Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,746 products)
- Apoptosis(6,181 products)
- Cell Cycle/Checkpoint(4,806 products)
- Chromatin/Epigenetics(2,567 products)
- Cytoskeletal Signaling(1,498 products)
- DNA Damage/DNA Repair(2,897 products)
- Endocrinology/Hormones(3,701 products)
- Enzyme(3,671 products)
- GPCR/G-Protein(8,960 products)
- Immunology and Inflammation(3,692 products)
- Influenza Virus(296 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,244 products)
- Membrane Transporter/Ion Channel(3,135 products)
- Metabolism(10,101 products)
- Microbiology/Virology(7,550 products)
- Neuroscience(10,300 products)
- Other Inhibitors(35,772 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,400 products)
- Proteases/Proteasome(1,670 products)
- Stem Cell and Derivatives(742 products)
- Tyrosine Kinase/Adaptors(1,922 products)
- Ubiquitination(1,715 products)
Show 16 more subcategories
Found 66578 products of "Inhibitors"
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CDC25B-IN-1
CAS:CDC25B-IN-1 is an inhibitor of CDC25B with a Ki of 8.5 μM. CDC25B-IN-1 increases the G2/M phase by inhibiting cell proliferation and colony formation.Formula:C20H19NO3Purity:97.05%Color and Shape:SolidMolecular weight:321.37Ref: TM-T10723
1mg72.00€5mg161.00€10mg245.00€25mg405.00€50mg572.00€100mg772.00€1mL*10mM (DMSO)126.00€R-932348 choline
CAS:R-932348 choline, a dual JAK/SYK inhibitor, is used potentially for treatment of dry eye disease.Formula:C28H35FN6O5SPurity:98%Color and Shape:SolidMolecular weight:586.68Alprenolol hydrochloride, (S)-
CAS:Alprenolol hydrochloride, (S)- is a nonselective β-blocker. It is also a serotonin 5HT1A receptor antagonist.Formula:C15H24ClNO2Color and Shape:SolidMolecular weight:285.81Antileishmanial agent-11
CAS:Antileishmanial agent-11: Potent against L. brazilensis (28.3 μM), L. infantum (24.8 μM), T. cruzi (13.0 μM) with strong antiprotozoal efficacy.Formula:C27H24ClN3O4Color and Shape:SolidMolecular weight:489.95Phenglutarimid
CAS:Phenglutarimid is an anticholinergic. It is used as an antiparkinsonian agent.Formula:C17H24N2O2Purity:98%Color and Shape:SolidMolecular weight:288.38Ocaphane Hydrochloride
CAS:Ocaphane Hydrochloride is a strong antitumor agent used on a number of animal tumors.Formula:C14H22Cl4N2O2Purity:98%Color and Shape:SolidMolecular weight:392.14GNE-1858
CAS:GNE-1858 inhibits HPK1; IC50: 1.9 nM for wild-type, 1.9 nM (HPK1-TSEE), 4.5 nM (HPK1-SA).Formula:C21H26F2N8Purity:99.36%Color and Shape:SolidMolecular weight:428.48Ref: TM-T11438
1mg163.00€5mg334.00€10mg500.00€25mg807.00€50mg1,099.00€100mg1,485.00€500mg2,962.00€1mL*10mM (DMSO)358.00€Braco-19 trihydrochloride
CAS:BRACO19 3HCl inhibits telomerase, blocking its capping function, and prevents HAdV viral replication.Formula:C35H46Cl3N7O2Purity:98.74%Color and Shape:SolidMolecular weight:703.1415-OxoETE
CAS:15-OxoETE is produced by oxidation of the 15-hydroxyl of 15-HETE. Whether this is a major pathway of 15-HETE metabolism is yet to be clearly established.Formula:C20H30O3Color and Shape:SolidMolecular weight:318.45Pozanicline
CAS:Pozanicline, a selective α4β2 nAChR partial agonist (Ki=16 nM), may treat nicotine addiction by reversing cognitive deficits.Formula:C11H16N2OPurity:98%Color and Shape:SolidMolecular weight:192.26Caspase-3/7 activator 2
Caspase-3/7 activator 2 triggers apoptosis with tumor selectivity and anti-proliferative properties.Formula:C32H34N2O7Color and Shape:SolidMolecular weight:558.62TRβ agonist 2
CAS:TRβ agonist 2 (Compound 1) is a highly potent agonist of TRβ.Formula:C22H27NO4Color and Shape:SolidMolecular weight:369.45(S)-Carvedilol
CAS:(S)-Carvedilol is a non-selective β/α-1 blocker.It exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).Formula:C24H26N2O4Purity:98%Color and Shape:Less Crystalline Solid Colourless Crystalline SolidMolecular weight:406.47DL-AP5 Sodium salt
CAS:DL-AP5 Sodium salt is a NMDA receptor antagonist.Formula:C5H12NNaO5PPurity:98%Color and Shape:SolidMolecular weight:220.12NCX-278
CAS:NCX-278 is a ROCK inhibitor and NO-donating anti-glaucoma agent.Formula:C14H21N3O9S3Color and Shape:SolidMolecular weight:471.53SRI-37240
CAS:SRI-37240 suppresses CFTR nonsense mutations, aids in fixing premature termination codons, works with G418.Formula:C24H23N3O2Purity:98.73%Color and Shape:SolidMolecular weight:385.46RO-61-3662
CAS:RO-61-3662 is a bioactive chemical.Formula:C14H13NO3Color and Shape:SolidMolecular weight:243.26Z36
CAS:Z36, a Bcl-xL inhibitor, boosts FAM134B/LC3/Atg9, inducing autophagy, cell death, ER stress, and UPR.Formula:C23H24FN3O2Color and Shape:SolidMolecular weight:393.45LY 186826
CAS:LY 186826 is an antibacterial agent with bicyclic pyrazolidinone properties.Formula:C15H16N6O6SPurity:98%Color and Shape:SolidMolecular weight:408.39NSC-70220
CAS:SOS1-IN-1 is an inhibitor of SOS1.Formula:C22H15NO2Purity:98%Color and Shape:SolidMolecular weight:325.36RIPK1-IN-12
CAS:RIPK1-IN-12: Strong RIPK1 blocker, hinders necroptosis; EC50=1.6 nM (human), 2.9 nM (mouse).Formula:C24H26N4O3SColor and Shape:SolidMolecular weight:450.55FGFR2-IN-1
CAS:FGFR2-IN-1 is an FGFR inhibitor that inhibits FGFR1, FGFR2, and FGFR3, and can be used to study FGFR2-associated cancers.Formula:C22H19N3O2Purity:98.71%Color and Shape:SolidMolecular weight:357.41Org-13011 fumarate
CAS:Org-13011 fumarate1 is an agonist of the 5-HT1A receptor and can be used to study neurological disorders.Formula:C22H29F3N4O5Purity:98.92%Color and Shape:SolidMolecular weight:486.48ST101036
CAS:MC activators have recently been described as safe and effective vaccine adjuvants. ST101036 exhibited high degranulation potency in both human and mouse MCs.Formula:C18H21F3N4Color and Shape:SolidMolecular weight:350.38Dolutegravir SR Isomer
CAS:Dolutegravir SR Isomer, a potent HIV-1 inhibitor derivative, blocks virus replication in blood cells.Formula:C20H19F2N3O5Color and Shape:SolidMolecular weight:419.38S07-2001
CAS:S07-2001 boosts Doxorubicin's effect on cancer, targeting AKR1C3 with IC50 of 2.08 μM, may overcome drug resistance.Formula:C15H17N3O4SColor and Shape:SolidMolecular weight:335.38P2X7-IN-2
CAS:P2X7-IN-2 is a P2X7 receptor blocker, halts IL-Iβ release (IC50: 0.01 nM), researched for autoimmunity and heart issues.Formula:C22H21F4N3O2Color and Shape:SolidMolecular weight:435.41Caroxazone
CAS:Caroxazone is an antidepressant drug, monoamine oxidase inhibitor (MAOI) that is irreversible and nonselective meanwhile.Formula:C10H10N2O3Color and Shape:SolidMolecular weight:206.2LY 219057
CAS:LY 219057 is a potent, competitive, and specific antagonist of CCK receptor on the exocrine pancreas.Formula:C23H17ClF3N3OSColor and Shape:SolidMolecular weight:475.91CGS8216
CAS:CGS8216 shows analgesic activity at high doses, has anxiolytic activity, and can be used to study immune system disorders.Formula:C16H11N3OPurity:98.53%Color and Shape:SolidMolecular weight:261.28SYK-IN-II
CAS:SYK-IN-II is an inhibitor of the spleen tyrosine kinase (STK).Formula:C21H27FN6Color and Shape:SolidMolecular weight:382.48PD-85639
CAS:PD-85639 blocks Na+ channels in rat brain neurons (75% at 10 min, >95% at 25 min). Binds Nav1.2 with dual-affinity; competes with anesthetics and activators.Formula:C24H32N2OColor and Shape:SolidMolecular weight:364.52AChE/HDAC-IN-1
CAS:COX-2-IN-23 (A10) inhibits AChE & HDAC (IC50s: 0.12 & 0.23 nM), has antioxidant/metal-binding traits, and is used in Alzheimer's research.Formula:C26H27ClN4O3Color and Shape:SolidMolecular weight:478.97Glyoxalase I inhibitor 7
CAS:Glyoxalase I inhibitor 7 (Compound 6) is a potent inhibitor of glyoxalase I (Glo-I) with an IC50 of 3.65 μM. It exhibits potential as an anticancer agent [1].Formula:C17H16N4O3SColor and Shape:SolidMolecular weight:356.4VT103
CAS:VT103, an oral TEAD1 palmitoylation inhibitor, shows promise against various cancers by disrupting YAP/TAZ-TEAD interactions.Formula:C18H17F3N4O2SPurity:99.58%Color and Shape:SolidMolecular weight:410.41Ref: TM-T62077
1mg112.00€5mg268.00€10mg424.00€25mg735.00€50mg1,071.00€100mg1,549.00€200mg2,097.00€1mL*10mM (DMSO)295.00€JAK-IN-20
CAS:JAK-IN-20: potent oral JAK1,2,3 inhibitor with IC50s 7, 5, 14 nM respectively, good pharmacokinetics, anti-inflammatory in vivo.Formula:C28H30FN7O2Color and Shape:SolidMolecular weight:515.58KRAS inhibitor-17
CAS:KRAS inhibitor-17 blocks G12C mutation (IC50: 3.37μM) and p-ERK in MIA PaCA-2 (IC50: 9.25μM). Could target pancreatic, colorectal, lung cancers.Formula:C21H18Cl2FN3O2SColor and Shape:SolidMolecular weight:466.36SSTR4 agonist 3
CAS:SSTR4 agonist 3 activates SSTR4 in the hippocampus and neocortex, aiding memory and learning, and shows potent pain relief in rodents.Formula:C18H24N4OSColor and Shape:SolidMolecular weight:344.47EMD 66684
CAS:angiotensin AT1 receptor antagonistFormula:C28H31ClN8O2Purity:98%Color and Shape:SolidMolecular weight:547.06Ivacaftor-D9
CAS:CTP-656, a cystic fibrosis transmembrane conductance regulator (CFTR) channel activator, is used potentially for the treatment of cystic fibrosis.Formula:C24H19D9N2O3Color and Shape:SolidMolecular weight:401.55Cyclamidomycin
CAS:Cyclamidomycin is an antibiotic. It also functions as an inhibitor of nucleoside diphosphokinase of Escherichia coli.Formula:C7H10N2OColor and Shape:SolidMolecular weight:138.17Urease-IN-4
Urease-IN-4 inhibits urease (IC50: 1.64 µM), targets P. vulgaris (IC50: 15.27 µg/mL), and is low in cytotoxicity.Formula:C16H20N2O3SColor and Shape:SolidMolecular weight:320.41Vintoperol
CAS:Vintoperol, a calcium channel antagonist, is used potentially for the treatment of arterial occlusive disease and peripheral artery disease.Formula:C18H24N2OColor and Shape:SolidMolecular weight:284.44991W93
CAS:4991W93 is a 5HT(1B/1D) agonist that blocks neurogenic inflammation and inhibits CGRP release.Formula:C18H23N3O2Color and Shape:SolidMolecular weight:313.39Aminomenthylnorepinephrine
CAS:Aminomenthylnorepinephrine is a partial agonist of the beta-adrenoreceptor that causes irreversible inactivation.Formula:C18H30N2O3Color and Shape:SolidMolecular weight:322.44Epocholeone
CAS:Epocholeone is a growth regulator and can be used for the control of fungal or physiological diseases of crops.Formula:C35H56O7Color and Shape:SolidMolecular weight:588.81XMD-12
CAS:XMD-12, also known as DUN57447, Aurora inhibitor (compound 1) or Aurora-IN-1, is an Auroro inhibitor, which targets Aurora A/B/C. (5.6/18.4/24.6 nM).Formula:C24H26N6O2Color and Shape:SolidMolecular weight:430.5RORγt agonist 1
CAS:RORγt agonist 1 is a potent, orally bioavailable agonist of RORγt(EC50 of 20.8 nM).Formula:C24H17F6NO5SPurity:98%Color and Shape:SolidMolecular weight:545.45CEP-40125
CAS:CEP-40125 (RXDX-107) is a DNA alkylating agent for the study of advanced solid tumors.Formula:C28H45Cl2N3O2Purity:98.28%Color and Shape:SolidMolecular weight:526.58CP-101537
CAS:CP-101537 is a MMP inhibitor.Formula:C10H18N2O2Color and Shape:SolidMolecular weight:198.26
