Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,833 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,875 products)
- Chromatin/Epigenetics(2,612 products)
- Cytoskeletal Signaling(1,566 products)
- DNA Damage/DNA Repair(2,872 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,014 products)
- Immunology and Inflammation(3,901 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,256 products)
- Membrane Transporter/Ion Channel(3,154 products)
- Metabolism(10,139 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,377 products)
- Other Inhibitors(35,852 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,430 products)
- Proteases/Proteasome(1,691 products)
- Stem Cell and Derivatives(733 products)
- Tyrosine Kinase/Adaptors(1,983 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66522 products of "Inhibitors"
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L-AP4 monohydrate
CAS:L-AP4 (L-APB) is a group III mGluR agonist with EC50s: 0.13μM (mGlu4), 0.29μM (mGlu8), 1.0μM (mGlu6), 249μM (mGlu7).Formula:C4H12NO6PColor and Shape:SolidMolecular weight:201.115Milfasartan
CAS:Milfasartan: Potent AT1 antagonist, oral, effectively reduces blood pressure in hypertensive rats.Formula:C30H30N6O3SColor and Shape:SolidMolecular weight:554.66VPC03090
CAS:VPC03090 inhibits S1P receptors, is a FTY-720 analog, antagonizes S1PR1/S1PR3, reduces mouse mammary tumors, with a 30-hour oral bioavailability.Formula:C19H31NOColor and Shape:SolidMolecular weight:289.46Delequamine HCl
CAS:Delequamine HCl: potent, selective alpha 2-adrenoceptor blocker; pKi 9.45 in rat cortex, pA2 9.72 in guinea-pig ileum.Formula:C18H27ClN2O3SColor and Shape:SolidMolecular weight:386.94hGGPPS-IN-2
CAS:hGGPPS-IN-2, a C2-ThP-BP analogue, inhibits hGGPPS, targets MM cells, induces apoptosis, and has anti-myeloma effects.Formula:C20H18FN5O7P2SColor and Shape:SolidMolecular weight:553.4Kadsurenone
CAS:Kadsurenone, from haifenteng, blocks PAF/PTAFR pathway, promising for breast cancer bone metastases treatment.Formula:C21H24O5Color and Shape:SolidMolecular weight:356.41AJG-049 free base
CAS:AJG-049 free base is a calcium channel antagonist that inhibits L-type Ca2+ channels via diltiazem-binding site(s).Formula:C27H30N2O2Color and Shape:SolidMolecular weight:414.54Antimicrobial agent-6
Antimicrobial agent-6: MIC 4-8 μg/mL for gram+ & gram- bacteria, anti-inflammatory.Formula:C40H64N16Color and Shape:SolidMolecular weight:769.04PT4
CAS:PT4: treats CL, disrupts parasite mitochondria, kills Leishmania spp., IC50- L. amazonensis 125.18 μM, L. braziliensis 233.18 μM, anti-inflammatory.Formula:C18H14N4O2Color and Shape:SolidMolecular weight:318.33PI3K-IN-36
CAS:PI3K-IN-36 is a potent inhibitor of PI3K, suitable for research applications in follicular lymphoma (FL).Formula:C30H36F2N8OColor and Shape:SolidMolecular weight:562.66Flupirtine HCl
CAS:Flupirtine HCl, non-opioid central analgesic sold as Katadolon/others since 1984, opens potassium channels, modulates NMDA/GABAA receptors.Formula:C15H18ClFN4O2Color and Shape:SolidMolecular weight:340.78hCAXII-IN-3
CAS:hCAXII-IN-3 (Compound 6o) is a selective inhibitor of human carbonic anhydrase XII (hCAXII) (Ki: 10.0 nM).Formula:C26H20BrN5O3SColor and Shape:SolidMolecular weight:562.445-Hydroxylansoprazole sulfone
CAS:5-hydroxylansoprazole is an in vitro metabolism-dependent CYP2C19 inhibitor.Formula:C16H14F3N3O4SColor and Shape:SolidMolecular weight:401.36NSC-18725
CAS:NSC-18725 is a novel inhibitor of growth of intracellular Mycobacterium tuberculosis, inducing autophagy in differentiated THP-1 macrophages.Formula:C11H11N3OColor and Shape:SolidMolecular weight:201.22Anticancer agent 92
Anticancer agent 92 is an anticancer agent that is nontoxic against noncancerous cells .Formula:C21H23ClN4O3SColor and Shape:SolidMolecular weight:446.95ASP9133
CAS:ASP9133, a LAMA, selectively inhibits bronchoconstriction with a faster action than tiotropium.Formula:C18H21BrClN3O2SColor and Shape:SolidMolecular weight:458.8Methylsilanol ascorbate
CAS:Methylsilanol ascorbate is a silanol analogue and inhibitor of angiotensin-converting enzyme.Formula:C7H12O8SiColor and Shape:SolidMolecular weight:252.25PR-104
CAS:PR-104: hypoxia-activated DNA cross-linker, pre-prodrug for nitrogen mustard, converts to PR-104A in tumors.Formula:C14H20BrN4O12PSColor and Shape:SolidMolecular weight:579.27SHP2/HDAC-IN-1
CAS:SHP2/HDAC-IN-1: dual SHP2/HDAC inhibitor, IC50: 20.4 nM/25.3 nM, boosts antitumor immunity, aids cancer immunotherapy research.Formula:C34H35Cl2N7O3Color and Shape:SolidMolecular weight:660.59mGAT3/4-IN-1
CAS:mGAT3/4-IN-1 inhibits mGAT3/4 with pIC50: 5.31/5.24, reduces neuropathic pain in diabetic mice.Formula:C26H31ClN2O2S2Color and Shape:SolidMolecular weight:503.12MLKL-IN-5
CAS:MLKL-IN-5 is a potent MLKL inhibitor that mediates necroptosis .Formula:C18H20N6O4SColor and Shape:SolidMolecular weight:416.45pUL89 Endonuclease-IN-1
CAS:Compound 13d: potent pUL89 endonuclease inhibitor, IC50 0.88 μM, anti-HCMV activity.Formula:C10H8N2O4SColor and Shape:SolidMolecular weight:252.25PAPD5-IN-1
CAS:GNE-9278 is an NMDA receptor positive allosteric modulator. It acts via the transmembrane domain.Formula:C21H27N5O3SColor and Shape:SolidMolecular weight:429.54Pifoxime
CAS:Pifoxime: a NSAID with COX-1/2 inhibition, used in anti-inflammatory treatment and neuropsychiatric studies.Formula:C15H20N2O3Color and Shape:SolidMolecular weight:276.33AM404
CAS:AM404 is a cannabinoid reuptake inhibitor and a TRPV (1) activator with neuroprotective and anticancer activities that blocks anandamide transport.Formula:C26H37NO2Color and Shape:SolidMolecular weight:395.58STOCK2S-26016
CAS:WNK-IN-B, a cell-permeable diaminoacridine, selectively inhibits WNK signaling in mpkDCT/MOVAS by targeting SPAK/OSR1 CCT domain.Formula:C20H19N3O2Color and Shape:SolidMolecular weight:333.38Aspaminol
CAS:Aspaminol is a smooth muscle relaxant.Formula:C21H27NOColor and Shape:SolidMolecular weight:309.45Dexamethasone oxetanone
CAS:Dex-Ox, a selective glucocorticoid derivative of Dex, exhibits antiglucocorticoid and antiprogestin activities, targeting PR A/B isoforms.Formula:C22H27FO4Color and Shape:SolidMolecular weight:374.45BHF-177
CAS:BHF-177 is a positive allosteric modulator of the GABAB receptor. BHF-177 reduces self-administration of nicotine in animal studies.Formula:C19H20F3N3Color and Shape:SolidMolecular weight:347.38SARS-CoV-2 Mpro-IN-5
SARS-CoV-2 Mpro-IN-5: inhibits Mpro (IC50=1800nM) & CatL (IC50=145nM), antiviral, hinders replication in hACE2 A549 cells (IC50=14.7nM).Formula:C34H43FN4O7Color and Shape:SolidMolecular weight:638.73R78206
CAS:R 78206 is a pyridazinamine derivative that suppresses the formation of poliovirus eclipse particles.Formula:C22H29N3O3Purity:98%Color and Shape:SolidMolecular weight:383.48Arnolol
CAS:Arnolol, a beta blocker, slows heart rate, reduces force of beats, lowers blood pressure, and enhances blood flow.Formula:C14H23NO3Color and Shape:SolidMolecular weight:253.34MSD-D
CAS:MSD-D is an inhibitor of voltage-gated K(+) (Kv) channels Kv1.5.Formula:C20H17N3O2SColor and Shape:SolidMolecular weight:363.43Reverse transcriptase-IN-4
Reverse transcriptase-IN-4: potent, selective NNRT inhibitor; EC50 = 0.053 μM for HIV-1, 0.26 μM for E138K mutant.Formula:C17H21N5OSColor and Shape:SolidMolecular weight:343.45MRGPRX4 modulator-1
CAS:MRGPRX4 modulator-1 (compound 31-2), potent MRGPR X4 antagonist, IC50 < 100nM, for itch, pain, autoimmune research.Formula:C16H13ClF3NO3Color and Shape:SolidMolecular weight:359.73NVP018
CAS:NVP018 (BC 556) inhibits HBV, HCV, HIV-1 replication, barely affects drug transporters, and resists HCV/HIV-1 resistance development.Formula:C45H62FN5O11Color and Shape:SolidMolecular weight:868CEP-6800
CAS:CEP-6800: potent PARP inhibitor, potential anticancer, may enhance various chemotherapies.Formula:C18H15N3O2Color and Shape:SolidMolecular weight:305.33CYP3A4-IN-1
CAS:CYP3A4-IN-1 is a potent inhibitor of cytochrome P450 3A4 (CYP3A4) (IC50: 0.085 μM).Formula:C31H37N5O3SColor and Shape:SolidMolecular weight:559.72Mtb-cyt-bd oxidase-IN-4
Mtb-cyt-bd oxidase inhibitor; IC50=0.25μM; MIC=8μM against Mycobacterium tuberculosis; for TB research.Formula:C25H32FNOColor and Shape:SolidMolecular weight:381.53Sphaerobioside
CAS:Sphaerobioside is a useful organic compound for research related to life sciences. The catalog number is T125786 and the CAS number is 14988-20-6.Formula:C27H30O14Color and Shape:SolidMolecular weight:578.523Ruzotolimod
CAS:Ruzotolimod, an agonist of TLR7, exhibits promising potential for investigating HBV, COVID-19, and SARS-CoV-2 infections （WO2021130195A1）[1].Formula:C14H18N4O5SColor and Shape:SolidMolecular weight:354.38GW2433
CAS:GW2433 is an agonist of PPAR receptor.Formula:C28H28Cl3FN2O4Color and Shape:SolidMolecular weight:581.89FLT3/ITD-IN-3
CAS:FLT3/ITD-IN-3 (Compound 19) is a potent FLT3-ITD inhibitor with IC50 values: FLT3D835Y (0.3 nM), FLT3 (0.4 nM), inhibits AML cell proliferation.Formula:C22H26ClN7O2Color and Shape:SolidMolecular weight:455.94(R)-Bambuterol
CAS:Bambuterol is a β2-agonist prodrug for asthma and COPD, taken daily, with a good safety profile and reduces plasma LDL-C and cholesterol.Formula:C18H29N3O5Color and Shape:SolidMolecular weight:367.44Anti-Trypanosoma cruzi agent-4
CAS:Anti-Trypanosoma cruzi Agent-4 is a Trypanosoma cruzi inhibitor utilized for the investigation of infections caused by this parasite.Formula:C17H16N2O3Color and Shape:SolidMolecular weight:296.32Antileishmanial agent-9
CAS:Compound 16c: potent anti-Leishmania agent, IC50=4.01 μM, low toxicity in L-6 cells, IC50=40.1 μM.Formula:C23H26O4Color and Shape:SolidMolecular weight:366.45Enpp-1-IN-6
CAS:Enpp-1-IN-6, a potent enpp-1 inhibitor, may aid cancer and infectious disease studies (WO2021203772A1, compound 51).Formula:C22H28N4O5SColor and Shape:SolidMolecular weight:460.55Rho-Kinase-IN-2
CAS:Rho-Kinase-IN-2, an oral ROCK inhibitor (IC50=3nM), penetrates the CNS; potential in Huntington's research.Formula:C20H25FN4O2Color and Shape:SolidMolecular weight:372.44Pipradimadol
CAS:Pipradimadol is a 4,4-disubstituted piperidine derivative with antidepressive and serotonin antagonistic activity.Formula:C24H37ClN2O2Color and Shape:SolidMolecular weight:421.02Acetabuton
CAS:Acetabuton is an alpha-adrenergic blocker and a hemodynamic and sympathetic drug.Formula:C24H29FN2O2Color and Shape:SolidMolecular weight:396.5
