Signaling(1,259 products)
- Membrane Transporter/Ion Channel(3,162 products)
- Metabolism(10,149 products)
- Microbiology/Virology(7,672 products)
- Neuroscience(10,549 products)
- Other Inhibitors(35,857 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,435 products)
- Proteases/Proteasome(1,693 products)
- Stem Cell and Derivatives(734 products)
- Tyrosine Kinase/Adaptors(1,991 products)
- Ubiquitination(1,743 products)
Show 16 more subcategories
Found 66517 products of "Inhibitors"
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ALM301
CAS:ALM301: oral AKT inhibitor targeting AKT1, AKT2, AKT3; blocks AKT phosphorylation, curbs cancer cell growth.Formula:C25H25N3O3Color and Shape:SolidMolecular weight:415.48KRAS inhibitor-12
CAS:KRAS inhibitor-12 blocks KRAS G12C (IC50: 0.537 μM) and p-ERK in cancer cells; promising for pancreatic, colorectal, lung cancer study.Formula:C19H16Cl2FN5OSColor and Shape:SolidMolecular weight:452.33PIM1-IN-1
CAS:PIM1-IN-1 inhibits PIM1/3 with IC50s: PIM1 (7 nM), PIM2 (5530 nM), PIM3 (70 nM); it has anti-cancer properties.Formula:C25H30N8O2Purity:98.59%Color and Shape:SolidMolecular weight:474.56Ref: TM-T12474
10mgTo inquire1mL*10mM (DMSO)To inquire1mg117.00€5mg281.00€25mg858.00€50mg1,341.00€100mg2,125.00€PDK4-IN-1 hydrochloride
CAS:PDK4-IN-1 hydrochloride is an anthraquinone derivative and a potent and orally active inhibitor of pyruvate dehydrogenase kinase 4 (PDK4, IC50 value = 84 nM).Formula:C22H20ClN3O2Purity:99.67%Color and Shape:SolidMolecular weight:393.87Ref: TM-T12412L
1mg70.00€5mg150.00€1mL*10mM (DMSO)165.00€10mg215.00€25mg358.00€50mg515.00€100mg707.00€200mg1,009.00€IIIM-8
CAS:IIIM-8 is a melanogenesis inhibitor that suppresses pigment production in both in vitro and in vivo settings, exhibiting no cytotoxic effects on Human AdultFormula:C14H17NO4Purity:98%Color and Shape:SolidMolecular weight:263.29GALK1-IN-1
CAS:Compound 4, known as GALK1-IN-1, is a potent inhibitor of galactokinase, exhibiting an IC50 value of 4.2129 μM [1].Formula:C19H20N4O2Purity:98%Color and Shape:SolidMolecular weight:336.39ASP6432
CAS:ASP6432 is an antagonist of type 1 lysophosphatidic acid receptor (LPA1). For human LPA1 and rat LPA1, the IC50s are 11 nM and 30 nM , respectively.Formula:C26H32KN4O6S2Color and Shape:SolidMolecular weight:599.78mTOR inhibitor-3
CAS:mTOR inhibitor-3 is a selective mTOR inhibitor (Ki= 1.5 nM). mTOR inhibitor-3 inhibits mTORC1 and mTORC2 in cellular and in vivo experiments.Formula:C25H30N8O2Purity:99% - 99.64%Color and Shape:SolidMolecular weight:474.56Ref: TM-T12123
1mg57.00€5mg120.00€1mL*10mM (DMSO)128.00€10mg170.00€25mg290.00€50mg439.00€100mg620.00€500mg1,288.00€CLP257
CAS:CLP257 is a selective K+-Cl− cotransporter KCC2 activator (EC50: 616 nM) and it is inactive against NKCC1, GABAA receptors, KCC1, KCC3 or KCC4.Formula:C14H14FN3O2SPurity:99.5%Color and Shape:SolidMolecular weight:307.344E2RCat
CAS:4E2RCat is an inhibitor of eIF4E-eIF4G interaction (IC50 = 13.5 μM) and is capable of blocking coronavirus replication as monitored by viral protein expressionFormula:C22H14ClNO4S2Purity:98.44%Color and Shape:SolidMolecular weight:455.93(S)-Ceralasertib
CAS:(S)-Ceralasertib: Potent, selective ATR inhibitor with strong preclinical physicochemical and PK profiles.Formula:C20H24N6O2SColor and Shape:SolidMolecular weight:412.51CCT241533 hydrochloride
CAS:CCT241533 hydrochloride is an effective and selective ATP competitive inhibitor of CHK2 (Ki: 1.16 nM; IC50: 3 nM).Formula:C23H28ClFN4O4Purity:97.13%Color and Shape:SolidMolecular weight:478.95Ref: TM-T10718L
1mg70.00€2mg90.00€5mg150.00€1mL*10mM (DMSO)167.00€10mg227.00€25mg487.00€50mg807.00€100mg1,198.00€500mg2,412.00€BPI-9016M
CAS:BPI-9016M, an oral c-Met/AXL inhibitor, curbs growth and spread of lung cancer.Formula:C25H18F2N4O3Color and Shape:SolidMolecular weight:460.43WIN site inhibitor 1 TFA (2407457-36-5 free base)
WIN site inhibitor 1 TFA is a WIN site of chromatin-associated WD repeat-containing protein 5 (WDR5) inhibitor (Kd: 0.1 nM).Formula:C27H23Cl2F4N5O3Purity:98%Color and Shape:SolidMolecular weight:612.4L 366948
CAS:L 366948 is an antagonist of the oxytocin receptor.Formula:C42H54N8O6Purity:98%Color and Shape:SolidMolecular weight:766.93Lobenzarit sodium
CAS:Lobenzarit sodium (CCA) is an agent with the activity of antirheumatic and antioxidative.Formula:C14H8ClNNa2O4Purity:99.35%Color and Shape:SolidMolecular weight:335.65MDL-19744A
CAS:MDL-19744A is an alpha 1-adrenergic receptor antagonist and renal vasodilator.Formula:C21H25NO3SColor and Shape:SolidMolecular weight:371.49SCH-538415
CAS:SCH-538415: Microbial acyl carrier protein synthase inhibitor, IC50 4.19µM; anti-Staphylococcus aureus.Formula:C16H14N2O4Purity:98%Color and Shape:SolidMolecular weight:298.29Lepadin E
CAS:Lepadin E, a notably cytotoxic compound, effectively stimulates ferroptosis via the canonical p53-SLC7A11-GPX4 pathway.Formula:C26H47NO3Purity:98%Color and Shape:SolidMolecular weight:421.6658-G3
CAS:58-G3 is an agonist of methuselah (Mth)-specific that acts by inducing dose-dependent calcium elevation and membrane translocation of β-arrestin2.Formula:C14H12Cl2N4O5Purity:98%Color and Shape:SolidMolecular weight:387.17S-Me-DM4
CAS:S-Me-DM4 is an intracellular enzyme S-methylated metabolite of DM4, a maytansinoid with microtubule-depolymerizing properties and potent cytotoxicity, employedFormula:C39H56ClN3O10SColor and Shape:SolidMolecular weight:794.39GSK321
CAS:GSK321 is an IDH1 inhibitor that prevents cytoplasmic glutamine reductive carboxylation.GSK321 is used in the study of leukemia.Formula:C28H28FN5O3Purity:99.73%Color and Shape:SolidMolecular weight:501.55Edralbrutinib
CAS:Edralbrutinib (TG-1701) is a potent BTK inhibitor with anticancer activity and is used in the treatment of tumors, immune system disorders, and blood andFormula:C26H21F2N5O3Purity:99.41%Color and Shape:SolidMolecular weight:489.47Edaglitazone
CAS:Edaglitazone (R-483) is a PPARγ agonist with antiplatelet activity that can be used in studies of diabetes and obesity.Formula:C24H20N2O4S2Purity:98%Color and Shape:SolidMolecular weight:464.56MK-0493
CAS:MK-0493 is an effective and selective agonist of the melanocortin receptor 4 (MC4R). It also demonstrated significant reductions in energy intake.Formula:C30H38ClF2N3O2Purity:98%Color and Shape:SolidMolecular weight:546.09HDAC/BET-IN-1
CAS:HDAC/BET-IN-1 inhibits HDAC1 (IC50: 0.163 μM), HDAC6 (IC50: 0.067 μM), BRD4 (Ki: 0.076 μM), and fights leukemia.Formula:C29H40N4O8SPurity:98%Color and Shape:SolidMolecular weight:604.71PARP7-IN-16
CAS:PARP7-IN-16 (compound 36) is a potent, selective, and orally active PARP-1/2/7 inhibitor, exhibiting IC50 values of 0.94, 0.87, and 0.21 nM , respectively.Formula:C25H26FN4NaO4Purity:98%Color and Shape:SolidMolecular weight:488.49BILR-355
CAS:BILR-355 is a reverse transcriptase inhibitor.Formula:C25H23N5O3Purity:98%Color and Shape:SolidMolecular weight:441.48Etidocaine Hydrochloride
CAS:Etidocaine Hydrochloride (W19053) is a long-acting anesthetic and a blocker of the voltage-gated sodium channel.Formula:C17H29ClN2OPurity:99.86%Color and Shape:SolidMolecular weight:312.88Ref: TM-T31716
1mg89.00€5mg177.00€1mL*10mM (DMSO)178.00€10mg260.00€25mg416.00€50mg565.00€100mg735.00€200mg973.00€Activated T Subunit
CAS:Activated T Subunit is employed in synthesizing exon-jumping oligomer conjugates that target specific sites within the human anti-muscular atrophy protein geneFormula:C31H34ClN4O5PColor and Shape:SolidMolecular weight:609.05Cimicoxib
CAS:Cimicoxib (UR8880) is a potent and selective inhibitor of COX-2 with anti-inflammatory and analgesic activity.Formula:C16H13ClFN3O3SPurity:98.22%Color and Shape:SolidMolecular weight:381.81Ref: TM-T30937
1mg44.00€2mg55.00€5mg79.00€1mL*10mM (DMSO)96.00€10mg105.00€25mg170.00€50mg255.00€100mg379.00€LSD1-UM-109
CAS:LSD1-UM-109 is a highly potent and reversible inhibitor of LSD1, demonstrating an IC50 of 3.1 nM.Formula:C29H27FN6Purity:98%Color and Shape:SolidMolecular weight:478.56Nilofabicin
CAS:Nilofabicin (CG-400549) is a potent inhibitor of enoyl-(acyl-carrier-protein) reductase fall(FabI) and can be used in studies about the treatment of complicatedFormula:C19H20N2O2SPurity:98.66%Color and Shape:SolidMolecular weight:340.44NT-0796
CAS:NT-0796 is an inflammasome NLRP3 inhibitor that inhibits NLRP3 activation.NT-0796 is a potential NDT-19795 delivery vector.Formula:C23H27N3O4Purity:99.67%Color and Shape:SolidMolecular weight:409.48GSK3395879
CAS:GSK3395879 is a selective and orally bioavailable antagonist of transient receptor potential vanilloid-4 (TRPV4) (IC50: 1 nM for hTRPV4).Formula:C20H15F4N3O5SPurity:98%Color and Shape:SolidMolecular weight:485.413,4'-Dihydroxyflavone
CAS:3,4'-Dihydroxyflavone (3,4'-DHF) is an oral active flavonoid. 3,4'-Dihydroxyflavone (3,4'-DHF) shows antiviral activity against Influenza A virus.Formula:C15H10O4Purity:98.33%Color and Shape:SolidMolecular weight:254.24HIF-2α-IN-9
CAS:HIF-2α-IN-9 (compound 35r) serves as an HIF-2α inhibitor, effectively suppressing VEGF-A with an IC50 of 305 nM, and modulating growth-promoting genes withinFormula:C12H13F5O4S2Purity:98%Color and Shape:SolidMolecular weight:380.35IPG7236
CAS:IPG7236, a selective CCR8 antagonist, demonstrates notable tumor suppression in a mouse xenograft model of human breast cancer and is applicable in cancerFormula:C23H31N3O3SPurity:98%Color and Shape:SolidMolecular weight:429.58MY-673
CAS:MY-673, a colchicine binding site inhibitor (CBSI), impedes tubulin polymerization and disrupts the ERK signaling pathway, consequently modulating SMAD4 proteinFormula:C18H14N2O4Color and Shape:SolidMolecular weight:322.31ALK-IN-6
CAS:ALK-IN-6 is an orally bioavailable inhibitor of anaplastic lymphoma kinase (ALK, IC50s: 71 nM, 18.72 nM, and 36.81 nM for ALK wild, ALK F1196M and ALK F1174L).Formula:C26H29ClD3N5O3SPurity:98%Color and Shape:SolidMolecular weight:533.1KRAS G12C inhibitor 13
CAS:KRAS G12C inhibitor 13 is a KRAS G12C inhibitor .Formula:C40H46F3N7O4Purity:98%Color and Shape:SolidMolecular weight:745.83RP 70676
CAS:RP 70676 is a potent ACAT inhibitor(rat and rabbit ACAT with IC50 of 25 and 44 nM ).Formula:C25H28N4SPurity:99.92%Color and Shape:SolidMolecular weight:416.58Ref: TM-T12767
1mg58.00€5mg128.00€1mL*10mM (DMSO)141.00€10mg187.00€25mg338.00€50mg475.00€100mg665.00€200mg893.00€GPR40 Agonist 2
CAS:GPR40 Agonist 2 is a GPR40 agonist. It can be used in the research of diabetes.Formula:C24H30O3Purity:98%Color and Shape:SolidMolecular weight:366.49RK-682
CAS:RK-682 is a natural selective inhibitor of protein tyrosine phosphatases (PTPases).Formula:C21H36O5Color and Shape:SolidMolecular weight:368.51Licostinel
CAS:Licostinel (CGP 63446) is a glutamate receptor antagonist. Licostinel protects against permanent focal cerebral ischemia.Formula:C8H3Cl2N3O4Purity:98.02%Color and Shape:SolidMolecular weight:276.03ddUTP
CAS:ddUTP (2′,3′-Dideoxyuridine-5′-triphosphate) serves as a selective inhibitor of HIV and AMV reverse transcriptases with Ki values of 0.05 µM for HIV and 1 µMFormula:C9H15N2O13P3Purity:98%Color and Shape:SolidMolecular weight:448.111JTK-853
CAS:JTK-853: novel non-nucleoside HCV polymerase inhibitor with strong antiviral activity (EC50: 0.38 μM genotype 1a, 0.035 μM 1b).Formula:C28H23F7N6O4S2Purity:98%Color and Shape:SolidMolecular weight:704.64CCPG
CAS:CCPG is an agonist of excitatory Amino Acid.Formula:C6H9NO4Purity:98%Color and Shape:SolidMolecular weight:159.14I-287
CAS:I-287 is a selective, orally active PAR2 inhibitor that functions as a negative allosteric modulator of Gαq and Gα12/13 activity and their downstream effectors.Formula:C30H30ClFN4O4Color and Shape:SolidMolecular weight:565.04Ro 24-5098
CAS:Ro 24-5098 is an anti-HIV inhibitory effects of isoddA pronucleotides.Formula:C10H13N5O2Purity:98%Color and Shape:SolidMolecular weight:235.24
