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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66627 products of "Inhibitors"

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  • WZ4002

    CAS:
    <p>WZ4002 is a mutant-selective EGFR inhibitor for EGFR(L858R) and EGFR(T790M) with IC50 of 2 nM/8 nM.</p>
    Formula:C25H27ClN6O3
    Purity:97.51%
    Color and Shape:Solid
    Molecular weight:494.97
  • AG-120 (racemic)

    CAS:
    <p>AG-120 (racemic) is an oral IDH1 inhibitor with potential anti-cancer effects.</p>
    Formula:C28H22ClF3N6O3
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:582.96
  • RS-25344 hydrochloride

    CAS:
    <p>RS 25344 hydrochloride is a phosphodiesterase (PDE) 4 inhibitor</p>
    Formula:C19H14ClN5O4
    Purity:99.25%
    Color and Shape:Solid
    Molecular weight:411.8
  • Oxytocin C-terminal tripeptide Acetate


    <p>Oxytocin C-terminal tripeptide Acetate: a mammalian hormone's end segment, binds to oxytocin receptors.</p>
    Formula:C15H28N4O5
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:344.41
  • VE-821

    CAS:
    <p>VE-821 (ATR Inhibitor IV) is a selective ATP competitive inhibitor of ATR( Ki/IC50: 13/26 nM in cell-free assays).</p>
    Formula:C18H16N4O3S
    Purity:97.19% - 99.97%
    Color and Shape:Solid
    Molecular weight:368.41
  • MID-1

    CAS:
    <p>MID-1 is an inhibitor of MG53-IRS-1 (Mitsugumin 53-Insulin Receptor Substrate-1) interaction.</p>
    Formula:C12H11N3O4S
    Purity:99.39%
    Color and Shape:Solid
    Molecular weight:293.3
  • Gentiopicroside

    CAS:
    <p>Gentiopicroside, an iridoid from Gentiana manshurica, inhibits CYP2A6 (IC50=61μM, Ki=22.8μM), and has anti-inflammatory and antioxidant properties.</p>
    Formula:C16H20O9
    Purity:98% - 99.99%
    Color and Shape:White Powder
    Molecular weight:356.32
  • Kyotorphin acetate


    <p>Kyotorphin acetate is an endogenous peptide with analgesia activity and can be used as a biomarker of Alzheimer disease.</p>
    Formula:C17H27N5O6
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:397.43
  • CPI-455 analogue


    <p>CPI-455 analogue (CPI-455 analogue) is an analogue of CPI-455 which is a KDM5 inhibitor.</p>
    Formula:C16H14N4O
    Purity:98% - 98.13%
    Color and Shape:Solid
    Molecular weight:278.31
  • Cangrelor free acid

    CAS:
    <p>Cangrelor, a reversible P2Y12 inhibitor for IV use, was approved in June 2015; it rapidly blocks ADP-induced platelet aggregation.</p>
    Formula:C17H25Cl2F3N5O12P3S2
    Color and Shape:Solid
    Molecular weight:776.36
  • Niraparib hydrochloride

    CAS:
    <p>Niraparib hydrochloride (MK-4827) is a PARP inhibitor with potential cancer treatment effects, causing DNA damage and apoptosis.</p>
    Formula:C19H21ClN4O
    Purity:99.26%
    Color and Shape:Solid
    Molecular weight:356.85
  • Leuphasyl TFA

    CAS:
    <p>Leuphasyl TFA: a long-lasting, degradation-resistant peptide &amp; δ-opioid receptor agonist for signaling research.</p>
    Formula:C31H40F3N5O9
    Purity:98.79%
    Color and Shape:Solid
    Molecular weight:683.67
  • Delsoline

    CAS:
    <p>Delsoline reduces blood pressure, prevents arrhythmias, and increases fibrillation threshold in rabbits.</p>
    Formula:C25H41NO7
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:467.6
  • BMS-986242

    CAS:
    <p>BMS-986242 is an orally active, potent and selective inhibitor of indoleamine-2,3-dioxygenase 1 (IDO1), and it can be used for the research of cancer.</p>
    Formula:C24H24ClFN2O
    Purity:98.9%
    Color and Shape:Solid
    Molecular weight:410.91
  • Nardosinone

    CAS:
    <p>Nardosinone inhibits H9c2 cell hypertrophy, protects neurons from OGD, and boosts neurite outgrowth by modifying key signaling pathways.</p>
    Formula:C15H22O3
    Purity:98.82% - 99%
    Color and Shape:Solid
    Molecular weight:250.33
  • 8-Azaadenosine

    CAS:
    <p>8-Azaadenosine inhibits ADAR1, blocks RNA editing, and reduces thyroid cancer cell proliferation and spread.</p>
    Formula:C9H12N6O4
    Purity:99.39%
    Color and Shape:Solid
    Molecular weight:268.23
  • DS-7423

    CAS:
    <p>DS-7423: a dual PI3K/mTOR inhibitor; IC50s—PI3Kα: 15.6 nM, mTOR: 34.9 nM, PI3Kβ: 1,143 nM, PI3Kγ: 249 nM, PI3Kδ: 262 nM.</p>
    Formula:C22H27F3N10O2
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:520.51
  • KU-0060648

    CAS:
    <p>KU-0060648 is a dual inhibitor of DNA-PK and PI3Kα, PI3Kβ, PI3Kδ with IC50 of 8.6 nM and 4 nM, 0.5 nM, 0.1 nM respectively, less inhibition of PI3Kγ.</p>
    Formula:C33H34N4O4S
    Purity:98.75%
    Color and Shape:Solid
    Molecular weight:582.71
  • Oct3/4-inducer-1

    CAS:
    <p>Oct3/4-inducer-1 (2-(4-(4-methoxybenzyloxy)phenyl)acetonitrile) is an OCT3/4 inducer that promotes the expression and stabilization of OCT3/4.</p>
    Formula:C15H12FNO
    Purity:97.42% - ≥98%
    Color and Shape:Solid
    Molecular weight:241.26
  • Theaflavin-3'-Gallate

    CAS:
    <p>Theaflavin-3'-Gallate (Theaflavin 2B) usually comes from the leaves of Camellia sinensis (L.) O. Kuntze,which act as prooxidants and induce oxidative stress.</p>
    Formula:C36H28O16
    Purity:99.21% - 99.89%
    Color and Shape:Solid
    Molecular weight:716.6
  • NLS PKKKRKV acetate(95088-49-6 free base)


    <p>NLS PKKKRKV acetate, a peptide from SV40 big T antigen, boosts nuclear entry for gene transfer research.</p>
    Formula:C42H82N14O10
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:943.21
  • Vonafexor

    CAS:
    <p>Vonafexor (EYP001) is a farnesoid X receptor (FXR, NR1H4) agonist, with anti-HBV effects</p>
    Formula:C19H15Cl3N2O5S
    Purity:98.74%
    Color and Shape:Solid
    Molecular weight:489.76
  • TVB-3166

    CAS:
    <p>TVB-3166: reversible, selective FASN inhibitor, induces apoptosis, hinders xenograft growth (IC50: 42 nM FASN, 81 nM palmitate synthesis).</p>
    Formula:C24H24N4O
    Purity:99.53% - 99.57%
    Color and Shape:Solid
    Molecular weight:384.47
  • TH-263

    CAS:
    <p>TH-263 is inactive toward both LIMK1 and LIMK2 and thus can be used as negative control for TH-257, and is a diaryl sulfonamide derivative.</p>
    Formula:C21H20N2O3S
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:380.46
  • Mexiletine

    CAS:
    <p>Mexiletine is a non-selective voltage-gated sodium channel blocker.</p>
    Formula:C11H17NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:179.26
  • SU 5402

    CAS:
    <p>SU 5402 is a potent multi-targeted receptor tyrosine kinase inhibitor with IC50 of 20 nM, 30 nM, and 510 nM for VEGFR2, FGFR1, and PDGF-Rβ, respectively.</p>
    Formula:C17H16N2O3
    Purity:98.91% - 99.64%
    Color and Shape:Yellow-Green Solid
    Molecular weight:296.32
  • YM-750

    CAS:
    <p>YM-750 is a potent inhibitor of acyl-CoA:cholesterol acyltransferase (ACAT), with an IC50 value of 0.18 μM.</p>
    Formula:C31H36N2O
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:452.63
  • Disodium succinate

    CAS:
    <p>Disodium succinate is a sodium salt of succinate, key in metabolism and reactive oxygen species regulation.</p>
    Formula:C4H4Na2O4
    Purity:97.162%
    Color and Shape:White Solid Crystalline Powder
    Molecular weight:162.05
  • Darunavir Ethanolate

    CAS:
    <p>Darunavir Ethanolate (UIC 94017) is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS.</p>
    Formula:C29H43N3O8S
    Purity:99.84% - 99.86%
    Color and Shape:Solid
    Molecular weight:593.74
  • GSK805

    CAS:
    <p>GSK805 is a potent, orally bioavailable and CNS-penetrant RORγt inhibitor.Cost-effective and quality-assured.</p>
    Formula:C23H18Cl2F3NO4S
    Purity:98% - ≥95%
    Color and Shape:Solid
    Molecular weight:532.36
  • Deoxylapachol

    CAS:
    <p>Deoxylapachol combats wood rot, blocking Gloeophyllum spp., Merulius tremellosus, Phlebia brevispora, and induces fungal cell wall stress.</p>
    Formula:C15H14O2
    Purity:98.05%
    Color and Shape:Solid
    Molecular weight:226.27
  • Mitiglinide

    CAS:
    <p>Mitiglinide (KAD-1229), an insulinotropic ATP-sensitive K+ channel antagonist, targets Kir6.2/SUR1; used in type 2 diabetes research.</p>
    Formula:C19H25NO3
    Color and Shape:Solid
    Molecular weight:315.41
  • Gardenin B

    CAS:
    <p>Gardenin B exhibits superior antiproliferative activity against lung, breast, colon, hepatic and leukaemia cell lines as well as in keratinocytes .</p>
    Formula:C19H18O7
    Purity:98.80% - 99.74%
    Color and Shape:Solid
    Molecular weight:358.34
  • Phosphocreatine disodium

    CAS:
    <p>Phosphocreatine disodium: a phosphorylated creatine for quick energy storage in muscle and brain.</p>
    Formula:C4H8N3Na2O5P
    Purity:97.52% - 97.62%
    Color and Shape:White Powder
    Molecular weight:255.08
  • L-Cysteinesulfinic acid monohydrate

    CAS:
    <p>L-Cysteinesulfinic acid monohydrate activates rat mGluR1/2/4/5/6/8 with pEC50s of 3.92, 3.9, 2.7, 4.6, 4.0, 3.94 respectively.</p>
    Formula:C3H9NO5S
    Purity:≥98%
    Color and Shape:Solid
    Molecular weight:171.17
  • N4-benzyl-N2-methylquinazoline-2,4-diamine hydrochloride

    CAS:
    <p>N4-benzyl-N2-methylquinazoline-2,4-diamine hydrochloride is an inhibitor of TRPC4.</p>
    Formula:C16H17ClN4
    Purity:99.25%
    Color and Shape:Solid
    Molecular weight:300.79
  • Ginsenoside Rd

    CAS:
    <p>Ginsenoside Rd (Gypenoside VIII) may have properties that inhibit or prevent the growth of tumors.</p>
    Formula:C48H82O18
    Purity:99.13% - 99.92%
    Color and Shape:Solid
    Molecular weight:947.15
  • Acipimox sodium

    CAS:
    <p>Acipimox sodium is an antilipolytic, enhancing leptin, curbing lipolysis and FFAs, and boosting insulin sensitivity.</p>
    Formula:C6H5N2NaO3
    Color and Shape:Solid
    Molecular weight:176.11
  • Polymyxin B nonapeptide acetate


    <p>Polymyxin B nonapeptide acetate, a low toxicity derivative of polymyxin B, disrupts Gram-negative bacteria membranes.</p>
    Formula:C45H78N14O13
    Purity:97.63% - 98.55%
    Color and Shape:Solid
    Molecular weight:1023.19
  • TFMB-(R)-2-HG

    CAS:
    <p>TFMB-(R)-2-HG, a carcinogen in AML, hinders SCF ER-Hoxb8 differentiation after estrogen loss.</p>
    Formula:C13H11F3O4
    Purity:97.15%
    Color and Shape:Solid
    Molecular weight:288.22
  • SRT1720 hydrochloride

    CAS:
    <p>SRT1720 hydrochloride (SRT1720 HCl) is a selective activator of SIRT1 (EC1.5: 0.16 μM) and shows less potent activities on SIRT2/SIRT3 (EC1.5s: 37 μM/300 μM).</p>
    Formula:C25H24ClN7OS
    Purity:98% - 99.93%
    Color and Shape:Solid
    Molecular weight:506.22
  • NVP-TAE 684

    CAS:
    <p>NVP-TAE 684 (TAE684) is a excellently effective and specific ALK inhibitor(IC50=3 nM).</p>
    Formula:C30H40ClN7O3S
    Purity:98% - 99.82%
    Color and Shape:Solid
    Molecular weight:614.2
  • ARRY 520 hydrochloride

    CAS:
    <p>'ARRY 520 hydrochloride: a KSP inhibitor causing apoptosis and strong anti-proliferative effects.'</p>
    Formula:C20H23ClF2N4O2S
    Purity:98.06% - 99.62%
    Color and Shape:Solid
    Molecular weight:456.94
  • MBP146-78

    CAS:
    <p>MBP146-78 is a potent and selective cGMP inhibitor dependent protein kinases.</p>
    Formula:C21H22FN3
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:335.42
  • 3-(Methylthio)propionic acid

    CAS:
    <p>3-(Methylthio)propionic acid forms from D-methionine metabolism. Streptomyces lincolnensis produces it proportionally to methionine levels.</p>
    Formula:C4H8O2S
    Purity:99.63%
    Color and Shape:Solid
    Molecular weight:120.17
  • Tomatidine

    CAS:
    <p>Tomatidine serves as an anti-inflammatory agent by inhibiting NF-κB and JNK signaling pathways.</p>
    Formula:C27H45NO2
    Purity:99.94% - 99.98%
    Color and Shape:Solid
    Molecular weight:415.65
  • β-Elemonic Acid

    CAS:
    <p>β-Elemonic Acid (3-Oxotirucallenoic Acid) exhibits anti-inflammatory effects, which inhibits proliferation by inducing hypoploid cells and cell apoptosis.</p>
    Formula:C30H46O3
    Purity:99.61% - 99.8%
    Color and Shape:Solid
    Molecular weight:454.68
  • Fructo-oligosaccharide DP9/GF8

    CAS:
    <p>Fructo-oligosaccharide DP9/GF8 (Fructo-oligosaccharide DP9 / GF8) belongs to fructooligosaccharides (FOS) with the degree of polymerization (DP=9).</p>
    Formula:C54H92O46
    Purity:98.82% - 99.8%
    Color and Shape:Solid
    Molecular weight:1477.28
  • Sertaconazole

    CAS:
    <p>Sertaconazole is a broad-spectrum antifungal.</p>
    Formula:C20H15Cl3N2OS
    Purity:99.483%
    Color and Shape:Solid
    Molecular weight:437.77
  • Pitstop 2

    CAS:
    <p>Pitstop2 is an amphipathic protein-bound inhibitor of the clathrin terminal domain. Pitstop2 has antitumor activity. Cost-effective, quality assurance.</p>
    Formula:C20H13BrN2O3S2
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:473.36