Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,787 products)
- Apoptosis(6,257 products)
- Cell Cycle/Checkpoint(4,835 products)
- Chromatin/Epigenetics(2,591 products)
- Cytoskeletal Signaling(1,534 products)
- DNA Damage/DNA Repair(2,880 products)
- Endocrinology/Hormones(3,748 products)
- Enzyme(3,670 products)
- GPCR/G-Protein(8,978 products)
- Immunology and Inflammation(3,782 products)
- Influenza Virus(299 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,249 products)
- Membrane Transporter/Ion Channel(3,148 products)
- Metabolism(10,142 products)
- Microbiology/Virology(7,590 products)
- Neuroscience(10,343 products)
- Other Inhibitors(35,823 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,414 products)
- Proteases/Proteasome(1,680 products)
- Stem Cell and Derivatives(746 products)
- Tyrosine Kinase/Adaptors(1,950 products)
- Ubiquitination(1,719 products)
Show 16 more subcategories
Found 66564 products of "Inhibitors"
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TLR4/NF-κB/MAPK-IN-1
CAS:TLR4/NF-κB/MAPK-IN-1 is a novel antineuroinflammatory agent that functions by inhibiting the TLR4/NF-κB/MAPK pathways.Formula:C19H25BrO6Color and Shape:SolidMolecular weight:429.3FT3967385
FT3967385: New USP30 inhibitor boosts mitochondrial ubiquitylation via PINK1-PARKIN.Formula:C21H19N5O2Color and Shape:SolidMolecular weight:373.41Pulvomycin
CAS:Pulvomycin is a protein biosynthesis inhibitor preventing ternary complex formation between elongation factor Tu, GTP, and aminoacyl-tRNA.Formula:C47H66O13Purity:98%Color and Shape:SolidMolecular weight:839.032Protease-Activated Receptor-1 antagonist 1
Compound 13 is a PAR-1 antagonist with a 3 nM IC50, useful for thrombosis and heart disease research.Formula:C25H24F2N2O3Color and Shape:SolidMolecular weight:438.47PPARγ agonist 1
PPARγ agonist 1 is a potent agonist of PPARγ that efficiently activates hPPARγ without causing full agonism, thereby avoiding adverse effects.Formula:C34H39NO3Color and Shape:SolidMolecular weight:509.68AD012
AD012, a dual cACE/NEP inhibitor, leverages lenopril-tryptophan for potential anti-hypertensive and cardioprotective benefits.Formula:C25H32N2O6Color and Shape:SolidMolecular weight:456.53NNC-11-1585
CAS:NNC-11-1585 is an M(1) and M(2) muscarinic acetylcholine receptor (mAChR) agonist.Formula:C18H19N3OSColor and Shape:SolidMolecular weight:325.43Dot1L-IN-1
CAS:The Ki value of DOT1L-in-1 is 2pm.It is a highly effective, selective and novel Dot1L inhibitor.Formula:C32H36ClN9O2SPurity:98%Color and Shape:SolidMolecular weight:646.21Antifungal agent 39
CAS:Antifungal agent 39 (Compound 9h) is a broad-spectrum antifungal agent.Formula:C23H22ClN3O5Color and Shape:SolidMolecular weight:455.89MEK4 inhibitor-2
CAS:MEK4 Inhibitor-2, a novel MEK4 inhibitor, demonstrates efficacy against pancreatic adenocarcinoma, exhibiting an IC50 value of 83 nM.Formula:C20H15FN4O3SColor and Shape:SolidMolecular weight:410.42Udifitimod
CAS:Udifitimod (BMS-986166) is a potent, selective, and orally active modulator of the S1P1R receptor, showing potential for research in autoimmune diseases.Formula:C25H33NO2Color and Shape:SolidMolecular weight:379.54KRAS G12C inhibitor 37
CAS:KRAS G12C inhibitor 37 targets a key signaling protein, showing promise for cancer research involving KRAS G12C.Formula:C35H39F3N8O2Color and Shape:SolidMolecular weight:660.73T-3764518
CAS:T-3764518 is a novel and potent inhibitor of stearoyl coenzyme A desaturase (SCD)(IC50 of 4.7 nM).Formula:C20H17F6N5O2Purity:98%Color and Shape:SolidMolecular weight:473.37RU 52583
CAS:RU 52583 is an alpha 2-adrenergic receptor antagonist.Formula:C18H20N2Purity:98%Color and Shape:SolidMolecular weight:264.36RAD51-IN-8
RAD51-IN-8 inhibits RAD51-BRCA2 interaction and H4A4 with EC50 of 19 μM; a micromolar PPI inhibitor.Formula:C16H14Cl2FN3O2Color and Shape:SolidMolecular weight:370.21NR1H4 activator 1
CAS:NR1H4 activator 1 is a potent and selective agonist of Famesoid X Receptor (FXR).Formula:C34H53NO7SPurity:98%Color and Shape:SolidMolecular weight:619.85RSV-IN-5
CAS:RSV-IN-5: Dual inhibitor for RSV fusion proteins, effective on wild-type A2 and D486N mutant with EC50s of 2.0 nM & 8.1 nM. Potent anti-RSV.Formula:C28H37N7O2Color and Shape:SolidMolecular weight:503.64TAI-95
CAS:TAI-95 is an inhibitor of highly expressed cancer protein 1 (Hec1).Formula:C24H23N5O3S2Color and Shape:SolidMolecular weight:493.60Trypanothione synthetase-IN-4
Trypanothione synthetase-IN-4, an L. infantum inhibitor, has potent anti-leishmanicidal properties (EC50: 0.6 μM).Formula:C29H52INO2Color and Shape:SolidMolecular weight:573.63Anticancer agent 142
CAS:Compound 142 (also known as Compound 235) is a PTPN inhibitor with potential applications in cancer research [1].Formula:C13H14BrF2N2O7PS2Purity:98%Color and Shape:SolidMolecular weight:523.26DGY-08-097
CAS:DGY-08-097: potent HCV NS3 degrader, low resistance risk, strong inhibition in cells, DC50 of 50nM at 4h.Formula:C60H76N10O14Color and Shape:SolidMolecular weight:1161.3MCTR3
CAS:MCTR3, derived from DHA via maresin 1 in macrophages, hastens tissue healing and reduces inflammation and eicosanoids post-E. coli infection in mice.Formula:C25H37NO5SColor and Shape:SolidMolecular weight:463.63Fabimycin
CAS:Fabimycin, a FabI inhibitor, combats drug-resistant gram-negative bacterial infections effectively.Formula:C23H25ClN4O3Color and Shape:SolidMolecular weight:440.92Ceclazepide
CAS:Ceclazepide is an antagonist of cholecystokinin receptor.Formula:C30H32N6O5Purity:98%Color and Shape:SolidMolecular weight:556.61RXR antagonist 1
RXR antagonist 1 is a Retinoid X Receptor (RXR) modulator that exhibits high RXR antagonism (pA2: 8.06). RXR antagonist 1 can be used to study type 2 diabetes.Formula:C28H33F3N2O3Color and Shape:SolidMolecular weight:502.57E-3030 free acid
CAS:E-3030 free acid, a PPAR agonist, lowers blood glucose, triglycerides, and insulin; boosts adiponectin; reduces apo C-III; and raises lipoprotein lipase.Formula:C22H23ClFNO5Purity:98%Color and Shape:SolidMolecular weight:435.87FGFR4-IN-4
CAS:FGFR4-IN-4 is a FGFR4 inhibitor with anti-tumor activity.Formula:C28H32Cl2N6O5Purity:98%Color and Shape:SolidMolecular weight:603.5Flurdihydroergotamine
CAS:Flurdihydroergotamine, a serotonin 5HT1 receptor agonist, is used as an antimigraine drug.Formula:C34H36F3N5O5Purity:98%Color and Shape:SolidMolecular weight:651.68Neuraminidase-IN-7
Neuraminidase-IN-7, a thiophene, inhibits neuraminidase (IC50 0.03 μM), showing promise for flu research.Formula:C21H20N2O6SColor and Shape:SolidMolecular weight:428.46ORP-101
CAS:ORP-101: large, stable molecule with partial μ agonist, full κ antagonist properties.Formula:C60H84N2O8Color and Shape:SolidMolecular weight:961.32RSK4-IN-1
CAS:RSK4-IN-1 is a compound exhibiting potent inhibition of RSK4, demonstrated by an IC50 value of 9.5 nM.Formula:C19H20F2N4O3Color and Shape:SolidMolecular weight:390.38D4R antagonist-1
Potent, selective D4R antagonist; IC50 = 6.87 µM; potential in Parkinson’s disease research.Formula:C21H25F2NO2Color and Shape:SolidMolecular weight:361.43Anti-inflammatory agent 12
Pentacyclic triterpene, anti-inflammatory agent 12, inhibits LPS inflammation (IC50: 2.22 μM). May benefit inflammatory disease studies.Formula:C30H50O4Color and Shape:SolidMolecular weight:474.72YCW-E11
CAS:YCW-E11 is an antiapoptotic Bcl-2 family proteins inhibitor.Formula:C25H21Cl2N3O6S2Purity:98%Color and Shape:SolidMolecular weight:594.49BAY-364
CAS:BAY-364 (BAY-299N) functions as an inhibitor targeting the second bromine domain in TAF1, demonstrating inhibitory effects on TAF1 in Kasumi-1 cells, CD34+Formula:C23H19N3O4Color and Shape:SolidMolecular weight:401.41AL-6556
CAS:AL-6556 is a prostaglandin DP receptor agonist.Formula:C20H33ClO5Color and Shape:SolidMolecular weight:388.93HIV-1 inhibitor-41
HIV-1 inhibitor-41 (B23): Oral non-nucleoside reverse transcriptase blocker, EC50 of 50 nM (E138K), 20.8 nM (WT), low hERG/CYP impact, non-toxic.Formula:C16H15F2N3OSColor and Shape:SolidMolecular weight:335.37Zetomipzomib
CAS:KZR-616: Immunoproteasome inhibitor targeting LMP7 (IC50: 39/57 nM) & LMP2 (IC50: 131/179 nM), potential in autoimmune disease research.Formula:C30H42N4O8Color and Shape:SolidMolecular weight:586.68Clavicoronic acid
CAS:Clavicoronic acid, a β-lactamase inhibitor, boosts penicillin antibiotics against resistant bacteria.Formula:C15H18O4Color and Shape:SolidMolecular weight:262.3LSD1/ER-IN-1
LSD1/ER-IN-1 inhibits ER & LSD1 (IC50: 1.55 μM), and fights MCF-7 breast cancer (IC50: 8.79 μM).Formula:C23H18FNO6SColor and Shape:SolidMolecular weight:455.46Belatacept
CAS:Belatacept (BMS 224818), a T-cell costimulation inhibitor, targets CD80/86 for transplant immunosuppression.Color and Shape:LiquidL-Afegostat
CAS:L-Afegostat (5-epi-Isofagomine), an iminosugar, inhibits glycosidase and β-Glucosidase (K i 30 μM), aids in carbohydrate synthesis.Formula:C6H13NO3Color and Shape:SolidMolecular weight:147.17Dehydrocrenatidine
CAS:Dehydrocrenatidine (Kumujian G) is an inhibitor of JAK and induces cell apoptosis.Formula:C15H14N2O2Purity:98%Color and Shape:SolidMolecular weight:254.28Galidesivir
CAS:Galidesivir (BCX4430) is an antiviral compound that inhibits viral RNA-dependent RNA polymerase (RdRp) activity and reduces lung infections in infected animals.Formula:C11H15N5O3Purity:96.73% - 99.13%Color and Shape:SolidMolecular weight:265.27CDK4/6-IN-3
CAS:CDK4/6-IN-3 is a brain-penetrant CDK4/CDK6 inhibitor (Kis: <0.3 nM and 2.2 nM) used for the treatment of glioblastoma. It inhibits CDK1 with a Ki of 110 nM.Formula:C25H31FN8Purity:98%Color and Shape:SolidMolecular weight:462.57KRAS G12C inhibitor 33
CAS:KRAS G12C inhibitor 33 is a KRAS G12C inhibitor that can be used to study cancer.Formula:C30H33N7O3Color and Shape:SolidMolecular weight:539.63Antitumor agent-51
Antitumor agent-51 targets osteosarcoma with 21.9 nM IC50, high selectivity, and low toxicity.Formula:C23H25N5O2SColor and Shape:SolidMolecular weight:435.54PD 140376
CAS:PD 140376: Selective CCK-B/gastrin receptor antagonist radioligand for guinea pig stomach & brain.Formula:C33H40N4O5Purity:98%Color and Shape:SolidMolecular weight:572.69Rostratin A
CAS:Rostratin A, a disulfide from Exserohilum rostratum, is cytotoxic to HCT-116 cells with an IC50 of 8.5 μg/mL.Formula:C18H24N2O6S2Color and Shape:SolidMolecular weight:428.52
