Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,849 products)
- Apoptosis(6,366 products)
- Cell Cycle/Checkpoint(4,907 products)
- Chromatin/Epigenetics(2,622 products)
- Cytoskeletal Signaling(1,585 products)
- DNA Damage/DNA Repair(2,873 products)
- Endocrinology/Hormones(3,758 products)
- Enzyme(3,673 products)
- GPCR/G-Protein(9,049 products)
- Immunology and Inflammation(3,943 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(417 products)
- MAPK Signaling(1,259 products)
- Membrane Transporter/Ion Channel(3,164 products)
- Metabolism(10,149 products)
- Microbiology/Virology(7,673 products)
- Neuroscience(10,547 products)
- Other Inhibitors(35,859 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,435 products)
- Proteases/Proteasome(1,692 products)
- Stem Cell and Derivatives(734 products)
- Tyrosine Kinase/Adaptors(1,991 products)
- Ubiquitination(1,743 products)
Show 16 more subcategories
Found 66517 products of "Inhibitors"
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FAP Ligand 1
CAS:FAP Ligand 1 (FL), a high-affinity small molecule targeting fibroblast activation protein (FAP), facilitates the delivery of conjugated therapeutics to FAP-Formula:C15H17F2N5O2Color and Shape:SolidMolecular weight:337.32VEGFR-2-IN-37
CAS:VEGFR-2-IN-37 (compound 12), a VEGFR-2 inhibitor, exhibits an inhibition rate of approximately 56.9 μM at a concentration of 200 μM.Formula:C18H16N2O2SPurity:98%Color and Shape:SolidMolecular weight:324.4Nicotinamide, N-(5-(p-aminophenoxy)pentyl)-
CAS:Nicotinamide, N-(5-(p-aminophenoxy)pentyl)- is a bioactive chemical.Formula:C17H21N3O2Color and Shape:SolidMolecular weight:299.374WNY1613
CAS:WNY1613: Potent PI3Kδ inhibitor with anti-NHL properties, induces apoptosis in cells, affects phosphorylation in vitro/in vivo.Formula:C29H35N9O3Color and Shape:SolidMolecular weight:557.65HPK1-IN-37
CAS:HPK1-IN-37 (compound A85), with an IC50 value of 3.7 nM, is a potent inhibitor of HPK1.Formula:C27H35N7O4Color and Shape:SolidMolecular weight:521.61BM152054
CAS:BM152054 is a potent PPARγ ligand that induces glucose utilization in peripheral tissues by enhancing insulin action.Formula:C22H18N2O4S3Purity:99.56%Color and Shape:SolidMolecular weight:470.58(2S,3R)-Voruciclib
CAS:(2S,3R)-Voruciclib is the (2S,3R)-enantiomer of Voruciclib. It is an orally active CDK inhibitor.Formula:C22H19ClF3NO5Purity:98%Color and Shape:SolidMolecular weight:469.84RTI-13951-33
CAS:RTI-13951-33 is an effective and brain-penetrant GPR88 agonist (EC50: 25 nM, in GPR88 cAMP functional assay).Formula:C28H33N3O3Purity:98%Color and Shape:SolidMolecular weight:459.58Ras inhibitor 134
CAS:Ras inhibitor 134 can be used in studies about Ras.Formula:C23H21ClFN5O3Color and Shape:SoildMolecular weight:469.9AH13205
CAS:AH13205 is an agonist of EP2 prostanoid receptor.Formula:C24H36O4Purity:98%Color and Shape:SolidMolecular weight:388.54FLT3/ITD-IN-4
CAS:FLT3/ITD-IN-4 inhibits FLT3-ITD mutations in acute myeloid leukemia (IC50: 2.3 nM).Formula:C25H22N4O5Color and Shape:SolidMolecular weight:458.47α-HNJNAc
CAS:α-HNJNAc is a potent, competitive hexosaminidases inhibitor that does not interfer with other glycosidases [1].Formula:C9H18N2O5Color and Shape:SolidMolecular weight:234.25Arginase inhibitor 1
CAS:Arginase inhibitor 1 is a potent inhibitor of human arginases I and II (IC50s: 223 and 509 nM).Formula:C13H27BN2O4Color and Shape:SolidMolecular weight:286.18(R)-3,4-DCPG
CAS:AMPA receptor antagonist with weak activity at NMDA receptors and little activity at kainate receptorsFormula:C10H9NO6Purity:98%Color and Shape:SolidMolecular weight:239.18PRMT5-IN-29
CAS:PRMT5-IN-29 is a potent, orally active inhibitor of PRMT5, exhibiting an IC50 value of 1.5 μM, showing promise for use in advanced cancer research [1].Formula:C18H20Cl3N5O5Purity:98%Color and Shape:SolidMolecular weight:492.74TC-5115
CAS:TC-5115 inhibits MLL1 enzyme at 16 nM, promising for treating MLL leukemia.Formula:C23H32N8O5SColor and Shape:SolidMolecular weight:532.62JYL-1511
CAS:JYL-1511 is the TRPV1 channel partial agonist.Formula:C21H29N3O3S2Purity:98%Color and Shape:SolidMolecular weight:435.6BO-1158
CAS:BO-1158 is an antibacteria agent.Formula:C13H16FN5O8S2Purity:98%Color and Shape:SolidMolecular weight:453.42LY 213024
CAS:LY 213024 is an antagonist of leukotriene B4 receptor.Formula:C27H34O6Color and Shape:SolidMolecular weight:454.56JAK-IN-31
CAS:JAK-IN-31 (Example 75), a JAK inhibitor, demonstrates IC50 values of ≤0.01 µM for JAK1, ≤0.01 µM for JAK2, 0.01-0.1 µM for JAK3, and ≤0.01 µM for Tyk2,Formula:C21H19N7O2S2Purity:98%Color and Shape:SolidMolecular weight:465.55Antibacterial agent 94
CAS:Compound 5b, an antibacterial, effectively targets MRSA and disrupts bacterial membranes and PG synthesis.Formula:C21H21FO4Color and Shape:SolidMolecular weight:356.39GSK3532795
CAS:GSK3532795: potent oral HIV-1 maturation inhibitor; EC50: 1.9-13 nM for various strains.Formula:C42H62N2O4SPurity:98%Color and Shape:SolidMolecular weight:691.02CycLuc2
CAS:CycLuc2, a cyclic luciferin for firefly luciferase, outshines aminoluciferin and D-luciferin by 4.7x and 2.6x, respectively.Formula:C14H13N3O2S2Color and Shape:SolidMolecular weight:319.4INX-SM-6
CAS:INX-SM-6, a chemical compound, serves as a targeted delivery vehicle for anti-inflammatory agents and has shown efficacy in suppressing LPS-induced IL-1βFormula:C32H36N2O6SColor and Shape:SolidMolecular weight:576.7WAY-608119
CAS:WAY-608119 is an active molecule.Formula:C13H9N3OColor and Shape:SolidMolecular weight:223.23Dusquetide TFA (931395-42-5 free base)
Dusquetide TFA is an IDR, reduces inflammation, enhances bacterial clearance, and modulates immune response to PAMPs/DAMPs via P62.Formula:C27H48F3N9O7Purity:98%Color and Shape:SolidMolecular weight:667.72S1P5 receptor agonist-1
CAS:S1P5 Receptor Agonist-1 (example 6) is a highly potent and selective agonist for the S1P5 receptor, exhibiting an EC50 value of 20 nM.Formula:C20H24F3NO3Color and Shape:SolidMolecular weight:383.4Risevistinel
CAS:Risevistinel (NYX-783), a positive allosteric modulator of the N-methyl-D-aspartate (NMDA) receptor, may mitigate cognitive deficits in neurodegenerativeFormula:C14H23N3O4Purity:98%Color and Shape:SolidMolecular weight:297.35Azaconazole
CAS:Azaconazole, an agricultural fungicide, is used for controlling powdery mildew on crops and bean rust.Formula:C12H11Cl2N3O2Color and Shape:SolidMolecular weight:300.14PF3845yne
CAS:PF3845yne is an alkyne analogue of PF-3845 maintaining high potency for FAAH.Formula:C25H24N4O2Color and Shape:SolidMolecular weight:412.48JGK-068S
CAS:Compound I (JGK-068S) is a potent inhibitor of the epidermal growth factor receptor (EGFR) [1].Formula:C22H23BrFN5O2Purity:98%Color and Shape:SolidMolecular weight:488.35Clocortolone pivalate
CAS:Clocortolone pivalate, a synthetic steroid, treats dermatitis and psoriasis.Formula:C27H36ClFO5Color and Shape:SolidMolecular weight:495.02SB-649701
CAS:SB-649701 is a potent antagonist of the human CCR8 receptor, exhibiting a pIC50 value of 7.7, and is utilized in asthma research [1].Formula:C27H28N4O3Purity:98%Color and Shape:SolidMolecular weight:456.54Dothiepin
CAS:Dothiepin (Dosulepin; Dothep), an antidepressant with sedative/anxiolytic properties, preferentially inhibits noradrenaline over serotonin uptake, enhancingFormula:C19H21NSPurity:98%Color and Shape:SolidMolecular weight:295.44PSMA-Val-Cit-PAB-MMAE
CAS:PSMA-Val-Cit-PAB-MMAE is a novel PSMA-targeted small-molecule conjugate leveraging monomethyl auristatin E (MMAE) for prostate cancer chemotherapy.Formula:C114H165ClN20O26Color and Shape:SolidMolecular weight:2267.1WAY-354436
CAS:WAY-354436 is an active molecule.Formula:C19H22FN3SColor and Shape:SolidMolecular weight:343.46A 53693
CAS:A 53693 is a rigid catecholamine and a selective adrenergic agonist. A 53693 has affinity to certain alpha receptor subtypes in rat alpha-2 receptors.Formula:C13H17NO2Purity:98%Color and Shape:SolidMolecular weight:219.28Anticancer agent 93
CAS:Anticancer Agent 93, a 4-Hydroxycoumarin derivative, inhibits the invasion and migration of lung cancer cells through modulation of epithelial-mesenchymalFormula:C16H10ClNO4Color and Shape:SolidMolecular weight:315.71DYRKs-IN-2
CAS:DYRKs-IN-2 has antitumor activity. DYRKs-IN-2 is a potent DYRKs inhibitor with IC50s of 30.6 nM and 12.8 nM for DYRK1B and DYRK1A, respectively.Formula:C32H38ClN9O3Purity:98%Color and Shape:SolidMolecular weight:632.16CJ-42794
CAS:CJ-42794 (CJ-042794) is a selective antagonist of prostaglandin E receptor subtype 4 (EP4).Formula:C22H17ClFNO4Purity:99.92%Color and Shape:SolidMolecular weight:413.83Deleobuvir sodium
CAS:Deleobuvir sodium (BI207127), a hepatitis C NS5B inhibitor, showed promise in some trials but was discontinued in 2013 due to insufficient efficacy.Formula:C34H32BrN6NaO3Color and Shape:SolidMolecular weight:675.56Aurora Kinases-IN-4
CAS:Aurora Kinases-IN-4 (Compound 11c) is a covalent, ATP-competitive inhibitor of aurora kinase A with an IC50 value of 1.7 nM.Formula:C26H28N8OPurity:98%Color and Shape:SolidMolecular weight:468.55MurA-IN-4
CAS:MurA-IN-4 exhibits antibacterial properties as a MurA inhibitor, impeding the synthesis of bacterial cell walls [1].Formula:C8H12ClNO3Color and Shape:SolidMolecular weight:205.64N-5984 Hydrochloride
CAS:N-5984 Hydrochloride is a beta3-AR agonist.Formula:C20H23Cl2NO5Color and Shape:SolidMolecular weight:428.31SQ 32970
CAS:SQ 32970 is a potent Endothia aspartic proteinase inhibitor.Formula:C33H51N5O4SColor and Shape:SolidMolecular weight:613.85Setipafant
CAS:Setipafant is an antagonist of the platelet-activating factor.Formula:C26H23ClN6O2SPurity:98%Color and Shape:SolidMolecular weight:519.022-Methyl-5-HT
CAS:2-Methyl-5-HT (2-Methyl-5-hydroxytryptamine) is a potent and selective 5-HT3 receptor agonist with anti-depressive-like effects.Formula:C11H14N2OPurity:97.18%Color and Shape:SolidMolecular weight:190.24Ref: TM-T10075
5mg48.00€1mL*10mM (DMSO)50.00€10mg84.00€25mg177.00€50mg334.00€100mg500.00€500mg1,099.00€Antiproliferative agent-40
CAS:Antiproliferative agent-40 (Compound 9) effectively inhibits the proliferation of HT1080 and MCF-7 cancer cells, displaying IC50 values of 52 μM and 8.2 μM,Formula:C20H18N4O3Color and Shape:SolidMolecular weight:362.38AY 31906
CAS:AY 31906: High ceiling diuretic, boosts sodium/chloride excretion without affecting potassium, GFR, or renal flow in dogs.Formula:C15H24N6O3SColor and Shape:SolidMolecular weight:368.45HD-2a
CAS:HA-2a inhibits the JAK2/STAT3 pathway by downregulating circDcbld2 expression in RAW264.7 cells [1].Formula:C18H18O6Color and Shape:SolidMolecular weight:330.33
