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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66669 products of "Inhibitors"

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  • SR 142948

    CAS:
    SR 142948 is a neurotensin (NT) receptor antagonist.
    Formula:C39H51N5O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:685.85
  • Mutant IDH1-IN-2

    CAS:
    Mutant IDH1-IN-2 is a inhibitor of mutant Isocitrate dehydrogenase (IDH) proteins, with IC50 of 16.6 nM in Fluorescence biochemical assay, IC50 of <22 nM in LS-
    Formula:C24H31F2N5O2
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:459.53
  • Lumateperone

    CAS:
    <p>Lumateperone (ITI 722) is a 5HT2A receptor antagonist and a dopamine receptor phosphoprotein modulator (DPPM).</p>
    Formula:C24H28FN3O
    Purity:99.68% - 99.91%
    Color and Shape:Solid
    Molecular weight:393.5
  • Y06137

    CAS:
    <p>Y06137, selective BET inhibitor, Kd 81 nM for BRD4(1), researched for castration-resistant prostate cancer treatment.</p>
    Formula:C27H32N4O2
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:444.57
  • AMG2850

    CAS:
    AMG2850 is a potent, orally bioavailable, and selective antagonist of transient receptor potential melastatin 8 (TRPM8).
    Formula:C19H17F6N3O
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:417.35
  • CeMMEC1

    CAS:
    CeMMEC1 is an inhibitor of BRD4, and also has a great affinity for TAF1(IC50=0.9 μM).
    Formula:C19H16N2O4
    Purity:98.9% - 99.92%
    Color and Shape:Solid
    Molecular weight:336.34
  • VBY-825

    CAS:
    VBY-825 is a reversible inhibitor of cathepsin with high potency against cathepsins B, L, S and V.
    Formula:C23H29F4N3O5S
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:535.55
  • PKC-IN-1

    CAS:
    PKC-IN-1 is an ATP-competitive and reversible conventional PKC enzymes inhibitor (PKCα, PKCβI, PKCβII, PKCθ, PKCγ, PKC mu and PKCε with IC50s of 2.3, 8.1, 7.6,
    Formula:C25H37FN8O2
    Purity:98% - 98.79%
    Color and Shape:Solid
    Molecular weight:500.61
  • Src Inhibitor 3

    CAS:
    Src Inhibitor 3 blocks c-Src kinase (IC50 <3 nM CSK HTRF, <4 nM Caliper), boosting T cell growth from receptor signals.
    Formula:C34H32ClFN8O4
    Purity:98.35%
    Color and Shape:Solid
    Molecular weight:671.12
  • SB-616234-A

    CAS:
    SB-616234-A is a selective and orally bioavailable antagonist of 5-HT1B receptor, with anxiolytic and antidepressant activity.
    Formula:C32H36ClN5O3
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:574.11
  • AZ-23

    CAS:
    AZ-23 is an inhibitor of ATP-competitive and Trk kinase A/B/C.
    Formula:C17H19ClFN7O
    Purity:99.4%
    Color and Shape:Solid
    Molecular weight:391.83
  • PXS-5120A

    CAS:
    PXS-5120A is an irreversible fluoroallylamine Lysyl Oxidase-like 2/3 (LOXL2/3) inhibitor with anti-fibrotic activity.
    Formula:C22H25ClFN3O4S
    Purity:97.02%
    Color and Shape:Solid
    Molecular weight:481.97
  • PKI-402

    CAS:
    PKI-402 is a potent PI3K and mTOR inhibitor. PKI-402 inhibits PI3Kα, mTOR, PI3Kβ, PI3Kδ and PI3Kγ with IC50s of 2, 3, 7, 14 and 16 nM, respectively.
    Formula:C29H34N10O3
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:570.65
  • PF-04979064

    CAS:
    <p>PF-04979064 is a potent and selective PI3K and mTOR dual kinase inhibitor(Ki of 0.13 nM and 1.42 nM,respectively).</p>
    Formula:C24H26N6O3
    Purity:98.20% - ≥98%
    Color and Shape:Solid
    Molecular weight:446.5
  • HM43239

    CAS:
    HM43239: oral FLT3 inhibitor; IC50: FLT3 WT 1.1nM, ITD 1.8nM, D835Y 1.0nM; blocks p-STAT5/p-ERK; affects SYK, JAK1/2, TAK1; halts leukemia cell growth.
    Formula:C29H33ClN6
    Purity:99.7%
    Color and Shape:Solid
    Molecular weight:501.07
  • GSK-3 inhibitor 1

    CAS:
    GSK-3 inhibitor 1 is a GSK-3 inhibitor.
    Formula:C22H17ClFN5O2
    Purity:98.42%
    Color and Shape:Solid
    Molecular weight:437.85
  • Lomibuvir

    CAS:
    Lomibuvir (VCH-222, VX-222) is an allosteric inhibitor of HCV NS5B with Kd 17 nM, blocks RNA elongation, EC50 5.2 nM for 1b/Con1.
    Formula:C25H35NO4S
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:445.61
  • GSK-F1

    CAS:
    GSK-F1 (PI4KA inhibitor-F1) is a novel potent PI4KA inhibitor.
    Formula:C27H18F5N5O4S
    Purity:97.03%
    Color and Shape:Solid
    Molecular weight:603.52
  • EGFR-IN-8

    CAS:
    <p>EGFR-IN-8, a dual inhibitor targeting both EGFR and c-Met, shows potential as a promising candidate for further development in treating EGFR TKI-resistant NSCLC</p>
    Formula:C32H23ClF3N7O4
    Purity:99.51%
    Color and Shape:Solid
    Molecular weight:662.02
  • GDC-0349

    CAS:
    <p>GDC-0349 (RG-7603) is a potent and selective ATP-competitive inhibitor of mTOR, 790-fold inhibitory effect against PI3Kα and other 266 kinases. Phase 1.</p>
    Formula:C24H32N6O3
    Purity:96.00% - 98.17%
    Color and Shape:Solid
    Molecular weight:452.55