Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,785 products)
- Apoptosis(6,253 products)
- Cell Cycle/Checkpoint(4,833 products)
- Chromatin/Epigenetics(2,588 products)
- Cytoskeletal Signaling(1,532 products)
- DNA Damage/DNA Repair(2,883 products)
- Endocrinology/Hormones(3,747 products)
- Enzyme(3,670 products)
- GPCR/G-Protein(8,977 products)
- Immunology and Inflammation(3,777 products)
- Influenza Virus(299 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,248 products)
- Membrane Transporter/Ion Channel(3,147 products)
- Metabolism(10,143 products)
- Microbiology/Virology(7,585 products)
- Neuroscience(10,341 products)
- Other Inhibitors(35,820 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,413 products)
- Proteases/Proteasome(1,680 products)
- Stem Cell and Derivatives(747 products)
- Tyrosine Kinase/Adaptors(1,948 products)
- Ubiquitination(1,719 products)
Show 16 more subcategories
Found 66565 products of "Inhibitors"
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PqsR-IN-1
PqsR-IN-1, potent PqsR inhibitor, curbs pyocyanin in Pseudomonas aeruginosa with low cytotoxicity.Formula:C17H18ClN3OSColor and Shape:SolidMolecular weight:347.86SHP2-IN-9
SHP2-IN-9: Potent SHP2 inhibitor, IC50=1.174 μM, 85x SHP1 selectivity, crosses blood-brain barrier, hampers cancer growth.Formula:C20H20FN3O2SColor and Shape:SolidMolecular weight:385.46Saprisartan potassium
CAS:Saprisartan potassium is an Angiotensin II Type 1 receptor antagonist and antihypertensive agent.Formula:C25H21BrF3KN4O4SColor and Shape:SolidMolecular weight:649.52Oral antiplatelet agent 1
CAS:Oral antiplatelet agent 1 is a potent antiplatelet agent with an IC50 of 2.94 μM in vitro.Formula:C23H24N4O5SPurity:98%Color and Shape:SolidMolecular weight:468.5320S Proteasome-IN-4
CAS:20S Proteasome-IN-4: brain-penetrant, parasite-specific, oral, inhibits T.b. brucei proteasome (IC50: 6.3nM), for HAT research.Formula:C20H18ClF2N3O3Color and Shape:SolidMolecular weight:421.83Mt KARI-IN-1
Mt KARI-IN-1 inhibits Mtb KARI with a 3.06 μM Ki, targeting tuberculosis.Formula:C14H11N5O4S2Color and Shape:SolidMolecular weight:377.4PTP1B-IN-21
PTP1B-IN-21 inhibits PTP1B (IC50=1.56μM) selectively over TCPTP, a type 2 diabetes target.Formula:C22H22O11Color and Shape:SolidMolecular weight:462.4Oncopterin
CAS:Oncopterin is found in urine from patients with solid and blood cancers.Formula:C12H18N6O3Color and Shape:SolidMolecular weight:294.31Anticancer agent 26
Anticancer agent 26 is a promising candidate for cancer therapy and deserves further development.Formula:C28H33NO5Color and Shape:SolidMolecular weight:463.57CYP1B1-IN-2
CYP1B1-IN-2 (compound 9j) is a highly potent and selective inhibitor of CYP1B1, a cytochrome P450 enzyme. It exhibits an IC50 value of 0.52 nM [1].Formula:C20H11F3O2Color and Shape:SolidMolecular weight:340.3TA-316
CAS:Agent induces megakaryocytes/platelets from stem cells to treat thrombopenia.Formula:C28H25BrN4O5S2Purity:98%Color and Shape:SolidMolecular weight:641.56Trilobolide
CAS:Trilobolide is a natural counterpart of thapsigargin and an activator of cytokine secretion.Formula:C27H38O10Color and Shape:SolidMolecular weight:522.58Orvepitant
CAS:Orvepitant is a potent and selective NK1 antagonist, which may be potentially useful for patients with major depressive disorder (MDD), anxiety and insomnia.Formula:C31H35F7N4O2Color and Shape:SolidMolecular weight:628.62GC 14
CAS:GC 14 is a selective thyroid hormone receptor antagonist, with IC50 values of 200 nM and 35 nM for hTRα and hTRβ, respectively.Formula:C26H27NO6Purity:98%Color and Shape:SolidMolecular weight:449.5Carnostatine
Carnostatine (SAN9812), a potent CN1 inhibitor with 11 nM K i, may boost renal carnosine to treat DN.Formula:C10H16N4O4Purity:98%Color and Shape:SolidMolecular weight:256.26ACT-777991
CAS:ACT-777991: oral CXCR3 blocker, stable in microsomes/hepatocytes, inhibits T-cell migration to CXCL11.Formula:C20H20F6N8O2SColor and Shape:SolidMolecular weight:550.48ART615
ART615 is a related isomer of ART558. ART615 inhibits Polθ by <10% at 12 μM and is able to act as a control for ART558 (IC50:7.9 nM).Formula:C21H21F3N4O2Color and Shape:SolidMolecular weight:418.41Cdc7-IN-10
CAS:Cdc7-IN-10 is a potent inhibitor of Cdc7 (IC50 ≤ 1 nM) and can be used in studies of proliferative diseases.Formula:C20H22F2N4O2SColor and Shape:SolidMolecular weight:420.48Cap-dependent endonuclease-IN-5
CAS:Cap-dependent endonuclease-IN-5 inhibits CEN and fights influenza with low toxicity and good in vivo properties.Formula:C27H21F2N3O4S2Color and Shape:SolidMolecular weight:553.60Ornoprostil
CAS:Ornoprostil, a prostaglandin E1 analogue, acts as a mucosal protectant.Formula:C23H38O6Purity:98%Color and Shape:SolidMolecular weight:410.54CI 992
CAS:CI 992 is a novel potent inhibitor of primate renin.Formula:C33H52N6O7S2Color and Shape:SolidMolecular weight:708.93FGFR4-IN-6
FGFR4-IN-6: covalent, reversible FGFR4 blocker, 5.4 nM IC50, good oral bioavailability, reduces Hep3B2.1-7 tumors in mice, low toxicity.Formula:C31H33N7O4Color and Shape:SolidMolecular weight:567.64MM-589 TFA
CAS:MM-589 TFA is a potent WD repeat domain 5 (WDR5)inhibitor and mixed lineage leukemia (MLL) protein-protein interaction.Formula:C30H45F3N8O7Purity:98%Color and Shape:SolidMolecular weight:686.72SSR-182289A (Free)
CAS:SSR-182289A (Free) is a thrombin inhibitor.Formula:C30H33F2N5O4SPurity:98%Color and Shape:SolidMolecular weight:597.68VEGFR-2-IN-18
VEGFR-2-IN-18 is a potent VEGFR-2 inhibitor with a 60 nM IC50, promoting cell apoptosis and anticancer effects.Formula:C20H13ClN4O2Color and Shape:SolidMolecular weight:376.8S-8510 phosphate
CAS:S-8510 phosphate is an agonist of inverse Benzodiazepine (BDZ) receptor(Kis of 34.6 nM, 36.2 nM for –GABA and +GABA respectively).Formula:C12H13N4O6PPurity:98%Color and Shape:SolidMolecular weight:340.23Namitecan
CAS:Namitecan is an effective inhibitor of topoisomerase I. It has antitumor property.Formula:C23H22N4O5Purity:98%Color and Shape:SolidMolecular weight:434.44BRL-42715
CAS:BRL-42715 is an effective inhibitor of bacterial beta-lactamases.Formula:C10H7N4NaO3SPurity:98%Color and Shape:SolidMolecular weight:286.24HDAC6-IN-12
HDAC6-IN-12 is a potent inhibitor of HDAC6 that binds in the DNA chain, causing DNA damage and exhibiting anticancer effects that can be used in cancer researchFormula:C24H39F2N3O5Color and Shape:SolidMolecular weight:487.58TD-0212
CAS:TD-0212: Oral dual antagonist for AT1 (pKi 8.9) & NEP inhibitor (pIC50 9.2).Formula:C28H34FN3O4SPurity:98%Color and Shape:SolidMolecular weight:527.65FGFR3-IN-4
CAS:FGFR3-IN-4 is a selective inhibitor targeting FGFR3, demonstrating an IC50 value of under 50 nM.Formula:C26H24ClN7OColor and Shape:SolidMolecular weight:485.97RMS5
CAS:RMS5: hambanine analogue, inhibits P-gp, anti-cancer with cytotoxic, anti-proliferative effects, reduces Bcl-2 proteins, cleaves PARP.Formula:C35H38N2O5SColor and Shape:SolidMolecular weight:598.75Tribenuron
CAS:Tribenuron, a slow acting sulfonylurea herbicide, controls broadleaf weed.Formula:C14H15N5O6SColor and Shape:SolidMolecular weight:381.36BTK inhibitor 18
BTK inhibitor 18 is a selective, potent, covalent, orally active Btk inhibitor (IC50: 142 nM) that exhibits anti-inflammatory effects.Formula:C29H25N5O4S2Color and Shape:SolidMolecular weight:571.67MAP855
CAS:MAP855: potent, selective, oral MEK1/2 inhibitor; IC50=3 nM, pERKEC50=5 nM; effective on wild-type/mutant MEK1/2.Formula:C28H23ClF2N6O3Color and Shape:SolidMolecular weight:564.97Sucistil
Sucistil is an active biochemical. hemoglobin sucistil (bovine) is an oxygen carrier [1].Formula:C9H15NO4SColor and Shape:SolidMolecular weight:233.28AMG-369
CAS:AMG-369 (AMG 247) is an S1P1/S1P5 dual agonist that delays the development of experimental autoimmune encephalomyelitis in rats.Formula:C26H22FN3O2SPurity:98.04% - 98.92%Color and Shape:SolidMolecular weight:459.54Macropa-NCS
CAS:Macropa-NCS is a macropa bifunctional analog with antitumor activity and can be used to study prostate cancer.Formula:C27H35N5O8SPurity:98%Color and Shape:SolidMolecular weight:589.66SX 3202
CAS:SX 3202 is an aldose reductase inhibitor being developed for the treatment of diabetic neuropathy.Formula:C17H11BrFN3O4Color and Shape:SolidMolecular weight:420.19Anticancer agent 142
CAS:Compound 142 (also known as Compound 235) is a PTPN inhibitor with potential applications in cancer research [1].Formula:C13H14BrF2N2O7PS2Purity:98%Color and Shape:SolidMolecular weight:523.26α-Amylase-IN-1
CAS:α-Amylase-IN-1 is an α-Amylase inhibitor (IC50: 0.5509 μM).Formula:C18H18N2O3Purity:99.92%Color and Shape:SoildMolecular weight:310.35HSV-TK substrate
CAS:HSV-TK substrate is a substrate for HSV-TK with antitumor activity. It induces multi-log cytotoxicity in HSV-TK-expressing and bystander cells.Formula:C11H15N5O4Purity:98%Color and Shape:SolidMolecular weight:281.27DC41SMe
CAS:DC41SMe, a DC1 derivative and CC-1065 analogue, targets cancer with 18-25 pM IC50 against Ramos, Namalwa, HL60/s cells.Formula:C38H36ClN5O4S2Purity:98%Color and Shape:SolidMolecular weight:726.31DS-9300
CAS:DS-9300, an orally administered potent and selective inhibitor of EP300/CBP HAT, exhibits a significant inhibitory activity with an IC50 value of 28 nM.Formula:C25H26F3N5O3Color and Shape:SolidMolecular weight:501.50ZK118182 isopropyl ester
CAS:ZK118182 isopropyl ester is a PG analog with potent DP-agonist activity (EC50 = 16.5 nM) and high affinity for the DP receptor (Ki = 74 nM).Formula:C23H37ClO5Purity:98%Color and Shape:SolidMolecular weight:428.99MA242 free base
CAS:MA242 free base is a dual MDM2/NFAT1 inhibitor that triggers apoptosis in pancreatic cancer cells.Formula:C24H20ClN3O3SColor and Shape:SolidMolecular weight:465.95CYP2C9/CYP2C19-IN-1
CYP2C9/CYP2C19-IN-1 is a potent inhibitor of CYP2C9/CYP2C19 without liver toxicity or genotoxicity and can be used to study Zika virus (ZIKV) infection.Formula:C27H28N2O6SColor and Shape:SolidMolecular weight:508.59HIV-1 inhibitor-52
CAS:HIV-1 inhibitor-52: potent, broad-spectrum with EC50s 1.6-6.4 nM against various HIV-1 strains.Formula:C46H72FNO5SColor and Shape:SolidMolecular weight:770.13Glutamate-5-kinase-IN-1
Glutamate-5-kinase-IN-1 is a potent G5K inhibitor with a 4.1 μM MIC, showing promise in anti-TB research.Formula:C20H18N2OColor and Shape:SolidMolecular weight:302.37CDK4/6-IN-13
CAS:Compounds 10B and 10C: potent cdk4/6 inhibitors with low nM activity, great antiproliferative effects, excellent metabolism, and good pharmacokinetics.Formula:C25H29N7OColor and Shape:SolidMolecular weight:443.54
