Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,834 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,878 products)
- Chromatin/Epigenetics(2,613 products)
- Cytoskeletal Signaling(1,568 products)
- DNA Damage/DNA Repair(2,871 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,021 products)
- Immunology and Inflammation(3,904 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,258 products)
- Membrane Transporter/Ion Channel(3,157 products)
- Metabolism(10,131 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,484 products)
- Other Inhibitors(35,844 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,429 products)
- Proteases/Proteasome(1,689 products)
- Stem Cell and Derivatives(731 products)
- Tyrosine Kinase/Adaptors(1,982 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66514 products of "Inhibitors"
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LY3295668
CAS:LY3295668 (AK-01) is a selective inhibitor of Aurora A with Kis of 0.8 nM and 1038 nM for Aurora A and B, respectively.Formula:C24H26ClF2N5O2Purity:99.68%Color and Shape:SolidMolecular weight:489.95IACS-52825
CAS:IACS-52825 is a DLK inhibitor that reverses para-mechanical aberrant pain in a CIPN mouse model and can be used to study neurological disorders.Formula:C16H13F7N4O2Purity:99.77%Color and Shape:SolidMolecular weight:426.29EGFR-IN-87
CAS:EGFR-IN-87 is an EGFR tyrosine kinase inhibitor with potent inhibitory activity, exhibiting IC50 values of 3.1 nM, 1.3 nM, and 7.1 nM against EGFR_d746-750,Formula:C28H33N7O2Purity:98.64%Color and Shape:SolidMolecular weight:499.61Oditrasertib
CAS:Oditrasertib, a RIPK1 inhibitor characterized by an IC50 value below 100 nM, is employed in inflammation research.Formula:C14H15F2N3O2Purity:98.65% - 99.65%Color and Shape:SolidMolecular weight:295.28Ref: TM-T69726
1mg70.00€1mL*10mM (DMSO)138.00€5mg150.00€10mg215.00€25mg358.00€50mg517.00€100mg707.00€500mg1,431.00€Ac-YVAD-AOM
CAS:Ac-YVAD-AOM is a selective and potent caspase-1 inhibitor showing antitumor activity and potential analgesic activity.Formula:C33H42N4O10Purity:98%Color and Shape:SolidMolecular weight:654.71Funapide
CAS:Funapide (TV 45070) is a potent Nav1.7 inhibitor, potentially treating inflammation and various pains.Formula:C22H14F3NO5Purity:99.91%Color and Shape:SolidMolecular weight:429.35Ref: TM-T15358
1mg120.00€5mg289.00€1mL*10mM (DMSO)318.00€10mg439.00€25mg708.00€50mg954.00€100mg1,288.00€Rilapladib
CAS:Rilapladib (SB 659032) is a selective inhibitor of Lipoprotein-Associated Phospholipase A2(Lp-PLA2, IC50 = 230 pM) and an antagonist of the platelet activatingFormula:C40H38F5N3O3SPurity:99.92%Color and Shape:SolidMolecular weight:735.8Ref: TM-T16751
1mg87.00€5mg215.00€10mg349.00€1mL*10mM (DMSO)349.00€25mg537.00€50mg745.00€100mg1,108.00€200mg1,504.00€TZ3O
CAS:TZ3O is an anticholinergic compound with neuroprotective activity.TZ3O ameliorates memory impairment in Scopolamine-induced Alzheimer's type model in rats.Formula:C18H13NO4SPurity:99.84%Color and Shape:SolidMolecular weight:339.37γ-Glu-Tyr
CAS:gamma-Glu-Tyr (gamma-Glutamyltyrosine) is a kokumi peptide against dipeptidyl peptidase-IV (DPP-IV) and is used in the study of diabetes mellitus.Formula:C14H18N2O6Purity:98.92%Color and Shape:SolidMolecular weight:310.3ERDRP-0519
CAS:ERDRP-0519 is an oral measles polymerase inhibitor, preventing disease in monkeys, with potent nanomolar efficacy against morbilliviruses.Formula:C23H30F3N5O4SPurity:98.64% - 98.71%Color and Shape:SolidMolecular weight:529.58Ref: TM-T24040
1mg130.00€5mg313.00€1mL*10mM (DMSO)344.00€10mg439.00€25mg707.00€50mg1,009.00€100mg1,333.00€WAY-297848
CAS:WAY-297848 is a novel glucokinase activator for the prevention or treatment of hyperglycemia, diabetes mellitus, obesity, dyslipidemia, and metabolic syndrome.Formula:C13H13ClN2O2SPurity:98.19%Color and Shape:SolidMolecular weight:296.77Cis-N-Feruloyltyramine
CAS:Cis-N-Feruloyltyramine is a naturally occurring compound found in various plants that shows cytotoxicity against the P-388 cancer cell line.Formula:C18H19NO4Purity:97.43%Color and Shape:SolidMolecular weight:313.35Supercinnamaldehyde
CAS:Supercinnamaldehyde is a potent activator of transient receptor potential ankyrin 1 (TRPA1), exhibiting an EC50 of 0.8 μM, and induces activation of TRPA1 ionFormula:C12H11NO2Purity:98.89%Color and Shape:SolidMolecular weight:201.22TP-10
CAS:TP-10 is a selective inhibitor of PDE10A against other PDEs with IC50 of 0.8 nM.Formula:C26H19F3N4OPurity:99.21%Color and Shape:SolidMolecular weight:460.45Ref: TM-T13189
1mg87.00€2mg114.00€5mg177.00€1mL*10mM (DMSO)178.00€10mg264.00€25mg460.00€50mg668.00€100mg945.00€500mg1,783.00€αvβ1 integrin-IN-1
CAS:αvβ1 integrin-IN-1 is a potent and selective inhibitor of αvβ1 integrin (IC50 of 0.63 nM) with antifibrotic effects.Formula:C26H34N6O6SPurity:99.39% - 99.69%Color and Shape:SolidMolecular weight:558.65Ref: TM-T13473
1mg109.00€5mg260.00€1mL*10mM (DMSO)319.00€10mg409.00€25mg660.00€50mg888.00€100mg1,224.00€200mg1,648.00€ML400
CAS:ML400 (CID73050863) is an allosteric inhibitor of LMPTP with an EC50 of 1μM. ML400 displays good cell-based activity and rodent pharmacokinetics.Formula:C24H29N3OPurity:99.95%Color and Shape:SolidMolecular weight:375.51Ref: TM-T25824
1mg92.00€5mg172.00€1mL*10mM (DMSO)222.00€10mg281.00€25mg447.00€50mg618.00€100mg853.00€500mg1,701.00€Moracin C
CAS:Moracin C, a natural compound found in Morus mesozygia, Morus alba var.Formula:C19H18O4Purity:99.77% - >99.99%Color and Shape:SolidMolecular weight:310.34Aneratrigine hydrochloride
CAS:Aneratrigine hydrochloride is a Nav 1.9 blocker that may be used to prevent or treat sodium channel blocker-related disorders.Formula:C19H21Cl2F2N5O2S2Purity:98.37% - 99.16%Color and Shape:SolidMolecular weight:524.43Sembragiline
CAS:Sembragiline (EVT-302) is a selective MAO-B inhibitor for the study of Alzheimer's disease (AD).Formula:C19H19FN2O3Purity:99.49% - 99.49%Color and Shape:SolidMolecular weight:342.36Dechloro Rivaroxaban
CAS:Dechloro Rivaroxaban is a Factor Xa inhibitor that inhibits free FXa and plasminogen and fibrin-associated FXa activity in humans.Formula:C19H19N3O5SPurity:98.63%Color and Shape:SolidMolecular weight:401.44Ref: TM-T78215
5mg40.00€1mL*10mM (DMSO)44.00€10mg63.00€25mg107.00€50mg170.00€100mg264.00€200mg418.00€CF53
CAS:CF53: potent, selective oral BET inhibitor; Ki <1 nM, Kd 2.2 nM, IC50 2 nM for BRD4 BD1; high affinity for BRD2/3/4/BRDT; effective anti-tumor agent.Formula:C24H25N7O2Purity:99.72%Color and Shape:SolidMolecular weight:443.5Ref: TM-T10773
1mg92.00€5mg200.00€1mL*10mM (DMSO)215.00€10mg299.00€25mg484.00€50mg658.00€100mg892.00€DGAT-1 inhibitor 2
CAS:DGAT-1 inhibitor 2: effective against obesity, targets enzyme in triglyceride synthesis for diabetes treatment.Formula:C24H28N4O3Purity:98.36%Color and Shape:SolidMolecular weight:420.5Ref: TM-T11016
1mg62.00€5mg133.00€1mL*10mM (DMSO)147.00€10mg205.00€25mg378.00€50mg580.00€100mg798.00€Ertugliflozin L-pyroglutamic acid
CAS:Ertugliflozin is a potent oral hSGLT2 inhibitor (IC50: 0.877 nM) for type 2 diabetes treatment studies.Formula:C27H32ClNO10Purity:99.88% - 99.94%Color and Shape:SolidMolecular weight:566Ref: TM-T15244
5mg44.00€1mL*10mM (DMSO)50.00€10mg57.00€25mg85.00€50mg90.00€100mg133.00€200mg188.00€500mg323.00€GNE-7883
CAS:GNE-7883 is an inhibitor targeting TEAD transcription factor, inhibits cell proliferation and suppresses YAP/TAZ activation, and can be used to study YAP/TAZ-dependent tumors.Formula:C28H29FN6O2Purity:97.61%Color and Shape:SolidMolecular weight:500.57Ref: TM-T78558
1mg116.00€5mg283.00€1mL*10mM (DMSO)310.00€10mg455.00€25mg747.00€50mg1,026.00€100mg1,444.00€200mg1,882.00€Iptacopan
CAS:Iptacopan (LNP023) is an inhibitor with high affinity to factor B, with a KD value of 7.9 nM and an IC50 value of 10 nM. Cost-effective and quality-assured.Formula:C25H30N2O4Purity:99.07% - >99.99%Color and Shape:SolidMolecular weight:422.52Ref: TM-T11864
1mg56.00€5mg120.00€1mL*10mM (DMSO)133.00€10mg195.00€25mg351.00€50mg588.00€100mg969.00€200mg1,311.00€PKC-IN-1
CAS:PKC-IN-1 is an ATP-competitive and reversible conventional PKC enzymes inhibitor (PKCα, PKCβI, PKCβII, PKCθ, PKCγ, PKC mu and PKCε with IC50s of 2.3, 8.1, 7.6,Formula:C25H37FN8O2Purity:98% - 98.79%Color and Shape:SolidMolecular weight:500.61SR 142948
CAS:SR 142948 is a neurotensin (NT) receptor antagonist.Formula:C39H51N5O6Purity:98%Color and Shape:SolidMolecular weight:685.85INCB3344
CAS:INCB3344 is an effective, specific and orally bioavailable CCR2 antagonist with IC50 values of 9.5 nM (mCCR2) and 5.1 nM (hCCR2) in binding antagonism and 7.8Formula:C29H34F3N3O6Purity:98% - 98.2%Color and Shape:SolidMolecular weight:577.59Ref: TM-TQ0103
1mg66.00€5mg144.00€1mL*10mM (DMSO)178.00€10mg230.00€25mg358.00€50mg512.00€100mg707.00€200mg973.00€PKI-402
CAS:PKI-402 is a potent PI3K and mTOR inhibitor. PKI-402 inhibits PI3Kα, mTOR, PI3Kβ, PI3Kδ and PI3Kγ with IC50s of 2, 3, 7, 14 and 16 nM, respectively.Formula:C29H34N10O3Purity:99.94%Color and Shape:SolidMolecular weight:570.65EGFR-IN-8
CAS:EGFR-IN-8, a dual inhibitor targeting both EGFR and c-Met, shows potential as a promising candidate for further development in treating EGFR TKI-resistant NSCLCFormula:C32H23ClF3N7O4Purity:99.51%Color and Shape:SolidMolecular weight:662.02PF-04979064
CAS:PF-04979064 is a potent and selective PI3K and mTOR dual kinase inhibitor(Ki of 0.13 nM and 1.42 nM,respectively).
Formula:C24H26N6O3Purity:98.20% - ≥98%Color and Shape:SolidMolecular weight:446.5Src Inhibitor 3
CAS:Src Inhibitor 3 blocks c-Src kinase (IC50 <3 nM CSK HTRF, <4 nM Caliper), boosting T cell growth from receptor signals.Formula:C34H32ClFN8O4Purity:98.35%Color and Shape:SolidMolecular weight:671.12Ref: TM-T13000
100mgTo inquire1mg96.00€5mg177.00€1mL*10mM (DMSO)264.00€10mg304.00€25mg480.00€50mg665.00€CeMMEC1
CAS:CeMMEC1 is an inhibitor of BRD4, and also has a great affinity for TAF1(IC50=0.9 μM).Formula:C19H16N2O4Purity:98.9% - 99.92%Color and Shape:SolidMolecular weight:336.34Lumateperone
CAS:Lumateperone (ITI 722) is a 5HT2A receptor antagonist and a dopamine receptor phosphoprotein modulator (DPPM).Formula:C24H28FN3OPurity:99.68% - 99.91%Color and Shape:SolidMolecular weight:393.5GDC-0349
CAS:GDC-0349 (RG-7603) is a potent and selective ATP-competitive inhibitor of mTOR, 790-fold inhibitory effect against PI3Kα and other 266 kinases. Phase 1.Formula:C24H32N6O3Purity:96.00% - 98.49%Color and Shape:SolidMolecular weight:452.55Sorivudine
CAS:Sorivudine (BV-araU) is an antiviral blocking DNA synthesis in viruses like varicella, HSV-1, and Epstein-Barr.Formula:C11H13BrN2O6Purity:99.74%Color and Shape:SolidMolecular weight:349.13PSB 1115
CAS:PSB 1115 is an A2B receptor antagonist and can counteract the inhibitory effect of NECA.Formula:C14H14N4O5SPurity:98.69% - >99.99%Color and Shape:SolidMolecular weight:350.35CAY10781
CAS:CAY10781 inhibits NRP-1/VEGF-A binding by 43% at 12.5μM and blocks VEGFR2 phosphorylation in CAD cells.Formula:C11H9N3O3Purity:99.49%Color and Shape:SolidMolecular weight:231.21Ref: TM-T37424
2mg39.00€5mg54.00€10mg77.00€1mL*10mM (DMSO)79.00€25mg124.00€50mg172.00€100mg316.00€200mg442.00€Mutant IDH1-IN-2
CAS:Mutant IDH1-IN-2 is a inhibitor of mutant Isocitrate dehydrogenase (IDH) proteins, with IC50 of 16.6 nM in Fluorescence biochemical assay, IC50 of ＜22 nM in LS-Formula:C24H31F2N5O2Purity:99.88%Color and Shape:SolidMolecular weight:459.53Ref: TM-T12128
1mg60.00€1mL*10mM (DMSO)137.00€5mg138.00€10mg224.00€25mg374.00€50mg532.00€100mg718.00€200mg964.00€Pan-RAS-IN-1
CAS:Pan-RAS-IN-1 is an inhibitor of pan-Ras. It disrupts the interaction of Ras proteins and their effectors.Formula:C36H41Cl2F3N6O2Purity:99.77%Color and Shape:SolidMolecular weight:717.65Ref: TM-T16432
1mg75.00€2mg92.00€5mg137.00€10mg205.00€1mL*10mM (DMSO)210.00€25mg416.00€50mg625.00€100mg888.00€500mg1,783.00€HM43239
CAS:HM43239: oral FLT3 inhibitor; IC50: FLT3 WT 1.1nM, ITD 1.8nM, D835Y 1.0nM; blocks p-STAT5/p-ERK; affects SYK, JAK1/2, TAK1; halts leukemia cell growth.Formula:C29H33ClN6Purity:99.7%Color and Shape:SolidMolecular weight:501.07Ref: TM-T9428
1mg50.00€5mg99.00€1mL*10mM (DMSO)109.00€10mg158.00€25mg309.00€50mg464.00€100mg647.00€200mg855.00€MK-8353
CAS:MK-8353 (SCH900353) is a potent, selective and orally available inhibitor of ERK1/2 (IC50s of 23.0 nM and 8.8 nM, respectively)Formula:C37H41N9O3SPurity:96.15% - 97.19%Color and Shape:SolidMolecular weight:691.84Ref: TM-T12069
1mg77.00€2mg92.00€5mg147.00€1mL*10mM (DMSO)217.00€10mg258.00€25mg557.00€50mg888.00€100mg1,341.00€BMS-986176
CAS:AAK1-IN-1 is a highly selective and potent inhibitor of adaptor associated kinase 1 (AAK1, IC50 = 2 nM).
Formula:C19H23F4N3OPurity:98.58% - 98.7%Color and Shape:SolidMolecular weight:385.4MDR-1339
CAS:MDR-1339 is a blood-brain-barrier-permeable inhibitor of amyloid-β (Aβ) aggregation.Formula:C20H22O4Purity:98.57%Color and Shape:SolidMolecular weight:326.39AMG2850
CAS:AMG2850 is a potent, orally bioavailable, and selective antagonist of transient receptor potential melastatin 8 (TRPM8).Formula:C19H17F6N3OPurity:99.84%Color and Shape:SolidMolecular weight:417.35Ref: TM-T10300
1mg71.00€5mg161.00€1mL*10mM (DMSO)172.00€10mg235.00€25mg423.00€50mg627.00€100mg803.00€AZ-23
CAS:AZ-23 is an inhibitor of ATP-competitive and Trk kinase A/B/C.Formula:C17H19ClFN7OPurity:99.4%Color and Shape:SolidMolecular weight:391.83GSK-F1
CAS:GSK-F1 (PI4KA inhibitor-F1) is a novel potent PI4KA inhibitor.Formula:C27H18F5N5O4SPurity:97.03%Color and Shape:SolidMolecular weight:603.52Ref: TM-T19840
1mg104.00€5mg215.00€1mL*10mM (DMSO)304.00€10mg318.00€25mg510.00€50mg692.00€100mg888.00€200mg1,251.00€AMG 837 calcium hydrate
CAS:AMG 837 calcium hydrate is a potent GPR40 agonist with an EC50 of 13 nM.Formula:C52H44CaF6O8Purity:98.07%Color and Shape:SolidMolecular weight:950.97PXS-5120A
CAS:PXS-5120A is an irreversible fluoroallylamine Lysyl Oxidase-like 2/3 (LOXL2/3) inhibitor with anti-fibrotic activity.Formula:C22H25ClFN3O4SPurity:97.02%Color and Shape:SolidMolecular weight:481.97Ref: TM-T12584
1mg205.00€2mg293.00€5mg462.00€1mL*10mM (DMSO)502.00€10mg612.00€25mg893.00€50mg1,224.00€100mg1,639.00€SB-616234-A
CAS:SB-616234-A is a selective and orally bioavailable antagonist of 5-HT1B receptor, with anxiolytic and antidepressant activity.Formula:C32H36ClN5O3Purity:99.72%Color and Shape:SolidMolecular weight:574.11
