Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,833 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,875 products)
- Chromatin/Epigenetics(2,612 products)
- Cytoskeletal Signaling(1,566 products)
- DNA Damage/DNA Repair(2,872 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,014 products)
- Immunology and Inflammation(3,900 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,256 products)
- Membrane Transporter/Ion Channel(3,154 products)
- Metabolism(10,139 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,369 products)
- Other Inhibitors(35,852 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,430 products)
- Proteases/Proteasome(1,691 products)
- Stem Cell and Derivatives(733 products)
- Tyrosine Kinase/Adaptors(1,983 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66522 products of "Inhibitors"
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4'-Azidothymidine
CAS:4'-Azidothymidine exhibits potent and selective activity against the human immunodeficiency virus.Formula:C10H13N5O5Color and Shape:SolidMolecular weight:283.24L 699333
CAS:L 699333 is an effective inhibitor of 5-lipoxygenase.Formula:C36H35ClN2O4SColor and Shape:SolidMolecular weight:627.19LB-60-OF61
CAS:LB-60-OF61 is a NAMPT inhibitor, a NAMPT inhibitor that displays antiproliferative activity against MYC oncogene-dependent cancer cell lines.Formula:C29H30N6O2Purity:99.47%Color and Shape:SolidMolecular weight:494.59Ref: TM-T11823
1mg154.00€5mg371.00€10mg612.00€25mg1,189.00€50mg2,008.00€100mg3,132.00€1mL*10mM (DMSO)404.00€CHF 2819
CAS:CHF 2819 is a novel orally active acetylcholinesterase inhibitor (AChE) developed for the treatment of Alzheimer's disease (AD).Formula:C21H26ClN3O3Color and Shape:SolidMolecular weight:403.9hCAIX-IN-15
CAS:hCAIX-IN-15 is a potent inhibitor of human carbonic anhydrase IX (hCA IX) with an inhibition constant (Ki) of 38.8 nM, exhibiting broad-spectrum anticancerFormula:C18H14FN7O2SPurity:98%Color and Shape:SolidMolecular weight:411.41DUB-IN-7
CAS:DUB-IN-7 (compound 43), a deubiquitinating enzyme (DUB) inhibitor, has utility in researching diseases driven by aberrant JAK2 activity, including leukemia [1].Formula:C17H19N5OColor and Shape:SolidMolecular weight:309.37GSK3532795
CAS:GSK3532795: potent oral HIV-1 maturation inhibitor; EC50: 1.9-13 nM for various strains.Formula:C42H62N2O4SPurity:98%Color and Shape:SolidMolecular weight:691.02ICMT-IN-32
CAS:ICMT-IN-32 (compound 70) acts as an inhibitor of isoprenylcysteine carboxyl methyltransferase (ICMT), demonstrating an IC50 value of 0.777 µM [1].Formula:C20H25NO2Color and Shape:SolidMolecular weight:311.42PF-05241328
CAS:PF-05241328 is an effective and selective inhibitor of human Nav1.7 voltage-dependent sodium channels (IC50: 31 nM).Formula:C19H21ClN4O4SPurity:98%Color and Shape:SolidMolecular weight:436.91Aβ/tau aggregation-IN-3
CAS:Aβ/tau aggregation-IN-3 is a potent inhibitor of amyloid protein aggregation, exhibiting an IC50 value of 0.85 µM in an Aβ-Thioflavin T (Aβ-ThT) functionalFormula:C23H22N4O3Color and Shape:SolidMolecular weight:402.45Chitin synthase inhibitor 14
CAS:Chitin Synthase Inhibitor 14 (compound 4n), a potent chitin synthase (CHS) inhibitor, exhibits antifungal activity and is effective against drug-resistantFormula:C25H26ClN5O5Color and Shape:SolidMolecular weight:511.96ICMT-IN-7
CAS:ICMT-IN-7 (compound 74), with an IC50 value of 0.015 µM, functions as an ICMT inhibitor, promotes cytoplasmic accumulation of ICMT in HCT-116 cells in a dose-Formula:C23H31NOColor and Shape:SolidMolecular weight:337.5GGFG-amide-glycol-amide-Exatecan
CAS:Exatecan (Intermediate 2), a derivative of GGFG-amide-glycol-amide-Exatecan, facilitates the synthesis of antibody-drug conjugates (ADCs) [1].Formula:C43H47FN8O11Color and Shape:SolidMolecular weight:870.88Muraglitazar glucuronide
CAS:Muraglitazar glucuronide is a Peroxime Proliferator Activated (PPAR) Agonist that has glucose- and lipid-lowering activities.Formula:C35H36N2O13Color and Shape:SolidMolecular weight:692.67CGS 21680
CAS:CGS 21680 is a chemical compound that acts as a selective agonist for both adenosine and its A2A receptor, demonstrating a binding affinity (K i) of 27 nM.Formula:C23H29N7O6Color and Shape:SolidMolecular weight:499.52TLR7/8 agonist 4 hydroxy-PEG6-acid
CAS:TLR7/8 agonist 4 hydroxy-PEG6-acid, a Drug-Linker Conjugate for ADCs, comprises the TLR7/8 agonist 4 and a hydroxy-PEG6-acid linker, suitable for the synthesisFormula:C33H52N6O8Color and Shape:SolidMolecular weight:660.8CFTR corrector 12
CAS:CFTR corrector 12 is a CFTR corrector that rescues all mutant proteins except M760R ABCA3 and can be used to study cystic fibrosis.Formula:C19H21ClN4O2S2Purity:99.47%Color and Shape:SolidMolecular weight:436.982,7-Bis(alloxycarbonylamino)-9-chloroacridine
CAS:2,7-Bis(alloxycarbonylamino)-9-chloroacridine serves as a fluorescent label.Formula:C21H18ClN3O4Color and Shape:SolidMolecular weight:411.84OY-201
CAS:OY-201 is a promising anti-ischemic stroke agent capable of crossing the blood-brain barrier (BBB).Formula:C25H33Cl2NColor and Shape:SolidMolecular weight:418.44BMS-983970
CAS:BMS-983970 is an oral inhibitor of pan-Notch, and for the treatment of multiplecancers.Formula:C26H26F4N4O3Color and Shape:SolidMolecular weight:518.5pan-KRAS-IN-2
CAS:Pan-KRAS-IN-2 (compound 6) is a broad-spectrum KRAS inhibitor exhibiting potent activity with IC50 values of ≤10 nM against KRAS wild type and its mutants (G12DFormula:C34H34F2N4O3Purity:98%Color and Shape:SolidMolecular weight:584.66EMD638683 S-Form
CAS:EMD638683 is a highly selective SGK1 inhibitor with IC50 of 3 μM. EMD638683 S-Form is the S-form of EMD638683.Formula:C18H18F2N2O4Color and Shape:SolidMolecular weight:364.34BO 2367
CAS:BO 2367, a topoisomerase inhibitor, is used to suppress the growth of tumor .Formula:C21H22ClF2N3O3Color and Shape:SolidMolecular weight:437.87AZD-1175
CAS:AZD-1175 is a cannabinoid receptor CB1 antagonist and highly lipophilic compound for the treatment of type 2 diabetes and obesity.Formula:C25H25Cl2F3N4O4SColor and Shape:SolidMolecular weight:605.46Anticancer agent 3
CAS:Anticancer agent 3 (Compound 4) is a anti-cancer agent.Formula:C20H25N3OSPurity:98%Color and Shape:SolidMolecular weight:355.5Emzadirib
CAS:Emzadirib (RAD51-IN-2) is a potent RAD51 inhibitor with potential anticancer activity for the study of DNA damage repair.Formula:C27H40N4O6S2Purity:99.79% - 99.9%Color and Shape:SolidMolecular weight:580.76Ref: TM-T12682
1mg147.00€2mg212.00€5mg356.00€10mg595.00€25mg954.00€50mg1,269.00€1mL*10mM (DMSO)393.00€FEN1-IN-5
CAS:FEN1-IN-5 (compound 12A) is a potent Flap endonuclease-1 (FEN1) inhibitor with an IC50 value of 12 nM, playing a role in DNA repair mechanisms [1].Formula:C21H17N3O4SPurity:98%Color and Shape:SolidMolecular weight:407.44GNE-6468
CAS:GNE-6468 is a potent and selective agonist of RORγ(RORc) (EC50: 13 nM for HEK-293 cell).Formula:C23H16ClN3O4Color and Shape:SolidMolecular weight:433.84R1498
CAS:R1498 inhibits CDK2, targets angiogenesis and mitosis, and is an oral treatment for liver and stomach cancer.
Formula:C18H15ClN4OPurity:98%Color and Shape:SolidMolecular weight:338.79TASP0412098
CAS:TASP0412098 is a potent, selective CRTH2 antagonist with oral activity.Formula:C27H23ClN2O3Purity:98%Color and Shape:SolidMolecular weight:458.94c-Fms-IN-14
CAS:c-Fms-IN-14 (Example 76) is a potent inhibitor of the c-Fms kinase with an IC50 of 4 nM, utilized in cancer and autoimmune disease research [1].Formula:C26H24N6OPurity:98%Color and Shape:SolidMolecular weight:436.51CC-90005
CAS:CC-90005 is a potent, selective oral PKC-θ inhibitor with an IC50 of 8 nM, preferential over PKC-δ, and inhibits T cell activation.Formula:C21H27F2N7O2Color and Shape:SolidMolecular weight:447.48Oloctinebart
CAS:Oloctinebart, a humanized immunoglobulin G4-kappa (IgG4-κ) monoclonal antibody targeting LGALS3, is utilized to decrease the formation of amyloid beta oligomersColor and Shape:Liquidvc-PABC-DM1
CAS:vc-PABC-DM1 is a chemical compound utilized for the synthesis of an antibody-drug conjugate (ADC) that incorporates a disulfide linker.Formula:C53H75ClN8O13SColor and Shape:SolidMolecular weight:1099.73SR 2595
CAS:SR2595 is an inverse agonist of nuclear receptor PPARγ with an IC 50 of 30 nM [1].Formula:C37H38N2O3Color and Shape:SolidMolecular weight:558.71Xeniafaraunol A
CAS:Xeniafaraunol A (compound 31) is a potent inhibitor of the transient receptor potential melastatin 7 (TRPM7) channel [1].Formula:C20H28O2Color and Shape:SolidMolecular weight:300.44Mal-PEG2-Val-Cit-PABA
CAS:Mal-PEG2-Val-Cit-PABA is a cleavable linker utilized in the construction of antibody-drug conjugates (ADCs), facilitating their synthesis by allowing forFormula:C27H38N6O9Purity:99.72%Color and Shape:SolidMolecular weight:590.631,2-Diheptadecanoyl-sn-glycero-3-phosphorylcholine
CAS:1,2-Diheptadecanoyl-sn-glycero-3-phosphorylcholine (DHPC) is a derivative of phosphatidylcholine (PC) that exhibits biological activity, functioning as aFormula:C42H84NO8PColor and Shape:SolidMolecular weight:762.09HBV-IN-8
CAS:HBV-IN-6 is a potent inhibitor of HBV (EC50: 287.9 nM).Formula:C21H25ClFN5O5S2Color and Shape:SolidMolecular weight:546.04Iganidipine HCl
CAS:NKY-722 (HCl), also known as Iganidipine, is a calcium channel blocker potentially for the treatment of glaucoma.Formula:C28H40Cl2N4O6Color and Shape:SolidMolecular weight:599.55Sigma-1 receptor antagonist 3
CAS:Sigma-1 receptor antagonist 3 is a more potent and selective antagonist of Sigma-1 (σ1) receptor (Ki = 1.14 nM) than σ2 receptor(Ki = 1239 nM).Formula:C19H23ClFN3OPurity:99.95%Color and Shape:SolidMolecular weight:363.86YXG-158
CAS:YXG-158 (Compound 23-h), an orally active androgen receptor (AR) degrader and cytochrome P450 17A1 (CYP17A1) inhibitor, exhibits AR degradation with a DC50 of 1Formula:C30H36FN3OPurity:98%Color and Shape:SolidMolecular weight:473.62(R)-FT671
CAS:(R)-FT671 is the R-isomer of FT671. FT671 is a potent, non-covalent and selective inhibitor of USP7 (IC50 of 52 nM)Formula:C24H23F4N7O3Purity:98%Color and Shape:SolidMolecular weight:533.48Bisindolylmaleimide X hydrochloride
CAS:Bisindolylmaleimide X hydrochloride (BIM-X hydrochloride) is a potent and selective PKC inhibitor. It is also a potent CDK2 antagonist (IC50: 200 nM).Formula:C26H25ClN4O2Purity:99.23%Color and Shape:SolidMolecular weight:460.96Afizagabar
CAS:Afizagabar, a first-in-class α5-GABAAR antagonist, IC50: 585 nM, Ki: 66 nM, may boost memory.Formula:C19H12FN3O2SColor and Shape:SolidMolecular weight:365.38RCB16007
CAS:RCB16007 is a Yellow Fever Virus (YFV) inhibitor that also demonstrates inhibitory action against the West Nile virus with an effective concentration (EC50) ofFormula:C18H14ClN5O2SColor and Shape:SolidMolecular weight:399.85Cergutuzumab amunaleukin
CAS:Cergutuzumab amunaleukin (CEA-IL2v) is a CEA-targeted IL-2 variant immunocytokine for combination cancer immunotherapy with anti-tumor activity.Purity:98% (SDS-PAGE); 99.7% (SEC-HPLC) - 98% (SDS-PAGE); 99.7% (SEC-HPLC)Color and Shape:LiquidMolecular weight:162.05 kDaUbrogepant
CAS:Ubrogepant (MK-1602) is an antagonist of calcitonin gene-related peptide receptor that can be used in the acute treatment of migraine studies.Formula:C29H26F3N5O3Purity:99.452% - 99.78%Color and Shape:SolidMolecular weight:549.54Ref: TM-T17194
1mg144.00€5mg358.00€10mg565.00€25mg880.00€50mg1,161.00€100mg1,594.00€1mL*10mM (DMSO)432.00€BGB-102
CAS:BGB-102 (JNJ-26483327) is a kinase inhibitor targeting FLT3 and YES1 and an antagonist targeting EGFR and VEGFR3.Formula:C22H25BrN4O2Purity:99.02%Color and Shape:SolidMolecular weight:457.365(S)-HpEPE
CAS:5(S)-HpEPE, derived from EPA by 5-LO, forms LTA5 for leukotrienes or is reduced to 5(S)-HEPE by peroxidases.Formula:C20H30O4Color and Shape:SolidMolecular weight:334.45
