Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
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Subcategories of "Inhibitors"
Angiogenesis
Apoptosis
Cell Cycle/Checkpoint
Chromatin/Epigenetics
Cytoskeletal Signaling
DNA Damage/DNA Repair
Endocrinology/Hormones
Enzyme
GPCR/G-Protein
Immunology and Inflammation
Influenza Virus
JAK/STAT signaling
MAPK Signaling
Membrane Transporter/Ion Channel
Metabolism
Microbiology/Virology
Neuroscience
Other Inhibitors
Oxidation-Reduction
PI3K/Akt/mTOR Signaling
Proteases/Proteasome
Stem Cell and Derivatives
Tyrosine Kinase/Adaptors
Ubiquitination
Show 16 more subcategories
Products of "Inhibitors"
PSB 1115
CAS:152529-79-8
PSB 1115 is an A2B receptor antagonist and can counteract the inhibitory effect of NECA.
Formula:
C14H14N4O5S
Purity:
100% - 99.24%
Color and Shape:
Solid
Molecular weight:
350.35
Ref: TM-T23201
| 1mg | 66.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Tuesday 28 Jan 2025
MDR-1339
CAS:1018946-38-7
MDR-1339 is a blood-brain-barrier-permeable inhibitor of amyloid-β (Aβ) aggregation.
Formula:
C20H22O4
Purity:
98.57%
Color and Shape:
Solid
Molecular weight:
326.39
Ref: TM-TQ0026
| 1mg | 58.00 € | ||
| 5mg | 122.00 € | ||
| 10mg | 182.00 € | ||
| 25mg | 365.00 € | ||
| 50mg | 551.00 € | ||
| 100mg | 828.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
INCB3344
CAS:1262238-11-8
INCB3344 is an effective, specific and orally bioavailable CCR2 antagonist with IC50 values of 9.5 …
Formula:
C29H34F3N3O6
Purity:
98.00% - 98.2%
Color and Shape:
Solid
Molecular weight:
577.59
Ref: TM-TQ0103
| 1mg | 69.00 € | ||
| 5mg | 150.00 € | ||
| 10mg | 237.00 € | ||
| 25mg | 402.00 € | ||
| 50mg | 596.00 € | ||
| 100mg | 852.00 € | ||
| 1mL*10mM (DMSO) | 187.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
AMG 837 calcium hydrate
CAS:1259389-38-2
AMG 837 calcium hydrate is a potent GPR40 agonist with an EC50 of 13 nM.
Formula:
C52H44CaF6O8
Purity:
98.07%
Color and Shape:
Solid
Molecular weight:
950.97
Ref: TM-TQ0020
| 2mg | 36.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 145.00 € | ||
| 50mg | 282.00 € | ||
| 100mg | 400.00 € | ||
| 200mg | 547.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
SB-616234-A
CAS:908601-49-0
SB-616234-A is a selective and orally bioavailable antagonist of 5-HT1B receptor, with anxiolytic and antidepressant …
Formula:
C32H36ClN5O3
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
574.11
Ref: TM-T12847
| 1mg | 103.00 € | ||
| 5mg | 248.00 € | ||
| 10mg | 358.00 € | ||
| 25mg | 542.00 € | ||
| 50mg | 732.00 € | ||
| 100mg | 1,007.00 € | ||
| 200mg | 1,358.00 € | ||
| 1mL*10mM (DMSO) | 313.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
CAY10781
CAS:1210360-87-4
CAY10781 inhibits NRP-1/VEGF-A binding by 43% at 12.5μM and blocks VEGFR2 phosphorylation in CAD cells.
Formula:
C11H9N3O3
Purity:
98.69%
Color and Shape:
Solid
Molecular weight:
231.21
Ref: TM-T37424
| 2mg | 41.00 € | ||
| 5mg | 55.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 174.00 € | ||
| 100mg | 322.00 € | ||
| 200mg | 451.00 € | ||
| 1mL*10mM (DMSO) | 81.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
GSK-F1
CAS:1402345-92-9
GSK-F1 (PI4KA inhibitor-F1) is a novel potent PI4KA inhibitor.
Formula:
C27H18F5N5O4S
Purity:
95.5%
Color and Shape:
Solid
Molecular weight:
603.52
Ref: TM-T19840
| 1mg | 106.00 € | ||
| 5mg | 218.00 € | ||
| 10mg | 323.00 € | ||
| 25mg | 519.00 € | ||
| 50mg | 703.00 € | ||
| 100mg | 903.00 € | ||
| 200mg | 1,272.00 € | ||
| 1mL*10mM (DMSO) | 309.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
HM43239
CAS:2294874-49-8
HM43239: oral FLT3 inhibitor; IC50: FLT3 WT 1.1nM, ITD 1.8nM, D835Y 1.0nM; blocks p-STAT5/p-ERK; affects …
Formula:
C29H33ClN6
Purity:
98.56%
Color and Shape:
Solid
Molecular weight:
501.07
Ref: TM-T9428
| 1mg | 69.00 € | ||
| 5mg | 150.00 € | ||
| 10mg | 221.00 € | ||
| 25mg | 434.00 € | ||
| 50mg | 620.00 € | ||
| 100mg | 862.00 € | ||
| 1mL*10mM (DMSO) | 186.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Pan-RAS-IN-1
CAS:1835283-94-7
Pan-RAS-IN-1 is an inhibitor of pan-Ras. It disrupts the interaction of Ras proteins and their …
Formula:
C36H41Cl2F3N6O2
Purity:
98.57%
Color and Shape:
Solid
Molecular weight:
717.65
Ref: TM-T16432
| 1mg | 80.00 € | ||
| 2mg | 96.00 € | ||
| 5mg | 144.00 € | ||
| 10mg | 215.00 € | ||
| 25mg | 437.00 € | ||
| 50mg | 655.00 € | ||
| 100mg | 931.00 € | ||
| 500mg | 1,866.00 € | ||
| 1mL*10mM (DMSO) | 220.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
VBY-825
CAS:1310340-58-9
VBY-825 is a reversible inhibitor of cathepsin with high potency against cathepsins B, L, S …
Formula:
C23H29F4N3O5S
Purity:
98.99%
Color and Shape:
Solid
Molecular weight:
535.55
Ref: TM-T13288
| 1mg | 260.00 € | ||
| 2mg | 384.00 € | ||
| 5mg | 644.00 € | ||
| 10mg | 915.00 € | ||
| 25mg | 1,356.00 € | ||
| 50mg | 1,821.00 € | ||
| 100mg | 2,476.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
BMS-986176
CAS:1815613-42-3
AAK1-IN-1 is a highly selective and potent inhibitor of adaptor associated kinase 1 (AAK1, IC50 …
Formula:
C19H23F4N3O
Purity:
98.6%
Color and Shape:
Solid
Molecular weight:
385.4
Ref: TM-T35856
| 1mg | 169.00 € | ||
| 5mg | 346.00 € | ||
| 10mg | 519.00 € | ||
| 25mg | 832.00 € | ||
| 50mg | 1,133.00 € | ||
| 100mg | 1,532.00 € | ||
| 500mg | 5,761.00 € | ||
| 1mL*10mM (DMSO) | 375.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
PKI-402
CAS:1173204-81-3
PKI-402 is a potent PI3K and mTOR inhibitor. PKI-402 inhibits PI3Kα, mTOR, PI3Kβ, PI3Kδ and …
Formula:
C29H34N10O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
570.65
Ref: TM-T3656
| 1mg | 35.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 221.00 € | ||
| 50mg | 328.00 € | ||
| 100mg | 460.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
EGFR-IN-8
CAS:2407957-87-1
EGFR-IN-8, a dual inhibitor targeting both EGFR and c-Met, shows potential as a promising candidate …
Formula:
C32H23ClF3N7O4
Purity:
97.45%
Color and Shape:
Solid
Molecular weight:
662.02
Ref: TM-T11162
| 1mg | 74.00 € | ||
| 5mg | 166.00 € | ||
| 10mg | 266.00 € | ||
| 25mg | 440.00 € | ||
| 50mg | 602.00 € | ||
| 100mg | 825.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Mutant IDH1-IN-2
CAS:1429176-69-1
Mutant IDH1-IN-2 is a inhibitor of mutant Isocitrate dehydrogenase (IDH) proteins, with IC50 of 16.6 …
Formula:
C24H31F2N5O2
Purity:
99.11%
Color and Shape:
Solid
Molecular weight:
459.53
Ref: TM-T12128
| 1mg | 62.00 € | ||
| 5mg | 141.00 € | ||
| 10mg | 228.00 € | ||
| 25mg | 381.00 € | ||
| 50mg | 542.00 € | ||
| 100mg | 732.00 € | ||
| 200mg | 982.00 € | ||
| 1mL*10mM (DMSO) | 140.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
AMG2850
CAS:1470018-52-0
AMG2850 is a potent, orally bioavailable, and selective antagonist of transient receptor potential melastatin 8 …
Formula:
C19H17F6N3O
Purity:
99.05%
Color and Shape:
Solid
Molecular weight:
417.35
Ref: TM-T10300
| 1mg | 72.00 € | ||
| 5mg | 164.00 € | ||
| 10mg | 239.00 € | ||
| 25mg | 430.00 € | ||
| 50mg | 638.00 € | ||
| 100mg | 818.00 € | ||
| 1mL*10mM (DMSO) | 175.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
SR 142948
CAS:184162-64-9
SR 142948 is a neurotensin (NT) receptor antagonist.
Formula:
C39H51N5O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
685.85
Ref: TM-T23386
| 10mg | 878.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Y06137
CAS:2226534-49-0
Y06137, selective BET inhibitor, Kd 81 nM for BRD4(1), researched for castration-resistant prostate cancer treatment.
Formula:
C27H32N4O2
Purity:
97.27%
Color and Shape:
Solid
Molecular weight:
444.57
Ref: TM-T13363
| 1mg | 60.00 € | ||
| 2mg | 86.00 € | ||
| 5mg | 126.00 € | ||
| 10mg | 201.00 € | ||
| 25mg | 374.00 € | ||
| 1mL*10mM (DMSO) | 140.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
PXS-5153A
CAS:2125956-82-1
PXS-5153A rapidly inhibits lysyl oxidase 2/3 enzymes, blocks activity in 15 mins, and reduces fibrosis.
Formula:
C20H25Cl2FN4O2S
Purity:
99.71%
Color and Shape:
Solid
Molecular weight:
475.41
Ref: TM-T12585
| 1mg | 182.00 € | ||
| 5mg | 406.00 € | ||
| 10mg | 603.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
MK-8353
CAS:1184173-73-6
MK-8353 (SCH900353) is a potent, selective and orally available inhibitor of ERK1/2 (IC50s of 23.0 …
Formula:
C37H41N9O3S
Purity:
96.15% - 99.89%
Color and Shape:
Solid
Molecular weight:
691.84
Ref: TM-T12069
| 1mg | 79.00 € | ||
| 5mg | 153.00 € | ||
| 10mg | 268.00 € | ||
| 25mg | 451.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 229.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
DN02
DN02: a potent, selective BRD8(1) bromodomain probe; Ki=32 nM; 30x more affine than BRD8(2).
Formula:
C22H24FN3O3
Purity:
99.11% - 99.42%
Color and Shape:
Solid
Molecular weight:
397.44
Ref: TM-T61874
| 1mg | 145.00 € | ||
| 5mg | 352.00 € | ||
| 10mg | 625.00 € | ||
| 25mg | 1,284.00 € | ||
| 50mg | 1,869.00 € | ||
| 100mg | 2,359.00 € |
Estimated delivery in United States, on Tuesday 11 Feb 2025
