Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,850 products)
- Apoptosis(6,367 products)
- Cell Cycle/Checkpoint(4,909 products)
- Chromatin/Epigenetics(2,631 products)
- Cytoskeletal Signaling(1,586 products)
- DNA Damage/DNA Repair(2,868 products)
- Endocrinology/Hormones(3,765 products)
- Enzyme(3,673 products)
- GPCR/G-Protein(9,053 products)
- Immunology and Inflammation(3,946 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(417 products)
- MAPK Signaling(1,259 products)
- Membrane Transporter/Ion Channel(3,163 products)
- Metabolism(10,156 products)
- Microbiology/Virology(7,671 products)
- Neuroscience(10,551 products)
- Other Inhibitors(35,855 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,435 products)
- Proteases/Proteasome(1,692 products)
- Stem Cell and Derivatives(733 products)
- Tyrosine Kinase/Adaptors(1,989 products)
- Ubiquitination(1,744 products)
Show 16 more subcategories
Found 66515 products of "Inhibitors"
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Maropitant citrate anhydrous
CAS:Maropitant citrate anhydrous is a neurokinin (NK1) receptor antagonist.Formula:C38H48N2O8Color and Shape:SolidMolecular weight:660.8THRX-144644
CAS:THRX-144644: lung-specific ALK5 inhibitor, 0.14 nM IC50, no systemic TGFβ toxicity.Formula:C26H28ClF2N7Color and Shape:SolidMolecular weight:512eIF4A i28
CAS:eIF4A i28, an inhibitor of the eukaryotic initiation factor-4A (eIF4A) with an IC50 of 8.60 μM in an eIF4A ATPase assay, effectively reduces the viability ofFormula:C24H20N2O5Color and Shape:SolidMolecular weight:416.4310-Chloroestra-1,4-diene-3,17-dione
CAS:10-Chloroestra-1,4-diene-3,17-dione acts as an estrogen receptor α (ERα) agonist, enhancing reporter gene expression in S.Formula:C18H21ClO2Color and Shape:SolidMolecular weight:304.80C6 Urea Ceramide
CAS:C6 urea ceramide blocks neutral ceramidase, boosts ceramide levels, halts HT-29 cancer cell growth, and shrinks HT-29 tumors in mice when dosed.Formula:C25H50N2O3Color and Shape:SolidMolecular weight:426.68NVP-ABJ688
CAS:NVP-ABJ688 is the cysteine protease cathepsin K inhibitor.Formula:C25H32N8OPurity:98%Color and Shape:SolidMolecular weight:460.57CD73-IN-10
CAS:CD73-IN-10, a potent inhibitor of CD73, aids in creating cancer drugs by hindering adenosine synthesis, which fosters tumor growth.Formula:C15H13F2N5O2Color and Shape:SolidMolecular weight:333.29LONP1-IN-2
CAS:LONP1-IN-2: Potent LONP1 inhibitor, IC50=0.187μM; weak on 20S proteasome (>10μM); for cancer research.Formula:C16H27BN4O4Color and Shape:SolidMolecular weight:350.22Tolterodine Dimer
CAS:Tolterodine Dimer is a derivative of Tolterodine -- a muscarinic receptor antagonist that is used to treat patients with overactive bladder.Formula:C35H41NO2Color and Shape:SolidMolecular weight:507.71IR415
CAS:IR415 selectively interacts with Hepatitis B virus X protein (HBx, Kd = 2 nM) and blocks HBV-mediated RNAi suppression, reverses the inhibitory effect of HBxFormula:C13H14F2N4SPurity:99.85%Color and Shape:SolidMolecular weight:296.34Ref: TM-T11669
5mg43.00€1mL*10mM (DMSO)47.00€10mg71.00€25mg128.00€50mg215.00€100mg318.00€200mg444.00€Amotosalen hydrochloride
CAS:Amotosalen hydrochloride (S-59) is a light-activated, RNA-, DNA-crosslinking psoralen compound and is used to neutralize pathogens.Formula:C17H20ClNO4Color and Shape:SolidMolecular weight:337.8MMP-9-IN-8
CAS:MMP-9-IN-8 (Compound 3), an MMP-9 inhibitor, exhibits inhibitory activities of 42.16% at 10 μM and 58.28% at 50 μM.Formula:C20H21F4N7OColor and Shape:SolidMolecular weight:451.42AR453588
CAS:AR453588 is an orally bioavailable anti-diabetic glucokinase activator (EC50: 42 nM) with anti-hyperglycemic activity.Formula:C25H25N7O2S2Color and Shape:SolidMolecular weight:519.64SHP2-IN-20
CAS:SHP2-IN-20 (compound 193), a potent SHP2 inhibitor, exhibits an IC50 of 3 nM, making it suitable for glioblastoma research [1].Formula:C25H24F2N6Color and Shape:SolidMolecular weight:446.5α-Glucosidase-IN-29
CAS:α-Glucosidase-IN-29 (compound 19) is an inhibitor of α-glucosidases, exhibiting an IC50 value of 1.21 μM and a Ki of 1.80 μM.Formula:C33H30Br2O7Purity:98%Color and Shape:SolidMolecular weight:698.4PYZD-4409
CAS:PYZD-4409 is a selective UBA1 inhibitor with an IC50 of 20 μM.
Formula:C14H7ClFN3O5Purity:99.71%Color and Shape:SolidMolecular weight:351.67Sophorose
CAS:Sophorose, a disaccharide within sophorolipids synthesized by yeast, functions as a biosurfactant owing to its hydrophobic properties.Formula:C12H22O11Color and Shape:SolidMolecular weight:342.3Flesinoxan
CAS:Flesinoxan is a hypotensive agent and is an effective, high affinity, and selective 5-hydroxytryptamine1A receptor agonist (EC50: 24 nM).Formula:C22H26FN3O4Color and Shape:SolidMolecular weight:415.46WAY-221060-A
CAS:WAY-221060-A is an active molecule.Formula:C17H18N4OColor and Shape:SolidMolecular weight:294.35Cyclopropavir
CAS:Cyclopropavir (Filociclovir; MBX-400) is a broad-spectrum anti-herpes drug effective against CMV and HHV-6/8 (EC50: 0.7-8 μM).Formula:C11H13N5O3Purity:98%Color and Shape:SolidMolecular weight:263.25Lysyl-aspartyl-glutamyl-leucine
CAS:Lysyl-aspartyl-glutamyl-leucine maintains type II surface membrane proteins in the endoplasmic reticulum.Formula:C21H37N5O9Color and Shape:SolidMolecular weight:503.55PD 114595
CAS:PD 114595 is a Benzothiopyrano-indazole cpd.Formula:C23H31N5O2SColor and Shape:SolidMolecular weight:441.59Antitumor agent-92
CAS:Antitumor Agent-92, a derivative of Icaritin, halts cell cycle, triggers cell death, and is promising for liver cancer study.Formula:C33H41NO10Purity:98%Color and Shape:SolidMolecular weight:611.68A 74704
CAS:A 74704 is a pseudo C2-symmetric inhibitor of HIV-1 protease and its diester analog.Formula:C43H52N4O7Purity:98%Color and Shape:SolidMolecular weight:736.9ZIKV-IN-1
CAS:ZIKV-IN-1 blocks Zika virus effectively (EC50: 2.8 μM, EC90: 6.8 μM), targets the RdRp domain, and is low-toxic.Formula:C21H18BrF2N3O3Color and Shape:SolidMolecular weight:478.29PBB3
CAS:PBB3 is a tau-specific PET tracer.Formula:C17H15N3OSColor and Shape:SolidMolecular weight:309.39Sigma-1 receptor antagonist 2
CAS:Sigma-1 receptor antagonist 2 is a more potent and selective antagonist of sigma 1 receptor (σ1 R, Ki = 3.88 nM) than σ2 receptor (Ki = 1288 nM).Formula:C20H26ClN3O2Purity:99.6%Color and Shape:SolidMolecular weight:375.89Ref: TM-T12911
1mg46.00€5mg96.00€1mL*10mM (DMSO)105.00€10mg161.00€25mg261.00€50mg371.00€100mg504.00€200mg675.00€L-736380
CAS:L-736380, a CCK-B antagonist, reduces gastric acid (ID50: 0.064mg/kg) and blocks [(125)I]CCK-8S in mouse brains (ED50: 1.7mg/kg).Formula:C25H29N9O2Color and Shape:SolidMolecular weight:487.56HQ005
CAS:HQ005, a potent CCNK degrader, exhibits an impressive DC50 value of 0.041 µM and functions as a molecular-glue degrader.Formula:C15H15N5O2S2Color and Shape:SolidMolecular weight:361.44Deltakephalin
CAS:Deltakephalin is a synthetic, potent specific opiate delta receptors agonist.Formula:C34H48N6O10Purity:98%Color and Shape:SolidMolecular weight:700.782-Furoyl-LIGRLO-amide TFA
CAS:2-Furoyl-LIGRLO-amide TFA is a potent and selective agonist of the proteinase-activated receptor 2 (PAR2), exhibiting a pD2 value of 7.0 [1] [2].Formula:C38H64F3N11O10Color and Shape:SolidMolecular weight:891.98CBP-IN-1
CAS:CBP-IN-1 (compound 12) acts as a potent CBP inhibitor exhibiting an IC50 of 1.5 nM and additionally suppresses CBP BRET and BRD4(1) with IC50 values of 690 nMFormula:C27H33F2N7OPurity:98%Color and Shape:SolidMolecular weight:509.59FM26
CAS:FM26, an isoxazole-based RORγt inverse agonist, cuts EL4 IL-17a mRNA; potent with 264 nM IC50.Formula:C22H15ClF3N3O3Purity:98%Color and Shape:SolidMolecular weight:461.82Dibutepinephrine
CAS:Dibutylephrine is a sympathomimetic agent.Formula:C17H25NO5Color and Shape:SolidMolecular weight:323.38GIV3727
CAS:GIV3727, a bitter taste receptor hTAS2R antagonist, inhibits the activation of hTAS2R31 by saccharin and acesulfame potassium, effectively diminishing theFormula:C12H22O2Color and Shape:SolidMolecular weight:198.3DAM-IN-1
CAS:DMA-IN-1 is a DNA adenine methyltransferase (DAM) inhibitor with an IC50 value of 48 μM.Formula:C16H17NO4Purity:98%Color and Shape:SolidMolecular weight:287.313-Hydroxy-2-(palmitoyloxy)propyl stearat
CAS:3-Hydroxy-2-(palmitoyloxy)propyl stearate is a non-volatile compound isolated from the less polar fractions of the brown macroalga Fucus virsoides J.Formula:C37H72O5Color and Shape:SolidMolecular weight:596.96BMS-561392
CAS:BMS-561392 (DPC333) is a tumor necrosis factor-α ( TNF-α) Invertase inhibitor.Formula:C27H32N4O4Purity:99.16%Color and Shape:SolidMolecular weight:476.57IIIM-8
CAS:IIIM-8 is a melanogenesis inhibitor that suppresses pigment production in both in vitro and in vivo settings, exhibiting no cytotoxic effects on Human AdultFormula:C14H17NO4Purity:98%Color and Shape:SolidMolecular weight:263.29VER-00158411
CAS:VER-00158411 is a checkpoint kinase 1 and CHK2 inhibitor (IC50: 4.4 nM and 4.5 nM, respectively).Formula:C31H34N6O3Purity:98%Color and Shape:SolidMolecular weight:538.64MU-380
CAS:MU-380 is an effective and selective inhibitor of CHK1.Formula:C15H15BrF3N7Color and Shape:SolidMolecular weight:430.23KW-7158
CAS:KW-7158, a potassium channel activator, is used potentially for the treatment of urinary urgency and frequency.Formula:C16H12F3NO5S2Color and Shape:SolidMolecular weight:419.4NK007
CAS:NK007 is a novel anti-SARS-CoV-2 agent with an EC 50 value of 30 nM.Formula:C28H33NO9Color and Shape:SolidMolecular weight:527.56Siguazodan
CAS:Siguazodan (SKF 94836) is an effective, selective, orally active phosphodiesterase III ((PDE-III)) inhibitor with an IC50 of 117 nM.Formula:C14H16N6OPurity:99.62% - 99.87%Color and Shape:SolidMolecular weight:284.32Ref: TM-T12913
2mg38.00€5mg59.00€1mL*10mM (DMSO)64.00€10mg94.00€25mg175.00€50mg280.00€100mg434.00€200mg612.00€AMG 837
CAS:Prinaberel (ERB 041) is an ERβ agonist with anticancer activity and anti-inflammatory activity that inhibits the NFκB pro-inflammatory signaling pathway.Formula:C26H21F3O3Purity:98%Color and Shape:SolidMolecular weight:438.44FAS-IN-1 Tosylate
FAS-IN-1 Tosylate is an effective fatty acid synthase inhibitor;Has an IC50 of 10 nM.
Formula:C33H35N3O7S2Purity:98%Color and Shape:SolidMolecular weight:649.78PF-06807656
PF-06807656 remains effective against ROMK with N171D mutation, unlike other inhibitors; it has an IC50 of 160 nM for Tl+ flux.Formula:C19H20ClN5O4SPurity:98%Color and Shape:SolidMolecular weight:449.91Fiduxosin
CAS:Fiduxosin is a selective and potent α1-adrenoceptor antagonist with inhibitory effects on α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, with KiFormula:C30H29N5O4SPurity:99.73%Color and Shape:SolidMolecular weight:555.65Trithiozine
CAS:Trithiozine is used in peptic ulcer and hypersecretory disorder research for its antiulcer and antisecretory properties.Formula:C14H19NO4SPurity:90% - 99.47%Color and Shape:SolidMolecular weight:297.37Droxinavir Free Base
CAS:Droxinavir Free Base is an experimental protease inhibitor researched by Pharmacia as a treatment for HIV infection.Formula:C29H51N5O4Color and Shape:SolidMolecular weight:533.75
