Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,834 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,877 products)
- Chromatin/Epigenetics(2,613 products)
- Cytoskeletal Signaling(1,568 products)
- DNA Damage/DNA Repair(2,871 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,020 products)
- Immunology and Inflammation(3,905 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,257 products)
- Membrane Transporter/Ion Channel(3,155 products)
- Metabolism(10,133 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,473 products)
- Other Inhibitors(35,846 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,429 products)
- Proteases/Proteasome(1,689 products)
- Stem Cell and Derivatives(732 products)
- Tyrosine Kinase/Adaptors(1,982 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66515 products of "Inhibitors"
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AZ-23
CAS:AZ-23 is an inhibitor of ATP-competitive and Trk kinase A/B/C.Formula:C17H19ClFN7OPurity:99.4%Color and Shape:SolidMolecular weight:391.83SR 142948
CAS:SR 142948 is a neurotensin (NT) receptor antagonist.Formula:C39H51N5O6Purity:98%Color and Shape:SolidMolecular weight:685.85PSB 1115
CAS:PSB 1115 is an A2B receptor antagonist and can counteract the inhibitory effect of NECA.Formula:C14H14N4O5SPurity:98.69% - >99.99%Color and Shape:SolidMolecular weight:350.35INCB3344
CAS:INCB3344 is an effective, specific and orally bioavailable CCR2 antagonist with IC50 values of 9.5 nM (mCCR2) and 5.1 nM (hCCR2) in binding antagonism and 7.8Formula:C29H34F3N3O6Purity:98% - 98.2%Color and Shape:SolidMolecular weight:577.59Ref: TM-TQ0103
1mg66.00€5mg144.00€1mL*10mM (DMSO)178.00€10mg230.00€25mg358.00€50mg512.00€100mg707.00€200mg973.00€Lomibuvir
CAS:Lomibuvir (VCH-222, VX-222) is an allosteric inhibitor of HCV NS5B with Kd 17 nM, blocks RNA elongation, EC50 5.2 nM for 1b/Con1.Formula:C25H35NO4SPurity:99.83%Color and Shape:SolidMolecular weight:445.61AMG2850
CAS:AMG2850 is a potent, orally bioavailable, and selective antagonist of transient receptor potential melastatin 8 (TRPM8).Formula:C19H17F6N3OPurity:99.84%Color and Shape:SolidMolecular weight:417.35Ref: TM-T10300
1mg71.00€5mg161.00€1mL*10mM (DMSO)172.00€10mg235.00€25mg423.00€50mg627.00€100mg803.00€Butaprost
CAS:Butaprost: EP2 receptor agonist, EC50=33 nM, Ki=2.4 μM (murine), reduces fibrosis via TGF-β/Smad2.Formula:C24H40O5Purity:98%Color and Shape:SolidMolecular weight:408.57MALT1-IN-11
CAS:MALT1-IN-11: MALT1 inhibitor, IC50 <10-100 nM, reduces IL10, for cancer/autoimmune research.Formula:C20H16F4N8OColor and Shape:SolidMolecular weight:460.39α-Glucosidase-IN-18
α-Glucosidase-IN-18 (7B) is an orally active inhibitor of α-glucosidase, displaying an IC 50 value of 3.96 μM.Formula:C23H19NO2SColor and Shape:SolidMolecular weight:373.47Fusarisetin A
CAS:Fusarisetin A, a pentacyclic fungal metabolite, is an acinar morphogenesis inhibitor .Formula:C22H31NO5Color and Shape:SolidMolecular weight:389.49MDL-100173
CAS:MDL-100173 is a dual angiotensin-converting enzyme (ACE)/neutral endopeptidase (NEP) inhibitor.Formula:C24H26N2O4SColor and Shape:SolidMolecular weight:438.54CCR7 Ligand 1
CAS:CCR7-Cmp2105 is a thiadiazole-dioxide allosteric antagonist for CCR7 with a Kd of 3 nM and IC50 of 7.3 μM against arrestin binding.Formula:C22H29N5O5SColor and Shape:SolidMolecular weight:475.56Top/HDAC-IN-1
Top/HDAC-IN-1: Dual Top/HDAC inhibitor, potent against HDAC1-3,6,8 and HCT116 cells; blocks G2 phase, induces apoptosis.Formula:C29H27N5O4Color and Shape:SolidMolecular weight:509.56ALK5-IN-7
CAS:ALK5-IN-7 inhibits ALK5, useful in TGF-β disease research like cancer, fibrosis, and autoimmune disorders. See WO2021129621A1.Formula:C26H28N4O3SColor and Shape:SolidMolecular weight:476.59FAK-IN-4
FAK-IN-4 (Compound 7d) has anticancer activities that can induce cell apoptosis. FAK-IN-4 is potential inhibitor of FAK [1].Formula:C20H22N4OColor and Shape:SolidMolecular weight:334.41(R)-ONO-2952
(R)-ONO-2952 is the R-enantiomer of ONO-2952. ONO-2952 is selective and oral effective TSPO antagonist, with Kis of 0.330-9.30 nM inhibiting rat and human TSPO.Formula:C22H20ClFN2O2Color and Shape:SolidMolecular weight:398.86Nolpitantium Free Base
CAS:Nolpitantium is a potent, selective NK1 receptor antagonist that inhibits substance P without affecting NK2/NK3 receptors.Formula:C37H45Cl2N2O2Color and Shape:SolidMolecular weight:620.67CDK4-IN-1
CAS:CDK4 inhibitor is a novel and specific CDK4/Cyclin D1 inhibitor with an IC50 of 10 nM; 1500 and 500 fold than CDK1/Cyclin B (IC50>15 uM) and CDK2/Cyclin A (IC50Formula:C22H29ClN8Purity:98%Color and Shape:SolidMolecular weight:440.97Pateamine A
CAS:Pateamine A: marine-sourced macrolide from Mycale hentscheli; anticancer, antiviral, and translation inhibitor.Formula:C31H45N3O4SColor and Shape:SolidMolecular weight:555.77ATUX-1215
CAS:ATUX-1215, a protein phosphatase 2A (PP2A) activator, diminishes the phosphorylation of ERK, p38, JNK, and Akt, as well as decreases the secretion of IL-12p70,Formula:C27H24F5NO4SColor and Shape:SolidMolecular weight:553.54UAWJ9-36-1
CAS:UAWJ9-36-1: potent broad-spectrum coronavirus Protease inhibitor; IC50 = 51 nM.Formula:C23H29N3O5Color and Shape:SolidMolecular weight:427.49MGAT2-IN-1
CAS:MGAT2-IN-1 is an orally active monoacylglycerol acyltransferase (MGAT2)inhibitor (human and mouse MGAT2 with IC50 of 7.8 and 2.4 nM , respectively).Formula:C27H21ClF5N7O3SColor and Shape:SolidMolecular weight:654.01PAD-IN-2
CAS:PAD-IN-2, potent PAD4 inhibitor, IC50 <1 μM; targets autoimmune/cancer disorders.Formula:C27H28ClN5O2Color and Shape:SolidMolecular weight:490GLS1 Inhibitor-6
GLS1 Inhibitor-6: IC50=68nM, 220x more selective for GLS2, has anti-tumor and pro-apoptosis effects.Formula:C37H52N6O3SColor and Shape:SolidMolecular weight:660.91Org-31710
CAS:Org-31710 is a progesterone receptor antagonist potentially for contraception.Formula:C30H39NO2Purity:98%Color and Shape:SolidMolecular weight:445.64MB-7133
CAS:MB-7133 is an inhibitor of DNA synthesis.Formula:C17H21N4O8PPurity:98%Color and Shape:SolidMolecular weight:440.34KRAS G12C inhibitor 20
CAS:KRAS G12C inhibitor 20 is a KRAS G12C inhibitor.Formula:C33H37ClFN7O3Color and Shape:SolidMolecular weight:634.14S100A2-p53-IN-1
CAS:S100A2-p53-IN-1 inhibits S100A2-p53 in pancreatic cancer, stunting MiaPaCa-2 cell growth at 1.2-3.4 μM.Formula:C20H20F6N2O4SColor and Shape:SolidMolecular weight:498.44CEP-2563
CAS:CEP-2563 is a prodrug of CEP-751. It also used as an antitumor agent, inhibiting protein kinases.Formula:C36H41ClN6O6Purity:98%Color and Shape:SolidMolecular weight:689.20Teoprolol
CAS:Teoprolol is a blocker of β-adrenergic receptor.Formula:C23H30N6O4Purity:98%Color and Shape:SolidMolecular weight:454.52EGFR-IN-58
EGFR-IN-58 is a potent, selective, ATP-competitive inhibitor of EGFR. EGFR-IN-58 exhibits significant cytotoxicity against melanoma, colon and blood cancers.Formula:C31H30FN7OColor and Shape:SolidMolecular weight:535.61Antibacterial agent 62
Novel anti-TB agent 62 is a redox compound with bactericidal activity against active and dormant bacteria.Formula:C24H33BrN2O2Color and Shape:SolidMolecular weight:461.44RXR antagonist 2
RXR antagonist 2 is a potent antagonist of RXR (Ki: 0.391 μM, Kd: 0.281 μM). RXR antagonist 2 has shown research potential for RXR-related diseases.Formula:C29H35F3N2O3Color and Shape:SolidMolecular weight:516.6Antibacterial agent 76
Antibacterial agent 76 (compound 9) is a potent antibacterial agent.Formula:C23H27N3O2SColor and Shape:SolidMolecular weight:409.54Uprosertib hydrochloride
CAS:Uprosertib hydrochloride is a potent and selective inhibitor of pan-Akt (IC50: 180/328/38 nM for Akt1/Akt2/Akt3, respectively).Formula:C18H17Cl3F2N4O2Purity:98%Color and Shape:SolidMolecular weight:465.71PI3K-IN-35
CAS:PI3K-IN-35 (6l) selectively inhibits PI3K-α, β, δ (IC50: 13.98, 7.22, 10.94 μM), blocks G2/M phase, induces apoptosis, and is useful in leukemia research.Formula:C25H23N7O2Color and Shape:SolidMolecular weight:453.5Aurora inhibitor 1
CAS:Aurora inhibitor 1 is a potent Aurora inhibitor (IC50: ≤ 4 nM and ≤13 nM for Aurora A and Aurora B kinase).Formula:C23H25N9SPurity:98%Color and Shape:SolidMolecular weight:459.57Tubulin inhibitor 19
Tubulin inhibitor 19 (9b), a potent indole chalcone, strongly blocks tubulin, valuable in cancer studies.Formula:C21H23NO5Color and Shape:SolidMolecular weight:369.41Gusperimus
CAS:Gusperimus was synthesized by chemical modification of spergualin and in combination with cyclosporine A to prevent diabetes in susceptible NOD mice.Formula:C17H37N7O3Color and Shape:SolidMolecular weight:387.52TSWV-IN-1
TSWV-IN-1 is an anti-TSWV drug with potential TSWV N.Formula:C26H31FO4S2Color and Shape:SolidMolecular weight:490.65Tzc 5665
CAS:Tzc 5665 is a pyridazinone derivative with vasodilatory and beta-adrenergic blocking activities and type III phosphodiesterase inhibitory action.Formula:C31H38ClN5O7Color and Shape:SolidMolecular weight:628.12Rodatristat
CAS:Rodatristat is an effective tryptophan hydroxylase 1 and TPH2 inhibitor (IC50s: 33 nM and 7 nM, respectively).Formula:C27H27ClF3N5O3Purity:98%Color and Shape:SolidMolecular weight:561.98Protopine hydrochloride
CAS:Protopine inhibits thromboxane, lowers intracellular calcium, and reduces cell adhesion by altering adhesive factors.Formula:C20H20ClNO5Purity:98%Color and Shape:Prisms From Alc SolidMolecular weight:389.83Monoamine oxidase/Aromatase-IN-1
Compound 2q: Dual MAO/aromatase inhibitor; IC50: 39 nM (MAO-B), 31 nM (aromatase). Useful in neurological/breast cancer research.Formula:C19H19N3O3SColor and Shape:SolidMolecular weight:369.44TIM-3-IN-1
TIM-3-IN-1 is a useful tool to enable further studies on the biology of TIM-3 immunoregulation in cancer.Formula:C20H16ClN7O3SColor and Shape:SolidMolecular weight:469.9Leustroducsin B
CAS:Leustroducsin B is a novel colony-stimulating factor (CSF) inducer extracted from Streptomyces platensis SANK 60191.Formula:C34H56NO10PColor and Shape:SolidMolecular weight:669.78LP 12 hydrochloride hydrate
LP 12 hydrochloride hydrate: potent, selective 5-HT7 agonist (Ki: 0.13 nM); less affinity for D2, 5-HT1A/2A receptors.Formula:C32H39N3O·HCl·xH2OColor and Shape:SolidMDL-43291
CAS:MDL-43291 is a leukotriene receptor antagonist.Formula:C25H42O4SColor and Shape:SolidMolecular weight:438.66LY367385 hydrochloride
CAS:LY367385 hydrochloride: selective mGluR1a antagonist, IC50 = 8.8 μM, neuroprotective, anticonvulsant, antiepileptic.Formula:C10H12ClNO4Color and Shape:SolidMolecular weight:245.66C5aR-IN-3
CAS:C5aR-IN-3, a potent C5aR inhibitor, may treat autoimmune and inflammatory diseases.Formula:C36H40FN5O3Color and Shape:SolidMolecular weight:609.73
