Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,939 products)
- Apoptosis(6,643 products)
- Cell Cycle/Checkpoint(4,917 products)
- Chromatin/Epigenetics(2,633 products)
- Cytoskeletal Signaling(1,595 products)
- DNA Damage/DNA Repair(2,868 products)
- Endocrinology/Hormones(3,765 products)
- Enzyme(3,675 products)
- GPCR/G-Protein(9,484 products)
- Immunology and Inflammation(3,958 products)
- Influenza Virus(301 products)
- JAK/STAT signaling(417 products)
- MAPK Signaling(1,272 products)
- Membrane Transporter/Ion Channel(3,404 products)
- Metabolism(10,179 products)
- Microbiology/Virology(7,953 products)
- Neuroscience(11,146 products)
- Other Inhibitors(35,858 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,439 products)
- Proteases/Proteasome(1,692 products)
- Stem Cell and Derivatives(733 products)
- Tyrosine Kinase/Adaptors(1,992 products)
- Ubiquitination(1,745 products)
Show 16 more subcategories
Found 66510 products of "Inhibitors"
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GKA50 quarterhydrate
GKA50 quarterhydrate: glucokinase activator, EC50 of 33 nM, boosts insulin, cuts glucose in rats.Formula:C26H30N2O7Color and Shape:SolidMolecular weight:469.01Top/HDAC-IN-2
Top/HDAC-IN-2 (45b) is a dual inhibitor of Top and HDAC that induces apoptosis and exhibits significant anti-tumour effects.Formula:C30H32N8O4Color and Shape:SolidMolecular weight:568.63AMG-548 dihydrochloride
AMG-548 dihydrochloride, an oral p38α inhibitor (Ki: 0.5 nM), selectively targets p38β, γ, δ, inhibits TNFα (IC50: 3 nM), and suppresses Wnt signaling.Formula:C29H29Cl2N5OColor and Shape:SolidMolecular weight:534.488-Deazafolic acid
CAS:8-Deazafolic acid inhibits folate-dependent bacteria S. faecium & L. casei, and fights lymphoid leukemia L1210 in mice.Formula:C20H20N6O6Purity:98%Color and Shape:SolidMolecular weight:440.41Anti-inflammatory agent 19
Anti-inflammatory agent 19: NO inhibitor (IC50: 36μM), blocks HMGB1, for late-stage inflammation, relevant for COVID-19, sepsis.Formula:C30H50O7Color and Shape:SolidMolecular weight:522.71MGAT2-IN-1
CAS:MGAT2-IN-1 is an orally active monoacylglycerol acyltransferase (MGAT2)inhibitor (human and mouse MGAT2 with IC50 of 7.8 and 2.4 nM , respectively).Formula:C27H21ClF5N7O3SColor and Shape:SolidMolecular weight:654.01GSK3527497
CAS:GSK3527497 is a novel potent and selective inhibitor of transient receptor potential vanilloid-4 (TRPV4).Formula:C17H16ClFN4O4SColor and Shape:SolidMolecular weight:426.85AS2521780
CAS:AS2521780 is an inhibitor of PKCθ (IC50: 0.48 nM).Formula:C30H41N7OSPurity:98%Color and Shape:SolidMolecular weight:547.76Dyrk1A/α-synuclein-IN-2
Dyrk1A/α-synuclein-IN-2 (Compound b20) is a dual inhibitor of Dyrk1A and α-synuclein aggregation that acts on α-synuclein (IC50: 7.8 μM).Formula:C21H16N4O4SColor and Shape:SolidMolecular weight:420.44Lometrexol disodium
CAS:Lometrexol disodium: Inhibits hSHMT1/2 and GARFT, anticancer by blocking purine synthesis, induces apoptosis and cell cycle arrest.Formula:C21H23N5Na2O6Color and Shape:SolidMolecular weight:487.424Detajmium
CAS:Detajmium is an anti-arrhythmia compound. It is an Na(+)-channel-blocking drug with an extremely long recovery from use-dependent sodium channel block.Formula:C27H42N3O3Purity:98%Color and Shape:SolidMolecular weight:456.64Antibacterial agent 70
Antibacterial agent 70 is a new dihydropyrimidinone-imidazole hybrid antimicrobial agent (MIC: 0.5 μg/ml).Formula:C25H32ClN7O6SColor and Shape:SolidMolecular weight:594.08PROTAC CDK12/13 Degrader-1
PROTAC CDK12/13 Degrader-1 (7f) selectively degrades CDK12/13 at nanomolar potency, targeting breast cancer.Color and Shape:SolidAM-9514
CAS:AM-9514: a potent Glucokinase activator with strong in vitro results, good pharmacokinetics, and efficacy in diabetes.Formula:C18H25N5O4Color and Shape:SolidMolecular weight:375.42LEO 134310
CAS:LEO 134310: Selective, non-steroidal GR agonist with 14 nM EC50, for topical skin disease treatment.Formula:C34H40N2O8Color and Shape:SolidMolecular weight:604.69Mu opioid receptor antagonist 3
Potent, selective MOR antagonist (compound 26); crosses blood-brain barrier. Ki: 0.24 nM, EC50: 0.54 nM; for studying OUD.Formula:C25H28N2O4SColor and Shape:SolidMolecular weight:452.57MtTMPK-IN-2
CAS:MtTMPK-IN-2 inhibits M. tuberculosis TMPK (IC50: 1.1 μM), Mtb H37Rv (MIC: 12.5 μM), and is cytotoxic in MRC-5 cells (EC50: 6.1 μM).Formula:C23H24ClN3O3Color and Shape:SolidMolecular weight:425.91AMPK Activator SC4
CAS:SC4 is a potent, direct AMPK activator. SC4 preferentially activates α2 complexes and stimulates skeletal muscle glucose uptake.Formula:C26H18ClN3O4Color and Shape:SolidMolecular weight:471.89Indinavir monohydrate
CAS:Indinavir monohydrate is a potent and specific HIV protease inhibitor that appears to have good oral bioavailability.Formula:C36H49N5O5Color and Shape:SolidMolecular weight:631.82sEH inhibitor-4
Compound B15: potent sEH inhibitor (0.03 nm), reduces inflammation & pain.Formula:C27H28Cl2N4O3Color and Shape:SolidMolecular weight:527.44
